DK0738269T5 - Piperidinderivater med PAF-antagonistaktivitet - Google Patents
Piperidinderivater med PAF-antagonistaktivitetInfo
- Publication number
- DK0738269T5 DK0738269T5 DK95932668T DK95932668T DK0738269T5 DK 0738269 T5 DK0738269 T5 DK 0738269T5 DK 95932668 T DK95932668 T DK 95932668T DK 95932668 T DK95932668 T DK 95932668T DK 0738269 T5 DK0738269 T5 DK 0738269T5
- Authority
- DK
- Denmark
- Prior art keywords
- pct
- antagonist activity
- piperidine derivatives
- paf antagonist
- paf
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ES09402291A ES2087038B1 (es) | 1994-11-07 | 1994-11-07 | Nuevas piperidinas con actividad antagonista del paf. |
PCT/EP1995/003487 WO1996014317A1 (en) | 1994-11-07 | 1995-09-05 | Novel piperidine derivatives with paf antagonist activity |
Publications (2)
Publication Number | Publication Date |
---|---|
DK0738269T3 DK0738269T3 (da) | 2000-08-28 |
DK0738269T5 true DK0738269T5 (da) | 2000-12-18 |
Family
ID=8287905
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK95932668T DK0738269T5 (da) | 1994-11-07 | 1995-09-05 | Piperidinderivater med PAF-antagonistaktivitet |
Country Status (13)
Country | Link |
---|---|
US (1) | US5705504A (da) |
EP (1) | EP0738269B1 (da) |
JP (1) | JP4018137B2 (da) |
KR (1) | KR100514201B1 (da) |
AT (1) | ATE192152T1 (da) |
AU (1) | AU3563695A (da) |
DE (1) | DE69516503T2 (da) |
DK (1) | DK0738269T5 (da) |
ES (2) | ES2087038B1 (da) |
GR (1) | GR3033528T3 (da) |
NO (1) | NO306345B1 (da) |
PT (1) | PT738269E (da) |
WO (1) | WO1996014317A1 (da) |
Families Citing this family (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE69611598T2 (de) * | 1995-09-08 | 2001-06-07 | Uriach & Cia Sa J | Azoderivate von 5-aminosalicylsäure zur behandlung von enzündlichen darmerkrankungen |
ES2165803B1 (es) * | 2000-04-10 | 2003-09-16 | Uriach & Cia Sa J | Nueva sal de un derivado azo del acido 5-aminosalicilico |
GB0013060D0 (en) | 2000-05-31 | 2000-07-19 | Astrazeneca Ab | Chemical compounds |
US6638950B2 (en) | 2000-06-21 | 2003-10-28 | Bristol-Myers Squibb Pharma Company | Piperidine amides as modulators of chemokine receptor activity |
CA2774959C (en) * | 2000-08-04 | 2016-05-31 | Dmi Biosciences, Inc. | Method of using diketopiperazines and composition containing them |
GB0021670D0 (en) | 2000-09-04 | 2000-10-18 | Astrazeneca Ab | Chemical compounds |
GB0117899D0 (en) | 2001-07-23 | 2001-09-12 | Astrazeneca Ab | Chemical compounds |
JP2007500747A (ja) | 2003-05-15 | 2007-01-18 | ディーエムアイ バイオサイエンシズ インコーポレイテッド | T細胞媒介性疾患の処置 |
FR2860514A1 (fr) * | 2003-10-03 | 2005-04-08 | Sanofi Synthelabo | Derives d'arylalkylcarbamates, leur preparation et leur application en therapeutique |
WO2007101270A1 (en) * | 2006-03-02 | 2007-09-07 | Incyte Corporation | MODULATORS OF 11-β HYDROXYL STEROID DEHYDROGENASE TYPE 1, PHARMACEUTICAL COMPOSITIONS THEREOF, AND METHODS OF USING THE SAME |
CA2658913C (en) * | 2006-07-24 | 2015-07-21 | Ucb Pharma S.A. | Substituted aniline derivatives |
KR100737397B1 (ko) | 2007-01-31 | 2007-07-09 | 한국교세라정공(주) | 밀링 커터 |
JP5856843B2 (ja) | 2008-05-27 | 2016-02-10 | アンピオ ファーマシューティカルズ,インコーポレイテッド | ジケトピペラジンを用いた医薬組成物 |
FR2962649A1 (fr) | 2010-07-19 | 2012-01-20 | Conservatoire Nat Arts Et Metiers | Traitement d'une pathologie liee a un effet excessif du tnf par un compose de benzene sulfonamide |
GB201101517D0 (en) * | 2011-01-28 | 2011-03-16 | Proximagen Ltd | Receptor antagonists |
SG10201608087WA (en) | 2011-10-10 | 2016-11-29 | Ampio Pharmaceuticals Inc | Implantable medical devices with increased immune tolerance, and methods for making and implanting |
