DK97884A - 1,3-bis(1h-1,2,4-triazol-1-yl)-1-fluor-propan-2-ol-forb. og farmaceutisk og landbrugsmaessigt acceptable salte deraf, fremg. til fremst. deraf, farmaceutiske praeparater og fungicider indeh. disse forb. og fremg. til behand. af planter eller froe, som har en svampeinfektion - Google Patents

1,3-bis(1h-1,2,4-triazol-1-yl)-1-fluor-propan-2-ol-forb. og farmaceutisk og landbrugsmaessigt acceptable salte deraf, fremg. til fremst. deraf, farmaceutiske praeparater og fungicider indeh. disse forb. og fremg. til behand. af planter eller froe, som har en svampeinfektion

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Publication number
DK97884A
DK97884A DK97884A DK97884A DK97884A DK 97884 A DK97884 A DK 97884A DK 97884 A DK97884 A DK 97884A DK 97884 A DK97884 A DK 97884A DK 97884 A DK97884 A DK 97884A
Authority
DK
Denmark
Prior art keywords
pharmaceutical
indeh
forb
forever
triazol
Prior art date
Application number
DK97884A
Other languages
English (en)
Other versions
DK97884D0 (da
DK160823B (da
DK160823C (da
Inventor
Kenneth Richardson
Geoffrey Edward Gymer
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DK97884D0 publication Critical patent/DK97884D0/da
Publication of DK97884A publication Critical patent/DK97884A/da
Publication of DK160823B publication Critical patent/DK160823B/da
Application granted granted Critical
Publication of DK160823C publication Critical patent/DK160823C/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/45—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by condensation
    • C07C45/46—Friedel-Crafts reactions
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/63—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by introduction of halogen; by substitution of halogen atoms by other halogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK097884A 1983-02-25 1984-02-24 1,3-bis(1h-1,2,4-triazol-1-yl)-1-fluorpropan-2-ol-forbindelser, farmaceutiske praeparater og landbrugs fungicider indeholdende forbindelserne og fremgangsmaade til behandling af planter eller froe, som har en svampeinfektion DK160823C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB838305377A GB8305377D0 (en) 1983-02-25 1983-02-25 Antifungal agents
GB8305377 1983-02-25

Publications (4)

Publication Number Publication Date
DK97884D0 DK97884D0 (da) 1984-02-24
DK97884A true DK97884A (da) 1984-08-26
DK160823B DK160823B (da) 1991-04-22
DK160823C DK160823C (da) 1991-10-07

Family

ID=10538659

Family Applications (2)

Application Number Title Priority Date Filing Date
DK097884A DK160823C (da) 1983-02-25 1984-02-24 1,3-bis(1h-1,2,4-triazol-1-yl)-1-fluorpropan-2-ol-forbindelser, farmaceutiske praeparater og landbrugs fungicider indeholdende forbindelserne og fremgangsmaade til behandling af planter eller froe, som har en svampeinfektion
DK369889A DK171233B1 (da) 1983-02-25 1989-07-27 1-Fluor-1-(1H-1,2,4-triazol-1-yl)-2-(oxo eller methylen)ethanforbindelser

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK369889A DK171233B1 (da) 1983-02-25 1989-07-27 1-Fluor-1-(1H-1,2,4-triazol-1-yl)-2-(oxo eller methylen)ethanforbindelser

Country Status (28)

Country Link
US (1) US4960782A (da)
EP (1) EP0118245B1 (da)
JP (1) JPS59193877A (da)
KR (1) KR870000356B1 (da)
AU (1) AU545660B2 (da)
CA (1) CA1257276A (da)
CS (1) CS241047B2 (da)
DD (1) DD216457A5 (da)
DE (1) DE3463655D1 (da)
DK (2) DK160823C (da)
ES (1) ES8506653A1 (da)
FI (1) FI80683C (da)
GB (1) GB8305377D0 (da)
GR (1) GR79816B (da)
HK (1) HK32389A (da)
HU (1) HU190545B (da)
IE (1) IE57056B1 (da)
IL (1) IL71042A (da)
IN (1) IN161372B (da)
NO (1) NO161559C (da)
NZ (1) NZ207256A (da)
PH (1) PH20060A (da)
PL (1) PL142674B1 (da)
PT (1) PT78128B (da)
SG (1) SG6589G (da)
SU (1) SU1405701A3 (da)
YU (1) YU42634B (da)
ZA (1) ZA841322B (da)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5142053A (en) * 1990-04-20 1992-08-25 Adir Et Compagnie Process for the preparation of 1-(2,3,4-trimethoxybenzyl)piperazine by reductive animation

