EA201001368A1 - Гетероциклические производные мочевины и способы их применения-211 - Google Patents
Гетероциклические производные мочевины и способы их применения-211Info
- Publication number
- EA201001368A1 EA201001368A1 EA201001368A EA201001368A EA201001368A1 EA 201001368 A1 EA201001368 A1 EA 201001368A1 EA 201001368 A EA201001368 A EA 201001368A EA 201001368 A EA201001368 A EA 201001368A EA 201001368 A1 EA201001368 A1 EA 201001368A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- methods
- application
- urea derivatives
- heterocyclic urea
- heterocyclic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Abstract
Описываются соединения формулы (I) и их фармацевтически приемлемые соли. Также описываются способы их получения, содержащие их фармацевтические композиции, их применение в качестве лекарственных средств и их применение при лечении бактериальных инфекций.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US3162108P | 2008-02-26 | 2008-02-26 | |
PCT/GB2009/050187 WO2009106885A1 (en) | 2008-02-26 | 2009-02-25 | Heterocyclic urea derivatives and methods of use thereof-211 |
Publications (1)
Publication Number | Publication Date |
---|---|
EA201001368A1 true EA201001368A1 (ru) | 2011-04-29 |
Family
ID=40474753
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201001368A EA201001368A1 (ru) | 2008-02-26 | 2009-02-25 | Гетероциклические производные мочевины и способы их применения-211 |
Country Status (23)
Country | Link |
---|---|
US (1) | US20120101100A1 (ru) |
EP (1) | EP2262801A1 (ru) |
JP (1) | JP2011513216A (ru) |
KR (1) | KR20100117681A (ru) |
CN (1) | CN102015699A (ru) |
AR (1) | AR070493A1 (ru) |
AU (1) | AU2009219883A1 (ru) |
BR (1) | BRPI0907562A2 (ru) |
CA (1) | CA2716365A1 (ru) |
CL (1) | CL2009000426A1 (ru) |
CO (1) | CO6290656A2 (ru) |
CR (1) | CR11641A (ru) |
DO (1) | DOP2010000259A (ru) |
EA (1) | EA201001368A1 (ru) |
EC (1) | ECSP10010419A (ru) |
IL (1) | IL207731A0 (ru) |
MX (1) | MX2010009163A (ru) |
PE (1) | PE20091573A1 (ru) |
SA (1) | SA109300138B1 (ru) |
TW (1) | TW200940537A (ru) |
UY (1) | UY31673A1 (ru) |
WO (1) | WO2009106885A1 (ru) |
ZA (1) | ZA201005997B (ru) |
Families Citing this family (64)
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EP2250160B1 (en) | 2008-01-25 | 2015-11-11 | Millennium Pharmaceuticals, Inc. | Thiophenes and their use as phosphatidylinositol 3-kinase (pi3k) inhibitors |
AU2012203026B2 (en) * | 2008-03-21 | 2014-06-12 | Novartis Ag | Novel heterocyclic compounds and uses thereof |
US8865732B2 (en) | 2008-03-21 | 2014-10-21 | Novartis Ag | Heterocyclic compounds and uses thereof |
KR20110014710A (ko) * | 2008-06-04 | 2011-02-11 | 아스트라제네카 아베 | 박테리아 감염의 치료를 위한 헤테로시클릭 우레아 유도체 |
WO2010052448A2 (en) * | 2008-11-05 | 2010-05-14 | Ucb Pharma S.A. | Fused pyrazine derivatives as kinase inhibitors |
CN102264721B (zh) | 2008-11-10 | 2015-12-09 | 沃泰克斯药物股份有限公司 | 用作atr激酶抑制剂的化合物 |
RS56995B1 (sr) | 2008-12-19 | 2018-05-31 | Vertex Pharma | Derivati pirazina korisni kao inhibitori atr kinaze |
CA2750935A1 (en) | 2009-01-30 | 2010-08-12 | Millennium Pharmaceuticals, Inc. | Heteroaryls and their use as pi3k inhibitors |
US9090601B2 (en) * | 2009-01-30 | 2015-07-28 | Millennium Pharmaceuticals, Inc. | Thiazole derivatives |
US8796314B2 (en) | 2009-01-30 | 2014-08-05 | Millennium Pharmaceuticals, Inc. | Heteroaryls and uses thereof |
