DK521786D0 - Substituerede benzoatestere af estrogener - Google Patents

Substituerede benzoatestere af estrogener

Info

Publication number
DK521786D0
DK521786D0 DK521786A DK521786A DK521786D0 DK 521786 D0 DK521786 D0 DK 521786D0 DK 521786 A DK521786 A DK 521786A DK 521786 A DK521786 A DK 521786A DK 521786 D0 DK521786 D0 DK 521786D0
Authority
DK
Denmark
Prior art keywords
estrogenes
testers
substituted benzo
estradiol
substituted
Prior art date
Application number
DK521786A
Other languages
English (en)
Other versions
DK521786A (da
Inventor
Bruce Jeffrey Aungst
Munir Alwan Hussain
Original Assignee
Du Pont
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Du Pont filed Critical Du Pont
Publication of DK521786D0 publication Critical patent/DK521786D0/da
Publication of DK521786A publication Critical patent/DK521786A/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0066—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa
    • C07J1/007—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0081—Substituted in position 17 alfa and 17 beta
    • C07J1/0088—Substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
    • C07J1/0096—Alkynyl derivatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0072—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the A ring of the steroid being aromatic

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Silver Salt Photography Or Processing Solution Therefor (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DK521786A 1985-11-01 1986-10-31 Substituerede benzoatestere af estrogener DK521786A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/793,892 US4757062A (en) 1985-11-01 1985-11-01 Substituted benzoate ester prodrugs of estrogens

Publications (2)

Publication Number Publication Date
DK521786D0 true DK521786D0 (da) 1986-10-31
DK521786A DK521786A (da) 1987-05-02

Family

ID=25161090

Family Applications (1)

Application Number Title Priority Date Filing Date
DK521786A DK521786A (da) 1985-11-01 1986-10-31 Substituerede benzoatestere af estrogener

Country Status (12)

Country Link
US (1) US4757062A (da)
EP (1) EP0221506B1 (da)
JP (1) JPS62120398A (da)
AT (1) ATE49216T1 (da)
AU (1) AU583160B2 (da)
CA (1) CA1255295A (da)
DE (1) DE3667982D1 (da)
DK (1) DK521786A (da)
ES (1) ES2002058A6 (da)
GR (1) GR862633B (da)
IL (1) IL79710A0 (da)
ZA (1) ZA868272B (da)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6702705B1 (en) 1988-05-04 2004-03-09 Igen International, Inc. Prodrugs activated by targeted catalytic proteins
DK24089D0 (da) * 1989-01-20 1989-01-20 Hans Bundgaard Novel prodrug derivatives of biologically active agents containing hydroxyl groups or nh-acidic groups
US4909563A (en) * 1989-04-12 1990-03-20 Phillip E. Walker Automatically deployable covering device
US6258360B1 (en) * 1989-05-04 2001-07-10 Igen International, Inc. Prodrugs activated by targeted catalytic proteins
KR100334696B1 (ko) * 1991-08-05 2002-04-27 리차아드제이마세이 표적화된 촉매 단백질에 의해 활성화되는 선구 약제
AR039224A1 (es) * 2002-04-02 2005-02-09 Chugai Pharmaceutical Co Ltd Derivados de estrona y procedimientos para producirlos
RU2720677C1 (ru) * 2017-01-25 2020-05-12 Чжуншань Офтальмик Сентер, Сунь Ятсен Юниверсити Соединение, представляющее собой пролекарство ланостерина, а также способ его получения и его применение
BR112021001172A2 (pt) * 2018-07-25 2021-04-27 Guangzhou Ocusun Ophthalmic Biotechnology Co., Ltd. forma cristalina do composto do pró-fármaco lanosterol e aplicação do mesmo