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3461637D1 (en) * 1983-02-16 1987-01-22 Pfizer Ltd Triazole antifungal agents
US4690942A (en) * 1983-12-20 1987-09-01 Ciba-Geigy Corporation 1-aryl-2-fluoro-2-azolyl alkanones, alkanols, esters, and ethers, composition containing them, and use of them to control phytopathogenic microorganisms
IE58738B1 (en) * 1984-09-05 1993-11-03 Ici Plc Antifungal azole compounds
EP0228995A1 (de) * 1985-12-20 1987-07-15 Ciba-Geigy Ag Mikrobizide
DE3825841A1 (de) * 1988-07-29 1990-02-01 Basf Ag 1-halogen-1-azolypropene und -methyloxirane und diese enthaltende fungizide
DE4034352A1 (de) * 1990-10-29 1992-04-30 Basf Ag 1-halogen-1-azolylmethanderivate und diese enthaltende fungizide
TW210334B (da) * 1990-12-12 1993-08-01 Ciba Geigy Ag
US5488035A (en) * 1991-12-06 1996-01-30 Pioneer Hi-Bred International, Inc. Peptide with inhibitory activity towards plant pathogenic fungi
JP3471831B2 (ja) 1991-12-09 2003-12-02 富山化学工業株式会社 新規なトリアゾール誘導体およびその塩
US5360612A (en) * 1992-10-13 1994-11-01 Pfizer Inc. Pharmaceutical compositions containing triazole derivatives for rectal administration
GB9516121D0 (en) * 1995-08-05 1995-10-04 Pfizer Ltd Organometallic addition to ketones
JP6223329B2 (ja) * 2011-06-23 2017-11-01 ヴィアメット ファーマスーティカルズ，インコーポレイテッド 金属酵素化合物
JP6189865B2 (ja) 2012-01-20 2017-08-30 ヴィアメット ファーマスーティカルズ，インコーポレイテッド 金属酵素阻害薬化合物
TWI646088B (zh) * 2012-03-16 2019-01-01 維愛美製藥公司 金屬酶抑制劑化合物

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2918894A1 (de) * 1979-05-10 1980-11-20 Bayer Ag Fluorierte 1-triazolyl-butan-derivate, verfahren zu ihrer herstellung und ihre verwendung als fungizide
DE2938534A1 (de) * 1979-09-24 1981-04-23 Bayer Ag, 5090 Leverkusen Acylierte triazolyl-(gamma)-fluorpinakolyl-derivate, verfahren zu ihrer herstellung und ihre verwendung als fungizide
GB2078719B (en) * 1980-06-02 1984-04-26 Ici Ltd Heterocyclic compounds
DE3033592A1 (de) * 1980-09-06 1982-04-22 Bayer Ag, 5090 Leverkusen Fluorierte 1-azolyl-butan-derivate, verfahren zu ihrer herstellung und ihre verwendung als fungizide
EP0069442B1 (en) * 1981-06-06 1985-02-20 Pfizer Limited Antifungal agents, processes for their preparation, and pharmaceutical compositions containing them
DE3210570A1 (de) * 1982-03-23 1983-10-06 Hoechst Ag 3-azolyl-1,2-diaryl-1-halogen-1-propene, ihre herstellung, ihre verwendung als pflanzenschutzmittel und diese verbindungen enthaltende praeparate
GR79307B (da) * 1982-06-09 1984-10-22 Pfizer
US4510148A (en) * 1982-06-12 1985-04-09 Pfizer Inc. 2-Heterocyclic-1,3-bis(1H-1,2,4-triazol-1-yl)-propan-2-ols as antifungal agents
US4518604A (en) * 1983-07-25 1985-05-21 Pfizer Inc. Antifungal 1-aryl-2-(1H-1,2,4-triazol-1yl)-1-perfluoroalkylethyl halides
US4690942A (en) * 1983-12-20 1987-09-01 Ciba-Geigy Corporation 1-aryl-2-fluoro-2-azolyl alkanones, alkanols, esters, and ethers, composition containing them, and use of them to control phytopathogenic microorganisms

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5142053A (en) * 1990-04-20 1992-08-25 Adir Et Compagnie Process for the preparation of 1-(2,3,4-trimethoxybenzyl)piperazine by reductive animation

Also Published As

Publication number Publication date
DK369889D0 (da) 1989-07-27
NO840721L (no) 1984-08-27
YU42634B (en) 1988-10-31
FI840764L (fi) 1984-08-26
KR870000356B1 (ko) 1987-03-05
IE57056B1 (en) 1992-04-08
DE3463655D1 (en) 1987-06-19
US4960782A (en) 1990-10-02
CS241047B2 (en) 1986-03-13
NO161559B (no) 1989-05-22
AU545660B2 (en) 1985-07-25
JPS6411631B2 (da) 1989-02-27
EP0118245A1 (en) 1984-09-12
GR79816B (da) 1984-10-31
ES529992A0 (es) 1985-07-16
KR840008018A (ko) 1984-12-12
CS127684A2 (en) 1985-06-13
GB8305377D0 (en) 1983-03-30
HU190545B (en) 1986-09-29
DK369889A (da) 1989-07-27
ZA841322B (en) 1985-10-30
DK97884D0 (da) 1984-02-24
SG6589G (en) 1989-06-09
IE840451L (en) 1984-08-25
DK171233B1 (da) 1996-08-05
DK160823B (da) 1991-04-22
EP0118245B1 (en) 1987-05-13
SU1405701A3 (ru) 1988-06-23
IN161372B (da) 1987-11-21
PT78128A (en) 1984-03-01
YU33584A (en) 1986-08-31
CA1257276A (en) 1989-07-11
FI840764A0 (fi) 1984-02-24
PL142674B1 (en) 1987-11-30
PL246356A1 (en) 1985-02-27
DK160823C (da) 1991-10-07
DD216457A5 (de) 1984-12-12
JPS59193877A (ja) 1984-11-02
AU2504084A (en) 1984-08-30
FI80683C (fi) 1990-07-10
HK32389A (en) 1989-04-28
NO161559C (no) 1989-08-30
PH20060A (en) 1986-09-18
HUT34012A (en) 1985-01-28
IL71042A0 (en) 1984-05-31
ES8506653A1 (es) 1985-07-16
FI80683B (fi) 1990-03-30
PT78128B (en) 1986-07-17
NZ207256A (en) 1986-07-11
IL71042A (en) 1987-07-31

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