DK72686A - Aminosyrederivat og antikonvulsant praeparat som indeholder derivatet - Google Patents

Aminosyrederivat og antikonvulsant praeparat som indeholder derivatet Download PDF

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Publication number
DK72686A
DK72686A DK72686A DK72686A DK72686A DK 72686 A DK72686 A DK 72686A DK 72686 A DK72686 A DK 72686A DK 72686 A DK72686 A DK 72686A DK 72686 A DK72686 A DK 72686A
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DK
Denmark
Prior art keywords
anticonvulsant
derivative
lower alkyl
amino acid
preparation containing
Prior art date
Application number
DK72686A
Other languages
English (en)
Other versions
DK173553B1 (da
DK72686D0 (da
Inventor
Harold L Kohn
Darrell Watson
Original Assignee
Research Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Research Corp filed Critical Research Corp
Publication of DK72686D0 publication Critical patent/DK72686D0/da
Publication of DK72686A publication Critical patent/DK72686A/da
Application granted granted Critical
Publication of DK173553B1 publication Critical patent/DK173553B1/da

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Epidemiology (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
DK198600726A 1985-02-15 1986-02-14 Aminosyrederivater, antikonvulsant præparat som indeholder aminosyrederivat samt anvendelse af aminosyrederivater til frems DK173553B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US70219585A 1985-02-15 1985-02-15
US70219585 1985-02-15

Publications (3)

Publication Number Publication Date
DK72686D0 DK72686D0 (da) 1986-02-14
DK72686A true DK72686A (da) 1986-08-16
DK173553B1 DK173553B1 (da) 2001-03-12

Family

ID=24820226

Family Applications (1)

Application Number Title Priority Date Filing Date
DK198600726A DK173553B1 (da) 1985-02-15 1986-02-14 Aminosyrederivater, antikonvulsant præparat som indeholder aminosyrederivat samt anvendelse af aminosyrederivater til frems

Country Status (11)

Country Link
EP (1) EP0194464B1 (da)
JP (1) JPH06104649B2 (da)
AT (1) ATE62222T1 (da)
AU (1) AU596573B2 (da)
CA (1) CA1340902C (da)
DE (1) DE3678469D1 (da)
DK (1) DK173553B1 (da)
ES (1) ES8708142A1 (da)
GR (1) GR860455B (da)
IE (1) IE58422B1 (da)
PT (1) PT82032B (da)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2569186B1 (fr) * 1984-08-20 1986-09-05 Lafon Labor Derives de 1-(n-(a-amino-a-methylacetyl)-aminophenyl)-2-amino-propanone, procede de preparation et utilisation en therapeutique
US5654301A (en) * 1985-02-15 1997-08-05 Research Corporation Technologies, Inc. Amino acid derivative anticonvulsant
US5378729A (en) 1985-02-15 1995-01-03 Research Corporation Technologies, Inc. Amino acid derivative anticonvulsant
NZ222045A (en) * 1986-08-21 1989-10-27 Res Corp Technologies Inc From diamides up to tetrapeptides for use as anticanvulsants
WO1990015069A2 (en) * 1989-05-19 1990-12-13 Research Corporation Technologies, Inc. Amino acid derivative anticonvulsant
JPH06509090A (ja) * 1991-07-10 1994-10-13 メルク シヤープ エンド ドーム リミテツド 芳香族化合物、それらを含む組成物、及び治療におけるそれらの使用
GB9211193D0 (en) * 1992-05-27 1992-07-08 Merck Sharp & Dohme Therapeutic agents
WO1994003429A1 (en) * 1992-07-31 1994-02-17 Merck Sharp & Dohme Limited Substituted amines as tachykinin receptor antagonists
US5773475A (en) 1997-03-17 1998-06-30 Research Corporation Technologies, Inc. Anticonvulsant enantiomeric amino acid derivatives
ES2157567T3 (es) * 1996-03-15 2001-08-16 Res Corp Technologies Inc Derivados de aminoacidos enantiomericos que tienen efecto anticonvulsivo.
US6048899A (en) * 1997-03-17 2000-04-11 Research Corporation Tech., Inc. Anticonvulsant enantiomeric amino acid derivatives
ATE320249T1 (de) 1997-07-08 2006-04-15 Ono Pharmaceutical Co Aminosäurederivate
US6028102A (en) * 1998-02-24 2000-02-22 Yissum Research Development Company Of The Hebrew University Of Jerusalem Anticonvulsant drugs and pharmaceutical compositions thereof
TWI245035B (en) 1998-06-26 2005-12-11 Ono Pharmaceutical Co Amino acid derivatives and a pharmaceutical composition comprising the derivatives
EP1097929A4 (en) 1998-07-14 2005-12-21 Ono Pharmaceutical Co AMINO ACID DERIVATIVES AND MEDICAMENTS IN WHICH THESE DERIVATIVES ARE THE ACTIVE INGREDIENTS
ES2190305B1 (es) * 2000-05-24 2004-07-01 Medichem S.A. Compuestos intermedios para la preparacion de mirtazapina y sus procedimientos de obtencion.
EP1604656A1 (en) 2004-06-09 2005-12-14 Schwarz Pharma Ag Novel use of peptide compounds for treating amyotrophic lateral sclerosis (ALS)

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2676188A (en) * 1950-12-16 1954-04-20 American Home Prod Acylated glycinamides
GB1051220A (da) * 1963-03-21
IE33790B1 (en) * 1968-06-04 1974-10-30 Beecham Group Ltd Derivatives of n-acylaminoacid amides
US3707559A (en) * 1971-05-14 1972-12-26 Searle & Co N-acyl phenylalanine amides
JPS557242A (en) * 1978-06-30 1980-01-19 Tanabe Seiyaku Co Ltd Phenethylamine derivative
FR2480747A1 (fr) * 1980-04-17 1981-10-23 Roques Bernard Derives d'acides amines et leur application therapeutique
FR2489319A1 (fr) * 1980-08-27 1982-03-05 Clin Midy Derives de l'acide amino-4 butyrique et les medicaments, actifs notamment sur le systeme nerveux central, en contenant

Also Published As

Publication number Publication date
DE3678469D1 (de) 1991-05-08
GR860455B (en) 1986-06-18
ES8708142A1 (es) 1987-10-16
DK173553B1 (da) 2001-03-12
ES552348A0 (es) 1987-10-16
JPS61200950A (ja) 1986-09-05
PT82032A (en) 1986-03-01
DK72686D0 (da) 1986-02-14
EP0194464A1 (en) 1986-09-17
CA1340902C (en) 2000-02-22
IE58422B1 (en) 1993-09-22
IE860411L (en) 1986-08-15
ATE62222T1 (de) 1991-04-15
PT82032B (pt) 1988-07-01
JPH06104649B2 (ja) 1994-12-21
AU596573B2 (en) 1990-05-10
EP0194464B1 (en) 1991-04-03
AU5371186A (en) 1986-08-21

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Legal Events

Date Code Title Description
B1 Patent granted (law 1993)
PUP Patent expired