DK149591C - Analogifremgangsmaade til fremstilling af 2,5-diketopiperazinderivater eller syreadditionssalte deraf - Google Patents

Analogifremgangsmaade til fremstilling af 2,5-diketopiperazinderivater eller syreadditionssalte deraf

Info

Publication number
DK149591C
DK149591C DK274881A DK274881A DK149591C DK 149591 C DK149591 C DK 149591C DK 274881 A DK274881 A DK 274881A DK 274881 A DK274881 A DK 274881A DK 149591 C DK149591 C DK 149591C
Authority
DK
Denmark
Prior art keywords
dicetopiperazine
analogue
derivatives
preparation
acid addition
Prior art date
Application number
DK274881A
Other languages
English (en)
Other versions
DK149591B (da
DK274881A (da
Inventor
George Heavner
Foe-Siong Tjoeng
Gideon Goldstein
Original Assignee
Ortho Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ortho Pharma Corp filed Critical Ortho Pharma Corp
Publication of DK274881A publication Critical patent/DK274881A/da
Publication of DK149591B publication Critical patent/DK149591B/da
Application granted granted Critical
Publication of DK149591C publication Critical patent/DK149591C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/12—Cyclic peptides with only normal peptide bonds in the ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/06—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members
    • C07D241/08—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
    • C07K1/061—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Analytical Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Paper (AREA)
  • Coloring (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Steroid Compounds (AREA)
  • Cereal-Derived Products (AREA)
DK274881A 1980-06-23 1981-06-22 Analogifremgangsmaade til fremstilling af 2,5-diketopiperazinderivater eller syreadditionssalte deraf DK149591C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/162,228 US4289759A (en) 1980-06-23 1980-06-23 Immunoregulatory diketopiperazine compounds
US16222880 1980-06-23

Publications (3)

Publication Number Publication Date
DK274881A DK274881A (da) 1981-12-24
DK149591B DK149591B (da) 1986-08-04
DK149591C true DK149591C (da) 1987-02-09

Family

ID=22584724

Family Applications (1)

Application Number Title Priority Date Filing Date
DK274881A DK149591C (da) 1980-06-23 1981-06-22 Analogifremgangsmaade til fremstilling af 2,5-diketopiperazinderivater eller syreadditionssalte deraf

Country Status (19)

Country Link
US (1) US4289759A (da)
EP (1) EP0043219B1 (da)
JP (1) JPS5732272A (da)
AT (1) ATE4897T1 (da)
AU (1) AU544522B2 (da)
CA (1) CA1199024A (da)
DE (1) DE3161122D1 (da)
DK (1) DK149591C (da)
ES (1) ES503306A0 (da)
FI (1) FI75563C (da)
GR (1) GR74548B (da)
IE (1) IE51312B1 (da)
IL (1) IL63147A0 (da)
NO (1) NO157862C (da)
NZ (1) NZ197386A (da)
PH (1) PH17520A (da)
PT (1) PT73202B (da)
YU (1) YU42410B (da)
ZA (1) ZA814218B (da)

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Also Published As

Publication number Publication date
FI811950L (fi) 1981-12-24
ES8300718A1 (es) 1982-11-01
NO157862B (no) 1988-02-22
IE811383L (en) 1981-12-23
NO157862C (no) 1988-06-01
YU157281A (en) 1984-02-29
EP0043219A1 (en) 1982-01-06
IE51312B1 (en) 1986-11-26
NZ197386A (en) 1984-07-06
AU544522B2 (en) 1985-06-06
AU7124681A (en) 1982-01-07
IL63147A0 (en) 1981-09-13
PT73202A (en) 1981-07-01
FI75563B (fi) 1988-03-31
NO812126L (no) 1981-12-28
JPS5732272A (en) 1982-02-20
FI75563C (fi) 1988-07-11
CA1199024A (en) 1986-01-07
ZA814218B (en) 1983-02-23
YU42410B (en) 1988-08-31
PT73202B (en) 1983-04-26
ES503306A0 (es) 1982-11-01
US4289759A (en) 1981-09-15
PH17520A (en) 1984-09-13
DE3161122D1 (en) 1983-11-10
DK149591B (da) 1986-08-04
EP0043219B1 (en) 1983-10-05
GR74548B (da) 1984-06-29
DK274881A (da) 1981-12-24
ATE4897T1 (de) 1983-10-15

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