DK133051C - Analogifremgangsmade til fremstilling af 1,3-oxygenerede 8alfa-ostratriener - Google Patents

Analogifremgangsmade til fremstilling af 1,3-oxygenerede 8alfa-ostratriener

Info

Publication number
DK133051C
DK133051C DK368074A DK368074A DK133051C DK 133051 C DK133051 C DK 133051C DK 368074 A DK368074 A DK 368074A DK 368074 A DK368074 A DK 368074A DK 133051 C DK133051 C DK 133051C
Authority
DK
Denmark
Prior art keywords
ostratriens
8alfa
oxygenated
preparation
analogical procedure
Prior art date
Application number
DK368074A
Other languages
Danish (da)
English (en)
Other versions
DK368074A (enrdf_load_stackoverflow
DK133051B (da
Inventor
K Prezewowsky
H Laurent
H Hofmeister
R Wiechert
F Neumann
Y Nishino
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE2336431A external-priority patent/DE2336431C2/de
Priority claimed from DE19742426777 external-priority patent/DE2426777A1/de
Application filed by Schering Ag filed Critical Schering Ag
Publication of DK368074A publication Critical patent/DK368074A/da
Publication of DK133051B publication Critical patent/DK133051B/da
Application granted granted Critical
Publication of DK133051C publication Critical patent/DK133051C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051Estrane derivatives
    • C07J1/0066Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa
    • C07J1/007Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
    • C07J1/0074Esters
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051Estrane derivatives
    • C07J1/0059Estrane derivatives substituted in position 17 by a keto group
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J15/00Stereochemically pure steroids containing carbon, hydrogen, halogen or oxygen having a partially or totally inverted skeleton, e.g. retrosteroids, L-isomers
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J31/00Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0072Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the A ring of the steroid being aromatic
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J43/00Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Catalysts (AREA)
DK368074A 1973-07-13 1974-07-09 Analogifremgangsmade til fremstilling af 1,3-oxygenerede 8alfa-ostratriener DK133051C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE2336431A DE2336431C2 (de) 1973-07-13 1973-07-13 1.3-oxygenierte 8 alpha-Östratriene, Verfahren zu deren Herstellung und diese enthaltende Arzneimittel
DE19742426777 DE2426777A1 (de) 1974-05-31 1974-05-31 1.3-oxygenierte 8 alpha-oestratriene

Publications (3)

Publication Number Publication Date
DK368074A DK368074A (enrdf_load_stackoverflow) 1975-03-17
DK133051B DK133051B (da) 1976-03-15
DK133051C true DK133051C (da) 1976-08-16

Family

ID=25765510

Family Applications (1)

Application Number Title Priority Date Filing Date
DK368074A DK133051C (da) 1973-07-13 1974-07-09 Analogifremgangsmade til fremstilling af 1,3-oxygenerede 8alfa-ostratriener

Country Status (18)

