DK603983A - 1-cyclopropyl-6-fluor-1,4-dihydro-4-oxo-7-(4-(oxoalkyl)-1-piperazinyl)-3-quinolincarboxylsyre og derivater deraf, fremgangsmaader til fremstilling deraf samt antibakterielle midler med indhold af disse forbindelser - Google Patents
1-cyclopropyl-6-fluor-1,4-dihydro-4-oxo-7-(4-(oxoalkyl)-1-piperazinyl)-3-quinolincarboxylsyre og derivater deraf, fremgangsmaader til fremstilling deraf samt antibakterielle midler med indhold af disse forbindelser Download PDFInfo
- Publication number
- DK603983A DK603983A DK603983A DK603983A DK603983A DK 603983 A DK603983 A DK 603983A DK 603983 A DK603983 A DK 603983A DK 603983 A DK603983 A DK 603983A DK 603983 A DK603983 A DK 603983A
- Authority
- DK
- Denmark
- Prior art keywords
- oxo
- piperazinyl
- cyclopropyl
- dihydro
- fluoro
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Quinoline Compounds (AREA)
- Fodder In General (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE3248505 | 1982-12-29 | ||
DE19823248505 DE3248505A1 (de) | 1982-12-29 | 1982-12-29 | 1-cyclopropyl-6-fluor-1,4-dihydro-4-oxo-7(4- (oxoalkyl)-1-piperazinyl/-3-chinolincarbonsaeuren und ihre derivate, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel |
Publications (4)
Publication Number | Publication Date |
---|---|
DK603983D0 DK603983D0 (da) | 1983-12-28 |
DK603983A true DK603983A (da) | 1984-06-30 |
DK159106B DK159106B (da) | 1990-09-03 |
DK159106C DK159106C (da) | 1991-02-25 |
Family
ID=6182077
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK603983A DK159106C (da) | 1982-12-29 | 1983-12-28 | 1-cyclopropyl-6-fluor-1,4-dihydro-4-oxo-7-(4-substitueret-1-piperazinyl)-3-quinolincarboxylsyrer og derivater deraf, antibakterielle midler med indhold af disse forbindelser samt fremgangsmaade til fremstilling af saadanne midler |
Country Status (20)
Country | Link |
---|---|
US (1) | US4547503A (da) |
EP (1) | EP0113092B1 (da) |
JP (1) | JPS59172471A (da) |
KR (1) | KR870000896B1 (da) |
AT (1) | ATE19876T1 (da) |
AU (1) | AU559519B2 (da) |
CA (1) | CA1218069A (da) |
DD (1) | DD216015A5 (da) |
DE (2) | DE3248505A1 (da) |
DK (1) | DK159106C (da) |
ES (1) | ES8500262A1 (da) |
FI (1) | FI79311C (da) |
GR (1) | GR79446B (da) |
HU (1) | HU192861B (da) |
IE (1) | IE56511B1 (da) |
IL (1) | IL70538A (da) |
NO (1) | NO161492C (da) |
NZ (1) | NZ206706A (da) |
PH (5) | PH20489A (da) |
ZA (1) | ZA839645B (da) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3306772A1 (de) * | 1983-02-25 | 1984-08-30 | Bayer Ag, 5090 Leverkusen | Chinolonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel |
DE3426482A1 (de) * | 1984-07-18 | 1986-01-30 | Bayer Ag, 5090 Leverkusen | Verfahren zur herstellung von halogenierten aroylessigestern |
DE3435392A1 (de) * | 1984-09-27 | 1986-04-03 | Bayer Ag, 5090 Leverkusen | Verfahren zur herstellung von 2,4-dichlor-5-fluor-benzoesaeure |
JPS6259263A (ja) * | 1985-09-10 | 1987-03-14 | Kyorin Pharmaceut Co Ltd | キノロンカルボン酸誘導体 |
DE3542002A1 (de) * | 1985-11-28 | 1987-06-04 | Bayer Ag | 1-cyclopropyl-6-fluor-1,4-dihydro-4-oxo-7- (1-piperazinyl)-3-chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel |
US4767762A (en) * | 1985-12-23 | 1988-08-30 | Abbott Laboratories | Tricyclic quinoline and naphthyride antibacterials |
JPS62192321A (ja) * | 1986-02-19 | 1987-08-22 | Bayer Japan Kk | 魚類用抗菌剤 |
DE3705621C2 (de) * | 1986-02-25 | 1997-01-09 | Otsuka Pharma Co Ltd | Heterocyclisch substituierte Chinoloncarbonsäurederivate |
