DK169676B1 - 4,5,6,7-Tetrahydroisothiazolo[4,5-c]pyridinderivater og farmaceutiske kompositioner deraf - Google Patents
4,5,6,7-Tetrahydroisothiazolo[4,5-c]pyridinderivater og farmaceutiske kompositioner deraf Download PDFInfo
- Publication number
- DK169676B1 DK169676B1 DK121789A DK121789A DK169676B1 DK 169676 B1 DK169676 B1 DK 169676B1 DK 121789 A DK121789 A DK 121789A DK 121789 A DK121789 A DK 121789A DK 169676 B1 DK169676 B1 DK 169676B1
- Authority
- DK
- Denmark
- Prior art keywords
- tetrahydroisothiazolo
- pyridine
- methyl
- propynyloxy
- formula
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Neurosurgery (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Hospice & Palliative Care (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Psychiatry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB888806013A GB8806013D0 (en) | 1988-03-14 | 1988-03-14 | Heterocyclic compounds |
| GB8806013 | 1988-03-14 | ||
| GB888822564A GB8822564D0 (en) | 1988-09-26 | 1988-09-26 | Heterocyclic compounds |
| GB8822564 | 1988-09-26 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| DK121789D0 DK121789D0 (da) | 1989-03-14 |
| DK121789A DK121789A (da) | 1989-09-15 |
| DK169676B1 true DK169676B1 (da) | 1995-01-09 |
Family
ID=26293631
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK121789A DK169676B1 (da) | 1988-03-14 | 1989-03-14 | 4,5,6,7-Tetrahydroisothiazolo[4,5-c]pyridinderivater og farmaceutiske kompositioner deraf |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US4923880A (fr) |
| EP (1) | EP0336555B1 (fr) |
| JP (1) | JPH01275585A (fr) |
| AT (1) | ATE81130T1 (fr) |
| AU (1) | AU630085B2 (fr) |
| CA (1) | CA1337201C (fr) |
| DE (1) | DE68903019T2 (fr) |
| DK (1) | DK169676B1 (fr) |
| ES (1) | ES2052901T3 (fr) |
| FI (1) | FI91411C (fr) |
| GR (1) | GR3006606T3 (fr) |
| IE (1) | IE62782B1 (fr) |
| IL (1) | IL89351A0 (fr) |
| NO (1) | NO177145C (fr) |
| NZ (1) | NZ228182A (fr) |
| PT (1) | PT89992B (fr) |
| ZA (1) | ZA891769B (fr) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2645862B1 (fr) * | 1989-04-18 | 1991-07-12 | Esteve Labor Dr | Derives d'isothiazolo-pyrydone azetidinyl substitues, leur preparation et leur application en tant que medicaments |
| US5574028A (en) * | 1994-10-31 | 1996-11-12 | Eli Lilly And Company | Method for treating anxiety |
| CZ174698A3 (cs) * | 1995-12-07 | 1998-10-14 | Eli Lilly And Company | Léčivo pro léčbu bolesti |
| US20050137222A1 (en) * | 2003-12-18 | 2005-06-23 | H. Lundbeck A/S | Treatment of insomnia in human patients |
| US20110098777A1 (en) * | 2009-10-23 | 2011-04-28 | Silverstone Leon M | Method and apparatus for treatment of neurodegenerative diseases including depression, mild cognitive impairment, and dementia |
| DK3274331T3 (da) | 2015-03-24 | 2020-03-23 | H Lundbeck As | Fremstilling af 4,5,6,7-tetrahydroisozaxolo[5,4-c]pyridin-3-ol |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8314391D0 (en) * | 1983-05-24 | 1983-06-29 | Kefalas As | Heterocyclic compounds |
| IL87709A (en) * | 1987-09-16 | 1992-11-15 | Pfizer | Process for preparing haloalkyl thiazoles and some such novel haloalkyl thiazoles |
| DE3820775A1 (de) * | 1988-06-20 | 1989-12-21 | Thomae Gmbh Dr K | Neue 4,5,7,8-tetrahydro-6h-thiazolo(5,4,-d)azepine, ihre herstellung und ihre verwendung als arzneimittel |
| JP3054738B2 (ja) * | 1988-07-22 | 2000-06-19 | 武田薬品工業株式会社 | チアゾロ［５，４―ｂ］アゼピン誘導体 |
-
1989
- 1989-02-21 IL IL89351A patent/IL89351A0/xx not_active IP Right Cessation
- 1989-02-28 ES ES89301996T patent/ES2052901T3/es not_active Expired - Lifetime
- 1989-02-28 IE IE64889A patent/IE62782B1/en not_active IP Right Cessation
- 1989-02-28 EP EP89301996A patent/EP0336555B1/fr not_active Expired - Lifetime
- 1989-02-28 AT AT89301996T patent/ATE81130T1/de not_active IP Right Cessation
- 1989-02-28 DE DE8989301996T patent/DE68903019T2/de not_active Expired - Lifetime
- 1989-03-01 NZ NZ228182A patent/NZ228182A/xx unknown