Country Link
JP (1) JPS5821639B2 (enrdf_load_stackoverflow)
AT (1) ATA575574A (enrdf_load_stackoverflow)
AU (1) AU477010B2 (enrdf_load_stackoverflow)
CA (1) CA1030951A (enrdf_load_stackoverflow)
CH (2) CH614217A5 (enrdf_load_stackoverflow)
CS (2) CS182300B2 (enrdf_load_stackoverflow)
DD (1) DD114066A5 (enrdf_load_stackoverflow)
DK (1) DK133051C (enrdf_load_stackoverflow)
ES (1) ES428226A1 (enrdf_load_stackoverflow)
FI (1) FI54131C (enrdf_load_stackoverflow)
FR (1) FR2236505B1 (enrdf_load_stackoverflow)
GB (1) GB1479934A (enrdf_load_stackoverflow)
HU (1) HU169791B (enrdf_load_stackoverflow)
IE (1) IE39872B1 (enrdf_load_stackoverflow)
IL (1) IL45259A (enrdf_load_stackoverflow)
NO (1) NO742546L (enrdf_load_stackoverflow)
SE (1) SE7409151L (enrdf_load_stackoverflow)
SU (1) SU626705A3 (enrdf_load_stackoverflow)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2551214C2 (de) * 1975-11-12 1984-07-12 Schering AG, 1000 Berlin und 4709 Bergkamen Verfahren zur Herstellung von 1,3-oxygenierten 8α-Östratrienen
JPS5862734U (ja) * 1981-10-22 1983-04-27 日工株式会社 型枠支持サボ−ト
JPS59146759A (ja) * 1984-01-06 1984-08-22 株式会社日立製作所 自動ねじ込み装置
JPS60155376A (ja) * 1984-01-24 1985-08-15 松下電器産業株式会社 ナツト浮き検出装置
DE3710728A1 (de) * 1987-03-31 1988-10-13 Schering Ag Verfahren zur herstellung von 17(alpha)-ethinyl-17ss-hydroxy-18-methyl-4,15-estradien-3-on und die neuen zwischenprodukte fuer dieses verfahren
US6011024A (en) 1991-08-28 2000-01-04 Imperial College Of Science Technology & Medicine Steroid sulphatase inhibitors
US6476011B1 (en) 1991-08-28 2002-11-05 Sterix Limited Methods for introducing an estrogenic compound
US6903084B2 (en) 1991-08-28 2005-06-07 Sterix Limited Steroid sulphatase inhibitors
US7335650B2 (en) 2000-01-14 2008-02-26 Sterix Limited Composition
GB0020498D0 (en) 2000-08-18 2000-10-11 Sterix Ltd Compound
RU2679625C1 (ru) * 2018-11-08 2019-02-12 Ильясов Шамиль Сионович ПРИМЕНЕНИЕ 3-О-СУЛЬФАМОИЛОКСИ-6-ОКСА-7β-МЕТИЛ-D-ГОМО-8α-ЭСТРА-1,3,5(10)-ТРИЕН-17а-ОНА ДЛЯ ЛЕЧЕНИЯ РАКА МОЛОЧНОЙ ЖЕЛЕЗЫ, ВКЛЮЧАЯ ТРИЖДЫ-НЕГАТИВНУЮ ФОРМУ, И СПОСОБ ЕГО ПОЛУЧЕНИЯ

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3436411A (en) * 1967-12-28 1969-04-01 American Home Prod Process for cleaving an a-ring ether group in 13-alkylgona (and 8-isogona)-1,3,5(10)-trienes and delta-7-,delta-8(9)-,and delta-8(9),14(15)-dehydro derivatives thereof

Also Published As

Publication number Publication date
AU477010B2 (en) 1976-10-14
GB1479934A (en) 1977-07-13
CA1030951A (en) 1978-05-09
CH609064A5 (en) 1979-02-15
FI54131C (fi) 1978-10-10
DK368074A (enrdf_load_stackoverflow) 1975-03-17
JPS5821639B2 (ja) 1983-05-02
JPS5032160A (enrdf_load_stackoverflow) 1975-03-28
SU626705A3 (ru) 1978-09-30
IE39872L (en) 1975-01-13
FR2236505B1 (enrdf_load_stackoverflow) 1977-07-08
DK133051B (da) 1976-03-15
SE7409151L (sv) 1975-01-14
FI54131B (fi) 1978-06-30
HU169791B (en) 1977-01-28
CS182260B2 (en) 1978-04-28
FR2236505A1 (enrdf_load_stackoverflow) 1975-02-07
DD114066A5 (enrdf_load_stackoverflow) 1975-07-12
IL45259A0 (en) 1974-10-22
ATA575574A (de) 1978-05-15
IE39872B1 (en) 1979-01-17
CS182300B2 (en) 1978-04-28
ES428226A1 (es) 1976-07-16
CH614217A5 (en) 1979-11-15
FI213974A7 (enrdf_load_stackoverflow) 1975-01-14
AU7112374A (en) 1976-01-15
IL45259A (en) 1977-10-31
NO742546L (enrdf_load_stackoverflow) 1975-02-10

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