DK1149831T3 - Fremgangsmåde til fremstilling af mesylatsalttrihydratet af 1-(4-hydroxyphenyl)-2-(4-hydroxy-4-phenylpiperidin-1-yl)-1-proponal og mellemprodukter nyttige dertil - Google Patents
Fremgangsmåde til fremstilling af mesylatsalttrihydratet af 1-(4-hydroxyphenyl)-2-(4-hydroxy-4-phenylpiperidin-1-yl)-1-proponal og mellemprodukter nyttige dertilInfo
- Publication number
- DK1149831T3 DK1149831T3 DK01303713T DK01303713T DK1149831T3 DK 1149831 T3 DK1149831 T3 DK 1149831T3 DK 01303713 T DK01303713 T DK 01303713T DK 01303713 T DK01303713 T DK 01303713T DK 1149831 T3 DK1149831 T3 DK 1149831T3
- Authority
- DK
- Denmark
- Prior art keywords
- proponal
- phenylpiperidin
- hydroxyphenyl
- hydroxy
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
- C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/40—Oxygen atoms
- C07D211/44—Oxygen atoms attached in position 4
- C07D211/52—Oxygen atoms attached in position 4 having an aryl radical as the second substituent in position 4
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Hydrogenated Pyridines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US20041700P | 2000-04-28 | 2000-04-28 |
Publications (1)
Publication Number | Publication Date |
---|---|
DK1149831T3 true DK1149831T3 (da) | 2004-12-06 |
Family
ID=22741639
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK01303713T DK1149831T3 (da) | 2000-04-28 | 2001-04-24 | Fremgangsmåde til fremstilling af mesylatsalttrihydratet af 1-(4-hydroxyphenyl)-2-(4-hydroxy-4-phenylpiperidin-1-yl)-1-proponal og mellemprodukter nyttige dertil |
Country Status (26)
Country | Link |
---|---|
US (1) | US6570018B2 (da) |
EP (1) | EP1149831B1 (da) |
JP (1) | JP2001354650A (da) |
KR (1) | KR100432841B1 (da) |
CN (1) | CN1211366C (da) |
AR (1) | AR028377A1 (da) |
AT (1) | ATE275130T1 (da) |
AU (1) | AU781715B2 (da) |
BR (1) | BR0101611A (da) |
CA (1) | CA2345286C (da) |
CZ (1) | CZ20011472A3 (da) |
DE (1) | DE60105221T2 (da) |
DK (1) | DK1149831T3 (da) |
ES (1) | ES2225425T3 (da) |
HK (1) | HK1040514B (da) |
HU (1) | HUP0101725A3 (da) |
ID (1) | ID30012A (da) |
IL (1) | IL142706A0 (da) |
IN (1) | IN191534B (da) |
PL (1) | PL347299A1 (da) |
PT (1) | PT1149831E (da) |
RU (1) | RU2192415C1 (da) |
SI (1) | SI1149831T1 (da) |
TW (1) | TWI222440B (da) |
YU (1) | YU27801A (da) |
ZA (1) | ZA200103321B (da) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6743921B2 (en) * | 2002-01-24 | 2004-06-01 | Dsm Catalytica Pharmaceuticals, Inc. | Process for the preparation of nonracemic syn-1-(4-hydroxy-phenyl)-2-(4-hydroxy-4-phenyl-piperidin-1-yl)-1-propanol compounds |
CN105037221B (zh) * | 2015-06-18 | 2017-05-10 | 吉林大学珠海学院 | 一种具有神经保护作用的化合物及其制备方法 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN1615861A (zh) | 1995-08-11 | 2005-05-18 | 美国辉瑞有限公司 | (1s,2s)-1-(4-羟基苯基)-2-(4-羟基-4-苯基哌啶-1-基)-1-丙醇甲磺酸盐三水合物 |
TW450807B (en) * | 1995-09-15 | 2001-08-21 | Pfizer | Pharmaceutical compositions for treating tinnitus comprising neuroprotective agents |
-
2001
- 2001-04-18 YU YU27801A patent/YU27801A/sh unknown
- 2001-04-19 IL IL14270601A patent/IL142706A0/xx not_active IP Right Cessation
- 2001-04-20 IN IN357BO2001 patent/IN191534B/en unknown
- 2001-04-23 TW TW090109679A patent/TWI222440B/zh not_active IP Right Cessation
- 2001-04-23 US US09/840,668 patent/US6570018B2/en not_active Expired - Fee Related
- 2001-04-24 DK DK01303713T patent/DK1149831T3/da active
- 2001-04-24 ES ES01303713T patent/ES2225425T3/es not_active Expired - Lifetime
- 2001-04-24 ZA ZA200103321A patent/ZA200103321B/xx unknown
- 2001-04-24 SI SI200130185T patent/SI1149831T1/ unknown
- 2001-04-24 AT AT01303713T patent/ATE275130T1/de not_active IP Right Cessation
- 2001-04-24 PT PT01303713T patent/PT1149831E/pt unknown
- 2001-04-24 EP EP01303713A patent/EP1149831B1/en not_active Expired - Lifetime
- 2001-04-24 DE DE60105221T patent/DE60105221T2/de not_active Expired - Fee Related
- 2001-04-25 CZ CZ20011472A patent/CZ20011472A3/cs unknown
- 2001-04-26 ID IDP20010344D patent/ID30012A/id unknown
- 2001-04-26 AU AU38897/01A patent/AU781715B2/en not_active Ceased
- 2001-04-26 CA CA002345286A patent/CA2345286C/en not_active Expired - Fee Related
- 2001-04-26 AR ARP010101972A patent/AR028377A1/es unknown
- 2001-04-26 BR BR0101611-3A patent/BR0101611A/pt not_active IP Right Cessation
- 2001-04-27 HU HU0101725A patent/HUP0101725A3/hu unknown
- 2001-04-27 CN CNB011171545A patent/CN1211366C/zh not_active Expired - Fee Related
- 2001-04-27 KR KR10-2001-0022856A patent/KR100432841B1/ko not_active IP Right Cessation
- 2001-04-27 PL PL01347299A patent/PL347299A1/xx not_active Application Discontinuation
- 2001-04-27 JP JP2001130684A patent/JP2001354650A/ja active Pending
- 2001-04-27 RU RU2001111948/04A patent/RU2192415C1/ru not_active IP Right Cessation
-
2002
- 2002-03-14 HK HK02101947.0A patent/HK1040514B/zh not_active IP Right Cessation
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