DK2101731T3 - ENDOXIFEN FOR USING CANCER TREATMENT - Google Patents

ENDOXIFEN FOR USING CANCER TREATMENT Download PDF

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Publication number
DK2101731T3
DK2101731T3 DK07871563.8T DK07871563T DK2101731T3 DK 2101731 T3 DK2101731 T3 DK 2101731T3 DK 07871563 T DK07871563 T DK 07871563T DK 2101731 T3 DK2101731 T3 DK 2101731T3
Authority
DK
Denmark
Prior art keywords
endoxifen
acid
examples
breast
cancer
Prior art date
Application number
DK07871563.8T
Other languages
Danish (da)
English (en)
Inventor
Ateeq Ahmad
Shoukath M Ali
Moghis U Ahmad
Saifuddin Sheikh
Imran Ahmad
Original Assignee
Jina Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39492975&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK2101731(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Jina Pharmaceuticals Inc filed Critical Jina Pharmaceuticals Inc
Application granted granted Critical
Publication of DK2101731T3 publication Critical patent/DK2101731T3/en

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/138Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/127Synthetic bilayered vehicles, e.g. liposomes or liposomes with cholesterol as the only non-phosphatidyl surfactant
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/19Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles lyophilised, i.e. freeze-dried, solutions or dispersions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D309/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D309/08Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/10Oxygen atoms

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dispersion Chemistry (AREA)
  • Dermatology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Pyrane Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK07871563.8T 2006-11-21 2007-11-21 ENDOXIFEN FOR USING CANCER TREATMENT DK2101731T3 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US86042006P 2006-11-21 2006-11-21
US86078806P 2006-11-22 2006-11-22
PCT/US2007/085443 WO2008070463A2 (en) 2006-11-21 2007-11-21 Endoxifen methods and compositions

Publications (1)

Publication Number Publication Date
DK2101731T3 true DK2101731T3 (en) 2018-04-16

Family

ID=39492975

Family Applications (1)

Application Number Title Priority Date Filing Date
DK07871563.8T DK2101731T3 (en) 2006-11-21 2007-11-21 ENDOXIFEN FOR USING CANCER TREATMENT

Country Status (11)

Country Link
US (2) US9333190B2 (enExample)
EP (1) EP2101731B1 (enExample)
JP (1) JP2010510327A (enExample)
CA (1) CA2669913C (enExample)
DK (1) DK2101731T3 (enExample)
ES (1) ES2665917T3 (enExample)
HU (1) HUE037109T2 (enExample)
IN (1) IN2014MN00139A (enExample)
PL (1) PL2101731T3 (enExample)
PT (1) PT2101731T (enExample)
WO (1) WO2008070463A2 (enExample)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2010510327A (ja) 2006-11-21 2010-04-02 ジャイナ ファーマシューティカルズ,インコーポレーテッド エンドキシフェンの方法および組成物
US20090291134A1 (en) 2006-11-21 2009-11-26 Jina Pharmaceuticals, Inc. Endoxifen methods and compositions in the treatment of psychiatric and neurodegenerative diseases
DK3202420T3 (da) * 2008-12-11 2020-04-06 Besins Healthcare Lu Sarl Transdermale farmaceutiske sammensætninger omfattende en serm
HUE060783T2 (hu) 2011-04-28 2023-04-28 Oncopeptides Ab Citotoxikus dipeptidek liofilizált készítménye
EP2668945A1 (de) 2012-06-01 2013-12-04 Bayer Technology Services GmbH Genotyp- bzw. Phänotyp-basierte Arzeimittelformulierungen
KR102205592B1 (ko) * 2012-10-26 2021-01-20 온코펩타이드즈 아베 멜팔란 플루펜아미드의 동결건조 제제
EP3322406A4 (en) * 2015-07-14 2019-06-12 Atossa Genetics Inc. TRANSPAPILLARY METHOD AND COMPOSITION FOR THE TREATMENT OF BREAST DISEASES
DE102015222031A1 (de) 2015-11-10 2017-05-11 Robert Bosch Gesellschaft Für Medizinische Forschung Mbh Synthese von (Z)-Endoxifenhydrochlorid
US20170304232A1 (en) * 2016-04-20 2017-10-26 Northwestern University Endoxifen For Local Transdermal Therapy To The Breast
KR20200052349A (ko) 2017-09-11 2020-05-14 아토사 테라퓨틱스, 인크. 엔독시펜을 제조 및 사용하는 방법
CN111212631A (zh) * 2017-09-11 2020-05-29 阿托莎医疗公司 局部用组合物和治疗方法
JP7662204B2 (ja) * 2019-07-03 2025-04-15 アトッサ・セラピューティクス・インコーポレイテッド エンドキシフェンの徐放性組成物
WO2021205402A1 (en) 2020-04-10 2021-10-14 Jina Pharmaceuticals, Inc. Endoxifen for the treatment of bipolar i disorder
US12245997B2 (en) 2020-04-10 2025-03-11 Jina Pharmaceuticals, Inc. Endoxifen for the treatment of bipolar I disorder
TW202302073A (zh) * 2021-03-18 2023-01-16 予宇生技股份有限公司 包含帶電脂質的脂質製劑的組合物及製備方法
TW202340135A (zh) 2022-01-12 2023-10-16 美商阿托薩醫療公司 (z)—因多昔芬之組合物及其富集方法
CN119300811A (zh) * 2022-04-26 2025-01-10 阿托萨治疗学公司 高剂量因多昔芬制剂和使用方法

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2817157A1 (de) * 1978-04-17 1979-10-25 Schering Ag Verwendung von antioestrogenen und antigonadotrop wirkenden antiandrogenen zur prophylaxe und therapie der prostatahyperplasie
SK283026B6 (sk) * 1994-08-04 2003-02-04 Quadrant Holdings Cambridge Limited Tuhý časticový prostriedok na terapeutické použitie a spôsob jeho prípravy
US6290991B1 (en) * 1994-12-02 2001-09-18 Quandrant Holdings Cambridge Limited Solid dose delivery vehicle and methods of making same
WO1997040679A1 (en) * 1996-05-01 1997-11-06 Imarx Pharmaceutical Corp. Methods for delivering compounds into a cell
US6090407A (en) * 1997-09-23 2000-07-18 Research Development Foundation Small particle liposome aerosols for delivery of anti-cancer drugs
US7968532B2 (en) 2003-12-15 2011-06-28 Besins Healthcare Luxembourg Treatment of gynecomastia with 4-hydroxy tamoxifen
CA2666322C (en) 2006-10-10 2013-04-23 Jina Pharmaceuticals, Inc. Aqueous systems for the preparation of lipid-based pharmaceutical compounds; compositions, methods, and uses thereof
WO2008048194A1 (en) 2006-10-20 2008-04-24 Yesilogluj Aysegul Yildiz Use of the protein kinase c inhibitor tamoxifen for the treatment of bipolar disorder
CA2669355C (en) 2006-11-06 2012-10-30 Jina Pharmaceuticals, Inc. Guggulphospholipid methods and compositions
US20090291134A1 (en) 2006-11-21 2009-11-26 Jina Pharmaceuticals, Inc. Endoxifen methods and compositions in the treatment of psychiatric and neurodegenerative diseases
JP2010510327A (ja) 2006-11-21 2010-04-02 ジャイナ ファーマシューティカルズ,インコーポレーテッド エンドキシフェンの方法および組成物
JP5720881B2 (ja) 2011-01-31 2015-05-20 東芝ライテック株式会社 Ledランプ点灯装置および照明装置

Also Published As

Publication number Publication date
US9333190B2 (en) 2016-05-10
CA2669913A1 (en) 2008-06-12
US20100112041A1 (en) 2010-05-06
JP2010510327A (ja) 2010-04-02
WO2008070463A3 (en) 2008-11-06
US20160346230A1 (en) 2016-12-01
US10376479B2 (en) 2019-08-13
EP2101731A4 (en) 2011-04-20
CA2669913C (en) 2012-09-18
ES2665917T3 (es) 2018-04-30
WO2008070463A9 (en) 2008-09-18
EP2101731B1 (en) 2018-01-31
EP2101731A2 (en) 2009-09-23
IN2014MN00139A (enExample) 2015-06-19
PT2101731T (pt) 2018-04-18
WO2008070463A2 (en) 2008-06-12
PL2101731T3 (pl) 2018-07-31
HUE037109T2 (hu) 2018-08-28

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