DK159852C - Fremgangsmaade til fremstilling af penicillansyre-1,1-dioxid eller basesalte eller in vivo let hydrolyserbare estre deraf - Google Patents

Fremgangsmaade til fremstilling af penicillansyre-1,1-dioxid eller basesalte eller in vivo let hydrolyserbare estre deraf

Info

Publication number
DK159852C
DK159852C DK092680A DK92680A DK159852C DK 159852 C DK159852 C DK 159852C DK 092680 A DK092680 A DK 092680A DK 92680 A DK92680 A DK 92680A DK 159852 C DK159852 C DK 159852C
Authority
DK
Denmark
Prior art keywords
hydraulizable
vivo
esters
dioxide
procedure
Prior art date
Application number
DK092680A
Other languages
Danish (da)
English (en)
Other versions
DK92680A (da
DK159852B (da
Inventor
Bernard Shields Moore
Ronnie D Carroll
Robert Alfred Volkmann
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DK92680A publication Critical patent/DK92680A/da
Publication of DK159852B publication Critical patent/DK159852B/da
Application granted granted Critical
Publication of DK159852C publication Critical patent/DK159852C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cosmetics (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
DK092680A 1979-03-05 1980-03-04 Fremgangsmaade til fremstilling af penicillansyre-1,1-dioxid eller basesalte eller in vivo let hydrolyserbare estre deraf DK159852C (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US1780879A 1979-03-05 1979-03-05
US1781079A 1979-03-05 1979-03-05
US1781079 1979-03-05
US1780879 1979-03-05

Publications (3)

Publication Number Publication Date
DK92680A DK92680A (da) 1980-09-06
DK159852B DK159852B (da) 1990-12-17
DK159852C true DK159852C (da) 1991-05-06

Family

ID=26690337

Family Applications (2)

Application Number Title Priority Date Filing Date
DK092680A DK159852C (da) 1979-03-05 1980-03-04 Fremgangsmaade til fremstilling af penicillansyre-1,1-dioxid eller basesalte eller in vivo let hydrolyserbare estre deraf
DK145690A DK166353C (da) 1979-03-05 1990-06-14 Penicillansyre-1,1-dioxid-derivater

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK145690A DK166353C (da) 1979-03-05 1990-06-14 Penicillansyre-1,1-dioxid-derivater

Country Status (36)

Country Link
KR (1) KR850001339B1 (de)
AR (1) AR225031A1 (de)
AT (1) AT366693B (de)
AU (1) AU522572B2 (de)
BG (1) BG33292A3 (de)
CH (1) CH644608A5 (de)
CS (1) CS215130B2 (de)
DD (1) DD149367A5 (de)
DE (1) DE3008257C2 (de)
DK (2) DK159852C (de)
EG (1) EG14437A (de)
ES (1) ES489185A0 (de)
FI (1) FI70024C (de)
FR (1) FR2450836B1 (de)
GB (1) GB2045755B (de)
GR (1) GR67234B (de)
HK (1) HK66587A (de)
HU (1) HU186304B (de)
IE (1) IE49535B1 (de)
IL (1) IL59515A (de)
IN (1) IN153685B (de)
IT (1) IT1130300B (de)
KE (1) KE3464A (de)
LU (1) LU82215A1 (de)
MX (1) MX6032E (de)
MY (1) MY8500319A (de)
NL (1) NL180317C (de)
NO (2) NO800618L (de)
PL (1) PL125197B1 (de)
PT (1) PT70897A (de)
RO (1) RO80112A (de)
SE (2) SE449103B (de)
SG (1) SG55884G (de)
SU (1) SU1192626A3 (de)
UA (1) UA6342A1 (de)
YU (1) YU42328B (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IN159362B (de) * 1981-03-23 1987-05-09 Pfizer
US4419284A (en) * 1981-03-23 1983-12-06 Pfizer Inc. Preparation of halomethyl esters (and related esters) of penicillanic acid 1,1-dioxide
PT76526B (en) * 1982-04-19 1986-01-21 Gist Brocades Nv Preparation of 6-alpha-bromo- and/or 6,6-dibromopenicillanic acid 1,1-dioxides
IT1190897B (it) * 1982-06-29 1988-02-24 Opos Biochimica Srl Procedimento per la preparazione dell'estere 1-etossicarbonilossietilico dell'acido 6-(d(-)-alfa aminoalfa fenilacetamido)-penicillanico
US4606865A (en) * 1982-09-20 1986-08-19 Astra Lakemedel Aktiebolag Methods for the preparation of α-bromodiethylcarbonate
EP0139048A1 (de) * 1983-10-18 1985-05-02 Gist-Brocades N.V. Verfahren zur Dehalogenierung von 6,6-Dibromopenicillansäure-1,1-Dioxyd
EP0139047A1 (de) * 1983-10-18 1985-05-02 Gist-Brocades N.V. Verfahren zur Herstellung von 6,6-Dibromopenicillansäure-1,1-Dioxyd
US4596677A (en) * 1984-04-06 1986-06-24 Bristol-Myers Company Anhydropenicillin intermediates

