EA200400597A1 - 5-фенилпиримидины, способ их получения, содержащие их средства и их применение - Google Patents

5-фенилпиримидины, способ их получения, содержащие их средства и их применение

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Publication number
EA200400597A1
EA200400597A1 EA200400597A EA200400597A EA200400597A1 EA 200400597 A1 EA200400597 A1 EA 200400597A1 EA 200400597 A EA200400597 A EA 200400597A EA 200400597 A EA200400597 A EA 200400597A EA 200400597 A1 EA200400597 A1 EA 200400597A1
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EA
Eurasian Patent Office
Prior art keywords
saturated
nrr
crr
nrc
alkylthio
Prior art date
Application number
EA200400597A
Other languages
English (en)
Other versions
EA010628B1 (ru
Inventor
Андреас Гипзер
Томас Гроте
Аня Швёглер
Йоахим Райнхаймер
Франк Шивек
Хорди Тормо И Бласко
Инго Розе
Петер Шэфер
Маркус Гевер
Вассилиос Грамменос
Бернд МЮЛЛЕР
Эберхард Аммерманн
Зигфрид Штратманн
Гизела Лоренц
Райнхард Штирль
Original Assignee
Басф Акциенгезельшафт
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Application filed by Басф Акциенгезельшафт filed Critical Басф Акциенгезельшафт
Publication of EA200400597A1 publication Critical patent/EA200400597A1/ru
Publication of EA010628B1 publication Critical patent/EA010628B1/ru

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/42—One nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52—Two oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

5-Фенилпиримидины формулы Iгде заместители и индекс имеют следующее значение:R, Rозначают водород, алкил, галогеналкил, циклоалкил, галогенциклоалкил, алкенил, галогеналкенил, алкинил или галогеналкинил, Rи Rмогут также вместе с атомом азота, с которым они связаны, образовывать насыщенный или ненасыщенный цикл, который может быть прерван эфиро-, тио-, сульфоксил- или сульфонилгруппой и может быть замещен посредством одной до четырех групп Rи/или R;Rозначает водород, галоген, циано, алкил, галогеналкил, алкокси, галогеналкокси или алкенилокси;Rозначает водород, галоген, циано, гидрокси, меркапто, азидо, алкил, алкенил, алкинил, галогеналкил, алкокси, алкенилокси, алкинилокси, галогеналкокси, алкилтио, алкенилтио, алкинилтио, галогеналкилтио, -ON=CRR, -CR=NOR, -NRN=CRR, -NRR, -NRNRR, -NOR, -NRC(=NR)NRR, -NRC(=O)NRR, -NRC(=O)R, -NRC(=NOR)R', -OC(=O)R, -C(=NOR)NRR, -CR(=NNRR), -C(=O)NRRили -C(=O)R;где R,R,Rимеют приведенное в описании значение, X означает галоген, алкил, алкокси или галогеналкил; и m равно целому числу от 1 до 5.Изобретение относится к методам получения вышеприведенных соединений, агентам, содержащим эти соединения, и применению их для борьбы с фитопатогенными грибами.Международная заявка была опубликована вместе с отчетом о международном поиске.
EA200400597A 2001-11-19 2002-11-15 5-фенилпиримидины, способ их получения, содержащие их средства и их применение EA010628B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10156279 2001-11-19
PCT/EP2002/012807 WO2003043993A1 (de) 2001-11-19 2002-11-15 5-phenylpyrimidine, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung

Publications (2)

Publication Number Publication Date
EA200400597A1 true EA200400597A1 (ru) 2004-12-30
EA010628B1 EA010628B1 (ru) 2008-10-30

Family

ID=7705956

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200400597A EA010628B1 (ru) 2001-11-19 2002-11-15 5-фенилпиримидины, способ их получения, содержащие их средства и их применение

Country Status (17)

