DK141992D0 - 2-(3-oxocycloalken-1-yl)-aminobenzonitril-derivater - Google Patents

2-(3-oxocycloalken-1-yl)-aminobenzonitril-derivater

Info

Publication number
DK141992D0
DK141992D0 DK921419A DK141992A DK141992D0 DK 141992 D0 DK141992 D0 DK 141992D0 DK 921419 A DK921419 A DK 921419A DK 141992 A DK141992 A DK 141992A DK 141992 D0 DK141992 D0 DK 141992D0
Authority
DK
Denmark
Prior art keywords
oxocycloalken
aminobenzonitril
derivatives
Prior art date
Application number
DK921419A
Other languages
English (en)
Other versions
DK141992A (da
DK168704B1 (da
Inventor
Gregory M Shutske
Frank A Pierrat
Original Assignee
Hoechst Roussel Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/664,731 external-priority patent/US4631286A/en
Priority claimed from US06/781,155 external-priority patent/US4695573A/en
Application filed by Hoechst Roussel Pharma filed Critical Hoechst Roussel Pharma
Publication of DK141992D0 publication Critical patent/DK141992D0/da
Publication of DK141992A publication Critical patent/DK141992A/da
Application granted granted Critical
Publication of DK168704B1 publication Critical patent/DK168704B1/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D219/00—Heterocyclic compounds containing acridine or hydrogenated acridine ring systems
    • C07D219/04—Heterocyclic compounds containing acridine or hydrogenated acridine ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
    • C07D219/08—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D219/00—Heterocyclic compounds containing acridine or hydrogenated acridine ring systems
    • C07D219/04—Heterocyclic compounds containing acridine or hydrogenated acridine ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
    • C07D219/08—Nitrogen atoms
    • C07D219/10—Nitrogen atoms attached in position 9
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D219/00—Heterocyclic compounds containing acridine or hydrogenated acridine ring systems
    • C07D219/04—Heterocyclic compounds containing acridine or hydrogenated acridine ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
    • C07D219/08—Nitrogen atoms
    • C07D219/10—Nitrogen atoms attached in position 9
    • C07D219/12—Amino-alkylamino radicals attached in position 9
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04—Ortho- or peri-condensed ring systems
    • C07D221/06—Ring systems of three rings
    • C07D221/16—Ring systems of three rings containing carbocyclic rings other than six-membered
DK141992A 1984-10-25 1992-11-26 N-(3-Oxocyclohexen-1-yl)-2-aminobenzonitrilderivater DK168704B1 (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US06/664,731 US4631286A (en) 1984-10-25 1984-10-25 9-amino-1,2,3,4-tetrahydroacridin-1-ol and related compounds
US66473184 1984-10-25
US06/781,155 US4695573A (en) 1984-10-25 1985-10-01 9-amino-1,2,3,4-tetrahydroacridin-1-ol and related compounds
US78115585 1985-10-01

Publications (3)

Publication Number Publication Date
DK141992D0 true DK141992D0 (da) 1992-11-26
DK141992A DK141992A (da) 1992-11-26
DK168704B1 DK168704B1 (da) 1994-05-24

Family

ID=27099040

Family Applications (2)

Application Number Title Priority Date Filing Date
DK488885A DK167250B1 (da) 1984-10-25 1985-10-24 9-amino-acridinderivater, fremgangsmaade til deres fremstilling, farmaceutiske praeparater deraf og deres anvendelse til fremstilling af laegemidler
DK141992A DK168704B1 (da) 1984-10-25 1992-11-26 N-(3-Oxocyclohexen-1-yl)-2-aminobenzonitrilderivater

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DK488885A DK167250B1 (da) 1984-10-25 1985-10-24 9-amino-acridinderivater, fremgangsmaade til deres fremstilling, farmaceutiske praeparater deraf og deres anvendelse til fremstilling af laegemidler

Country Status (20)

Country Link
US (1) US4839364A (da)
EP (1) EP0179383B1 (da)
JP (1) JPH01125362A (da)
KR (1) KR900007624B1 (da)
AR (1) AR247394A1 (da)
AT (1) ATE63903T1 (da)
AU (2) AU589141B2 (da)
CA (1) CA1292744C (da)
DE (1) DE3582995D1 (da)
DK (2) DK167250B1 (da)
ES (3) ES8701165A1 (da)
FI (1) FI86421C (da)
GR (1) GR852555B (da)
HU (1) HU196183B (da)
IE (1) IE58696B1 (da)
IL (3) IL76796A (da)
NO (1) NO172847C (da)
NZ (2) NZ229248A (da)
PH (1) PH22614A (da)
PT (1) PT81362B (da)

