DK0995747T3 - Substituterede sulfonylphenylheterocykler som cyclooxygenase-2- og 5-lipoxygenase-inhibitorer - Google Patents

Substituterede sulfonylphenylheterocykler som cyclooxygenase-2- og 5-lipoxygenase-inhibitorer

Info

Publication number
DK0995747T3
DK0995747T3 DK00100201T DK00100201T DK0995747T3 DK 0995747 T3 DK0995747 T3 DK 0995747T3 DK 00100201 T DK00100201 T DK 00100201T DK 00100201 T DK00100201 T DK 00100201T DK 0995747 T3 DK0995747 T3 DK 0995747T3
Authority
DK
Denmark
Prior art keywords
cyclooxygenase
heterocycles
lipoxygenase inhibitors
sulfonylphenyl
substituted
Prior art date
Application number
DK00100201T
Other languages
Danish (da)
English (en)
Inventor
James A Sikorski
Balekudru Devadas
Matthew J Graneto
Jeffery S Carter
Bryan H Norman
Roland S Rogers
Kathy L Rogers
Hwang-Fun Lu
David L Brown
John Jeffrey Talley
Original Assignee
Searle & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23828245&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK0995747(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Searle & Co filed Critical Searle & Co
Application granted granted Critical
Publication of DK0995747T3 publication Critical patent/DK0995747T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Rheumatology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
DK00100201T 1995-06-02 1996-05-31 Substituterede sulfonylphenylheterocykler som cyclooxygenase-2- og 5-lipoxygenase-inhibitorer DK0995747T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US08/460,324 US5643933A (en) 1995-06-02 1995-06-02 Substituted sulfonylphenylheterocycles as cyclooxygenase-2 and 5-lipoxygenase inhibitors

Publications (1)

Publication Number Publication Date
DK0995747T3 true DK0995747T3 (da) 2002-11-25

Family

ID=23828245

Family Applications (2)

Application Number Title Priority Date Filing Date
DK00100201T DK0995747T3 (da) 1995-06-02 1996-05-31 Substituterede sulfonylphenylheterocykler som cyclooxygenase-2- og 5-lipoxygenase-inhibitorer
DK96917888T DK0828736T3 (da) 1995-06-02 1996-05-31 Substituerede sulfonylphenylheterocycler som cyclooxygenase-2- og 5-lipoxygenase-inhibitorer

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK96917888T DK0828736T3 (da) 1995-06-02 1996-05-31 Substituerede sulfonylphenylheterocycler som cyclooxygenase-2- og 5-lipoxygenase-inhibitorer

Country Status (11)

Country Link
US (1) US5643933A (de)
EP (2) EP0828736B1 (de)
AT (2) ATE246188T1 (de)
AU (1) AU6027996A (de)
CA (1) CA2223091A1 (de)
DE (2) DE69629290T2 (de)
DK (2) DK0995747T3 (de)
ES (2) ES2181614T3 (de)
HK (1) HK1027802A1 (de)
PT (2) PT828736E (de)
WO (1) WO1996038442A1 (de)

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Also Published As

Publication number Publication date
CA2223091A1 (en) 1996-12-05
EP0995747B1 (de) 2002-08-07
HK1027802A1 (en) 2001-01-23
PT828736E (pt) 2003-12-31
DE69622894D1 (de) 2002-09-12
EP0995747A1 (de) 2000-04-26
PT995747E (pt) 2002-12-31
ES2181614T3 (es) 2003-03-01
US5643933A (en) 1997-07-01
ATE221885T1 (de) 2002-08-15
EP0828736A1 (de) 1998-03-18
EP0828736B1 (de) 2003-07-30
DK0828736T3 (da) 2003-11-24
DE69622894T2 (de) 2003-04-30
WO1996038442A1 (en) 1996-12-05
DE69629290T2 (de) 2004-04-22
AU6027996A (en) 1996-12-18
ATE246188T1 (de) 2003-08-15
DE69629290D1 (en) 2003-09-04
ES2205035T3 (es) 2004-05-01

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