DK130480A - Fremgangsmaade til fremstilling af analgiteske pentapeptider - Google Patents
Fremgangsmaade til fremstilling af analgiteske pentapeptiderInfo
- Publication number
- DK130480A DK130480A DK130480A DK130480A DK130480A DK 130480 A DK130480 A DK 130480A DK 130480 A DK130480 A DK 130480A DK 130480 A DK130480 A DK 130480A DK 130480 A DK130480 A DK 130480A
- Authority
- DK
- Denmark
- Prior art keywords
- sup
- sub
- methyl
- pentapeptides
- hydrogen
- Prior art date
Links
- 229910052739 hydrogen Inorganic materials 0.000 abstract 3
- 239000001257 hydrogen Substances 0.000 abstract 3
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 2
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 125000004432 carbon atom Chemical group C* 0.000 abstract 2
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 2
- 125000006045 2-methyl-1-pentenyl group Chemical group 0.000 abstract 1
- 125000006049 2-methyl-2-pentenyl group Chemical group 0.000 abstract 1
- 241001465754 Metazoa Species 0.000 abstract 1
- 230000000202 analgesic effect Effects 0.000 abstract 1
- 125000004850 cyclobutylmethyl group Chemical group C1(CCC1)C* 0.000 abstract 1
- 125000004186 cyclopropylmethyl group Chemical group [H]C([H])(*)C1([H])C([H])([H])C1([H])[H] 0.000 abstract 1
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 abstract 1
- 150000002431 hydrogen Chemical class 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 125000001436 propyl group Chemical group [H]C([*])([H])C([H])([H])C([H])([H])[H] 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000007790 solid phase Substances 0.000 abstract 1
- 238000010189 synthetic method Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/665—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
- C07K14/70—Enkephalins
- C07K14/702—Enkephalins with at least 1 amino acid in D-form
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Zoology (AREA)
- Genetics & Genomics (AREA)
- Medicinal Chemistry (AREA)
- Gastroenterology & Hepatology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Toxicology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Hydrogenated Pyridines (AREA)
- Measurement Of Radiation (AREA)
- Curing Cements, Concrete, And Artificial Stone (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US05/932,089 US4278596A (en) | 1978-08-08 | 1978-08-08 | Analgesic pentapeptides |
| PCT/US1979/000531 WO1980000342A1 (en) | 1978-08-08 | 1979-07-23 | Analgesic pentapeptides |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK130480A true DK130480A (da) | 1980-03-26 |
Family
ID=25461755
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK130480A DK130480A (da) | 1978-08-08 | 1980-03-26 | Fremgangsmaade til fremstilling af analgiteske pentapeptider |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US4278596A (da) |
| EP (1) | EP0008196B1 (da) |
| JP (1) | JPS55500551A (da) |
| AT (1) | ATE4590T1 (da) |
| AU (1) | AU528223B2 (da) |
| CA (1) | CA1138440A (da) |
| DE (1) | DE2966134D1 (da) |
| DK (1) | DK130480A (da) |
| GB (1) | GB2027034B (da) |
| IE (1) | IE49056B1 (da) |
| PH (1) | PH15696A (da) |
| WO (1) | WO1980000342A1 (da) |
| ZA (1) | ZA793983B (da) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FI770219A7 (da) | 1976-02-02 | 1977-08-03 | Sandoz Ag | |
| FR2488253A1 (fr) * | 1980-08-08 | 1982-02-12 | Roques Bernard | Nouveaux peptides et leur application en therapeutique |
| EP0076557B1 (en) * | 1981-06-22 | 1985-11-13 | Imperial Chemical Industries Plc | Peptides and pseudopeptides in which the n terminus bears two substituents |
| JPH0742313B2 (ja) * | 1988-03-28 | 1995-05-10 | 日立化成工業株式会社 | 新規ペプチド、その塩及びペプチド性抗アレルギー剤 |
| JPH0449298A (ja) * | 1990-06-19 | 1992-02-18 | Univ New York State | 新規なエンケファリン誘導体および鎮痛剤 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5291839A (en) * | 1976-01-26 | 1977-08-02 | Wellcome Found | Peptide and derivatives |
| GB1523812A (en) * | 1976-04-08 | 1978-09-06 | Ici Ltd | Polypeptide |
| NZ183712A (en) * | 1976-04-08 | 1979-10-25 | Ici Ltd | Polypeptide analogues of enkephalins, and pharmaceutical compositions |
| DK386677A (da) * | 1976-09-01 | 1978-03-02 | D H Y | Methioninencephalinderivater deres fremstilling og anvendelsesamt mellemprodukter til fremstillingen |
| US4128541A (en) * | 1976-12-27 | 1978-12-05 | American Home Products Corporation | Pentapeptide with morphine- like activity |
-
1978
- 1978-08-08 US US05/932,089 patent/US4278596A/en not_active Expired - Lifetime
-
1979
- 1979-07-23 JP JP50127379A patent/JPS55500551A/ja active Pending
- 1979-07-23 WO PCT/US1979/000531 patent/WO1980000342A1/en not_active Ceased
- 1979-07-24 PH PH22811A patent/PH15696A/en unknown
- 1979-08-01 GB GB7926809A patent/GB2027034B/en not_active Expired
- 1979-08-01 EP EP79301542A patent/EP0008196B1/en not_active Expired
- 1979-08-01 DE DE7979301542T patent/DE2966134D1/de not_active Expired
- 1979-08-01 AT AT79301542T patent/ATE4590T1/de not_active IP Right Cessation
- 1979-08-02 ZA ZA00793983A patent/ZA793983B/xx unknown
- 1979-08-03 CA CA000333192A patent/CA1138440A/en not_active Expired
- 1979-08-03 AU AU49556/79A patent/AU528223B2/en not_active Ceased
- 1979-08-08 IE IE1473/79A patent/IE49056B1/en unknown
-
1980
- 1980-03-26 DK DK130480A patent/DK130480A/da not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| EP0008196A1 (en) | 1980-02-20 |
| GB2027034A (en) | 1980-02-13 |
| AU4955679A (en) | 1980-02-14 |
| EP0008196B1 (en) | 1983-09-07 |
| GB2027034B (en) | 1982-07-21 |
| IE791473L (en) | 1980-02-08 |
| ATE4590T1 (de) | 1983-09-15 |
| CA1138440A (en) | 1982-12-28 |
| AU528223B2 (en) | 1983-04-21 |
| WO1980000342A1 (en) | 1980-03-06 |
| ZA793983B (en) | 1981-03-25 |
| PH15696A (en) | 1983-03-14 |
| US4278596A (en) | 1981-07-14 |
| DE2966134D1 (en) | 1983-10-13 |
| IE49056B1 (en) | 1985-07-24 |
| JPS55500551A (da) | 1980-08-21 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AHS | Application shelved for other reasons than non-payment |