DK149753C - Analogifremgangsmaade til fremstilling af morfinderivater - Google Patents

Analogifremgangsmaade til fremstilling af morfinderivater

Info

Publication number
DK149753C
DK149753C DK129978A DK129978A DK149753C DK 149753 C DK149753 C DK 149753C DK 129978 A DK129978 A DK 129978A DK 129978 A DK129978 A DK 129978A DK 149753 C DK149753 C DK 149753C
Authority
DK
Denmark
Prior art keywords
preparation
morphine derivatives
analogy procedure
analogy
procedure
Prior art date
Application number
DK129978A
Other languages
Danish (da)
English (en)
Other versions
DK149753B (da
DK129978A (da
Inventor
Ryszard Jurek Kobylecki
Gordon William Kirby
Ian Geoffrey Guest
John William Lewis
Original Assignee
Reckitt & Colmann Prod Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Reckitt & Colmann Prod Ltd filed Critical Reckitt & Colmann Prod Ltd
Publication of DK129978A publication Critical patent/DK129978A/da
Publication of DK149753B publication Critical patent/DK149753B/da
Application granted granted Critical
Publication of DK149753C publication Critical patent/DK149753C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D489/00Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
    • C07D489/06Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: with a hetero atom directly attached in position 14
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12Antidiarrhoeals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK129978A 1977-03-23 1978-03-22 Analogifremgangsmaade til fremstilling af morfinderivater DK149753C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB1234277 1977-03-23
GB12342/77A GB1587831A (en) 1977-03-23 1977-03-23 Morphine derivatives

Publications (3)

Publication Number Publication Date
DK129978A DK129978A (da) 1978-09-24
DK149753B DK149753B (da) 1986-09-22
DK149753C true DK149753C (da) 1987-07-06

Family

ID=10002756

Family Applications (1)

Application Number Title Priority Date Filing Date
DK129978A DK149753C (da) 1977-03-23 1978-03-22 Analogifremgangsmaade til fremstilling af morfinderivater

Country Status (25)

Country Link
US (1) US4241067A (sv)
JP (1) JPS53121798A (sv)
AR (1) AR218296A1 (sv)
AT (1) AT360664B (sv)
AU (1) AU518614B2 (sv)
BE (1) BE865182A (sv)
CA (1) CA1089455A (sv)
CH (1) CH630629A5 (sv)
CS (1) CS199522B2 (sv)
DD (1) DD135081A5 (sv)
DE (1) DE2812581A1 (sv)
DK (1) DK149753C (sv)
ES (1) ES468170A1 (sv)
FR (1) FR2384775A1 (sv)
GB (1) GB1587831A (sv)
HU (1) HU177722B (sv)
IE (1) IE46442B1 (sv)
IT (1) IT1105172B (sv)
LU (1) LU79295A1 (sv)
NL (1) NL7803084A (sv)
NZ (1) NZ186693A (sv)
PL (1) PL111722B1 (sv)
SE (1) SE436132B (sv)
SU (1) SU856381A3 (sv)
ZA (1) ZA781525B (sv)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4362870A (en) * 1980-01-16 1982-12-07 Regents Of The University Of Minnesota Selective opioid receptor alkylating agents
US4401672A (en) * 1981-10-13 1983-08-30 Regents Of The University Of Minnesota Non-addictive narcotic antitussive preparation
DE3381877D1 (de) * 1982-03-16 1990-10-18 Univ Rockefeller Verwendung von opium antagonisten zur herstellung von arzneimitteln zur behebung gastro-intestinaler stoerungen.
GB8711558D0 (en) * 1987-05-15 1987-06-17 Reckitt & Colmann Prod Ltd Derivative of codeine
NZ246687A (en) * 1992-01-23 1996-12-20 Toray Industries Morphinan derivative and pharmaceutical compositions thereof
KR100341950B1 (ko) * 1993-07-19 2002-11-29 도레이 가부시끼가이샤 뇌세포보호제
NZ268969A (en) * 1993-07-23 1997-06-24 Toray Industries Morphinan derivatives and pharmaceutical compositions
US20060063792A1 (en) * 2004-09-17 2006-03-23 Adolor Corporation Substituted morphinans and methods of their use
EP1893616B1 (en) 2005-06-16 2010-12-29 Mallinckrodt, Inc. A synthetic route to 14-hydroxyl opiates through 1-halo-thebaine or analogs
WO2015082932A1 (en) 2013-12-05 2015-06-11 The University Of Bath Novel opioid compounds and their uses

