DK158786C - Analogifremgangsmaade til fremstilling af 1alfa-hydroxyvitamin d3 eller diacetatet deraf - Google Patents

Analogifremgangsmaade til fremstilling af 1alfa-hydroxyvitamin d3 eller diacetatet deraf

Info

Publication number
DK158786C
DK158786C DK009474A DK9474A DK158786C DK 158786 C DK158786 C DK 158786C DK 009474 A DK009474 A DK 009474A DK 9474 A DK9474 A DK 9474A DK 158786 C DK158786 C DK 158786C
Authority
DK
Denmark
Prior art keywords
1alfa
hydroxyvitamin
diacetate
analogue
preparation
Prior art date
Application number
DK009474A
Other languages
English (en)
Other versions
DK158786B (da
Inventor
Derek Harold Richard Barton
Ezzio Rizzardo
Robert Henry Hesse
Original Assignee
Res Inst Medicine Chem
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27348128&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK158786(C) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Res Inst Medicine Chem filed Critical Res Inst Medicine Chem
Priority claimed from KR7401148A external-priority patent/KR790000218B1/ko
Publication of DK158786B publication Critical patent/DK158786B/da
Application granted granted Critical
Publication of DK158786C publication Critical patent/DK158786C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C401/00—Irradiation products of cholesterol or its derivatives; Vitamin D derivatives, 9,10-seco cyclopenta[a]phenanthrene or analogues obtained by chemical preparation without irradiation

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicinal Preparation (AREA)
  • Feed For Specific Animals (AREA)
  • Fodder In General (AREA)
DK009474A 1973-01-10 1974-01-09 Analogifremgangsmaade til fremstilling af 1alfa-hydroxyvitamin d3 eller diacetatet deraf DK158786C (da)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US32246273A 1973-01-10 1973-01-10
US32246273 1973-01-10
US362339A US3901928A (en) 1973-01-10 1973-05-21 1' ,3' -dihydroxy steroid-5-enes method of preparing same and their use for preparing 1' -hydroxy-25-hydrogen vitamin d compounds
US36233973 1973-05-21
KR7401148A KR790000218B1 (en) 1973-01-10 1974-01-09 Process for preparation of 1 , 3 -dihy droxy steroid-5-enes
KR740001148 1974-01-09

Publications (2)

Publication Number Publication Date
DK158786B DK158786B (da) 1990-07-16
DK158786C true DK158786C (da) 1990-11-26

Family

ID=27348128

Family Applications (1)

Application Number Title Priority Date Filing Date
DK009474A DK158786C (da) 1973-01-10 1974-01-09 Analogifremgangsmaade til fremstilling af 1alfa-hydroxyvitamin d3 eller diacetatet deraf

Country Status (19)

Country Link
US (1) US3901928A (da)
JP (4) JPS5745740B2 (da)
AR (1) AR213608A1 (da)
BE (1) BE809578A (da)
CA (1) CA1055011A (da)
CH (1) CH603571A5 (da)
DE (2) DE2463203C2 (da)
DK (1) DK158786C (da)
ES (1) ES422140A1 (da)
FR (1) FR2213053B1 (da)
GB (1) GB1463985A (da)
HK (1) HK98589A (da)
IE (1) IE40496B1 (da)
LU (1) LU69133A1 (da)
MY (1) MY104375A (da)
NL (1) NL187010C (da)
PH (1) PH14419A (da)
SE (1) SE419981B (da)
SG (1) SG68389G (da)

