DK3630725T3 - Krystallinsk form af n-butyldeoxygalactonojirimycin - Google Patents

Krystallinsk form af n-butyldeoxygalactonojirimycin

Info

Publication number
DK3630725T3
DK3630725T3 DK18728624.0T DK18728624T DK3630725T3 DK 3630725 T3 DK3630725 T3 DK 3630725T3 DK 18728624 T DK18728624 T DK 18728624T DK 3630725 T3 DK3630725 T3 DK 3630725T3
Authority
DK
Denmark
Prior art keywords
butyldeoxygalactonojirimycin
crystalline form
crystalline
Prior art date
Application number
DK18728624.0T
Other languages
English (en)
Inventor
Vitor Oliveira
Ivan Pogorelic
Jean-Paul Roduit
Original Assignee
Idorsia Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Idorsia Pharmaceuticals Ltd filed Critical Idorsia Pharmaceuticals Ltd
Application granted granted Critical
Publication of DK3630725T3 publication Critical patent/DK3630725T3/da

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40Oxygen atoms
    • C07D211/44Oxygen atoms attached in position 4
    • C07D211/46Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Saccharide Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
DK18728624.0T 2017-06-01 2018-05-31 Krystallinsk form af n-butyldeoxygalactonojirimycin DK3630725T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP2017063287 2017-06-01
PCT/EP2018/064365 WO2018220131A1 (en) 2017-06-01 2018-05-31 Crystalline form of n-butyldeoxygalactonojirimycin

Publications (1)

Publication Number Publication Date
DK3630725T3 true DK3630725T3 (da) 2026-02-09

Family

ID=62492649

Family Applications (1)

Application Number Title Priority Date Filing Date
DK18728624.0T DK3630725T3 (da) 2017-06-01 2018-05-31 Krystallinsk form af n-butyldeoxygalactonojirimycin

Country Status (24)

Country Link
US (2) US11306058B2 (da)
EP (1) EP3630725B1 (da)
JP (2) JP6937850B2 (da)
KR (1) KR102612650B1 (da)
CN (1) CN110799497A (da)
AU (1) AU2018278247B2 (da)
CA (1) CA3065147A1 (da)
CL (1) CL2019003478A1 (da)
DK (1) DK3630725T3 (da)
EA (1) EA201992807A1 (da)
FI (1) FI3630725T3 (da)
HR (1) HRP20251697T1 (da)
IL (1) IL270961B2 (da)
LT (1) LT3630725T (da)
MA (1) MA48944B1 (da)
MX (1) MX2019014427A (da)
MY (1) MY201196A (da)
PH (1) PH12019502635A1 (da)
PT (1) PT3630725T (da)
RS (1) RS67675B1 (da)
SI (1) SI3630725T1 (da)
TW (1) TWI770184B (da)
UA (1) UA125938C2 (da)
WO (1) WO2018220131A1 (da)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK3630725T3 (da) * 2017-06-01 2026-02-09 Idorsia Pharmaceuticals Ltd Krystallinsk form af n-butyldeoxygalactonojirimycin
WO2021061701A1 (en) 2019-09-25 2021-04-01 Teva Pharmaceuticals International Gmbh Solid state forms of lucerastat salts and process for preparation thereof
WO2025017212A1 (en) 2023-07-20 2025-01-23 Katholieke Universiteit Leuven Udp-glucose ceramide glucosyltransferase synthase (ugcg) inhibitors in the treatment of cancer
WO2026043459A2 (en) * 2024-08-23 2026-02-26 Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi Capsule formulations comprising migalastat

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1992000277A1 (en) * 1990-06-29 1992-01-09 Nippon Shinyaku Co., Ltd. Piperidine derivative
US6291657B1 (en) 1993-05-13 2001-09-18 Monsanto Company Deoxygalactonojirimycin derivatives
US6274597B1 (en) 1998-06-01 2001-08-14 Mount Sinai School Of Medicine Of New York University Method of enhancing lysosomal α-Galactosidase A
GB0100889D0 (en) 2001-01-12 2001-02-21 Oxford Glycosciences Uk Ltd Compounds
GB0229476D0 (en) 2002-12-17 2003-01-22 Oxford Glycosciences Uk Ltd Novel process
FR2861991B1 (fr) * 2003-11-07 2008-01-18 Centre Nat Rech Scient Utilisation d'inhibiteurs de glucosidase pour une therapie de la mucoviscidose
WO2006037069A1 (en) 2004-09-28 2006-04-06 Allergan, Inc. Compositions comprising nb-dnj, ne-dnj or d-glucaro-delta-lactam and their uses for the treatment of pain and other neurological conditions
EP3782655A1 (en) 2005-05-17 2021-02-24 Amicus Therapeutics, Inc. A method for the treatment of pompe disease using 1-deoxynojirimycin and derivatives
AU2006272497B2 (en) 2005-07-27 2012-07-19 University Of Florida Research Foundation, Inc. Small compounds that correct protein misfolding and uses thereof
ATE479696T1 (de) 2006-04-24 2010-09-15 Amc Amsterdam Verbessertes verfahren zur behandlung von cystischer fibrose
GB0712494D0 (en) 2007-06-27 2007-08-08 Isis Innovation Substrate reduction therapy
ITMI20122090A1 (it) * 2012-12-06 2014-06-07 Dipharma Francis Srl Sintesi di un inibitore delle glicosiltransferasi
DK3630725T3 (da) * 2017-06-01 2026-02-09 Idorsia Pharmaceuticals Ltd Krystallinsk form af n-butyldeoxygalactonojirimycin

Also Published As

Publication number Publication date
WO2018220131A1 (en) 2018-12-06
IL270961A (en) 2020-01-30
TWI770184B (zh) 2022-07-11
AU2018278247B2 (en) 2022-07-28
KR102612650B1 (ko) 2023-12-11
KR20200011992A (ko) 2020-02-04
US11306058B2 (en) 2022-04-19
EP3630725A1 (en) 2020-04-08
PH12019502635A1 (en) 2020-07-13
TW201902876A (zh) 2019-01-16
RS67675B1 (sr) 2026-02-27
HRP20251697T1 (hr) 2026-02-27
JP2020521796A (ja) 2020-07-27
US20220002245A1 (en) 2022-01-06
FI3630725T3 (fi) 2026-01-27
BR112019025125A2 (pt) 2020-07-21
MA48944A (fr) 2020-04-08
IL270961B1 (en) 2024-11-01
AU2018278247A1 (en) 2020-01-16
US20200140385A1 (en) 2020-05-07
EP3630725B1 (en) 2025-10-29
MX2019014427A (es) 2020-02-05
CN110799497A (zh) 2020-02-14
MA48944B1 (fr) 2025-12-31
JP2021185184A (ja) 2021-12-09
JP6937850B2 (ja) 2021-09-22
UA125938C2 (uk) 2022-07-13
JP7373529B2 (ja) 2023-11-02
LT3630725T (lt) 2026-01-12
IL270961B2 (en) 2025-03-01
SI3630725T1 (sl) 2026-01-30
PT3630725T (pt) 2026-01-27
US11713297B2 (en) 2023-08-01
CA3065147A1 (en) 2018-12-06
CL2019003478A1 (es) 2020-06-05
MY201196A (en) 2024-02-09
EA201992807A1 (ru) 2020-05-20

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