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3332950A (en) * 1963-03-23 1967-07-25 Endo Lab 14-hydroxydihydronormorphinone derivatives
IL26896A (en) * 1966-01-19 1970-11-30 Endo Lab 14 - Hydroxynormorphinins and 14 - Hydroxynormorphinones
BE788478A (fr) * 1971-09-08 1973-03-06 Bristol Myers Co Procede de preparation de composes analgesiques
US4017497A (en) * 1975-11-18 1977-04-12 Bristol-Myers Company Process for the preparation of 14-hydroxymorphinan derivatives

Also Published As

Publication number Publication date
NZ186693A (en) 1979-10-25
HU177722B (en) 1981-12-28
BE865182A (fr) 1978-09-22
NL7803084A (nl) 1978-09-26
AR218296A1 (es) 1980-05-30
ES468170A1 (es) 1979-01-01
IT7848545A0 (it) 1978-03-22
FR2384775B1 (sv) 1981-04-30
AU3435678A (en) 1979-09-27
IE46442B1 (en) 1983-06-15
DK149753B (da) 1986-09-22
DD135081A5 (de) 1979-04-11
GB1587831A (en) 1981-04-08
JPS6259112B2 (sv) 1987-12-09
JPS53121798A (en) 1978-10-24
DK129978A (da) 1978-09-24
CH630629A5 (fr) 1982-06-30
AU518614B2 (en) 1981-10-08
CS199522B2 (en) 1980-07-31
IE780514L (en) 1978-09-23
SE7803329L (sv) 1978-09-24
SE436132B (sv) 1984-11-12
CA1089455A (en) 1980-11-11
ATA204378A (de) 1980-06-15
IT1105172B (it) 1985-10-28
US4241067A (en) 1980-12-23
PL205497A1 (pl) 1979-06-04
AT360664B (de) 1981-01-26
FR2384775A1 (fr) 1978-10-20
SU856381A3 (ru) 1981-08-15
PL111722B1 (en) 1980-09-30
DE2812581A1 (de) 1978-09-28
ZA781525B (en) 1979-04-25
LU79295A1 (fr) 1979-10-29

Similar Documents

Publication Publication Date Title
DK148280C (da) Analogifremgangsmaade til fremstilling af thienothiazinderivater
DK155367C (da) Analogifremgangsmaade til fremstilling af 2-nitroimidazolderivater
DK63178A (da) Fremgangsmaade til fremstilling af pyrrodinderivater
DK536178A (da) Fremgangsmaade til fremstilling af stilbenderivater
DK155603C (da) Analogifremgangsmaade til fremstilling af benzimidazolderivater
DK149858C (da) Analogifremgangsmaade til fremstilling af morfinderivater
DK110778A (da) Fremgangsmaade til fremstilling af 4-acylamino-phenyl-ethanolaminer
DK149954C (da) Analogifremgangsmaade til fremstilling af 18-umaettede prostacyklinderivater
DK153482C (da) Analogifremgangsmaade til fremstilling af 5-cyano-prostacyklinderivater
DK39778A (da) Fremgangsmaade til fremstilling af ethoxyquinderivater
DK154137C (da) Analogifremgangsmaade til fremstilling af meta-sulfonamido-benzamidderivater
DK30578A (da) Fremgangsmaade til fremstilling af aminoalkoxyphenylderivater
DK156568C (da) Analogifremgangsmaade til fremstilling af 3-indolderivater
DK145701C (da) Fremgangsmaade til fremstilling af ergotalkaloider
DK149753C (da) Analogifremgangsmaade til fremstilling af morfinderivater
DK50778A (da) Fremgangsmaade til fremstilling af oxadiazolopyrimidinderivater
DK154970C (da) Analogifremgangsmaade til fremstilling af carbostyrilderivater
DK309678A (da) Fremgangsmaade til fremstilling af tetralinderivater
DK154949C (da) Fremgangsmaade til fremstilling af trifluormethylphenoler
DK50878A (da) Fremgangsmaade til fremstilling af oxadiazolopyrimidinderivater
DK27178A (da) Fremgangsmaade til fremstilling af isoquinolinderivater
DK246878A (da) Fremgangsmaade til fremstilling af acylderivater
DK19278A (da) Fremgangsmaade til fremstilling af isoquinolinderivater
DK61778A (da) Fremgangsmaade til fremstilling af everninominderivater
DK147072C (da) Analogifremgangsmaade til fremstilling af ergolenderivater

Legal Events

Date Code Title Description
PBP Patent lapsed