DK72686A - Aminosyrederivat og antikonvulsant praeparat som indeholder derivatet - Google Patents
Aminosyrederivat og antikonvulsant praeparat som indeholder derivatet Download PDFInfo
- Publication number
- DK72686A DK72686A DK72686A DK72686A DK72686A DK 72686 A DK72686 A DK 72686A DK 72686 A DK72686 A DK 72686A DK 72686 A DK72686 A DK 72686A DK 72686 A DK72686 A DK 72686A
- Authority
- DK
- Denmark
- Prior art keywords
- anticonvulsant
- derivative
- lower alkyl
- amino acid
- preparation containing
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biomedical Technology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Epidemiology (AREA)
- Psychiatry (AREA)
- Anesthesiology (AREA)
- Pain & Pain Management (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US70219585A | 1985-02-15 | 1985-02-15 | |
US70219585 | 1985-02-15 |
Publications (3)
Publication Number | Publication Date |
---|---|
DK72686D0 DK72686D0 (da) | 1986-02-14 |
DK72686A true DK72686A (da) | 1986-08-16 |
DK173553B1 DK173553B1 (da) | 2001-03-12 |
Family
ID=24820226
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK198600726A DK173553B1 (da) | 1985-02-15 | 1986-02-14 | Aminosyrederivater, antikonvulsant præparat som indeholder aminosyrederivat samt anvendelse af aminosyrederivater til frems |
Country Status (11)
Country | Link |
---|---|
EP (1) | EP0194464B1 (da) |
JP (1) | JPH06104649B2 (da) |
AT (1) | ATE62222T1 (da) |
AU (1) | AU596573B2 (da) |
CA (1) | CA1340902C (da) |
DE (1) | DE3678469D1 (da) |
DK (1) | DK173553B1 (da) |
ES (1) | ES8708142A1 (da) |
GR (1) | GR860455B (da) |
IE (1) | IE58422B1 (da) |
PT (1) | PT82032B (da) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2569186B1 (fr) * | 1984-08-20 | 1986-09-05 | Lafon Labor | Derives de 1-(n-(a-amino-a-methylacetyl)-aminophenyl)-2-amino-propanone, procede de preparation et utilisation en therapeutique |
US5654301A (en) * | 1985-02-15 | 1997-08-05 | Research Corporation Technologies, Inc. | Amino acid derivative anticonvulsant |
US5378729A (en) | 1985-02-15 | 1995-01-03 | Research Corporation Technologies, Inc. | Amino acid derivative anticonvulsant |
NZ222045A (en) * | 1986-08-21 | 1989-10-27 | Res Corp Technologies Inc | From diamides up to tetrapeptides for use as anticanvulsants |
WO1990015069A2 (en) * | 1989-05-19 | 1990-12-13 | Research Corporation Technologies, Inc. | Amino acid derivative anticonvulsant |
JPH06509090A (ja) * | 1991-07-10 | 1994-10-13 | メルク シヤープ エンド ドーム リミテツド | 芳香族化合物、それらを含む組成物、及び治療におけるそれらの使用 |
GB9211193D0 (en) * | 1992-05-27 | 1992-07-08 | Merck Sharp & Dohme | Therapeutic agents |
WO1994003429A1 (en) * | 1992-07-31 | 1994-02-17 | Merck Sharp & Dohme Limited | Substituted amines as tachykinin receptor antagonists |
US5773475A (en) | 1997-03-17 | 1998-06-30 | Research Corporation Technologies, Inc. | Anticonvulsant enantiomeric amino acid derivatives |
ES2157567T3 (es) * | 1996-03-15 | 2001-08-16 | Res Corp Technologies Inc | Derivados de aminoacidos enantiomericos que tienen efecto anticonvulsivo. |
US6048899A (en) * | 1997-03-17 | 2000-04-11 | Research Corporation Tech., Inc. | Anticonvulsant enantiomeric amino acid derivatives |
