DK0874815T3 - 17-Sidekæde alkynyl og 20-oxopregna-derivater af vitamin D, Fremgangsmåder til deres fremstilling og farmaceutiske præparater deraf - Google Patents

17-Sidekæde alkynyl og 20-oxopregna-derivater af vitamin D, Fremgangsmåder til deres fremstilling og farmaceutiske præparater deraf

Info

Publication number
DK0874815T3
DK0874815T3 DK96943236T DK96943236T DK0874815T3 DK 0874815 T3 DK0874815 T3 DK 0874815T3 DK 96943236 T DK96943236 T DK 96943236T DK 96943236 T DK96943236 T DK 96943236T DK 0874815 T3 DK0874815 T3 DK 0874815T3
Authority
DK
Denmark
Prior art keywords
derivatives
oxopregna
vitamin
preparation
methods
Prior art date
Application number
DK96943236T
Other languages
English (en)
Inventor
Robert Henry Hesse
Maurice Murdoch Pechet
Sundara Katugam Srinivas Setty
Original Assignee
Res Inst Medicine Chem
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Res Inst Medicine Chem filed Critical Res Inst Medicine Chem
Application granted granted Critical
Publication of DK0874815T3 publication Critical patent/DK0874815T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C401/00Irradiation products of cholesterol or its derivatives; Vitamin D derivatives, 9,10-seco cyclopenta[a]phenanthrene or analogues obtained by chemical preparation without irradiation
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/59Compounds containing 9, 10- seco- cyclopenta[a]hydrophenanthrene ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Transplantation (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicinal Preparation (AREA)
DK96943236T 1995-12-21 1996-12-23 17-Sidekæde alkynyl og 20-oxopregna-derivater af vitamin D, Fremgangsmåder til deres fremstilling og farmaceutiske præparater deraf DK0874815T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9526208.5A GB9526208D0 (en) 1995-12-21 1995-12-21 Chemical compounds
PCT/GB1996/003218 WO1997023453A1 (en) 1995-12-21 1996-12-23 17-side chain alkynyl-and 20-oxopregna-derivatives of vitamin d, methods for their production and pharmaceutical compositions thereof

Publications (1)

Publication Number Publication Date
DK0874815T3 true DK0874815T3 (da) 2002-03-04

Family

ID=10785847

Family Applications (1)

Application Number Title Priority Date Filing Date
DK96943236T DK0874815T3 (da) 1995-12-21 1996-12-23 17-Sidekæde alkynyl og 20-oxopregna-derivater af vitamin D, Fremgangsmåder til deres fremstilling og farmaceutiske præparater deraf

Country Status (21)

Country Link
US (2) US6372926B2 (da)
EP (1) EP0874815B1 (da)
JP (1) JP2000503636A (da)
KR (1) KR19990076664A (da)
CN (1) CN1086694C (da)
AT (1) ATE200663T1 (da)
AU (1) AU710680B2 (da)
CA (1) CA2241011A1 (da)
CZ (1) CZ290930B6 (da)
DE (1) DE69612568T2 (da)
DK (1) DK0874815T3 (da)
ES (1) ES2155948T3 (da)
GB (1) GB9526208D0 (da)
GR (1) GR3036132T3 (da)
HU (1) HUP9903786A3 (da)
IL (1) IL125027A0 (da)
NO (1) NO982816L (da)
NZ (1) NZ324775A (da)
PT (1) PT874815E (da)
WO (1) WO1997023453A1 (da)
ZA (1) ZA9610874B (da)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003087048A2 (en) * 2002-04-11 2003-10-23 Instytut Farmaceutyczny Preparation of 24 alkyl analogs of cholecalciferol and non-racemic compounds
US7253293B2 (en) * 2004-01-06 2007-08-07 Andrzej Slominski Enzymatic method to produce 7-dehydropregnenolone, vitamin D3-like compounds and derivatives thereof
CA2571710A1 (en) 2004-06-24 2006-11-02 Nicholas Valiante Small molecule immunopotentiators and assays for their detection
US20080280860A1 (en) * 2005-03-23 2008-11-13 Bioxell S.P.A. Use of Vitamin D Compounds to Treat Endometriosis
TW200714580A (en) * 2005-10-14 2007-04-16 Formosa Lab Inc Process for preparing vitamin D analogs
SG173119A1 (en) * 2009-01-27 2011-08-29 Berg Biosystems Llc Vitamin d3 and analogs thereof for alleviating side effects associated with chemotherapy
BR112012003372A2 (pt) 2009-08-14 2019-09-24 Berg Biosystems Llc vitamina d3 e análogos da mesma para o tratamento de alopecia.
JP5563324B2 (ja) * 2010-02-03 2014-07-30 フォーモサ・ラボラトリーズ・インコーポレーテッド マキサカルシトール中間体およびその製造方法
EP3003497B1 (en) 2013-05-29 2024-02-14 BPGbio, Inc. Preventing or mitigating chemotherapy induced alopecia using vitamin d

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6034543B2 (ja) 1977-07-01 1985-08-09 中外製薬株式会社 ビタミンd誘導体
GB9214202D0 (en) * 1992-07-03 1992-08-12 Leo Pharm Prod Ltd Chemical compounds
GB9220439D0 (en) * 1992-09-28 1992-11-11 Leo Pharm Prod Ltd Chemical compounds
US5397776A (en) * 1993-08-20 1995-03-14 Wisconsin Alumni Research Foundation Vitamin D compounds with anti-progesterone activity

Also Published As

Publication number Publication date
ZA9610874B (en) 1997-06-18
NZ324775A (en) 1999-02-25
CZ194798A3 (cs) 1998-11-11
JP2000503636A (ja) 2000-03-28
CN1086694C (zh) 2002-06-26
ES2155948T3 (es) 2001-06-01
GR3036132T3 (en) 2001-09-28
US20020010163A1 (en) 2002-01-24
NO982816L (no) 1998-08-21
CN1209120A (zh) 1999-02-24
GB9526208D0 (en) 1996-02-21
US6372926B2 (en) 2002-04-16
CA2241011A1 (en) 1997-07-03
DE69612568D1 (de) 2001-05-23
EP0874815A1 (en) 1998-11-04
US20020188142A1 (en) 2002-12-12
EP0874815B1 (en) 2001-04-18
NO982816D0 (no) 1998-06-18
AU1202597A (en) 1997-07-17
ATE200663T1 (de) 2001-05-15
PT874815E (pt) 2001-07-31
IL125027A0 (en) 1999-01-26
KR19990076664A (ko) 1999-10-15
HUP9903786A3 (en) 2000-09-28
WO1997023453A1 (en) 1997-07-03
CZ290930B6 (cs) 2002-11-13
DE69612568T2 (de) 2001-09-06
AU710680B2 (en) 1999-09-30
HUP9903786A2 (hu) 2000-03-28

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