DK262782A - Fremgangsmaade til fremstilling af n-dihydrothiazolyl-3-quinolincarboxamidderivater - Google Patents
Fremgangsmaade til fremstilling af n-dihydrothiazolyl-3-quinolincarboxamidderivater Download PDFInfo
- Publication number
- DK262782A DK262782A DK262782A DK262782A DK262782A DK 262782 A DK262782 A DK 262782A DK 262782 A DK262782 A DK 262782A DK 262782 A DK262782 A DK 262782A DK 262782 A DK262782 A DK 262782A
- Authority
- DK
- Denmark
- Prior art keywords
- quinolincarboxamide
- dihydrothiazolyl
- derivatives
- preparing
- quinolincarboxamide derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR8111607A FR2507602A1 (fr) | 1981-06-12 | 1981-06-12 | Nouveau derive dihydrothiazole de la quinoleine, ses sels, procede de preparation, application a titre de medicaments et compositions les renfermant |
| FR8111607 | 1981-06-12 | ||
| FR8204331 | 1982-03-15 | ||
| FR8204331A FR2523130A1 (fr) | 1982-03-15 | 1982-03-15 | Nouveaux derives de la n-dihydrothiazolyl-3-quinoleine carboxamide, leurs sels, procede de preparation, application a titre de medicaments et compositions les renfermant |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| DK262782A true DK262782A (da) | 1982-12-13 |
| DK150070B DK150070B (da) | 1986-12-01 |
| DK150070C DK150070C (da) | 1987-11-09 |
Family
ID=26222434
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK262782A DK150070C (da) | 1981-06-12 | 1982-06-11 | Analogifremgangsmaade til fremstilling af n-dihydrothiazolyl-3-quinolincarboxamidderivater |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US4450166A (da) |
| EP (1) | EP0067772B1 (da) |
| KR (1) | KR880000808B1 (da) |
| AU (1) | AU552029B2 (da) |
| CA (1) | CA1216795A (da) |
| DE (1) | DE3262536D1 (da) |
| DK (1) | DK150070C (da) |
| ES (1) | ES8304567A1 (da) |
| FI (1) | FI78087C (da) |
| GR (1) | GR77201B (da) |
| HU (1) | HU190796B (da) |
| IE (1) | IE53520B1 (da) |
| IL (1) | IL65943A (da) |
| MA (1) | MA19488A1 (da) |
| NZ (1) | NZ200931A (da) |
| PT (1) | PT75023B (da) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2557570B1 (fr) * | 1984-01-04 | 1986-04-18 | Adir | Nouveaux derives de la quinoleine, leur procede de preparation et les compositions pharmaceutiques les renfermant |
| FR2566405B1 (fr) * | 1984-06-25 | 1986-09-26 | Roussel Uclaf | Nouveaux derives de l'acide 4-hydroxy 3-quinoleine carboxylique substitues en 2 par une fonction aminee, leur preparation, leur application comme medicaments, les compositions les renfermant et les intermediaires nouveaux obtenus |
| US4602014A (en) * | 1984-07-09 | 1986-07-22 | Ciba-Geigy Corporation | Ring-fused pyrazolo[3,4-d]-pyridin-3-one derivatives as benzodiazepine receptor modulators |
| US4560692A (en) * | 1984-07-18 | 1985-12-24 | Hoffmann-La Roche Inc. | 4-Piperidino-2-phenylquinolines |
| US4786644A (en) * | 1987-11-27 | 1988-11-22 | Hoechst-Roussel Pharmaceuticals Inc. | 1-aryl-3-quinolinecarboxamide |
| BR9908321A (pt) * | 1998-02-26 | 2001-12-18 | Neurogen Corp | Composto |
| MXPA01011173A (es) * | 1999-05-06 | 2002-04-24 | Neurogen Corp | 4-0x0-quinolin-3-carboxamidas sustituidas: ligandos del receptor cerebro de gaba. |
| US20100074949A1 (en) | 2008-08-13 | 2010-03-25 | William Rowe | Pharmaceutical composition and administration thereof |
| ES2656017T3 (es) * | 2004-06-24 | 2018-02-22 | Vertex Pharmaceuticals Incorporated | Moduladores de transportadores del casete de unión a ATP |
| US8354427B2 (en) * | 2004-06-24 | 2013-01-15 | Vertex Pharmaceutical Incorporated | Modulators of ATP-binding cassette transporters |
| JP2009521468A (ja) * | 2005-12-24 | 2009-06-04 | バーテックス ファーマシューティカルズ インコーポレイテッド | Ａｂｃ輸送体の調節因子としてのキノリン−４−オン誘導体 |
| PL1993360T3 (pl) | 2005-12-28 | 2017-08-31 | Vertex Pharmaceuticals Incorporated | Stałe postacie n-[2,4-bis(1,1-dimetyloetylo)-5-hydroksyfenylo]-1,4- dihydro-4-oksochinolino-3-karboksyamidu |
| PL2408750T3 (pl) | 2009-03-20 | 2016-02-29 | Vertex Pharma | Sposób otrzymywania modulatorów błonowego regulatora przewodnictwa swoistego dla mukowiscydozy |