ES2006977A6 (es) * | 1988-06-13 | 1989-05-16 | Union Quimico Farma | Procedimiento para la obtencion de ciprofloxacina. |
FR2657895A1 (fr) * | 1990-02-05 | 1991-08-09 | Inst Textile De France | Materiau antiseptique a greffons complexes par des ions metalliques et procede de preparation. |
TW584632B (en) * | 2000-01-12 | 2004-04-21 | Pharmaceutical Ind Tech & Dev | 6-fluoro-1,4-dihydro-7-[4-(2-hydroxyiminoethyl)-1-piperazinyl]-4-oxoquinoline-3-carboxylic acid derivatives, their preparation and pharmaceutical compositions |
CA2424402A1 (en) | 2000-12-21 | 2002-08-01 | Pharmacia & Upjohn Company | Antimicrobial quinolone derivatives and use of the same to treat bacterial infections |
KR100821894B1 (ko) * | 2004-07-02 | 2008-04-16 | 주식회사 코오롱 | 항균 염료 및 그를 이용한 항균 섬유 |
EP2957561A1 (en) * | 2014-06-18 | 2015-12-23 | Université Paris 6 Pierre et Marie Curie UPMC | Novel fluoroquinolones and use thereof to treat bacterial infections |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3149104A (en) * | 1961-01-03 | 1964-09-15 | Sterling Drug Inc | 4-hydroxy-7-styryl-1, 8-naphthyridine-3-carboxylic acids and esters |
DE2808070A1 (de) * | 1978-02-24 | 1979-08-30 | Bayer Ag | Verfahren zur herstellung von 4-pyridon-3-carbonsaeuren und/oder deren derivaten |
JPS5845426B2 (ja) * | 1978-09-29 | 1983-10-08 | 杏林製薬株式会社 | 置換キノリンカルボン酸誘導体 |
DE3033157A1 (de) * | 1980-09-03 | 1982-04-01 | Bayer Ag, 5090 Leverkusen | 7-amino-1-cyclopropyl-4-oxo-1,4-dihydro-naphthyridin-3-carbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel |
DE3142854A1 (de) * | 1981-10-29 | 1983-05-11 | Bayer Ag, 5090 Leverkusen | 1-cyclopropyl-6-fluor-1,4-dihydro-4-oxo-7-piperazino-chinolin-3-carbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel |
-
1982
- 1982-12-29 DE DE19823248505 patent/DE3248505A1/de not_active Withdrawn
-
1983
- 1983-12-09 US US06/560,026 patent/US4547503A/en not_active Expired - Lifetime
- 1983-12-15 NO NO834633A patent/NO161492C/no unknown
- 1983-12-17 AT AT83112724T patent/ATE19876T1/de active
- 1983-12-17 DE DE8383112724T patent/DE3363607D1/de not_active Expired
- 1983-12-17 EP EP83112724A patent/EP0113092B1/de not_active Expired
- 1983-12-19 AU AU22509/83A patent/AU559519B2/en not_active Ceased
- 1983-12-22 NZ NZ206706A patent/NZ206706A/en unknown
- 1983-12-22 IE IE3035/83A patent/IE56511B1/en not_active IP Right Cessation
- 1983-12-23 CA CA000444207A patent/CA1218069A/en not_active Expired
- 1983-12-26 IL IL70538A patent/IL70538A/xx not_active IP Right Cessation
- 1983-12-27 GR GR73354A patent/GR79446B/el unknown
- 1983-12-27 JP JP58244938A patent/JPS59172471A/ja active Granted
- 1983-12-27 FI FI834807A patent/FI79311C/fi not_active IP Right Cessation
- 1983-12-27 PH PH30029A patent/PH20489A/en unknown
- 1983-12-28 ES ES528496A patent/ES8500262A1/es not_active Expired
- 1983-12-28 DD DD83258779A patent/DD216015A5/de not_active IP Right Cessation
- 1983-12-28 DK DK603983A patent/DK159106C/da not_active IP Right Cessation
- 1983-12-28 HU HU834500A patent/HU192861B/hu not_active IP Right Cessation
- 1983-12-28 ZA ZA839645A patent/ZA839645B/xx unknown
- 1983-12-29 KR KR1019830006263A patent/KR870000896B1/ko not_active IP Right Cessation
-
1985
- 1985-03-21 PH PH32023A patent/PH22496A/en unknown
- 1985-03-21 PH PH32022A patent/PH23670A/en unknown
- 1985-03-21 PH PH32024A patent/PH23141A/en unknown
- 1985-06-24 PH PH32445A patent/PH22886A/en unknown
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PBP | Patent lapsed |