EA017170B1 - Модуляторы рецептора св1 - Google Patents
Модуляторы рецептора св1 Download PDFInfo
- Publication number
- EA017170B1 EA017170B1 EA200900838A EA200900838A EA017170B1 EA 017170 B1 EA017170 B1 EA 017170B1 EA 200900838 A EA200900838 A EA 200900838A EA 200900838 A EA200900838 A EA 200900838A EA 017170 B1 EA017170 B1 EA 017170B1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- chlorophenyl
- hydrogen
- pyrazole
- ethyl
- methyl
- Prior art date
Links
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Classifications
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Landscapes
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- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Endocrinology (AREA)
- Psychiatry (AREA)
- Emergency Medicine (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Addiction (AREA)
- Child & Adolescent Psychology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Gastroenterology & Hepatology (AREA)
- Reproductive Health (AREA)
- Nutrition Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0625197A GB0625197D0 (en) | 2006-12-18 | 2006-12-18 | Cannabinoid receptor modulators |
| GB0717998A GB0717998D0 (en) | 2007-09-14 | 2007-09-14 | Canabinoid receptor modulators |
| PCT/GB2007/004831 WO2008075012A1 (en) | 2006-12-18 | 2007-12-17 | Cb1 receptor modulators |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| EA200900838A1 EA200900838A1 (ru) | 2010-02-26 |
| EA017170B1 true EA017170B1 (ru) | 2012-10-30 |
Family
ID=39156232
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EA200900838A EA017170B1 (ru) | 2006-12-18 | 2007-12-17 | Модуляторы рецептора св1 |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US8148404B2 (enExample) |
| EP (2) | EP2121659B1 (enExample) |
| JP (2) | JP5222855B2 (enExample) |
| CN (1) | CN103145620A (enExample) |
| AU (2) | AU2007336068B2 (enExample) |
| BR (1) | BRPI0720732A2 (enExample) |
| CA (2) | CA2673359A1 (enExample) |
| EA (1) | EA017170B1 (enExample) |
| IL (2) | IL198990A0 (enExample) |
| MX (1) | MX2009006214A (enExample) |
| NZ (1) | NZ578063A (enExample) |
| WO (3) | WO2008075019A1 (enExample) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7923465B2 (en) | 2005-06-02 | 2011-04-12 | Glenmark Pharmaceuticals S.A. | Cannabinoid receptor ligands, pharmaceutical compositions containing them, and process for their preparation |
| US7977358B2 (en) | 2007-07-26 | 2011-07-12 | Hoffmann-La Roche Inc. | Pyrazol derivatives |
| WO2009074782A1 (en) | 2007-12-10 | 2009-06-18 | 7Tm Pharma A/S | Cannabinoid receptor modulators |
| GB0813142D0 (en) | 2008-07-17 | 2008-08-27 | Glaxo Group Ltd | Novel compounds |
| GB0813144D0 (en) | 2008-07-17 | 2008-08-27 | Glaxo Group Ltd | Novel compounds |
| US10022263B2 (en) | 2011-07-14 | 2018-07-17 | Cook Medical Technologies Llc | Sling-based treatment of obstructive sleep apnea |
| US9710644B2 (en) | 2012-02-01 | 2017-07-18 | Servicenow, Inc. | Techniques for sharing network security event information |
| JO3215B1 (ar) | 2012-08-09 | 2018-03-08 | Phenex Pharmaceuticals Ag | حلقات غير متجانسة بها 5 ذرات تحتوي على النيتروجين بها استبدال بكربوكساميد أو سلفوناميد كمعدلات لمستقبل نووي غير محمي RORy |
| WO2014189540A1 (en) | 2012-10-16 | 2014-11-27 | Catalano Peter J | Method and apparatus for treating obstructive sleep apnea (osa) |
| CA2919504A1 (en) | 2013-08-01 | 2015-02-05 | Christine BRONIKOWSKI | Tissue adjustment implant |
| JP6364078B2 (ja) | 2013-08-05 | 2018-07-25 | クック・メディカル・テクノロジーズ・リミテッド・ライアビリティ・カンパニーＣｏｏｋ Ｍｅｄｉｃａｌ Ｔｅｃｈｎｏｌｏｇｉｅｓ Ｌｌｃ | 解放可能なチューブ状部材を有する医療機器およびその使用方法 |
| EP2898920B1 (en) | 2014-01-24 | 2018-06-06 | Cook Medical Technologies LLC | Articulating balloon catheter |