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DD83130A (da) *
US2054271A (en) * 1932-05-17 1936-09-15 Schering Kahlbaum Ag Production of crystallized hormone esters
US2243887A (en) * 1935-11-09 1941-06-03 Schering Corp Tertiary carbinols of the cyclopentano-polyhydrophenanthrene series and a method of producing the same
US2251939A (en) * 1935-11-22 1941-08-12 Schering Corp Tertiary alcohols of the cyclopentano polyhydro phenanthrene series and a method of producing the same
CH202847A (de) * 1937-06-26 1939-02-15 Chem Ind Basel Verfahren zur Darstellung von Acetylen-Derivaten der Cyclopentanopolyhydrophenanthren-Reihe.
US2265976A (en) * 1937-10-25 1941-12-09 Schering Corp Tertiary alcohols of the estrane series and their derivatives and a process for their manufacture
US3347880A (en) * 1962-10-05 1967-10-17 Schering Corp 17alpha-halogenoethinylestranes
GB1039447A (en) * 1964-02-21 1966-08-17 Nicholas Gueritee Oestradiol derivatives
US3624113A (en) * 1968-12-11 1971-11-30 Warner Lambert Co Long-acting estradiol derivatives
US3634404A (en) * 1969-05-08 1972-01-11 American Home Prod 7alpha 8alpha-methyleneestrogens and preparation thereof
US3647784A (en) * 1970-02-02 1972-03-07 American Home Prod Preparation of steroidal formate esters
US4110324A (en) * 1974-02-26 1978-08-29 Nicolas Gueritee Nicotinic derivatives of estriol
DE2506548C2 (de) * 1975-02-17 1986-05-15 Theramex S.A., Paris Östriol-Nicotinsäurederivate, Verfahren zu ihrer Herstellung und diese enthaltende Arzneimittel
CA1076480A (en) * 1975-04-28 1980-04-29 John S. Kent Inert core implant pellet
FR2401173A1 (fr) * 1977-06-27 1979-03-23 Roussel Uclaf Nouveaux steroides, leur procede de preparation et leur application dans la synthese de steroides marques au tritium
DE2818164A1 (de) * 1978-04-21 1979-10-31 Schering Ag 1,3-dibenzoesaeureester des 17alpha- ethinyl-7 alpha -methyl-1,3,5(10)-oestratrien- 1,3,17 beta -triols, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische zusammensetzungen
US4318908A (en) * 1979-12-06 1982-03-09 Kureha Kagaku Kogyo Kabushiki Kaisha Methylated prostaglandin derivatives
DE3144049A1 (de) * 1981-11-03 1983-05-19 Schering Ag, 1000 Berlin Und 4619 Bergkamen 16(beta)-methyl-8(alpha)-oestradiole, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate
FI83087C (fi) * 1984-05-16 1991-05-27 Schering Ag Foerfarande foer framstaellning av terapeutiskt anvaendbara estriol-3,17-diestrar.

Also Published As

Publication number Publication date
CA1255295A (en) 1989-06-06
DE3667982D1 (de) 1990-02-08
AU583160B2 (en) 1989-04-20
JPS62120398A (ja) 1987-06-01
EP0221506B1 (en) 1990-01-03
EP0221506A1 (en) 1987-05-13
IL79710A0 (en) 1986-11-30
DK521786A (da) 1987-05-02
ZA868272B (en) 1988-07-27
US4757062A (en) 1988-07-12
AU6461686A (en) 1987-05-07
GR862633B (en) 1987-03-03
ATE49216T1 (de) 1990-01-15
ES2002058A6 (es) 1988-07-01

Similar Documents

Publication Publication Date Title
BR7604146A (pt) Conjunto aperfeicoado de quadro de distribuicao modular e sistema aperfeicoado de distribuicao de quadros
DK159375C (da) Depotplaster til transdermal administration af clonidin
DK263288A (da) Farmaceutisk praeparat af cefuroxim-axetil
IT1066085B (it) Composizione farmaceutica antinfiammatoria a base di corticosteroidi,particolarmente per il trattamento di manifestazioni infiammatorie di dermatosi,e procedimento per la sua preparazione
FI93350C (fi) Menetelmä uusien farmakologisesti aktiivisten katekolijohdoksien valmistamiseksi
DE3673664D1 (de) 13-substituierte derivate von avermectin-aglyconen.
DK520180A (da) Forankringsfod for eksempelvis trafikmarkeringsstolper
IT1061771B (it) Dispositivo per la somministrazione di anestetici
LU88790I2 (fr) Moxidectin et ses dérivés pharmaceutiquement acceptables
DK521786D0 (da) Substituerede benzoatestere af estrogener
SE7604317L (sv) Fast farmaceutisk doseringsform med fordrojd frigoring och sett att framstella desamma
DK312279A (da) Farmaceutisk formulering af guargummi
BE864124A (fr) Compositions pharmaceutiques analgesiques et anti-inflammatoires
BE862310A (fr) Compositions analgesiques et anti-inflammatoires
DK448587A (da) Stereoisomer form af visse phenylethanolamniderivater
DK522986D0 (da) Fremgangsmaade til indgift af ethanolaminderivater til husdyr
DE68927129T2 (de) Resistzusammensetzung, Phenolverbindung und Chinondiazidsulfonsäureester dieser Phenolverbindung
DK549586D0 (da) Fremgangsmaade til fremstilling af polymerbeton med lavt svind
DK142990C (da) Fremgangsmaade til fremstilling af antibakterielt virksomme aldehydderivater af clavulansyre
FR2336921A1 (fr) Compositions pharmaceutiques anti-inflammatoires
SE7701723L (sv) Analgetiska och anti-inflammatoriska kompositioner
IT1060651B (it) Procedimento ed apparecchiatura per la formatura di un alimentatore di effluente
BE842486A (fr) Compositions analgesiques de levo- ou dextro-propoxyphene et de benzodiazepines et leur preparation
DK150844C (da) Kirurgisk forankringsredskab
JPS5282836A (en) Power edge device for preventing sinking of building structure

Legal Events

Date Code Title Description
AHB Application shelved due to non-payment