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IN149747B (de) * 1977-06-07 1982-04-03 Pfizer
CA1158639A (en) * 1978-12-11 1983-12-13 Eric M. Gordon 6-bromopenicillanic acid sulfone
DE3068390D1 (en) * 1979-01-10 1984-08-09 Beecham Group Plc Penicillin derivatives, process for their preparation and pharmaceutical compositions containing certain of these compounds
IE49880B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd Penicillin derivatives

Also Published As

Publication number Publication date
GB2045755A (en) 1980-11-05
KR850001339B1 (ko) 1985-09-19
NL180317C (nl) 1987-02-02
MX6032E (es) 1984-10-04
AU5610480A (en) 1980-09-11
DK92680A (da) 1980-09-06
FI70024C (fi) 1986-09-12
AR225031A1 (es) 1982-02-15
FR2450836A1 (fr) 1980-10-03
SE8000512L (sv) 1980-09-06
LU82215A1 (fr) 1980-09-24
ATA119080A (de) 1981-09-15
HU186304B (en) 1985-07-29
AU522572B2 (en) 1982-06-17
PL125197B1 (en) 1983-04-30
UA6342A1 (uk) 1994-12-29
NO800618L (no) 1980-09-08
IL59515A (en) 1983-02-23
BG33292A3 (en) 1983-01-14
IT8020367A0 (it) 1980-03-05
IE49535B1 (en) 1985-10-16
DK145690A (da) 1990-06-14
SG55884G (en) 1985-03-08
CS215130B2 (en) 1982-07-30
FI70024B (fi) 1986-01-31
DK166353C (da) 1993-09-06
DK166353B (da) 1993-04-13
SE8603309L (sv) 1986-08-04
YU42328B (en) 1988-08-31
AT366693B (de) 1982-04-26
CH644608A5 (de) 1984-08-15
YU58580A (en) 1983-02-28
PT70897A (en) 1980-04-01
NL180317B (nl) 1986-09-01
NL8001285A (nl) 1980-09-09
ES8103094A1 (es) 1981-02-16
SE449103B (sv) 1987-04-06
DE3008257A1 (de) 1980-09-11
EG14437A (en) 1984-09-30
IE800429L (en) 1980-09-05
IL59515A0 (en) 1980-06-30
MY8500319A (en) 1985-12-31
GR67234B (de) 1981-06-25
GB2045755B (en) 1983-01-26
HK66587A (en) 1987-09-25
DE3008257C2 (de) 1984-03-01
FI800661A (fi) 1980-09-06
NO823127L (no) 1980-09-08
SE8603309D0 (sv) 1986-08-04
KE3464A (en) 1984-10-12
RO80112A (ro) 1982-10-26
DD149367A5 (de) 1981-07-08
FR2450836B1 (fr) 1986-03-21
DK145690D0 (da) 1990-06-14
IN153685B (de) 1984-08-04
PL222448A1 (de) 1981-01-02
SU1192626A3 (ru) 1985-11-15
ES489185A0 (es) 1981-02-16
DK159852B (da) 1990-12-17
IT1130300B (it) 1986-06-11

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PUP Patent expired