Country Link
US (2) US7465735B2 (ru)
EP (1) EP1448532A1 (ru)
JP (1) JP4450625B2 (ru)
KR (1) KR100950632B1 (ru)
CN (1) CN1312134C (ru)
AU (1) AU2002352015B2 (ru)
BR (1) BR0214253A (ru)
CA (1) CA2467683C (ru)
EA (1) EA010628B1 (ru)
HU (1) HUP0402385A3 (ru)
IL (1) IL161893A0 (ru)
MX (1) MXPA04004583A (ru)
NZ (1) NZ533265A (ru)
PL (1) PL371059A1 (ru)
UA (1) UA78255C2 (ru)
WO (1) WO2003043993A1 (ru)
ZA (1) ZA200404835B (ru)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2007502846A (ja) * 2003-05-20 2007-02-15 ビーエーエスエフ　アクチェンゲゼルシャフト ２−置換ピリミジン類
AU2004261373B8 (en) * 2003-07-24 2010-11-04 Basf Se 2-substituted pyrimidines
MXPA06000383A (es) * 2003-07-24 2006-04-05 Basf Ag Pirimidinas 2-sustituidas.
AU2004275733A1 (en) 2003-09-24 2005-04-07 Wyeth Holdings Corporation 5-arylpyrimidines as anticancer agents
JP2005232081A (ja) * 2004-02-19 2005-09-02 Bayer Cropscience Ag ベンジルピリミジン誘導体の農園芸用殺菌剤としての利用
AU2005245580A1 (en) 2004-05-19 2005-12-01 Basf Aktiengesellschaft 2-substituted pyrimidines and their use as pesticides
EP1761516B1 (de) * 2004-06-25 2007-11-28 Basf Aktiengesellschaft 2, 4, 5, 6-substituierte pyridine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen
JP2008505957A (ja) * 2004-07-14 2008-02-28 ビーエーエスエフ　アクチェンゲゼルシャフト ２−置換ピリミジン、その調製方法および有害菌類を防除するためのその使用
TW200637556A (en) 2005-01-31 2006-11-01 Basf Ag Substituted 5-phenyl pyrimidines I in therapy
TW200640881A (en) * 2005-02-15 2006-12-01 Du Pont Fungicidal pyrazine derivatives
DE102005046592A1 (de) * 2005-09-28 2007-03-29 Basf Ag 2-Substituierte Hydroxylaminopyrimidine, Verfahren zu ihrer Herstellung und ihre Verwendung als Pestizid
WO2007054472A1 (de) * 2005-11-11 2007-05-18 Basf Se Verhenkelte pyridin- und pyrimidinderivate, verfahren zu ihrer herstellung und ihre verwendung als pestizid
JP2009532327A (ja) * 2006-02-15 2009-09-10 ビーエーエスエフ ソシエタス・ヨーロピア ２−置換ピリミジン誘導体
AR060140A1 (es) * 2006-03-27 2008-05-28 Basf Ag 5-heteroaril-4-aminopirimidinas sustituidas
CL2007002231A1 (es) * 2006-08-02 2008-04-11 Basf Ag Uso de compuestos derivados de 5-(het) arilpirimidina para combatir hongos daninos; compuestos derivados de 5-(het) arilpirimidina; agente fungicida; y agente farmaceutico.
WO2008107398A2 (en) * 2007-03-02 2008-09-12 Basf Se Pyrazine compounds
US8981111B2 (en) * 2008-04-22 2015-03-17 Bayer Cropscience Ag Fungicide hydroximoyl-heterocycles derivatives
MA33932B1 (fr) * 2009-12-17 2013-01-02 Dow Agrosciences Llc Dérivés de 2-aldoximino-5-fluoropyrimidine
MX2012014304A (es) 2010-06-07 2013-05-30 Dow Agrosciences Llc Carboxamidas de pirazinilo como fungicidas.
EP2595965B1 (en) * 2010-07-20 2016-06-22 Vestaron Corporation Insecticidal triazines and pyrimidines

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US3919229A (en) * 1973-07-19 1975-11-11 Labaz Pyrimidine derivatives and process for preparing the same
DE3620841A1 (de) * 1986-06-21 1987-12-23 Basf Ag 4-aminopyrimidinderivate
DE3901084A1 (de) 1988-07-28 1990-02-01 Bayer Ag Substituierte 4-sulfonylamino-2-azinyl-1,2,4-triazol-3-one, verfahren sowie zwischenprodukte zu ihrer herstellung und ihre verwendung als herbizide
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JPH02200678A (ja) * 1989-01-28 1990-08-08 Kumiai Chem Ind Co Ltd ２―ヨードプロパルギルオキシピリミジン誘導体及び農園芸用殺菌剤
DE3922735A1 (de) 1989-07-11 1991-01-24 Hoechst Ag Aminopyrimidin-derivate, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung als fungizide
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Also Published As

Publication number Publication date
CA2467683C (en) 2011-09-27
US20060148764A1 (en) 2006-07-06
EP1448532A1 (de) 2004-08-25
WO2003043993A1 (de) 2003-05-30
HUP0402385A3 (en) 2005-10-28
AU2002352015A1 (en) 2003-06-10
MXPA04004583A (es) 2004-08-13
US20070149551A1 (en) 2007-06-28
HUP0402385A2 (hu) 2005-03-29
EA010628B1 (ru) 2008-10-30
NZ533265A (en) 2006-05-26
CN1606547A (zh) 2005-04-13
AU2002352015B2 (en) 2008-07-31
JP2005514363A (ja) 2005-05-19
JP4450625B2 (ja) 2010-04-14
CA2467683A1 (en) 2003-05-30
CN1312134C (zh) 2007-04-25
IL161893A0 (en) 2005-11-20
BR0214253A (pt) 2004-12-14
KR100950632B1 (ko) 2010-04-01
US7449471B2 (en) 2008-11-11
PL371059A1 (en) 2005-06-13
KR20040079901A (ko) 2004-09-16
UA78255C2 (en) 2007-03-15
US7465735B2 (en) 2008-12-16
ZA200404835B (en) 2005-06-20

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