DK1525198T3 - Acyloxypyrrolidinderivater og anvendelse af disse i egenskab af ligander for AVP's V1b-eller V1a-receptorer - Google Patents

Acyloxypyrrolidinderivater og anvendelse af disse i egenskab af ligander for AVP's V1b-eller V1a-receptorer

Info

Publication number
DK1525198T3
DK1525198T3 DK03753652T DK03753652T DK1525198T3 DK 1525198 T3 DK1525198 T3 DK 1525198T3 DK 03753652 T DK03753652 T DK 03753652T DK 03753652 T DK03753652 T DK 03753652T DK 1525198 T3 DK1525198 T3 DK 1525198T3
Authority
DK
Denmark
Prior art keywords
avp
ligands
receptors
acyloxypyrrolidine
derivatives
Prior art date
Application number
DK03753652T
Other languages
Danish (da)
English (en)
Inventor
Alain Aulombard
Georges Garcia
Antoine Pradines
Gal Claudine Serradeil-Le
Jean Wagnon
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Application granted granted Critical
Publication of DK1525198T3 publication Critical patent/DK1525198T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/06—Antiabortive agents; Labour repressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
DK03753652T 2002-07-19 2003-07-17 Acyloxypyrrolidinderivater og anvendelse af disse i egenskab af ligander for AVP's V1b-eller V1a-receptorer DK1525198T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0209242A FR2842527B1 (fr) 2002-07-19 2002-07-19 Derives d'acyloxypyrolidine, leur preparation et leur application en therapeutique

Publications (1)

Publication Number Publication Date
DK1525198T3 true DK1525198T3 (da) 2006-04-18

Family

ID=29797610

Family Applications (1)

Application Number Title Priority Date Filing Date
DK03753652T DK1525198T3 (da) 2002-07-19 2003-07-17 Acyloxypyrrolidinderivater og anvendelse af disse i egenskab af ligander for AVP's V1b-eller V1a-receptorer

Country Status (28)

Country Link
US (1) US7202267B2 (is)
EP (1) EP1525198B1 (is)
JP (1) JP4264414B2 (is)
CN (1) CN100425608C (is)
AR (1) AR040571A1 (is)
AT (1) ATE312092T1 (is)
AU (1) AU2003271815B8 (is)
BR (1) BR0312800A (is)
CA (1) CA2492224A1 (is)
DE (1) DE60302670T2 (is)
DK (1) DK1525198T3 (is)
EA (1) EA008444B1 (is)
ES (1) ES2254962T3 (is)
FR (1) FR2842527B1 (is)
HK (1) HK1074444A1 (is)
HR (1) HRP20041231A2 (is)
IL (1) IL165942A (is)
IS (1) IS2487B (is)
ME (1) MEP12408A (is)
MX (1) MXPA05000822A (is)
NO (1) NO20050292L (is)
NZ (1) NZ537615A (is)
PL (1) PL375309A1 (is)
RS (1) RS20050018A (is)
TW (1) TWI274751B (is)
UA (1) UA78805C2 (is)
WO (1) WO2004009585A2 (is)
ZA (1) ZA200500478B (is)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005021534A1 (ja) 2003-08-28 2005-03-10 Taisho Pharmaceutical Co., Ltd. １，３−ジヒドロ−２ｈ−インドール−２−オン誘導体
TW200643015A (en) 2005-03-11 2006-12-16 Akzo Nobel Nv 2-(4-oxo-4H-quinazolin-3-yl)acetamide derivatives
DE102005015957A1 (de) * 2005-03-31 2006-10-05 Abbott Gmbh & Co. Kg Substituierte Oxindol-Derivate, diese enthaltende Arzneimittel und deren Verwendung
AU2006255009B2 (en) 2005-06-07 2011-10-27 Pharmacopeia L.L.C. Azinone and diazinone V3 inhibitors for depression and stress disorders
JP5256202B2 (ja) 2006-09-11 2013-08-07 エム・エス・ディー・オス・ベー・フェー キナゾリノンおよびイソキノリノンアセトアミド誘導体
CN103864658B (zh) * 2014-03-06 2016-06-15 南京工业大学 氮杂环丁酮衍生物及其制备方法与应用
CN104447489B (zh) * 2014-12-29 2017-01-11 南京工业大学 3,4-二芳基马来酰亚胺衍生物及其制备方法与应用

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2804114B1 (fr) * 2000-01-25 2002-03-08 Sanofi Synthelabo Nouveaux derives de 1,3-dihydro-2h-indol-2-one, un procede pour leur preparation et les compositions pharmaceutiques en contenant

Also Published As

Publication number Publication date
IL165942A0 (en) 2006-01-15
US7202267B2 (en) 2007-04-10
US20050192335A1 (en) 2005-09-01
CN100425608C (zh) 2008-10-15
IS7641A (is) 2005-01-12
DE60302670D1 (de) 2006-01-12
CN1681806A (zh) 2005-10-12
CA2492224A1 (en) 2004-01-29
AU2003271815B8 (en) 2009-04-30
NZ537615A (en) 2006-11-30
WO2004009585A3 (fr) 2004-05-06
HK1074444A1 (en) 2005-11-11
IS2487B (is) 2008-12-15
AU2003271815A1 (en) 2004-02-09
MXPA05000822A (es) 2005-08-29
AR040571A1 (es) 2005-04-13
ZA200500478B (en) 2006-07-26
RS20050018A (en) 2007-06-04
NO20050292L (no) 2005-04-19
JP4264414B2 (ja) 2009-05-20
FR2842527B1 (fr) 2005-01-28
HRP20041231A2 (en) 2005-02-28
AU2003271815B2 (en) 2009-03-12
PL375309A1 (en) 2005-11-28
EA008444B1 (ru) 2007-06-29
TW200410957A (en) 2004-07-01
EP1525198A2 (fr) 2005-04-27
IL165942A (en) 2010-04-15
FR2842527A1 (fr) 2004-01-23
EP1525198B1 (fr) 2005-12-07
WO2004009585A2 (fr) 2004-01-29
UA78805C2 (en) 2007-04-25
MEP12408A (en) 2010-06-10
TWI274751B (en) 2007-03-01
ES2254962T3 (es) 2006-06-16
BR0312800A (pt) 2005-04-19
ATE312092T1 (de) 2005-12-15
JP2005537271A (ja) 2005-12-08
DE60302670T2 (de) 2006-09-07
EA200500032A1 (ru) 2005-08-25

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