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US4927820A (en) * 1988-11-25 1990-05-22 Hoechst Roussel Pharmaceuticals Inc. Fused heterocyclic derivatives of 1,2,3,4-tetrahydroacridine
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US5280032A (en) * 1989-02-14 1994-01-18 Toyama Chemical Co., Ltd. 1,2-ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same
US4916135A (en) * 1989-05-08 1990-04-10 Hoechst Roussel Pharmaceuticals Inc. N-heteroaryl-4-quinolinamines
US5053513A (en) * 1990-03-29 1991-10-01 Hoechst-Roussel Pharmaceuticals Incorporated Method of reducing a carbonyl containing acridine
US5210087A (en) * 1991-02-13 1993-05-11 Hoechst-Roussel Pharmaceuticals Inc. 9-aminotetrahydroacridines and related compounds
RU2024509C1 (ru) * 1991-05-07 1994-12-15 Всероссийский научный центр по безопасности биологически активных веществ Производные 9-аминоакридина или их соли с органическими или неорганическими кислотами, проявляющие психотропную, антиамнестическую и липидрегулирующую активность
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US5434165A (en) * 1991-11-18 1995-07-18 Sanawa Kagaku Kenkyusho Company, Ltd. Nootropic agents, compositions of, and method of use thereof
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ES2059263B1 (es) * 1992-10-27 1995-10-01 Vita Invest Sa Procedimiento para la obtencion del (+)-9-amino-1,2,3,4-tetrahidroacridin-1-ol.
CA2161538A1 (en) * 1993-07-22 1995-02-02 S. Shirley Yang Controlled release tacrine drug delivery systems and methods for preparing same
US5434170A (en) * 1993-12-23 1995-07-18 Andrulis Pharmaceuticals Corp. Method for treating neurocognitive disorders
US20100210590A1 (en) * 1995-09-27 2010-08-19 Northwestern University Compositions and treatments for seizure-related disorders
ES2144353B1 (es) * 1997-12-26 2001-01-01 Consejo Superior Investigacion Nuevos analogos de tacrina: potenciales agentes neuroprotectores para las enfermedades de alzheimer y parkinson. su procedimiento de obtencion.
KR100381716B1 (ko) * 2000-10-09 2003-04-26 한국화학연구원 항암활성을 가지는 아크리딘 유도체
US20050222123A1 (en) 2004-01-27 2005-10-06 North Shore-Long Island Jewish Research Institute Cholinesterase inhibitors for treating inflammation
US20080045500A1 (en) * 2004-07-01 2008-02-21 Eisai R&D Management Co., Ltd. Nerve Regeneration Stimulator
ATE523199T1 (de) * 2004-11-02 2011-09-15 Univ Northwestern Pyridazinverbindungen und verfahren
AU2005310986A1 (en) * 2004-11-12 2006-06-08 Bellus Health (International) Limited Methods and fluorinated compositions for treating amyloid-related diseases
US20080188510A1 (en) * 2005-05-23 2008-08-07 Eisai R & D Management Co., Ltd. Novel methods using zonisamide
WO2007127474A2 (en) * 2006-04-28 2007-11-08 Northwestern University Compositions and treatments using pyridazine compounds and cholinesterase inhibitors
JP2017503026A (ja) * 2014-01-15 2017-01-26 サントル ナシオナル ドゥ ラ ルシェルシュ シアンティフィーク（セーエヌエールエス） 水溶性４−アザポドフィルロトキシン類似体
KR101586473B1 (ko) * 2014-04-30 2016-01-19 (주)이컴프 스크롤 압축기
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Also Published As

Publication number Publication date
AU3823489A (en) 1989-10-26
PH22614A (en) 1988-10-17
AU4903885A (en) 1986-05-01
ES8801213A1 (es) 1988-01-01
FI854156A0 (fi) 1985-10-23
EP0179383A3 (en) 1987-01-28
NO904711D0 (no) 1990-10-30
ATE63903T1 (de) 1991-06-15
IL90300A0 (en) 1989-12-15
PT81362B (pt) 1987-11-30
NZ213932A (en) 1990-12-21
GR852555B (da) 1986-02-24
PT81362A (en) 1985-11-01
DK488885A (da) 1986-04-26
DK141992A (da) 1992-11-26
EP0179383A2 (en) 1986-04-30
HUT41009A (en) 1987-03-30
AR247394A1 (es) 1994-12-29
KR900007624B1 (ko) 1990-10-17
ES548137A0 (es) 1986-11-16
NO172847B (no) 1993-06-07
DE3582995D1 (de) 1991-07-04
US4839364A (en) 1989-06-13
ES554569A0 (es) 1988-01-01
HU196183B (en) 1988-10-28
JPH01125362A (ja) 1989-05-17
NO904711L (no) 1986-04-28
IE58696B1 (en) 1993-11-03
JPH0584306B2 (da) 1993-12-01
IL76796A0 (en) 1986-02-28
IL76796A (en) 1990-03-19
FI86421B (fi) 1992-05-15
FI854156L (fi) 1986-04-26
DK167250B1 (da) 1993-09-27
NZ229248A (en) 1990-12-21
DK488885D0 (da) 1985-10-24
KR860003227A (ko) 1986-05-21
IE852632L (en) 1986-04-25
AU615768B2 (en) 1991-10-10
EP0179383B1 (en) 1991-05-29
CA1292744C (en) 1991-12-03
NO172847C (no) 1993-09-15
IL90300A (en) 1990-11-29
DK168704B1 (da) 1994-05-24
ES8701165A1 (es) 1986-11-16
AU589141B2 (en) 1989-10-05
ES8802383A1 (es) 1988-05-16
ES554568A0 (es) 1988-05-16
FI86421C (fi) 1992-08-25

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Legal Events

Date Code Title Description
A0 Application filed
B1 Patent granted (law 1993)
PBP Patent lapsed

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