DK590586D0 - 5-amino- og 5-hydroxy-6,8-difluorquinoloner og salte deraf og farmaceutiske kompositioner indeholdende forbindelserne - Google Patents
5-amino- og 5-hydroxy-6,8-difluorquinoloner og salte deraf og farmaceutiske kompositioner indeholdende forbindelserneInfo
- Publication number
- DK590586D0 DK590586D0 DK590586A DK590586A DK590586D0 DK 590586 D0 DK590586 D0 DK 590586D0 DK 590586 A DK590586 A DK 590586A DK 590586 A DK590586 A DK 590586A DK 590586 D0 DK590586 D0 DK 590586D0
- Authority
- DK
- Denmark
- Prior art keywords
- difluoroquinolons
- hydroxy
- salts
- amino
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US80812285 | 1985-12-12 | ||
| US06/808,122 US4668680A (en) | 1985-12-12 | 1985-12-12 | 5-amino-6,8-difluoroquinolones as antibacterial agents |
| US91856886 | 1986-10-20 | ||
| US06/918,568 US4977154A (en) | 1985-12-12 | 1986-10-20 | 5-amino and 5-hydroxy-6-fluoroquinolones as antibacterial agents |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| DK590586D0 true DK590586D0 (da) | 1986-12-09 |
| DK590586A DK590586A (da) | 1987-06-13 |
| DK166493B1 DK166493B1 (da) | 1993-06-01 |
Family
ID=27123084
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK590586A DK166493B1 (da) | 1985-12-12 | 1986-12-09 | 5-amino-, 5-alkoxy- og 5-hydroxy-6-fluor-1,4-dihydro-4-oxo-quinolin-3-carboxylsyrederivater og farmaceutisk acceptable syreadditions- og basesalte deraf og farmaceutiske kompositioner indeholdende forbindelserne |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US4977154A (da) |
| EP (1) | EP0226961B1 (da) |
| KR (1) | KR900000555B1 (da) |
| CN (1) | CN1013114B (da) |
| AU (1) | AU591732B2 (da) |
| DE (1) | DE3679793D1 (da) |
| DK (1) | DK166493B1 (da) |
| ES (1) | ES2039198T3 (da) |
| FI (1) | FI865004A (da) |
| GR (1) | GR3002129T3 (da) |
| HU (1) | HU203231B (da) |
| IE (1) | IE59261B1 (da) |
| IL (1) | IL80933A (da) |
| NO (1) | NO865013L (da) |
| OA (1) | OA08561A (da) |
| PT (1) | PT83909B (da) |
Families Citing this family (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU594983B2 (en) * | 1985-10-29 | 1990-03-22 | Dainippon Pharmaceutical Co. Ltd. | Novel quinoline derivatives and processes for preparation thereof |
| EP0242789A3 (en) * | 1986-04-25 | 1990-09-05 | Dainippon Pharmaceutical Co., Ltd. | Novel quinoline derivates and processes for preparation thereof |
| DE3711193A1 (de) * | 1987-04-02 | 1988-10-13 | Bayer Ag | 5-substituierte chinolon- und naphthyridoncarbonsaeure-derivate |
| US4780468A (en) * | 1987-08-07 | 1988-10-25 | Warner-Lambert Company | 8-trifluoromethyl quinolones as antibacterial agents |
| US4933335A (en) * | 1987-08-07 | 1990-06-12 | Warner-Lambert Company | Quinolones as antibacterial agents |
| US4929613A (en) * | 1987-08-26 | 1990-05-29 | Warner-Lambert Company | Antibacterial agents |
| EP0339406A1 (en) * | 1988-04-19 | 1989-11-02 | Hokuriku Pharmaceutical Co.,Ltd | Quinoline-3-carboxylic acid derivatives, process for preparing the same, and composition exhibiting excellent antibacterial effect containing the same |
| JP2844079B2 (ja) * | 1988-05-23 | 1999-01-06 | 塩野義製薬株式会社 | ピリドンカルボン酸系抗菌剤 |
| FI95130C (fi) * | 1988-07-20 | 1995-12-27 | Sankyo Co | Menetelmä lääkeaineena käyttökelpoisten 4-oksokinoliini-3-karboksyylihapon johdannaisten valmistamiseksi |
| ATE193890T1 (de) | 1990-04-18 | 2000-06-15 | Procter & Gamble Pharma | Antimikrobielle chinolonyl-lactame |
