MX2009011577A - Composiciones y metodos para distribucion de domperidona a traves de la mucosa. - Google Patents

Composiciones y metodos para distribucion de domperidona a traves de la mucosa.

Info

Publication number
MX2009011577A
MX2009011577A MX2009011577A MX2009011577A MX2009011577A MX 2009011577 A MX2009011577 A MX 2009011577A MX 2009011577 A MX2009011577 A MX 2009011577A MX 2009011577 A MX2009011577 A MX 2009011577A MX 2009011577 A MX2009011577 A MX 2009011577A
Authority
MX
Mexico
Prior art keywords
methods
domperidone
compositions
transmucosal delivery
vomiting
Prior art date
Application number
MX2009011577A
Other languages
English (en)
Inventor
Craig A Aronchick
Original Assignee
Craig A Aronchick
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Craig A Aronchick filed Critical Craig A Aronchick
Publication of MX2009011577A publication Critical patent/MX2009011577A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/006Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/14Drugs for genital or sexual disorders; Contraceptives for lactation disorders, e.g. galactorrhoea

Abstract

Se proporcionan composiciones de domperidona para distribución a través de la mucosa. También se proporcionan métodos para el tratamiento de nausea, vómito y trastornos de motilidad gastrointestinal, y métodos para mejorar la producción de leche materna. Los métodos utilizan composiciones de domperidona formulados para la administración a través de la mucosa, administrados a pacientes en una cantidad efectiva para tratar nausea, vómito o trastornos de motilidad gastrointestinal, o para mejorar la producción de leche materna.
MX2009011577A 2007-04-26 2008-04-25 Composiciones y metodos para distribucion de domperidona a traves de la mucosa. MX2009011577A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US91413507P 2007-04-26 2007-04-26
PCT/US2008/061617 WO2008134540A1 (en) 2007-04-26 2008-04-25 Compositions and methods for transmucosal delivery of domperidone

Publications (1)

Publication Number Publication Date
MX2009011577A true MX2009011577A (es) 2010-03-10

Family

ID=39926093

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2009011577A MX2009011577A (es) 2007-04-26 2008-04-25 Composiciones y metodos para distribucion de domperidona a traves de la mucosa.

Country Status (6)

Country Link
US (1) US20100255096A1 (es)
EP (1) EP2142176A1 (es)
AU (1) AU2008245580A1 (es)
CA (1) CA2685362A1 (es)
MX (1) MX2009011577A (es)
WO (1) WO2008134540A1 (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102670830A (zh) * 2012-05-22 2012-09-19 徐州三源医药科技有限公司 一种催乳汤及制备方法
WO2014105655A1 (en) 2012-12-24 2014-07-03 Neurogastrx, Inc. Methods for treating gi tract disorders
US9844554B2 (en) 2014-06-24 2017-12-19 Neurogastrx, Inc. Prodrugs of metopimazine
CN108697700B (zh) 2016-02-04 2021-08-17 辛多美制药有限公司 氘代多潘立酮组合物和用于治疗病症的方法
US11364226B2 (en) 2017-06-30 2022-06-21 Cinrx Pharma, Llc Deuterated domperidone compositions, methods, and preparation
KR20230169456A (ko) * 2018-10-25 2023-12-15 신돔 파마, 인크. 중수소화 돔페리돈을 함유하는 제제
US10836757B1 (en) 2020-04-02 2020-11-17 Neurogastrx, Inc. Polymorphic forms of metopimazine

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW466119B (en) * 1994-02-28 2001-12-01 Janssen Pharmaceutica Nv Film coated tablet of paracetamol and domperidone
GB9710767D0 (en) * 1996-06-26 1997-07-23 On Ninh Analgesic and anti-inflamatory compositions comprising domperidone and methods of using same
GB9702392D0 (en) * 1997-02-06 1997-03-26 Boots Co Plc Therapeutic agents
US20040043071A1 (en) * 2002-06-21 2004-03-04 Pauletti Giovanni M. Intravaginal mucosal or transmucosal delivery of antimigraine and antinausea drugs
KR20030045473A (ko) * 2001-12-04 2003-06-11 대신제약주식회사 점막부착성을 가지는 의약품 조성물
ATE353635T1 (de) * 2004-09-09 2007-03-15 Medinfar Produtos Farmaceutico Schnell wasserdispergierbare und domperidon enthaltende tabletten

Also Published As

Publication number Publication date
EP2142176A1 (en) 2010-01-13
US20100255096A1 (en) 2010-10-07
AU2008245580A1 (en) 2008-11-06
WO2008134540A1 (en) 2008-11-06
CA2685362A1 (en) 2008-11-06

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal