DK171404B1 - C63-Amidderivater af 34-de-(acetylglucosaminyl)-34-deoxy-teicoplaniner, fremgangsmåde til fremstilling heraf, anvendelse af sådanne forbindelser til fremstilling af medikamenter samt farmaceutiske præparater indeholdende forbindelserne - Google Patents

C63-Amidderivater af 34-de-(acetylglucosaminyl)-34-deoxy-teicoplaniner, fremgangsmåde til fremstilling heraf, anvendelse af sådanne forbindelser til fremstilling af medikamenter samt farmaceutiske præparater indeholdende forbindelserne Download PDF

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Publication number
DK171404B1
DK171404B1 DK640489A DK640489A DK171404B1 DK 171404 B1 DK171404 B1 DK 171404B1 DK 640489 A DK640489 A DK 640489A DK 640489 A DK640489 A DK 640489A DK 171404 B1 DK171404 B1 DK 171404B1
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DK
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Prior art keywords
group
hydrogen
formula
decanoyl
branched
Prior art date
Application number
DK640489A
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Danish (da)
English (en)
Other versions
DK640489A (da
DK640489D0 (da
Inventor
Adriano Malabarba
Juergen Kurt Kettenring
Original Assignee
Lepetit Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Lepetit Spa filed Critical Lepetit Spa
Publication of DK640489D0 publication Critical patent/DK640489D0/da
Publication of DK640489A publication Critical patent/DK640489A/da
Application granted granted Critical
Publication of DK171404B1 publication Critical patent/DK171404B1/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/006—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
    • C07K9/008—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Genetics & Genomics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Communicable Diseases (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Cephalosporin Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Electric Stoves And Ranges (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK640489A 1988-12-27 1989-12-18 C63-Amidderivater af 34-de-(acetylglucosaminyl)-34-deoxy-teicoplaniner, fremgangsmåde til fremstilling heraf, anvendelse af sådanne forbindelser til fremstilling af medikamenter samt farmaceutiske præparater indeholdende forbindelserne DK171404B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP88121708 1988-12-27
EP88121708 1988-12-27

Publications (3)

Publication Number Publication Date
DK640489D0 DK640489D0 (da) 1989-12-18
DK640489A DK640489A (da) 1990-06-28
DK171404B1 true DK171404B1 (da) 1996-10-14

Family

ID=8199722

Family Applications (1)

Application Number Title Priority Date Filing Date
DK640489A DK171404B1 (da) 1988-12-27 1989-12-18 C63-Amidderivater af 34-de-(acetylglucosaminyl)-34-deoxy-teicoplaniner, fremgangsmåde til fremstilling heraf, anvendelse af sådanne forbindelser til fremstilling af medikamenter samt farmaceutiske præparater indeholdende forbindelserne

Country Status (19)

Country Link
EP (1) EP0376041B1 (fr)
JP (1) JPH02221298A (fr)
CN (1) CN1043941A (fr)
AT (1) ATE134646T1 (fr)
AU (1) AU629883B2 (fr)
CA (1) CA2006379A1 (fr)
DE (1) DE68925806T2 (fr)
DK (1) DK171404B1 (fr)
ES (1) ES2083374T3 (fr)
FI (1) FI91076C (fr)
GR (1) GR3020070T3 (fr)
HU (1) HU209939B (fr)
IE (1) IE71942B1 (fr)
IL (1) IL92827A (fr)
NO (1) NO178664C (fr)
NZ (1) NZ231863A (fr)
PT (1) PT92672B (fr)
RU (1) RU2068418C1 (fr)
ZA (1) ZA899772B (fr)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU647122B2 (en) * 1990-05-28 1994-03-17 Gruppo Lepetit S.P.A. C63-amide derivatives of 34-de(acetylglucosaminyl)-34-deoxy- teicoplanin and their use as medicaments against bacteria resistant to glycopeptide antibiotics
US5606036A (en) * 1991-03-27 1997-02-25 Gruppo Lepetit Spa Antibiotic A 40926 ester derivatives
WO1993003060A1 (fr) * 1991-07-29 1993-02-18 Gruppo Lepetit S.P.A. Derives amides de l'antibiotique a 40926
US5750509A (en) * 1991-07-29 1998-05-12 Gruppo Lepetit S.P.A. Amide derivatives of antibiotic A 40926
AR021964A1 (es) * 1998-12-23 2002-09-04 Theravance Inc Un compuesto glicopeptidico, composiciones farmaceuticas que los contienen y uso de dichos compuestos glicopeptidicos para la manufactura de un medicamento antibacteriano.
CZ301184B6 (cs) 1998-12-23 2009-12-02 Theravance, Inc. Glykopeptidový derivát a farmaceutické prostredky, které jej obsahují
TWI275594B (en) 2001-08-24 2007-03-11 Theravance Inc Process for preparing vancomycin phosphonate derivatives
TWI312785B (en) 2001-08-24 2009-08-01 Theravance Inc Process for preparing vancomycin derivatives
US20060074014A1 (en) 2002-11-18 2006-04-06 Vicuron Pharmaceuticals Inc. Dalbavancin compositions for treatment of bacterial infections
US7119061B2 (en) 2002-11-18 2006-10-10 Vicuron Pharmaceuticals, Inc. Dalbavancin compositions for treatment of bacterial infections
US6900175B2 (en) 2002-11-18 2005-05-31 Vicuron Pharmaceuticals Inc. Methods of administering dalbavancin for treatment of bacterial infections

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8522574D0 (en) * 1985-09-12 1985-10-16 Lepetit Spa Amides of teicoplanin compounds
GB8529272D0 (en) * 1985-11-28 1986-01-02 Lepetit Spa Teicoplanin derivatives
GB8704847D0 (en) * 1987-03-02 1987-04-08 Lepetit Spa Substituted alkylamides of teicoplanin compounds
GB8711066D0 (en) * 1987-05-11 1987-06-17 Lepetit Spa Teicoplanin derivatives
GB8827202D0 (en) * 1988-11-22 1988-12-29 Lepetit Spa Process for preparing 63-carboxyamides of teicoplanin antibiotics

Also Published As

Publication number Publication date
DE68925806T2 (de) 1996-09-26
IL92827A0 (en) 1990-09-17
ATE134646T1 (de) 1996-03-15
NO895123L (no) 1990-06-28
JPH02221298A (ja) 1990-09-04
DK640489A (da) 1990-06-28
NO178664C (no) 1996-05-08
AU4698489A (en) 1990-07-05
PT92672A (pt) 1990-06-29
ZA899772B (en) 1991-01-30
IE71942B1 (en) 1997-03-12
HUT53376A (en) 1990-10-28
NO178664B (no) 1996-01-29
CN1043941A (zh) 1990-07-18
DE68925806D1 (de) 1996-04-04
EP0376041A2 (fr) 1990-07-04
ES2083374T3 (es) 1996-04-16
NZ231863A (en) 1992-08-26
HU209939B (en) 1994-12-28
IE894143L (en) 1990-06-27
RU2068418C1 (ru) 1996-10-27
GR3020070T3 (en) 1996-08-31
EP0376041B1 (fr) 1996-02-28
CA2006379A1 (fr) 1990-06-27
FI896199A0 (fi) 1989-12-22
FI91076B (fi) 1994-01-31
AU629883B2 (en) 1992-10-15
FI91076C (fi) 1994-05-10
DK640489D0 (da) 1989-12-18
PT92672B (pt) 1996-09-30
NO895123D0 (no) 1989-12-19
HU896772D0 (en) 1990-03-28
IL92827A (en) 1994-08-26
EP0376041A3 (fr) 1991-11-13

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Legal Events

Date Code Title Description
B1 Patent granted (law 1993)
PBP Patent lapsed