TW201102065A (en) | 2009-05-29 | 2011-01-16 | Astrazeneca Ab | Heterocyclic urea derivatives and methods of use thereof |
FR2953519B1 (fr) * | 2009-12-08 | 2012-02-10 | Commissariat Energie Atomique | Nouveaux composes chimiques aptes a complexer au moins un element metallique et complexe de coordination a base de ces composes |
US20130096119A1 (en) | 2010-03-31 | 2013-04-18 | Daniel Bur | Isoquinolin-3-Ylurea Derivatives |
AR081626A1 (es) | 2010-04-23 | 2012-10-10 | Cytokinetics Inc | Compuestos amino-piridazinicos, composiciones farmaceuticas que los contienen y uso de los mismos para tratar trastornos musculares cardiacos y esqueleticos |
US9133123B2 (en) | 2010-04-23 | 2015-09-15 | Cytokinetics, Inc. | Certain amino-pyridines and amino-triazines, compositions thereof, and methods for their use |
AR081331A1 (es) | 2010-04-23 | 2012-08-08 | Cytokinetics Inc | Amino- pirimidinas composiciones de las mismas y metodos para el uso de los mismos |
WO2011143423A2 (en) | 2010-05-12 | 2011-11-17 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of atr kinase |
US9334244B2 (en) | 2010-05-12 | 2016-05-10 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of ATR kinase |
SG185524A1 (en) | 2010-05-12 | 2012-12-28 | Vertex Pharma | Compounds useful as inhibitors of atr kinase |
US8969356B2 (en) | 2010-05-12 | 2015-03-03 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of ATR kinase |
WO2011143419A1 (en) | 2010-05-12 | 2011-11-17 | Vertex Pharmaceuticals Incorporated | Pyrazines useful as inhibitors of atr kinase |
CN102947272A (zh) * | 2010-05-12 | 2013-02-27 | 沃泰克斯药物股份有限公司 | 用作atr激酶抑制剂的2-氨基吡啶衍生物 |
MX2013000103A (es) | 2010-06-23 | 2013-06-13 | Vertex Pharma | Derivados de pirrolo-pirazina utiles como inhibidores de cinasa art. |
WO2012021696A1 (en) | 2010-08-11 | 2012-02-16 | Millennium Pharmaceuticals, Inc. | Heteroaryls and uses thereof |
WO2012021611A1 (en) | 2010-08-11 | 2012-02-16 | Millennium Pharmaceuticals, Inc. | Heteroaryls and uses thereof |
WO2012021615A1 (en) | 2010-08-11 | 2012-02-16 | Millennium Pharmaceuticals, Inc. | Heteroaryls and uses thereof |
EP3590925B1 (en) | 2010-09-17 | 2022-03-30 | Purdue Pharma L.P. | Pyridine compounds and the uses thereof |
CN103237450A (zh) | 2010-10-13 | 2013-08-07 | 米伦纽姆医药公司 | 杂芳基化合物和其用途 |
AR088729A1 (es) | 2011-03-29 | 2014-07-02 | Actelion Pharmaceuticals Ltd | Derivados de 3-ureidoisoquinolin-8-ilo y una composicion farmaceutica |
EP2694498B1 (en) | 2011-04-05 | 2016-03-30 | Vertex Pharmaceuticals Incorporated | Aminopyrazine compounds useful as inhibitors of tra kinase |
WO2012178124A1 (en) | 2011-06-22 | 2012-12-27 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of atr kinase |
WO2012178123A1 (en) | 2011-06-22 | 2012-12-27 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of atr kinase |
EP2723746A1 (en) | 2011-06-22 | 2014-04-30 | Vertex Pharmaceuticals Inc. | Compounds useful as inhibitors of atr kinase |
MX2014001860A (es) * | 2011-09-12 | 2014-05-30 | Hoffmann La Roche | Hidrazidas del acido 3-piridin carboxilico como agentes elevadores del colesterol de lipoproteina de alta densidad (hdl). |
WO2013049719A1 (en) | 2011-09-30 | 2013-04-04 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of atr kinase |
US8853217B2 (en) | 2011-09-30 | 2014-10-07 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of ATR kinase |
