EA200870540A1 - Бензилфенильное глюкопиранозидное производное - Google Patents

Бензилфенильное глюкопиранозидное производное

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Publication number
EA200870540A1
EA200870540A1 EA200870540A EA200870540A EA200870540A1 EA 200870540 A1 EA200870540 A1 EA 200870540A1 EA 200870540 A EA200870540 A EA 200870540A EA 200870540 A EA200870540 A EA 200870540A EA 200870540 A1 EA200870540 A1 EA 200870540A1
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EA
Eurasian Patent Office
Prior art keywords
hydrogen atom
alkyl group
derivative
benzylphenylic
glucopiranoside
Prior art date
Application number
EA200870540A
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English (en)
Inventor
Такеси Хонда
Минору Огути
Масао ЙОСИДА
Рио Окуяма
Цунеаки Огата
Манабу Абе
Кендзиро Уеда
Дзун Осуми
Масанори Изуми
Original Assignee
Дайити Санкио Компани, Лимитед
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Publication date
Application filed by Дайити Санкио Компани, Лимитед filed Critical Дайити Санкио Компани, Лимитед
Publication of EA200870540A1 publication Critical patent/EA200870540A1/ru

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    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07H17/02—Heterocyclic radicals containing only nitrogen as ring hetero atoms

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Abstract

Настоящее изобретение относится к бензилфенилглюкопиранозидному производному, обладающему превосходным ингибирующим эффектом на активности человеческих SGLT1 и/или SGLT2, конкретно к соединению или его фармакологически приемлемой соли, представленным следующей общей формулой (I)где Rпредставляет атом водорода, аминогруппу, гидроксиС-Салкильную группу и т.д.; Rпредставляет атом водорода и т.д.; Rпредставляет C-Салкильную группу, гидроксиС-Салкильную группу и т.д.; Rпредставляет атом водорода, С-Сацильную группу и т.д.; R, R, Rи Rявляются одинаковыми или различными и каждый представляет атом водорода или C-Салкильную группу, при условии, если R, R, Rи Rне являются одновременно атомами водорода; n равно 0-4; и Х представляет СН или N.
EA200870540A 2006-08-04 2007-08-03 Бензилфенильное глюкопиранозидное производное EA200870540A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2006213600 2006-08-04
PCT/JP2007/065231 WO2008016132A1 (en) 2006-08-04 2007-08-03 Benzyl phenyl glucopyranoside derivative

Publications (1)

Publication Number Publication Date
EA200870540A1 true EA200870540A1 (ru) 2009-04-28

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Family Applications (1)

Application Number Title Priority Date Filing Date
EA200870540A EA200870540A1 (ru) 2006-08-04 2007-08-03 Бензилфенильное глюкопиранозидное производное

Country Status (15)

Country Link
US (1) US20090137499A1 (ru)
EP (1) EP2048150A4 (ru)
JP (3) JP4249256B2 (ru)
KR (1) KR20090040250A (ru)
CN (1) CN101472937A (ru)
AU (1) AU2007279616A1 (ru)
BR (1) BRPI0708521A2 (ru)
CA (1) CA2649044A1 (ru)
EA (1) EA200870540A1 (ru)
IL (1) IL194404A0 (ru)
MX (1) MX2008012481A (ru)
NO (1) NO20084127L (ru)
TW (1) TW200817424A (ru)
WO (1) WO2008016132A1 (ru)
ZA (1) ZA200809543B (ru)

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US20090137499A1 (en) 2009-05-28
TW200817424A (en) 2008-04-16
IL194404A0 (en) 2009-08-03
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AU2007279616A1 (en) 2008-02-07
JP4425318B2 (ja) 2010-03-03
JP2009024021A (ja) 2009-02-05
JP4249256B2 (ja) 2009-04-02
JP2009108105A (ja) 2009-05-21
CA2649044A1 (en) 2008-02-07
EP2048150A4 (en) 2011-06-29
ZA200809543B (en) 2010-03-31
NO20084127L (no) 2009-04-30
CN101472937A (zh) 2009-07-01
BRPI0708521A2 (pt) 2011-05-31
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MX2008012481A (es) 2008-10-10
JPWO2008016132A1 (ja) 2009-12-24

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