DK163519B - Analogifremgangsmaade til fremstilling af 17alfa-alkyl-17beta-hydroxy-1alfa-methyl-4-androsten-3-oner - Google Patents

Analogifremgangsmaade til fremstilling af 17alfa-alkyl-17beta-hydroxy-1alfa-methyl-4-androsten-3-oner Download PDF

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Publication number
DK163519B
DK163519B DK164182A DK164182A DK163519B DK 163519 B DK163519 B DK 163519B DK 164182 A DK164182 A DK 164182A DK 164182 A DK164182 A DK 164182A DK 163519 B DK163519 B DK 163519B
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DK
Denmark
Prior art keywords
androsten
methyl
hydroxy
alkyl
pentyl
Prior art date
Application number
DK164182A
Other languages
Danish (da)
English (en)
Other versions
DK164182A (da
Inventor
Henry Laurent
Annerose Schleusener
Manfred Albring
Rudolf Wiechert
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Publication of DK164182A publication Critical patent/DK164182A/da
Publication of DK163519B publication Critical patent/DK163519B/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J21/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J21/005—Ketals
    • C07J21/006—Ketals at position 3
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003—Androstane derivatives
    • C07J1/0033—Androstane derivatives substituted in position 17 alfa and 17 beta
    • C07J1/0037—Androstane derivatives substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being a saturated hydrocarbon group

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Obesity (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hematology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK164182A 1981-04-13 1982-04-13 Analogifremgangsmaade til fremstilling af 17alfa-alkyl-17beta-hydroxy-1alfa-methyl-4-androsten-3-oner DK163519B (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19813115996 DE3115996A1 (de) 1981-04-13 1981-04-13 17(alpha)-alkyl-17(beta)-hydroxy-1(alpha)- methyl-4-androsten-3-one-.verfahren zu ihrer herstellung und pharmazeutische praeparate, die diese verbindungen enthalten
DE3115996 1981-04-13

Publications (2)

Publication Number Publication Date
DK164182A DK164182A (da) 1982-10-14
DK163519B true DK163519B (da) 1992-03-09

Family

ID=6130599

Family Applications (1)

Application Number Title Priority Date Filing Date
DK164182A DK163519B (da) 1981-04-13 1982-04-13 Analogifremgangsmaade til fremstilling af 17alfa-alkyl-17beta-hydroxy-1alfa-methyl-4-androsten-3-oner

Country Status (10)

Country Link
US (1) US4673673A (fr)
EP (1) EP0062903B1 (fr)
JP (1) JPS57179197A (fr)
AT (1) ATE22085T1 (fr)
DE (2) DE3115996A1 (fr)
DK (1) DK163519B (fr)
ES (1) ES511253A0 (fr)
GB (1) GB2098991A (fr)
GR (1) GR75456B (fr)
IE (1) IE53012B1 (fr)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1989011543A1 (fr) * 1988-05-25 1989-11-30 Hyman Edward S Detection de bacteries dans l'urine du cheval
US5616670A (en) * 1993-11-10 1997-04-01 Minnesota Mining And Manufacturing Company Pressure sensitive adhesives with good oily surface adhesion
US5602221A (en) * 1993-11-10 1997-02-11 Minnesota Mining And Manufacturing Company Pressure sensitive adhesives with good low energy surface adhesion
US5683798A (en) * 1993-11-10 1997-11-04 Minnesota Mining And Manufacturing Company Tackified pressure sensitive adhesives
US5654387A (en) * 1993-11-10 1997-08-05 Minnesota Mining And Manufacturing Company Pressure sensitive adhesives
US5620795A (en) * 1993-11-10 1997-04-15 Minnesota Mining And Manufacturing Company Adhesives containing electrically conductive agents
DE69519368T2 (de) * 1994-01-06 2001-03-08 Stanford Res Inst Int Neue antiandrogenen mitteln pharmazeutische präparate und verwendungen davon

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1223837B (de) * 1963-04-17 1966-09-01 Schering Ag Verfahren zur Herstellung von 1alpha-Methyl-delta 4-3-ketosteroiden
US3391168A (en) * 1965-08-23 1968-07-02 Searle & Co 1, 17-dimethyl-5-androstane-3beta, 17beta-diol and esters thereof
DE2046640C3 (de) * 1970-09-14 1973-10-18 Schering Ag Verfahren zur Herstellung von Delta hoch 4 -3-Oxo-l alpha-methyl·Steroiden
US3705180A (en) * 1971-09-02 1972-12-05 Paul D Klimstra 17-oxygenate-2-alpha-methyl-2-methylen-5 alpha-androstan-3-ones and intermediates
US4039669A (en) * 1975-08-01 1977-08-02 Sterling Drug Inc. Composition for topical application and use thereof
DE2943776A1 (de) * 1979-10-26 1981-05-14 Schering Ag Berlin Und Bergkamen, 1000 Berlin 17 (alpha) -alkylsteroide, diese enthaltende praeparate sowie verfahren zu ihrer herstellung

Also Published As

Publication number Publication date
DK164182A (da) 1982-10-14
EP0062903B1 (fr) 1986-09-10
DE3273108D1 (en) 1986-10-16
IE820847L (en) 1982-10-13
JPS57179197A (en) 1982-11-04
JPH033677B2 (fr) 1991-01-21
GR75456B (fr) 1984-07-19
ES8303450A1 (es) 1983-02-16
DE3115996A1 (de) 1982-11-04
GB2098991A (en) 1982-12-01
US4673673A (en) 1987-06-16
ATE22085T1 (de) 1986-09-15
ES511253A0 (es) 1983-02-16
EP0062903A1 (fr) 1982-10-20
IE53012B1 (en) 1988-05-11

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Legal Events

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PHB Application deemed withdrawn due to non-payment or other reasons