CN108464983A (zh) | 2011-09-30 | 2018-08-31 | 沃泰克斯药物股份有限公司 | 用atr抑制剂治疗胰腺癌和非小细胞肺癌 |
PT2940017T (pt) | 2011-09-30 | 2019-10-31 | Vertex Pharma | Processos para a produção de compostos úteis como inibidores de atr quinase |
WO2013049722A1 (en) | 2011-09-30 | 2013-04-04 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of atr kinase |
PE20142282A1 (es) * | 2011-11-04 | 2015-01-08 | Hoffmann La Roche | Nuevos derivados de aril-quinolina |
WO2013071088A1 (en) | 2011-11-09 | 2013-05-16 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of atr kinase |
US8846918B2 (en) | 2011-11-09 | 2014-09-30 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of ATR kinase |
US8841337B2 (en) | 2011-11-09 | 2014-09-23 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of ATR kinase |
US8841450B2 (en) | 2011-11-09 | 2014-09-23 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of ATR kinase |
EP2776419B1 (en) | 2011-11-09 | 2016-05-11 | Vertex Pharmaceuticals Incorporated | Pyrazine compounds useful as inhibitors of atr kinase |
CN104125947A (zh) * | 2011-12-21 | 2014-10-29 | 生物区欧洲有限公司 | 杂环脲化合物 |
NZ700580A (en) | 2012-04-05 | 2016-07-29 | Vertex Pharma | Compounds useful as inhibitors of atr kinase and combination therapies thereof |
US9546155B2 (en) | 2012-06-15 | 2017-01-17 | Mitsubishi Tanabe Pharma Corporation | Aromatic heterocyclic compound |
DK2904406T3 (en) | 2012-10-04 | 2018-06-18 | Vertex Pharma | METHOD OF DETERMINING THE ATR INHIBITION, INCREASED DNA DAMAGE |
WO2014062604A1 (en) | 2012-10-16 | 2014-04-24 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of atr kinase |
US9340546B2 (en) | 2012-12-07 | 2016-05-17 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of ATR kinase |
US9242969B2 (en) | 2013-03-14 | 2016-01-26 | Novartis Ag | Biaryl amide compounds as kinase inhibitors |
WO2014143240A1 (en) | 2013-03-15 | 2014-09-18 | Vertex Pharmaceuticals Incorporated | Fused pyrazolopyrimidine derivatives useful as inhibitors of atr kinase |
ES2682040T3 (es) | 2013-09-06 | 2018-09-18 | Aurigene Discovery Technologies Limited | Derivados de 1,3,4-oxadiazol y 1,3,4-tiadiazol como inmunomoduladores |
HUE046727T2 (hu) | 2013-12-06 | 2020-03-30 | Vertex Pharma | Az ATR-kináz inhibitoraként használható vegyület, 2-amino-6-fluoro-N-[5-fluoro-piridin-3-IL]-pirazolo-[1,5-A]-pirimidin-3-karboxamid, ennek elõállítása, különbözõ szilárd formái és ezek radioaktív nyomjelzett származékai |
AU2015271030B2 (en) | 2014-06-05 | 2019-05-16 | Vertex Pharmaceuticals Incorporated | Radiolabelled derivatives of a 2-amino-6-fluoro-n-[5-fluoro-pyridin-3-yl]- pyrazolo [1,5-a] pyrimidin-3-carboxamide compound useful as ATR kinase inhibitor, the preparation of said compound and different solid forms thereof |
PL3157566T3 (pl) | 2014-06-17 | 2019-10-31 | Vertex Pharma | Metoda leczenia nowotworu przy użyciu kombinacji inhibitorów chk1 i atr |
UY36294A (es) | 2014-09-12 | 2016-04-29 | Novartis Ag | Compuestos y composiciones como inhibidores de quinasa |
JP2018507884A (ja) * | 2015-03-10 | 2018-03-22 | オーリジーン ディスカバリー テクノロジーズ リミテッドAurigene Discovery Technologies Limited | 免疫調節剤としての3−置換1,3,4−オキサジアゾールおよびチアジアゾール化合物 |
JP7187308B2 (ja) | 2015-09-30 | 2022-12-12 | バーテックス ファーマシューティカルズ インコーポレイテッド | Dna損傷剤とatr阻害剤との組み合わせを使用する、がんを処置するための方法 |
CN106866571B (zh) * | 2017-01-20 | 2018-06-29 | 中国药科大学 | 杂环脲类化合物及其药物组合物和应用 |