| US8802700B2 (en) | 2010-12-10 | 2014-08-12 | Vertex Pharmaceuticals Incorporated | Modulators of ATP-Binding Cassette transporters |
| CA2865519C (en) | 2012-02-27 | 2018-01-02 | Vertex Pharmaceuticals Incorporated | Pharmaceutical compositions comprising a solid dispersion of n-[2,4-bis(1,1-dimethylethyl0-5-hydroxyphenyl-1]-1,4-dihydro-4-oxoquinolone-3-carboxamide for treating cystic fibrosis |
| EP3204358B1 (en) | 2014-10-07 | 2018-09-19 | Vertex Pharmaceuticals Incorporated | Co-crystals of modulators of cystic fibrosis transmembrane conductance regulator |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR1364605A (fr) * | 1962-03-01 | 1964-06-26 | Procédé de préparation d'amides des acides carboxyliques | |
| FR2281761A1 (fr) * | 1974-08-13 | 1976-03-12 | Roussel Uclaf | Nouveaux derives de l'acide 3-quinoleine carboxylique, leur procede de preparation et leur application comme medicament |
| FR2324304A2 (fr) * | 1975-09-22 | 1977-04-15 | Roussel Uclaf | Nouveaux derives de l'acide 3-quinoleine carboxylique, leur procede de preparation et leur application comme medicament |
| FR2340735A1 (fr) * | 1976-02-11 | 1977-09-09 | Roussel Uclaf | Nouveaux derives de l'acide 3-quinoleine carboxylique, leur procede de preparation et leur application comme medicament |
| FR2377400A2 (fr) * | 1977-01-18 | 1978-08-11 | Roussel Uclaf | Nouveaux derives de l'acide 3-quinoleine carboxylique, leur procede de preparation et leur application comme medicament |
| FR2443467A1 (fr) * | 1978-12-08 | 1980-07-04 | Roussel Uclaf | Nouveaux derives de l'acide 3-quinoleine carboxylique, leur procede de preparation et leur application comme medicament |
| FR2482596A1 (fr) * | 1980-05-19 | 1981-11-20 | Roussel Uclaf | Nouveaux derives de l'acide 4-hydroxy 3-quinoleine carboxylique substitues en 2, leur procede de preparation et leur application comme medicament |
-
1982
- 1982-05-24 HU HU821657A patent/HU190796B/hu not_active IP Right Cessation
- 1982-05-26 MA MA19695A patent/MA19488A1/fr unknown
- 1982-06-01 IL IL65943A patent/IL65943A/xx unknown
- 1982-06-04 ES ES512852A patent/ES8304567A1/es not_active Expired
- 1982-06-08 PT PT75023A patent/PT75023B/pt not_active IP Right Cessation
- 1982-06-09 US US06/386,597 patent/US4450166A/en not_active Expired - Fee Related
- 1982-06-10 FI FI822067A patent/FI78087C/fi not_active IP Right Cessation
- 1982-06-10 GR GR68384A patent/GR77201B/el unknown
- 1982-06-11 NZ NZ200931A patent/NZ200931A/en unknown
- 1982-06-11 AU AU84827/82A patent/AU552029B2/en not_active Ceased
- 1982-06-11 EP EP82401062A patent/EP0067772B1/fr not_active Expired
- 1982-06-11 DK DK262782A patent/DK150070C/da not_active IP Right Cessation
- 1982-06-11 IE IE1394/82A patent/IE53520B1/en unknown
- 1982-06-11 DE DE8282401062T patent/DE3262536D1/de not_active Expired
- 1982-06-11 KR KR8202613A patent/KR880000808B1/ko active
- 1982-06-11 CA CA000405006A patent/CA1216795A/fr not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| FI78087B (fi) | 1989-02-28 |
| KR880000808B1 (ko) | 1988-05-11 |
| US4450166A (en) | 1984-05-22 |
| ES512852A0 (es) | 1983-03-01 |
| PT75023A (fr) | 1982-07-01 |
| ES8304567A1 (es) | 1983-03-01 |
| HU190796B (en) | 1986-11-28 |
| CA1216795A (fr) | 1987-01-20 |
| FI822067A0 (fi) | 1982-06-10 |
| FI78087C (fi) | 1989-06-12 |
| IE53520B1 (en) | 1988-12-07 |
| EP0067772B1 (fr) | 1985-03-13 |
| NZ200931A (en) | 1984-12-14 |
| KR840000541A (ko) | 1984-02-25 |
| AU552029B2 (en) | 1986-05-22 |
| AU8482782A (en) | 1982-12-16 |
| IL65943A (en) | 1985-12-31 |
| IL65943A0 (en) | 1982-09-30 |
| GR77201B (da) | 1984-09-11 |
| DK150070B (da) | 1986-12-01 |
| DE3262536D1 (en) | 1985-04-18 |
| DK150070C (da) | 1987-11-09 |
| IE821394L (en) | 1982-12-12 |
| MA19488A1 (fr) | 1982-12-31 |
| EP0067772A1 (fr) | 1982-12-22 |
| PT75023B (fr) | 1985-05-17 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PBP | Patent lapsed |