ATE320249T1 (de) | 1997-07-08 | 2006-04-15 | Ono Pharmaceutical Co | Aminosäurederivate |
US6028102A (en) * | 1998-02-24 | 2000-02-22 | Yissum Research Development Company Of The Hebrew University Of Jerusalem | Anticonvulsant drugs and pharmaceutical compositions thereof |
TWI245035B (en) | 1998-06-26 | 2005-12-11 | Ono Pharmaceutical Co | Amino acid derivatives and a pharmaceutical composition comprising the derivatives |
EP1097929A4 (en) | 1998-07-14 | 2005-12-21 | Ono Pharmaceutical Co | AMINO ACID DERIVATIVES AND MEDICAMENTS IN WHICH THESE DERIVATIVES ARE THE ACTIVE INGREDIENTS |
ES2190305B1 (es) * | 2000-05-24 | 2004-07-01 | Medichem S.A. | Compuestos intermedios para la preparacion de mirtazapina y sus procedimientos de obtencion. |
EP1604656A1 (en) | 2004-06-09 | 2005-12-14 | Schwarz Pharma Ag | Novel use of peptide compounds for treating amyotrophic lateral sclerosis (ALS) |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2676188A (en) * | 1950-12-16 | 1954-04-20 | American Home Prod | Acylated glycinamides |
GB1051220A (da) * | 1963-03-21 | |||
IE33790B1 (en) * | 1968-06-04 | 1974-10-30 | Beecham Group Ltd | Derivatives of n-acylaminoacid amides |
US3707559A (en) * | 1971-05-14 | 1972-12-26 | Searle & Co | N-acyl phenylalanine amides |
JPS557242A (en) * | 1978-06-30 | 1980-01-19 | Tanabe Seiyaku Co Ltd | Phenethylamine derivative |
FR2480747A1 (fr) * | 1980-04-17 | 1981-10-23 | Roques Bernard | Derives d'acides amines et leur application therapeutique |
FR2489319A1 (fr) * | 1980-08-27 | 1982-03-05 | Clin Midy | Derives de l'acide amino-4 butyrique et les medicaments, actifs notamment sur le systeme nerveux central, en contenant |
-
1986
- 1986-02-14 EP EP86101865A patent/EP0194464B1/en not_active Expired - Lifetime
- 1986-02-14 DK DK198600726A patent/DK173553B1/da not_active IP Right Cessation
- 1986-02-14 IE IE41186A patent/IE58422B1/en not_active IP Right Cessation
- 1986-02-14 CA CA000501869A patent/CA1340902C/en not_active Expired - Lifetime
- 1986-02-14 AT AT86101865T patent/ATE62222T1/de not_active IP Right Cessation
- 1986-02-14 DE DE8686101865T patent/DE3678469D1/de not_active Expired - Lifetime
- 1986-02-15 ES ES552348A patent/ES8708142A1/es not_active Expired
- 1986-02-15 JP JP61031742A patent/JPH06104649B2/ja not_active Expired - Lifetime
- 1986-02-17 PT PT82032A patent/PT82032B/pt not_active IP Right Cessation
- 1986-02-17 AU AU53711/86A patent/AU596573B2/en not_active Expired
- 1986-02-17 GR GR860455A patent/GR860455B/el unknown
Also Published As
Publication number | Publication date |
---|---|
DE3678469D1 (de) | 1991-05-08 |
GR860455B (en) | 1986-06-18 |
ES8708142A1 (es) | 1987-10-16 |
DK173553B1 (da) | 2001-03-12 |
ES552348A0 (es) | 1987-10-16 |
JPS61200950A (ja) | 1986-09-05 |
PT82032A (en) | 1986-03-01 |
DK72686D0 (da) | 1986-02-14 |
EP0194464A1 (en) | 1986-09-17 |
CA1340902C (en) | 2000-02-22 |
IE58422B1 (en) | 1993-09-22 |
IE860411L (en) | 1986-08-15 |
ATE62222T1 (de) | 1991-04-15 |
PT82032B (pt) | 1988-07-01 |
JPH06104649B2 (ja) | 1994-12-21 |
AU596573B2 (en) | 1990-05-10 |
EP0194464B1 (en) | 1991-04-03 |
AU5371186A (en) | 1986-08-21 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B1 | Patent granted (law 1993) | ||
PUP | Patent expired |