EP2766029B1 (en) | 2011-10-10 | 2020-03-25 | Ampio Pharmaceuticals, Inc. | Treatment of degenerative joint disease |
MX355446B (es) | 2011-10-28 | 2018-04-18 | Ampio Pharmaceuticals Inc | Tratamiento de rinitis. |
CA2906864A1 (en) | 2013-03-15 | 2014-09-18 | Ampio Pharmaceuticals, Inc. | Compositions for the mobilization, homing, expansion and differentiation of stem cells and methods of using the same |
KR20170045274A (ko) | 2014-08-18 | 2017-04-26 | 앰피오 파마슈티컬스 인코퍼레이티드 | 관절 징후의 치료 |
US11389512B2 (en) | 2015-06-22 | 2022-07-19 | Ampio Pharmaceuticals, Inc. | Use of low molecular weight fractions of human serum albumin in treating diseases |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0029707B1 (en) * | 1979-11-21 | 1984-02-01 | Kyowa Hakko Kogyo Co., Ltd | Novel piperidine derivatives, method for the preparation thereof and pharmaceutical compositions containing them |
IL85700A0 (en) * | 1987-03-24 | 1988-08-31 | Takeda Chemical Industries Ltd | 1,4-disubstituted piperazine compounds,their production and use |
EP0441226A1 (en) * | 1990-01-29 | 1991-08-14 | J. URIACH & CIA. S.A. | (cyanomethyl)pyridines useful as PAF antagonists |
GB9102997D0 (en) * | 1991-02-13 | 1991-03-27 | Pfizer Ltd | Therapeutic agents |
ES2036926B1 (es) * | 1991-08-08 | 1994-01-16 | Uriach & Cia Sa J | "procedimiento para la obtencion de derivados de la (2-alquil-3-piridil)metilpiperazina". |
US5268376A (en) * | 1991-09-04 | 1993-12-07 | Minnesota Mining And Manufacturing Company | 1-substituted 1H-imidazo[4,5-c]quinolin-4-amines |
US5283242A (en) * | 1991-10-24 | 1994-02-01 | American Home Products Corporation | Substituted benzimidazoles and quinazolines as antihypertensives |
-
1994
- 1994-11-07 ES ES09402291A patent/ES2087038B1/es not_active Expired - Fee Related
-
1995
- 1995-09-05 AU AU35636/95A patent/AU3563695A/en not_active Abandoned
- 1995-09-05 DK DK95932668T patent/DK0738269T5/da active
- 1995-09-05 KR KR1019960703655A patent/KR100514201B1/ko not_active IP Right Cessation
- 1995-09-05 AT AT95932668T patent/ATE192152T1/de not_active IP Right Cessation
- 1995-09-05 DE DE69516503T patent/DE69516503T2/de not_active Expired - Lifetime
- 1995-09-05 ES ES95932668T patent/ES2147616T3/es not_active Expired - Lifetime
- 1995-09-05 EP EP95932668A patent/EP0738269B1/en not_active Expired - Lifetime
- 1995-09-05 WO PCT/EP1995/003487 patent/WO1996014317A1/en active IP Right Grant
- 1995-09-05 JP JP51497296A patent/JP4018137B2/ja not_active Expired - Fee Related
- 1995-09-05 PT PT95932668T patent/PT738269E/pt unknown
- 1995-09-05 US US08/669,440 patent/US5705504A/en not_active Expired - Lifetime
-
1996
- 1996-07-05 NO NO962855A patent/NO306345B1/no not_active IP Right Cessation
-
2000
- 2000-05-29 GR GR20000401219T patent/GR3033528T3/el not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
PT738269E (pt) | 2000-08-31 |
ES2147616T3 (es) | 2000-09-16 |
MX9602559A (es) | 1997-07-31 |
DE69516503T2 (de) | 2001-03-15 |
ATE192152T1 (de) | 2000-05-15 |
DE69516503D1 (de) | 2000-05-31 |
AU3563695A (en) | 1996-05-31 |
NO962855L (no) | 1996-07-05 |
NO962855D0 (no) | 1996-07-05 |
GR3033528T3 (en) | 2000-09-29 |
DK0738269T3 (da) | 2000-08-28 |
JPH09507862A (ja) | 1997-08-12 |
EP0738269A1 (en) | 1996-10-23 |
NO306345B1 (no) | 1999-10-25 |
WO1996014317A1 (en) | 1996-05-17 |
ES2087038A1 (es) | 1996-07-01 |
EP0738269B1 (en) | 2000-04-26 |
JP4018137B2 (ja) | 2007-12-05 |
US5705504A (en) | 1998-01-06 |
ES2087038B1 (es) | 1997-03-16 |
KR100514201B1 (ko) | 2005-12-29 |
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