Families Citing this family (36)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA74158B (en) * 1973-01-10 1975-03-26 Res Inst Medicine Chem Chemical process
US4022891A (en) * 1974-06-18 1977-05-10 Teijin Limited Novel 1α,24-dihydroxycholecalciferol compositions, novel precursors thereof, and processes for preparing them
US4004003A (en) * 1974-08-28 1977-01-18 The Upjohn Company 25-Hydroxycalciferol compounds for treatment of steroid-induced osteoporosis
US3993675A (en) * 1975-02-24 1976-11-23 Hoffmann-La Roche Inc. Process for the preparation of 1α,25-dihydroxycholecalciferol
JPS5265261A (en) * 1975-11-27 1977-05-30 Teijin Ltd Synthesis of 1alpha-hyaroxy-provitamine d compounds
JPS5265262A (en) * 1975-11-27 1977-05-30 Teijin Ltd Synthesis of 1alpha acyloxy-provitamine d compounds
US4021423A (en) * 1976-03-08 1977-05-03 Hoffmann-La Roche Inc. Syntheses of 24R,25- and 24S,25-dihydroxycholecalciferol
CH626336A5 (en) * 1976-03-08 1981-11-13 Hoffmann La Roche Process for the preparation of cholecalciferol derivatives
GB1583749A (en) * 1976-06-03 1981-02-04 Res Inst Medicine Chem Vitamin d derivatives
US4046760A (en) * 1976-07-01 1977-09-06 Merck & Co., Inc. Process for preparing 1-α-hydroxy cholesterol derivatives
IT1088094B (it) * 1976-10-14 1985-06-04 Hoffmann La Roche Derivati del pregnano
US4098801A (en) * 1977-01-26 1978-07-04 Hoffmann-La Roche Inc. Synthesis of 1α-hydroxylated derivatives of cholesterol
CH638215A5 (de) * 1977-02-04 1983-09-15 Hoffmann La Roche Oxadiazolopyrimidin-derivate.
US4218489A (en) * 1977-06-08 1980-08-19 Z-L Limited Partnership Antioxidants, antioxidant compositions and methods of preparing and using same
US4157984A (en) * 1977-06-08 1979-06-12 Z-L Limited Antioxidants, antioxidant compositions and methods of preparing and using same
JPS5452717A (en) * 1977-09-29 1979-04-25 Chugai Pharmaceut Co Ltd Stable oily pharmaceuticals containing 1alpha-hydroxyvitamin d
US4260549A (en) * 1979-05-21 1981-04-07 Wisconsin Alumni Research Foundation Process for preparing 1α-hydroxylated compounds
US4195027A (en) * 1978-01-16 1980-03-25 Wisconsin Alumni Research Foundation Process for preparing 1α-hydroxylated compounds
US4199518A (en) * 1978-03-30 1980-04-22 Diamond Shamrock Corporation 1α,3β-Dihydroxy-steroid-5-enes from 1α,2α-epoxy-steroid-4,6-dien-3-ones
JPS557215A (en) * 1978-06-30 1980-01-19 Teijin Ltd Preparation of active vitamin d3 or its oh-protected derivative and/or its corresponding previtamin d3 or its oh-protected derivative
LU80545A1 (de) * 1978-11-17 1980-06-05 Hoffmann La Roche Verfahren zur herstellung von 1a,3s-dihydroxy->5-steroiden
US4284577A (en) * 1979-02-16 1981-08-18 Sachiko Yamada Novel vitamin D3 derivative and process for preparing the same
FR2457282A1 (fr) * 1979-05-23 1980-12-19 Roussel Uclaf Nouveau derive du 1a,25 dihydroxy cholecalciferol, son procede de preparation et son application comme medicament
EP0028484B1 (en) * 1979-10-23 1985-08-14 Teijin Limited Process for the preparation of active-type vitamin d3 compounds and of the cholesta-5,7-diene precursors, and products so obtained
ATE19623T1 (de) * 1981-07-17 1986-05-15 Duphar Int Res Verfahren zur herstellung von 1-alpha-hydroxy vitamin d oder 1-alpha hydroxy previtamin d derivaten und previtamin d oder tachysteroladdukten mit geeigneten dienophilen.
JPS5856646A (ja) * 1981-09-26 1983-04-04 Tatsuo Suda 産卵めんどりの初産促進方法、初産促進剤及びそのための飼料組成物
CA1272953A (en) 1984-10-08 1990-08-21 Yuji Makino Pharmaceutical composition for external use containing active-type vitamin d.sub.3
JPS61189229A (ja) * 1985-02-18 1986-08-22 Tokai Kapuseru Kk 安定な１α−ヒドロキシビタミンＤ類製剤
JPH0749435B2 (ja) * 1988-07-04 1995-05-31 帝人株式会社 １α，３β，２４−トリヒドロキシ−△▲上５▼−ステロイド類の製造方法
JP2525478B2 (ja) * 1989-03-01 1996-08-21 帝人株式会社 安定性の改良された活性型ビタミンｄ▲下３▼類固型製剤
KR960013798B1 (ko) * 1992-04-24 1996-10-10 재단법인 한국전자통신연구소 평면 도파로형 공간 스위치
AU666529B2 (en) * 1992-04-24 1996-02-15 Wisconsin Alumni Research Foundation Method of treating osteoporosis with 1 alpha, 24 (R)-dihydroxy-22 (E)-dehydro-vitamin D3
US5194431A (en) 1992-07-08 1993-03-16 Wisconsin Alumni Research Foundation 24-cyclopropane vitamin D derivatives
US7148211B2 (en) * 2002-09-18 2006-12-12 Genzyme Corporation Formulation for lipophilic agents
US20060270640A1 (en) * 2004-02-18 2006-11-30 Mercian Corporation Method of preventing, medicating, and/or treating hypocalcemia of domestic mammal
CN115785182B (zh) * 2022-11-29 2024-06-21 浙江工业大学 一种1α-羟基胆固醇的制备方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3697559A (en) * 1971-02-25 1972-10-10 Wisconsin Alumni Res Found 1,25-dihydroxycholecalciferol
US3741996A (en) * 1971-12-02 1973-06-26 Wisconsin Alumni Res Found 1{60 -hydroxycholecalciferol

Also Published As

Publication number Publication date
JPS581116B2 (ja) 1983-01-10
JPS50100045A (da) 1975-08-08
GB1463985A (en) 1977-02-09
HK98589A (en) 1989-12-22
DE2400931A1 (de) 1974-07-25
CA1055011A (en) 1979-05-22
IE40496L (en) 1974-07-10
NL187010B (nl) 1990-12-03
FR2213053A1 (da) 1974-08-02
DE2400931C2 (da) 1987-10-29
JPS4995956A (da) 1974-09-11
IE40496B1 (en) 1979-06-20
NL7400282A (da) 1974-07-12
DE2463203C2 (da) 1987-06-04
SG68389G (en) 1990-01-26
NL187010C (nl) 1993-12-16
MY104375A (en) 1994-03-31
ES422140A1 (es) 1976-08-01
JPS51110554A (da) 1976-09-30
JPS50100216A (da) 1975-08-08
DK158786B (da) 1990-07-16
FR2213053B1 (da) 1976-12-10
PH14419A (en) 1981-07-10
AU6434974A (en) 1975-07-10
CH603571A5 (da) 1978-08-31
LU69133A1 (da) 1974-04-02
SE419981B (sv) 1981-09-07
JPS5854160B2 (ja) 1983-12-02
BE809578A (fr) 1974-07-09
JPS5745740B2 (da) 1982-09-29
AR213608A1 (es) 1979-02-28
US3901928A (en) 1975-08-26

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