DK3411031T3 - Deutererede domperidonpræparater og fremgangsmåder til terapi af lidelser - Google Patents

Deutererede domperidonpræparater og fremgangsmåder til terapi af lidelser Download PDF

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Publication number
DK3411031T3
DK3411031T3 DK17748198.3T DK17748198T DK3411031T3 DK 3411031 T3 DK3411031 T3 DK 3411031T3 DK 17748198 T DK17748198 T DK 17748198T DK 3411031 T3 DK3411031 T3 DK 3411031T3
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DK
Denmark
Prior art keywords
disorders
preparations
therapy
methods
deuterated domperidone
Prior art date
Application number
DK17748198.3T
Other languages
Danish (da)
English (en)
Inventor
Catherine Pearce
Jon Isaacsohn
Piyush Patel
Original Assignee
Cindome Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cindome Pharma Inc filed Critical Cindome Pharma Inc
Application granted granted Critical
Publication of DK3411031T3 publication Critical patent/DK3411031T3/da

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41841,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0087Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4808Preparations in capsules, e.g. of gelatin, of chocolate characterised by the form of the capsule or the structure of the filling; Capsules containing small tablets; Capsules with outer layer for immediate drug release
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B59/00Introduction of isotopes of elements into organic compounds ; Labelled organic compounds per se
    • C07B59/002Heterocyclic compounds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/12Radicals substituted by oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/26Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/05Isotopically modified compounds, e.g. labelled

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Otolaryngology (AREA)
  • Hospice & Palliative Care (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Zoology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK17748198.3T 2016-02-04 2017-02-03 Deutererede domperidonpræparater og fremgangsmåder til terapi af lidelser DK3411031T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201662291198P 2016-02-04 2016-02-04
PCT/US2017/016334 WO2017136617A1 (en) 2016-02-04 2017-02-03 Deuterated domperidone compositions and methods for therapy of disorders

Publications (1)

Publication Number Publication Date
DK3411031T3 true DK3411031T3 (da) 2024-10-21

Family

ID=59501077

Family Applications (2)

Application Number Title Priority Date Filing Date
DK17748198.3T DK3411031T3 (da) 2016-02-04 2017-02-03 Deutererede domperidonpræparater og fremgangsmåder til terapi af lidelser
DK18743261.2T DK3644995T3 (da) 2016-02-04 2018-06-28 Deutererede domperidon-sammensætninger, fremgangsmåder og fremstilling

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK18743261.2T DK3644995T3 (da) 2016-02-04 2018-06-28 Deutererede domperidon-sammensætninger, fremgangsmåder og fremstilling

Country Status (11)

Country Link
US (2) US10266516B2 (enExample)
EP (2) EP3411031B1 (enExample)
JP (3) JP7296185B2 (enExample)
KR (2) KR102851614B1 (enExample)
CN (4) CN108697700B (enExample)
AU (2) AU2017213852B2 (enExample)
BR (2) BR112018016032B1 (enExample)
CA (2) CA3013123A1 (enExample)
DK (2) DK3411031T3 (enExample)
EA (2) EA035515B1 (enExample)
WO (2) WO2017136617A1 (enExample)

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KR20210082480A (ko) * 2018-10-25 2021-07-05 신돔 파마, 인크. 돔페리돈을 함유하는 제제
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US20220307004A1 (en) * 2021-03-29 2022-09-29 The Government Of The United States Of America, As Represented By The Secretary Of The Navy Multi-Enzyme Nanoparticle-Assisted Stable Isotope Incorporation Into Small Molecules by Channeling
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Also Published As

Publication number Publication date
CN111093653B (zh) 2023-06-23
JP2023052045A (ja) 2023-04-11
KR102695402B1 (ko) 2024-08-16
AU2017213852B2 (en) 2021-04-08
EP3644995B1 (en) 2025-05-07
WO2017136617A8 (en) 2017-10-05
DK3644995T3 (da) 2025-08-18
WO2017136617A1 (en) 2017-08-10
KR20180104662A (ko) 2018-09-21
JP2020534246A (ja) 2020-11-26
KR20200044790A (ko) 2020-04-29
CA3013123A1 (en) 2017-08-10
CN108697700A (zh) 2018-10-23
EA202090183A1 (ru) 2020-04-15
US20190241543A1 (en) 2019-08-08
AU2018290905A1 (en) 2020-02-13
CN111093653A (zh) 2020-05-01
JP7296185B2 (ja) 2023-06-22
BR112018016032A2 (pt) 2018-12-26
US20170298046A1 (en) 2017-10-19
KR102851614B1 (ko) 2025-08-29
CN113995755A (zh) 2022-02-01
EP3411031A1 (en) 2018-12-12
CA3055777A1 (en) 2019-01-03
BR112019028185A8 (pt) 2020-08-11
AU2017213852A1 (en) 2018-07-05
BR112018016032B1 (pt) 2024-03-05
JP2019504068A (ja) 2019-02-14
CN116712432A (zh) 2023-09-08
WO2019006078A1 (en) 2019-01-03
US10266516B2 (en) 2019-04-23
JP7602324B2 (ja) 2024-12-18
CN108697700B (zh) 2021-08-17
EP3644995A1 (en) 2020-05-06
AU2018290905B2 (en) 2022-10-06
EA201891727A1 (ru) 2018-12-28
EP3411031B1 (en) 2024-07-24
EP3411031A4 (en) 2019-08-07
BR112019028185A2 (pt) 2020-07-07
EA035515B1 (ru) 2020-06-29
US10590110B2 (en) 2020-03-17

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