DK1073447T3 - N1-modificerede glycopeptider - Google Patents

N1-modificerede glycopeptider

Info

Publication number
DK1073447T3
DK1073447T3 DK99909654T DK99909654T DK1073447T3 DK 1073447 T3 DK1073447 T3 DK 1073447T3 DK 99909654 T DK99909654 T DK 99909654T DK 99909654 T DK99909654 T DK 99909654T DK 1073447 T3 DK1073447 T3 DK 1073447T3
Authority
DK
Denmark
Prior art keywords
modified glycopeptides
glycopeptides
modified
compounds
useful
Prior art date
Application number
DK99909654T
Other languages
Danish (da)
English (en)
Inventor
Richard Craig Thompson
Stephen Charles Wilkie
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Application granted granted Critical
Publication of DK1073447T3 publication Critical patent/DK1073447T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K9/00Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/006Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
    • C07K9/008Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
DK99909654T 1998-05-01 1999-02-26 N1-modificerede glycopeptider DK1073447T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US8387998P 1998-05-01 1998-05-01
PCT/US1999/004306 WO1999056760A1 (en) 1998-05-01 1999-02-26 N1-modified glycopeptides

Publications (1)

Publication Number Publication Date
DK1073447T3 true DK1073447T3 (da) 2007-09-03

Family

ID=22181253

Family Applications (1)

Application Number Title Priority Date Filing Date
DK99909654T DK1073447T3 (da) 1998-05-01 1999-02-26 N1-modificerede glycopeptider

Country Status (10)

Country Link
US (3) US6670446B1 (enExample)
EP (1) EP1073447B1 (enExample)
JP (1) JP4307723B2 (enExample)
AT (1) ATE361931T1 (enExample)
AU (1) AU2881399A (enExample)
CA (1) CA2330619A1 (enExample)
DE (1) DE69936052T2 (enExample)
DK (1) DK1073447T3 (enExample)
ES (1) ES2283107T3 (enExample)
WO (1) WO1999056760A1 (enExample)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4307723B2 (ja) * 1998-05-01 2009-08-05 イーライ リリー アンド カンパニー N1−修飾グリコペプチド
US6392012B1 (en) 1998-12-23 2002-05-21 Advanced Medicine, Inc. Glycopeptide derivatives and pharmaceutical compositions containing the same
AU4054900A (en) * 1999-04-02 2000-10-23 Advanced Medicine East, Inc. Desleucyl glycopeptide antibiotics and methods of making same
US6699836B2 (en) 1999-04-02 2004-03-02 The Trustees Of Princeton University Vancomycin analogs
US7365053B2 (en) * 2000-02-11 2008-04-29 Eli Lilly And Company Selective N-acylation of A82846 glygopeptides analogs
UA90707C2 (en) 2005-04-06 2010-05-25 Астразенека Аб Novel 5-substituted 7-amino-[1,3]thiazolo[4,5-d]pyrimidine derivatives
AR053347A1 (es) 2005-04-06 2007-05-02 Astrazeneca Ab Derivados de [1,3]tiazolo[4,5-d]pirimidin-2(3h)-ona 5,7-sustituidos
JP5192384B2 (ja) 2005-09-22 2013-05-08 メディバス エルエルシー ビス−(α−アミノ)−ジオール−ジエステル含有ポリ(エステルアミド)およびポリ(エステルウレタン)組成物および使用の方法
JP5178520B2 (ja) 2005-09-22 2013-04-10 メディバス エルエルシー 固体ポリマー送達組成物およびその使用法
EP2260060A4 (en) 2008-04-01 2013-01-16 Univ Cornell ORGANIC SOLUBLE CHITOSA SALT AND CHITOSAN DERIVED BIOMATERIALS MANUFACTURED THEREFROM

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4698327A (en) 1985-04-25 1987-10-06 Eli Lilly And Company Novel glycopeptide derivatives
US4643987A (en) 1985-08-14 1987-02-17 Eli Lilly And Company Modified glycopeptides
US4639433A (en) 1985-08-14 1987-01-27 Eli Lilly And Company Glycopeptide derivatives
EG18377A (en) * 1986-09-19 1993-04-30 Lilly Co Eli Process for preparing glycopeptide antibiotics
US5534420A (en) 1988-07-28 1996-07-09 Eli Lilly And Company Biotransformation of glycopeptide antibiotics
CA2031803C (en) * 1989-12-13 2001-05-29 Ramakrishnan Nagarajan Improvements in or relating to glycopeptide deriveratives
AU703106B2 (en) 1994-01-28 1999-03-18 Eli Lilly And Company Glycopeptide antibiotic derivatives
US5952310A (en) * 1997-05-20 1999-09-14 Eli Lilly And Company Glycopeptide hexapeptides
JP4307723B2 (ja) 1998-05-01 2009-08-05 イーライ リリー アンド カンパニー N1−修飾グリコペプチド

Also Published As

Publication number Publication date
ES2283107T3 (es) 2007-10-16
AU2881399A (en) 1999-11-23
EP1073447A4 (en) 2001-10-04
EP1073447A1 (en) 2001-02-07
US20060128609A1 (en) 2006-06-15
US6670446B1 (en) 2003-12-30
WO1999056760A1 (en) 1999-11-11
JP2002513764A (ja) 2002-05-14
US20050037950A1 (en) 2005-02-17
US6939947B2 (en) 2005-09-06
DE69936052D1 (de) 2007-06-21
ATE361931T1 (de) 2007-06-15
DE69936052T2 (de) 2008-01-17
JP4307723B2 (ja) 2009-08-05
CA2330619A1 (en) 1999-11-11
EP1073447B1 (en) 2007-05-09

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