DK1132392T3 - Ketolid-antibiotika - Google Patents

Ketolid-antibiotika

Info

Publication number
DK1132392T3
DK1132392T3 DK01301966T DK01301966T DK1132392T3 DK 1132392 T3 DK1132392 T3 DK 1132392T3 DK 01301966 T DK01301966 T DK 01301966T DK 01301966 T DK01301966 T DK 01301966T DK 1132392 T3 DK1132392 T3 DK 1132392T3
Authority
DK
Denmark
Prior art keywords
compounds
formula
infections
relates
ketolide antibiotics
Prior art date
Application number
DK01301966T
Other languages
Danish (da)
English (en)
Inventor
Takushi Kaneko
William Thomas Mcmillen
Wei-Guo Su
Hongjuan Zhao
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Application granted granted Critical
Publication of DK1132392T3 publication Critical patent/DK1132392T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Public Health (AREA)
  • Biochemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Fats And Perfumes (AREA)
DK01301966T 2000-03-06 2001-03-05 Ketolid-antibiotika DK1132392T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US18697000P 2000-03-06 2000-03-06

Publications (1)

Publication Number Publication Date
DK1132392T3 true DK1132392T3 (da) 2004-06-07

Family

ID=22687057

Family Applications (1)

Application Number Title Priority Date Filing Date
DK01301966T DK1132392T3 (da) 2000-03-06 2001-03-05 Ketolid-antibiotika

Country Status (11)

Country Link
US (1) US6555524B2 (fr)
EP (1) EP1132392B1 (fr)
JP (1) JP2001261694A (fr)
AT (1) ATE260928T1 (fr)
BR (1) BR0100850A (fr)
CA (1) CA2339051A1 (fr)
DE (1) DE60102171T2 (fr)
DK (1) DK1132392T3 (fr)
ES (1) ES2214385T3 (fr)
PT (1) PT1132392E (fr)
TR (1) TR200400630T4 (fr)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5413293A (en) * 1992-12-22 1995-05-09 Hughes Aircraft Company Magnetic torque attitude control systems
US6555581B1 (en) 2001-02-15 2003-04-29 Jones Pharma, Inc. Levothyroxine compositions and methods
US6995143B2 (en) * 2002-02-28 2006-02-07 Basilea Pharmaceutica Ag Macrolides with antibacterial activity
AR043050A1 (es) 2002-09-26 2005-07-13 Rib X Pharmaceuticals Inc Compuestos heterociclicos bifuncionales y metodos para preparar y usar los mismos
ES2552682T3 (es) 2003-03-10 2015-12-01 Merck Sharp & Dohme Corp. Agentes antibacterianos novedosos
EP2716647A3 (fr) 2004-02-27 2014-08-20 Rib-X Pharmaceuticals, Inc. Composes Macrocycliques Et Leurs Procedes De Fabrication Et D'utilisation
BRPI0519135A2 (pt) 2004-12-21 2008-12-23 Pfizer Prod Inc macrolÍdeos
US7387972B2 (en) * 2006-03-01 2008-06-17 Promos Technologies Pte. Ltd. Reducing nitrogen concentration with in-situ steam generation
WO2009055557A1 (fr) * 2007-10-25 2009-04-30 Cempra Pharmaceuticals, Inc. Procédé pour la préparation d'agents antibactériens macrolides
WO2010048601A1 (fr) 2008-10-24 2010-04-29 Cempra Pharmaceuticals, Inc. Biodéfenses utilisant des macrolides contenant du triazole
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
AU2010292010B2 (en) * 2009-09-10 2016-01-07 Cempra Pharmaceuticals, Inc. Methods for treating malaria, tuberculosis and MAC diseases
SI2550286T1 (sl) 2010-03-22 2016-04-29 Cempra Pharmaceuticals, Inc. Kristalne oblike makrolida in njihove uporabe
RU2608390C2 (ru) 2010-05-20 2017-01-18 Семпра Фармасьютикалз, Инк. Способы получения макролидов и кетолидов, и промежуточных соединений для их получения
JP6042334B2 (ja) 2010-09-10 2016-12-14 センプラ ファーマシューティカルズ,インコーポレイテッド 疾患治療のための水素結合形成フルオロケトライド
RU2658050C2 (ru) 2012-03-27 2018-06-19 Семпра Фармасьютикалз, Инк. Парентеральные составы для введения макролидных антибиотиков
US9861616B2 (en) 2013-03-14 2018-01-09 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor
CN105188712A (zh) 2013-03-15 2015-12-23 森普拉制药公司 用于制备大环内酯抗菌剂的收敛方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL114589A (en) * 1990-11-21 1999-12-22 Roussel Uclaf Intermediates for the preparation of the history of erythromycin
FR2742757B1 (fr) * 1995-12-22 1998-01-30 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
CO4990960A1 (es) 1997-10-29 2000-12-26 Abbott Lab Derivados de cetolidos 2-halo-6-o sustituidos
FR2777282B1 (fr) 1998-04-08 2001-04-20 Hoechst Marion Roussel Inc Nouveaux derives de la 2-fluoro 3-de((2,6-dideoxy 3-c-methyl 3-0-methyl-alpha-l-ribohexopyranosyl) oxyl) 6-o-methyl 3-oxo erythromycine, leur procede de preparation et leur application a la synthese de principes actifs de medicaments

Also Published As

Publication number Publication date
EP1132392B1 (fr) 2004-03-03
ES2214385T3 (es) 2004-09-16
BR0100850A (pt) 2001-11-27
PT1132392E (pt) 2004-06-30
EP1132392A1 (fr) 2001-09-12
CA2339051A1 (fr) 2001-09-06
JP2001261694A (ja) 2001-09-26
US20020065235A1 (en) 2002-05-30
ATE260928T1 (de) 2004-03-15
TR200400630T4 (tr) 2004-05-21
US6555524B2 (en) 2003-04-29
DE60102171T2 (de) 2005-03-03
DE60102171D1 (de) 2004-04-08

Similar Documents

Publication Publication Date Title
EA200100623A1 (ru) Кетолидные антибиотики
ATE344269T1 (de) Carbamat und carbazat ketolid antibiotika
DK1132392T3 (da) Ketolid-antibiotika
BG105543A (en) Novel macrolide antibiotics
DE69917717D1 (de) C11-Carbamate von antibakteriellen Makroliden
DK1167376T3 (da) Makrolidantibiotika
YU66900A (sh) Derivati higromicina a
WO2002018353A3 (fr) Agents chimiotherapeutiques d'oxazolidinone
YU64300A (sh) Derivati 2"-deoksi higromicina
AP2001002154A0 (en) Hygromycin a derivatives (changed by the ISA to read hygromycin a derivatives as antibacterial agents.
EA200201167A1 (ru) Производные гигромицина а для лечения бактериальных и протозойных инфекций
AP2002002492A0 (en) Hygromycin a prodrugs.