| DE4019023A1 (de) * | 1990-06-14 | 1991-12-19 | Bayer Ag | Verfahren zur herstellung von chinolincarbonsaeuren |
| RU2140919C1 (ru) * | 1994-07-18 | 1999-11-10 | Убе Индастриз Лтд. | Производные 8-трифторметилхинолинкарбоновой кислоты, фармацевтическая композиция и способ ингибирования вируса иммунодефицита |
| US5866150A (en) * | 1996-03-20 | 1999-02-02 | Aquaculture Technology Incorporated | Antibacterially active extracts from the marine algae chaetoceros and methods of use |
| IN186245B (da) | 1997-09-19 | 2001-07-14 | Ranbaxy Lab Ltd | |
| CN1091103C (zh) * | 1999-04-02 | 2002-09-18 | 中国科学院上海药物研究所 | 一类喹诺酮类化合物及它的制备和其用途 |
| ATE407121T1 (de) * | 2000-02-09 | 2008-09-15 | Daiichi Sankyo Co Ltd | Gegen säurebeständige bakterien wirksame antibakterielle mittel die pyridincarbonsäuren als aktiven wirkstoff enthalten |
| DE102004035203A1 (de) * | 2004-07-21 | 2006-02-16 | Bayer Healthcare Ag | Substituierte Chinolone |
| US8524734B2 (en) | 2005-05-18 | 2013-09-03 | Mpex Pharmaceuticals, Inc. | Aerosolized fluoroquinolones and uses thereof |
| CN100415212C (zh) * | 2006-07-21 | 2008-09-03 | 哈药集团制药总厂 | 一种含乳酸卡德沙星的口服制剂 |
| CN102202649A (zh) | 2008-10-07 | 2011-09-28 | Mpex医药有限公司 | 用于改进的药物动力学的氟喹诺酮气雾剂制剂 |
| HUE050147T2 (hu) | 2008-10-07 | 2020-11-30 | Horizon Orphan Llc | Tüdõgyulladás csökkentése levofloxacin belélegzése útján |
| PT2473170T (pt) | 2009-09-04 | 2019-08-23 | Horizon Orphan Llc | Utilização de levofloxacina em aerossol para tratamento de fibrose cística |
| CN104557896A (zh) * | 2013-10-18 | 2015-04-29 | 沈敬山 | 布瑞哌唑、其关键中间体及其盐的制备方法 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2808070A1 (de) * | 1978-02-24 | 1979-08-30 | Bayer Ag | Verfahren zur herstellung von 4-pyridon-3-carbonsaeuren und/oder deren derivaten |
| DE3248506A1 (de) * | 1982-12-29 | 1984-07-05 | Bayer Ag, 5090 Leverkusen | 1-cyclopropyl-6-fluor-1,4-dihydro-4-oxo-7(alkyl-1-piperazinyl)-3-chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel |
| EP0160578B1 (en) * | 1984-02-17 | 1989-11-23 | Daiichi Seiyaku Co., Ltd. | 1,8-naphthyridine derivatives |
| US4604401A (en) * | 1984-07-20 | 1986-08-05 | Warner-Lambert Company | Antibacterial agents III |
| JPS61205258A (ja) * | 1985-03-08 | 1986-09-11 | Kyorin Pharmaceut Co Ltd | キノロンカルボン酸誘導体及びその製造方法 |
| AU594983B2 (en) * | 1985-10-29 | 1990-03-22 | Dainippon Pharmaceutical Co. Ltd. | Novel quinoline derivatives and processes for preparation thereof |
-
1986
- 1986-10-20 US US06/918,568 patent/US4977154A/en not_active Expired - Fee Related
- 1986-11-25 IE IE310486A patent/IE59261B1/en not_active IP Right Cessation
- 1986-12-02 AU AU65879/86A patent/AU591732B2/en not_active Ceased
- 1986-12-08 FI FI865004A patent/FI865004A/fi not_active Application Discontinuation
- 1986-12-09 DK DK590586A patent/DK166493B1/da not_active IP Right Cessation
- 1986-12-10 IL IL8680933A patent/IL80933A/xx not_active IP Right Cessation
- 1986-12-10 KR KR1019860010553A patent/KR900000555B1/ko not_active IP Right Cessation
- 1986-12-11 NO NO865013A patent/NO865013L/no unknown
- 1986-12-11 EP EP86117250A patent/EP0226961B1/en not_active Expired - Lifetime
- 1986-12-11 PT PT83909A patent/PT83909B/pt not_active IP Right Cessation
- 1986-12-11 HU HU865180A patent/HU203231B/hu not_active IP Right Cessation
- 1986-12-11 ES ES198686117250T patent/ES2039198T3/es not_active Expired - Lifetime
- 1986-12-11 DE DE8686117250T patent/DE3679793D1/de not_active Expired - Fee Related
- 1986-12-11 OA OA59014A patent/OA08561A/xx unknown