KR20190133667A (ko) | 2017-03-24 | 2019-12-03 | 다이쇼 세이야꾸 가부시끼가이샤 | 2(1h)-퀴놀리논 유도체 |
CN111116559A (zh) * | 2018-11-01 | 2020-05-08 | 复旦大学 | 吡啶脲类化合物及其制备方法和制药用途 |
WO2022147210A1 (en) * | 2020-12-31 | 2022-07-07 | Evrys Bio, Llc | Anti-tumor compositions and methods |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0014022D0 (en) * | 2000-06-08 | 2000-08-02 | Novartis Ag | Organic compounds |
AR042956A1 (es) * | 2003-01-31 | 2005-07-13 | Vertex Pharma | Inhibidores de girasa y usos de los mismos |
US7569591B2 (en) * | 2003-01-31 | 2009-08-04 | Vertex Pharmaceuticals Incorporated | Gyrase inhibitors and uses thereof |
CL2007003470A1 (es) * | 2006-12-04 | 2008-08-22 | Astrazeneca Ab | Compuestos derivados de urea; composicion farmaceutica que comprende a dichos compuestos; y su uso como antibacterianos. |
-
2009
- 2009-02-24 TW TW098105845A patent/TW200940537A/zh unknown
- 2009-02-25 SA SA109300138A patent/SA109300138B1/ar unknown
- 2009-02-25 EA EA201001368A patent/EA201001368A1/ru unknown
- 2009-02-25 JP JP2010547261A patent/JP2011513216A/ja active Pending
- 2009-02-25 KR KR1020107021270A patent/KR20100117681A/ko not_active Application Discontinuation
- 2009-02-25 UY UY031673A patent/UY31673A1/es not_active Application Discontinuation
- 2009-02-25 CL CL2009000426A patent/CL2009000426A1/es unknown
- 2009-02-25 CN CN2009801157676A patent/CN102015699A/zh active Pending
- 2009-02-25 CA CA2716365A patent/CA2716365A1/en not_active Abandoned
- 2009-02-25 AU AU2009219883A patent/AU2009219883A1/en not_active Abandoned
- 2009-02-25 BR BRPI0907562A patent/BRPI0907562A2/pt not_active IP Right Cessation
- 2009-02-25 EP EP09715006A patent/EP2262801A1/en not_active Withdrawn
- 2009-02-25 MX MX2010009163A patent/MX2010009163A/es unknown
- 2009-02-25 WO PCT/GB2009/050187 patent/WO2009106885A1/en active Application Filing
- 2009-02-25 US US12/392,730 patent/US20120101100A1/en not_active Abandoned
- 2009-02-26 AR ARP090100667A patent/AR070493A1/es not_active Application Discontinuation
- 2009-02-26 PE PE2009000289A patent/PE20091573A1/es not_active Application Discontinuation
-
2010
- 2010-08-19 IL IL207731A patent/IL207731A0/en unknown
- 2010-08-23 ZA ZA2010/05997A patent/ZA201005997B/en unknown
- 2010-08-24 DO DO2010000259A patent/DOP2010000259A/es unknown
- 2010-08-24 EC EC2010010419A patent/ECSP10010419A/es unknown
- 2010-08-24 CR CR11641A patent/CR11641A/es not_active Application Discontinuation
- 2010-08-24 CO CO10104182A patent/CO6290656A2/es not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
CL2009000426A1 (es) | 2011-02-11 |
TW200940537A (en) | 2009-10-01 |
PE20091573A1 (es) | 2009-11-12 |
MX2010009163A (es) | 2010-09-14 |
BRPI0907562A2 (pt) | 2017-05-23 |
CA2716365A1 (en) | 2009-09-03 |
DOP2010000259A (es) | 2010-09-15 |
ZA201005997B (en) | 2013-01-30 |
KR20100117681A (ko) | 2010-11-03 |
AU2009219883A1 (en) | 2009-09-03 |
US20120101100A1 (en) | 2012-04-26 |
CR11641A (es) | 2010-10-05 |
SA109300138B1 (ar) | 2012-11-03 |
EP2262801A1 (en) | 2010-12-22 |
CN102015699A (zh) | 2011-04-13 |
AR070493A1 (es) | 2010-04-07 |
IL207731A0 (en) | 2010-12-30 |
CO6290656A2 (es) | 2011-06-20 |
WO2009106885A1 (en) | 2009-09-03 |
UY31673A1 (es) | 2009-09-30 |
JP2011513216A (ja) | 2011-04-28 |
ECSP10010419A (es) | 2010-09-30 |
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