- 1989-03-08 ZA ZA891769A patent/ZA891769B/xx unknown
- 1989-03-10 FI FI891155A patent/FI91411C/fi not_active IP Right Cessation
- 1989-03-13 PT PT89992A patent/PT89992B/pt not_active IP Right Cessation
- 1989-03-13 CA CA000593449A patent/CA1337201C/fr not_active Expired - Fee Related
- 1989-03-13 US US07/322,632 patent/US4923880A/en not_active Expired - Fee Related
- 1989-03-13 NO NO891071A patent/NO177145C/no unknown
- 1989-03-14 JP JP1059860A patent/JPH01275585A/ja active Pending
- 1989-03-14 AU AU31262/89A patent/AU630085B2/en not_active Ceased
- 1989-03-14 DK DK121789A patent/DK169676B1/da active
-
1992
- 1992-12-21 GR GR920403014T patent/GR3006606T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| FI91411B (fi) | 1994-03-15 |
| DK121789A (da) | 1989-09-15 |
| PT89992A (pt) | 1989-11-10 |
| AU3126289A (en) | 1989-09-14 |
| IE62782B1 (en) | 1995-02-22 |
| AU630085B2 (en) | 1992-10-22 |
| DK121789D0 (da) | 1989-03-14 |
| NO177145C (no) | 1995-07-26 |
| ATE81130T1 (de) | 1992-10-15 |
| DE68903019T2 (de) | 1993-07-08 |
| EP0336555B1 (fr) | 1992-09-30 |
| FI891155A0 (fi) | 1989-03-10 |
| NO891071D0 (no) | 1989-03-13 |
| NZ228182A (en) | 1990-08-28 |
| FI891155A (fi) | 1989-09-15 |
| ES2052901T3 (es) | 1994-07-16 |
| GR3006606T3 (fr) | 1993-06-30 |
| FI91411C (fi) | 1994-06-27 |
| NO177145B (no) | 1995-04-18 |
| ZA891769B (en) | 1989-12-27 |
| NO891071L (no) | 1989-09-15 |
| DE68903019D1 (de) | 1992-11-05 |
| JPH01275585A (ja) | 1989-11-06 |
| CA1337201C (fr) | 1995-10-03 |
| IE890648L (en) | 1989-09-14 |
| PT89992B (pt) | 1994-05-31 |
| IL89351A0 (en) | 1989-09-10 |
| EP0336555A1 (fr) | 1989-10-11 |
| US4923880A (en) | 1990-05-08 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DE60316542T2 (de) | 7-azaindole als inhibitoren c-jun n-terminaler kinasen zur behandlung neurodegenerativer störungen | |
| JP2016535788A5 (fr) | ||
| JP2016535788A (ja) | Ｎ−ベンジルトリプタンスリン誘導体、ならびにその調製方法および利用 | |
| JP2009545594A (ja) | 改善された効能、安定性および安全性を有する疑似塩基ベンゾ［ｃ］フェナントリジン | |
| WO2010058314A1 (fr) | Hydroxyquinolin-2(1h)-ones et leurs dérivés | |
| JP2002513793A (ja) | 新規ｎ−オキシド | |
| JPH08311067A (ja) | 新規な複素環式スピロ化合物、それらの製造方法およびそれらを含有する医薬組成物 | |
| DK169676B1 (da) | 4,5,6,7-Tetrahydroisothiazolo[4,5-c]pyridinderivater og farmaceutiske kompositioner deraf | |
| TW201141873A (en) | 2,5,7-substituted oxazolopyrimidine derivatives | |
| JP2010095550A (ja) | キノリン誘導体 | |
| JPH064616B2 (ja) | ２−（ピペラジニル）−２−オキソエチレン−置換フラボノイド誘導体、その製法およびそれを含有する医薬組成物 | |
| KR20010042904A (ko) | 광학 활성 테트라하이드로벤즈인돌 유도체 | |
| KR20120112726A (ko) | ５?ｈｔ６ 수용체 리간드인 술폰 화합물 | |
| US9573921B2 (en) | Substituted N, N-dimethylaminoalkyl ethers of isoflavanone oximes as H1-receptor antagonists | |
| JPH08827B2 (ja) | 精神弛緩剤の２−置換パーヒドロ−１Ｈ−ピリド［１，２−ａピラジン | |
| DK166281B (da) | Tetrahydroisoxazoloe4,5-caapyridin derivater og farmaceutisk acceptable syreadditionssalte deraf, farmaceutiske praeparater indeholdende disse forbindelser, og fremgangsmaade til deres fremstilling | |
| CA2048959C (fr) | Les 3-(1,2-benzisoxazol-3-yl)-4-pyridinamines et leurs derives | |
| DK164913B (da) | 5,6,7,8-tetrahydro-4h-isoxazol oe4,5-caa azepin-derivater, isomere og farmaceutisk acceptable syreadditionssalte deraf, fremgangsmaader til deres fremstilling, og farmaceutiske praeparater indeholdende disse forbindelser | |
| JP2744224B2 (ja) | ビス−アザ−二環式抗不安薬の製法 | |
| CN110003033B (zh) | 氟比洛芬查尔酮曼尼希碱类化合物、其制备方法和用途 | |
| HU226059B1 (en) | Novel disubstituted trans-3,4,4a,5,6,10b-hexahydro-2h-naphto[1,2-b][1,4]oxazine derivatives, process for producing them and pharmaceutical compositions containing them | |
| FR2605008A1 (fr) | Derives d'imidazo (4,5-b)pyridinone-2, leur preparation et leur application en therapeutique | |
| DK158311B (da) | Analogifremgangsmaade til fremstilling af hexahydrobenzopyrano(3,2-c)pyridiner | |
| WO1992015553A1 (fr) | Derive de trialkylamine et adjuvant de motilite de l'appareil digestif le contenant | |
| CN117820309A (zh) | 一种哌嗪基-杂环化合物及其用途 |