- 1986-12-12 CN CN86108942A patent/CN1013114B/zh not_active Expired
-
1991
- 1991-06-13 GR GR91400732T patent/GR3002129T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| IL80933A0 (en) | 1987-03-31 |
| EP0226961B1 (en) | 1991-06-12 |
| ES2039198T3 (es) | 1993-09-16 |
| DK590586A (da) | 1987-06-13 |
| PT83909A (en) | 1987-01-01 |
| CN86108942A (zh) | 1987-11-04 |
| EP0226961A1 (en) | 1987-07-01 |
| FI865004A (fi) | 1987-06-13 |
| PT83909B (pt) | 1989-05-12 |
| NO865013L (no) | 1987-06-15 |
| HU203231B (en) | 1991-06-28 |
| AU6587986A (en) | 1987-06-18 |
| US4977154A (en) | 1990-12-11 |
| HUT42470A (en) | 1987-07-28 |
| KR900000555B1 (ko) | 1990-01-31 |
| KR870006034A (ko) | 1987-07-08 |
| AU591732B2 (en) | 1989-12-14 |
| OA08561A (en) | 1988-09-30 |
| IE863104L (en) | 1987-06-12 |
| IL80933A (en) | 1991-06-10 |
| GR3002129T3 (en) | 1992-12-30 |
| NO865013D0 (no) | 1986-12-11 |
| DK166493B1 (da) | 1993-06-01 |
| CN1013114B (zh) | 1991-07-10 |
| FI865004A0 (fi) | 1986-12-08 |
| IE59261B1 (en) | 1994-01-26 |
| DE3679793D1 (de) | 1991-07-18 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DK590586A (da) | 5-amino- og 5-hydroxy-6,8-difluorquinoloner og salte deraf og farmaceutiske kompositioner indeholdende forbindelserne | |
| IT8619625A0 (it) | Composizioni farmaceutiche per inalazione. | |
| DK364683D0 (da) | Sproejte, isaer til medicinsk anvendelse | |
| DK185685D0 (da) | 1,4-dihydro-4-oxonaphthyridinderivater og salte deraf, fremgangsmaade til fremstilling heraf og antibakterielle midler indeholdende saadanne forbindelser | |
| NO875419D0 (no) | Blandinger for farmasoeytisk tape. | |
| IT8820386A0 (it) | Composizioni farmaceutiche orosolubili contenti acetilcisteina. | |
| FI872733A0 (fi) | Farmaceutiska kompositioner. | |
| FI842927A (fi) | Nya 1,5-benzotiazepiner med foerdelaktig inverkan pao hjaertblodkaerlen, foerfarande foer deras framstaellning och dessa innehaollande farmaceutiska foereningar. | |
| FI861338A0 (fi) | Tvaettmedel innehaollande vaordmedel foer tyg. | |
| DK162221C (da) | Cinnolinforbindelser, fremgangsmaade til fremstilling deraf og farmaceutiske midler indeholdende forbindelserne | |
| FI872313A0 (fi) | Farmaceutiska kompositioner. | |
| IT1213453B (it) | Composizione farmaceutica. | |
| ES555778A0 (es) | Equipo para uso odontologico. | |
| DK133587D0 (da) | 2-heterocyclylthio-penemer, deres anvendelse og farmaceutisk komposition indeholdende forbindelserne | |
| FI860780A0 (fi) | Ortopedisk vaest. | |
| FI852706A0 (fi) | Skiktade kirurgiska utensilier av kompoundstruktur. | |
| DE3669656D1 (de) | Azanaphthalene enthaltende arzneimittelzusammensetzungen. | |
| ES554829A0 (es) | Procedimiento para preparar eteres 1,3-dioxano. | |
| DK164867C (da) | Pyrimidooe4,5-gaaquinolin-derivater eller salte deraf og farmaceutiske formuleringer indeholdende disse | |
| IT8520591A0 (it) | Formulazione farmaceutica. | |
| NO862593D0 (no) | Benzoyl-triazolyleddiksyre- eller -tioeddiksyrederivater, fremstilling derav og biocide midler inneholdende derivatene. | |
| DK17683A (da) | 2,5-benzodiazocinderivater og salte deraf | |
| IT1215261B (it) | Composizioni farmaceutiche adattivita' antigalattopoietica. | |
| DE68922225D1 (de) | Verdichtete pulverheilmittel. | |
| IT8421627A1 (it) | Composizione farmaceutica contenente come ingrediente attivo 24,25-diidrossicolecalciferolo |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B1 | Patent granted (law 1993) | ||
| PBP | Patent lapsed |