| US9974563B2 (en) | 2014-05-28 | 2018-05-22 | Cook Medical Technologies Llc | Medical devices having a releasable member and methods of using the same |
| US9913661B2 (en) | 2014-08-04 | 2018-03-13 | Cook Medical Technologies Llc | Medical devices having a releasable tubular member and methods of using the same |
| CN111093572A (zh) | 2017-06-29 | 2020-05-01 | 库克医学技术有限责任公司 | 用于重新定位组织的可植入医疗装置 |
| KR102880573B1 (ko) * | 2018-08-20 | 2025-11-04 | 베서, 파마 엘엘씨 | 칸나비노이드의 생성 공정 |
| CA3166630A1 (en) | 2020-01-03 | 2021-07-08 | Berg Llc | Polycyclic amides as ube2k modulators for treating cancer |
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| US20040192667A1 (en) * | 2001-08-31 | 2004-09-30 | University Of Connecticut | Novel pyrazole analogs acting on cannabinoid receptors |
| WO2004099157A1 (en) * | 2003-05-07 | 2004-11-18 | Pfizer Products Inc. | Cannabinoid receptor ligands and uses thereof |
| WO2005080343A2 (en) * | 2004-02-20 | 2005-09-01 | Astrazeneca Ab | 3-substituted 1,5-diphenylpyrazole derivatives useful as cb1 modulators |
| WO2006133926A1 (en) * | 2005-06-17 | 2006-12-21 | Carex Sa | Pyrazole derivates as cannabinoid receptor modulators |
| US20070213302A1 (en) * | 2006-03-10 | 2007-09-13 | Jenrin Discovery | Cannabinoid receptor antagonists/inverse agonists useful for treating obesity |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2692575B1 (fr) * | 1992-06-23 | 1995-06-30 | Sanofi Elf | Nouveaux derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant. |
| FR2741621B1 (fr) | 1995-11-23 | 1998-02-13 | Sanofi Sa | Nouveaux derives de pyrazole, procede pour leur preparation et compositions pharmaceutiques en contenant |
| FR2742148B1 (fr) | 1995-12-08 | 1999-10-22 | Sanofi Sa | Nouveaux derives du pyrazole-3-carboxamide, procede pour leur preparation et compositions pharmaceutiques les contenant |
| FR2789079B3 (fr) | 1999-02-01 | 2001-03-02 | Sanofi Synthelabo | Derive d'acide pyrazolecarboxylique, sa preparation, les compositions pharmaceutiques en contenant |
| CA2387892A1 (en) | 1999-10-18 | 2001-04-26 | University Of Connecticut | Pyrazole derivatives as cannabinoid receptor antagonists |
| EP1254115A2 (en) | 2000-02-11 | 2002-11-06 | Bristol-Myers Squibb Company | Cannabinoid receptor modulators, their processes of preparation, and use of cannabinoid receptor modulators for treating respiratory and non-respiratory diseases |
| HUP0204519A3 (en) * | 2000-03-23 | 2003-07-28 | Solvay Pharm Bv | 4,5-dihydro-1h-pyrazole derivatives having cb1-antagonistic activity, pharmaceutical compositions containing them and process for their preparations |
| JP4104983B2 (ja) * | 2001-02-28 | 2008-06-18 | メルク エンド カムパニー インコーポレーテッド | メラノコルチン−４受容体作動薬としてのアシル化ピペリジン誘導体 |
| JP2005507875A (ja) | 2001-08-31 | 2005-03-24 | ユニバーシティ オブ コネチカット | カンナビノイド受容体に作用する新規なピラゾール類似体 |
| FR2831883B1 (fr) * | 2001-11-08 | 2004-07-23 | Sanofi Synthelabo | Forme polymorphe du rimonabant, son procede de preparation et les compositions pharmaceutiques en contenant |
| US6825209B2 (en) * | 2002-04-15 | 2004-11-30 | Research Triangle Institute | Compounds having unique CB1 receptor binding selectivity and methods for their production and use |
| NZ540515A (en) * | 2002-12-02 | 2008-01-31 | Astellas Pharma Inc | Pyrazole derivatives useful as COX-I inhibitors |
| US7247628B2 (en) | 2002-12-12 | 2007-07-24 | Pfizer, Inc. | Cannabinoid receptor ligands and uses thereof |
| FR2856683A1 (fr) * | 2003-06-25 | 2004-12-31 | Sanofi Synthelabo | Derives de 4-cyanopyrazole-3-carboxamide, leur preparation et leur application en therapeutique |
| FR2867685B1 (fr) * | 2004-03-17 | 2008-05-23 | Sanofi Synthelabo | Utilisation d'un derive du pyrazole, pour la preparation de medicaments utiles dans la prevention et le traitement de la bronchite chronique et de la broncho-pneumopathie chronique obstructive |
| WO2006067443A1 (en) | 2004-12-23 | 2006-06-29 | Astrazeneca Ab | Therapeutic agents |
-
2007
- 2007-12-17 CA CA002673359A patent/CA2673359A1/en not_active Abandoned
- 2007-12-17 NZ NZ578063A patent/NZ578063A/en not_active IP Right Cessation
- 2007-12-17 CA CA002673177A patent/CA2673177A1/en not_active Abandoned
- 2007-12-17 EP EP07848579.4A patent/EP2121659B1/en not_active Not-in-force
- 2007-12-17 US US12/518,446 patent/US8148404B2/en not_active Expired - Fee Related
- 2007-12-17 WO PCT/GB2007/004842 patent/WO2008075019A1/en not_active Ceased
- 2007-12-17 JP JP2009542200A patent/JP5222855B2/ja not_active Expired - Fee Related
- 2007-12-17 WO PCT/GB2007/004831 patent/WO2008075012A1/en not_active Ceased
- 2007-12-17 CN CN2012103916453A patent/CN103145620A/zh active Pending
- 2007-12-17 EA EA200900838A patent/EA017170B1/ru not_active IP Right Cessation
- 2007-12-17 US US12/519,432 patent/US8124634B2/en not_active Expired - Fee Related
- 2007-12-17 WO PCT/GB2007/004835 patent/WO2008075013A1/en not_active Ceased
- 2007-12-17 JP JP2009542195A patent/JP5437812B2/ja not_active Expired - Fee Related
- 2007-12-17 BR BRPI0720732-8A patent/BRPI0720732A2/pt not_active IP Right Cessation
- 2007-12-17 AU AU2007336068A patent/AU2007336068B2/en not_active Ceased
- 2007-12-17 AU AU2007336061A patent/AU2007336061B2/en not_active Ceased
- 2007-12-17 MX MX2009006214A patent/MX2009006214A/es active IP Right Grant
- 2007-12-17 EP EP07848570.3A patent/EP2121617B1/en not_active Not-in-force
-
2009
- 2009-05-27 IL IL198990A patent/IL198990A0/en unknown
- 2009-05-27 IL IL198989A patent/IL198989A0/en unknown
Patent Citations (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0477049A1 (fr) * | 1990-08-20 | 1992-03-25 | Sanofi | Dérivés d'amido-3 pyrazole, procédé pour leur préparation et compositions pharmaceutiques les contenant |
| US20040192667A1 (en) * | 2001-08-31 | 2004-09-30 | University Of Connecticut | Novel pyrazole analogs acting on cannabinoid receptors |
| WO2004099157A1 (en) * | 2003-05-07 | 2004-11-18 | Pfizer Products Inc. | Cannabinoid receptor ligands and uses thereof |
| WO2005080343A2 (en) * | 2004-02-20 | 2005-09-01 | Astrazeneca Ab | 3-substituted 1,5-diphenylpyrazole derivatives useful as cb1 modulators |
| WO2006133926A1 (en) * | 2005-06-17 | 2006-12-21 | Carex Sa | Pyrazole derivates as cannabinoid receptor modulators |
| US20070213302A1 (en) * | 2006-03-10 | 2007-09-13 | Jenrin Discovery | Cannabinoid receptor antagonists/inverse agonists useful for treating obesity |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2008075019A1 (en) | 2008-06-26 |
| AU2007336061A1 (en) | 2008-06-26 |
| JP2010513435A (ja) | 2010-04-30 |
| WO2008075012A1 (en) | 2008-06-26 |
| US20100144701A1 (en) | 2010-06-10 |
| BRPI0720732A2 (pt) | 2014-04-08 |
| EP2121659B1 (en) | 2013-05-15 |
| AU2007336068B2 (en) | 2013-05-02 |
| EA200900838A1 (ru) | 2010-02-26 |
| EP2121617B1 (en) | 2014-01-22 |
| JP5222855B2 (ja) | 2013-06-26 |
| US8124634B2 (en) | 2012-02-28 |
| NZ578063A (en) | 2011-09-30 |
| JP2010513438A (ja) | 2010-04-30 |
| JP5437812B2 (ja) | 2014-03-12 |
| WO2008075013A1 (en) | 2008-06-26 |
| CN103145620A (zh) | 2013-06-12 |
| MX2009006214A (es) | 2009-06-22 |
| CA2673359A1 (en) | 2008-06-26 |
| CA2673177A1 (en) | 2008-06-26 |
| AU2007336061B2 (en) | 2013-06-27 |
| IL198990A0 (en) | 2010-02-17 |
| AU2007336068A1 (en) | 2008-06-26 |
| EP2121659A1 (en) | 2009-11-25 |
| IL198989A0 (en) | 2010-02-17 |
| US20100010061A1 (en) | 2010-01-14 |
| EP2121617A1 (en) | 2009-11-25 |
| US8148404B2 (en) | 2012-04-03 |
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| MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AM AZ BY KZ KG MD TJ TM RU |