DK0593520T3 - Forbindelser med indhold af steroider og deres anvendelse til behandling af glaucom - Google Patents

Forbindelser med indhold af steroider og deres anvendelse til behandling af glaucom

Info

Publication number
DK0593520T3
DK0593520T3 DK92912769T DK92912769T DK0593520T3 DK 0593520 T3 DK0593520 T3 DK 0593520T3 DK 92912769 T DK92912769 T DK 92912769T DK 92912769 T DK92912769 T DK 92912769T DK 0593520 T3 DK0593520 T3 DK 0593520T3
Authority
DK
Denmark
Prior art keywords
pct
glaucoma
treatment
content
date
Prior art date
Application number
DK92912769T
Other languages
Danish (da)
English (en)
Inventor
Gerard Schwadrohn
Original Assignee
Theramex
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR9109017A external-priority patent/FR2679139B1/fr
Priority claimed from FR9109015A external-priority patent/FR2679137B1/fr
Priority claimed from FR9109016A external-priority patent/FR2679138B1/fr
Priority claimed from FR9110160A external-priority patent/FR2680108B1/fr
Application filed by Theramex filed Critical Theramex
Application granted granted Critical
Publication of DK0593520T3 publication Critical patent/DK0593520T3/da

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/575Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of three or more carbon atoms, e.g. cholane, cholestane, ergosterol, sitosterol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J71/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005Oxygen-containing hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J9/00Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Ophthalmology & Optometry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
DK92912769T 1991-06-18 1992-06-18 Forbindelser med indhold af steroider og deres anvendelse til behandling af glaucom DK0593520T3 (da)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
FR9107412 1991-06-18
FR9109017A FR2679139B1 (fr) 1991-07-17 1991-07-17 Nouvelles compositions pharmaceutiques destinees a l'application oculaire renfermant un derive androstenique et leur procede de preparation.
FR9109015A FR2679137B1 (fr) 1991-07-17 1991-07-17 Nouvelles compositions pharmaceutiques a base d'un derive pregnenique et leur procede de preparation.
FR9109016A FR2679138B1 (fr) 1991-07-17 1991-07-17 Compositions pharmaceutiques anti-glaucomateuses et leur procede d'obtention.
FR9110160A FR2680108B1 (fr) 1991-08-09 1991-08-09 Nouvelles compositions pharmaceutiques a base de sterouides 6-hydroxymethyles et leur procede d'obtention.
PCT/FR1992/000549 WO1992022300A1 (fr) 1991-06-18 1992-06-18 Compositions oculaires contenant des steroïdes et leur utilisation pour le traitement du glaucome

Publications (1)

Publication Number Publication Date
DK0593520T3 true DK0593520T3 (da) 2000-04-03

Family

ID=27515565

Family Applications (1)

Application Number Title Priority Date Filing Date
DK92912769T DK0593520T3 (da) 1991-06-18 1992-06-18 Forbindelser med indhold af steroider og deres anvendelse til behandling af glaucom

Country Status (11)

Country Link
US (1) US5506220A (ja)
EP (1) EP0593520B1 (ja)
JP (1) JP3328729B2 (ja)
KR (1) KR100249555B1 (ja)
AT (1) ATE185071T1 (ja)
CA (1) CA2111699A1 (ja)
DE (1) DE69230069T2 (ja)
DK (1) DK0593520T3 (ja)
ES (1) ES2139602T3 (ja)
GR (1) GR3031967T3 (ja)
WO (1) WO1992022300A1 (ja)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2311465A1 (en) * 2003-04-18 2011-04-20 Advanced Medicine Research Institute Remedies for diseases to be applied to eye
WO2004093882A1 (ja) * 2003-04-18 2004-11-04 Advanced Medicine Research Institute 眼に適用する疾患治療剤
DK1919290T3 (da) * 2005-07-12 2014-04-22 Ampio Pharmaceuticals Inc Fremgangsmåder og produkter til behandling af sygdomme
SG2014008163A (en) 2009-06-22 2014-04-28 Ampio Pharmaceuticals Inc Method for treatment of diseases
EP2445350A4 (en) * 2009-06-22 2012-12-26 Dmi Acquisition Corp METHOD AND PRODUCTS FOR THE TREATMENT OF DISEASES
CN102134265B (zh) * 2009-12-29 2013-04-03 黄云生 一种合成6-甲基-17α-乙酰氧基-19-去甲孕甾-4,6-二烯-3,20-二酮的方法
CA2836612C (en) 2011-05-20 2018-06-12 Pier Vincenzo PIAZZA Antagonists of cb1 receptor
JP6335915B2 (ja) 2012-11-28 2018-05-30 アンスティチュ ナショナル ドゥ ラ サンテ エ ドゥ ラ ルシェルシュ メディカル プレグネノロンの3−(4’−置換)−ベンジル−エーテル誘導体
SG11201504380SA (en) 2012-12-19 2015-07-30 Ampio Pharmaceuticals Inc Method for treatment of diseases

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1515284A (en) * 1974-05-21 1978-06-21 Gastaud J Pharmaceutical compositions containing progestogens derived from the 17-alpha-hydroxy-19-nor-progesterone series
US4383992A (en) * 1982-02-08 1983-05-17 Lipari John M Water-soluble steroid compounds
US4617299A (en) * 1983-12-19 1986-10-14 Knepper Paul A Method for the prevention of ocular hypertension, treatment of glaucoma and treatment of ocular hypertension
US4863912A (en) * 1986-05-19 1989-09-05 New York Medical College Use of tetrahydrocortisol in glaucoma therapy
WO1987007141A1 (en) * 1986-05-23 1987-12-03 New England Medical Center Hospitals, Inc. Method for treating glaucoma
FR2622194B1 (fr) * 1987-10-27 1990-03-23 Theramex Laboratoire Nouveaux derives de la 19-nor progesterone, leur procede d'obtention et les compositions pharmaceutiques en contenant
US4876250A (en) * 1988-10-31 1989-10-24 Alcon Laboratories, Inc. Methods for controlling ocular hypertension with angiostatic steroids
FR2645864B1 (fr) * 1989-04-13 1991-07-12 Theramex Nouveaux derives alcoyles en 17/21 de la 19-nor progesterone, leurs procedes d'obtention et les compositions pharmaceutiques en renfermant
FR2679236B1 (fr) 1991-07-18 1997-01-24 Theramex Nouveaux sterouides substitues en position 6, leurs procedes d'obtention et des compositions pharmaceutiques en renfermant.

Also Published As

Publication number Publication date
ATE185071T1 (de) 1999-10-15
ES2139602T3 (es) 2000-02-16
US5506220A (en) 1996-04-09
WO1992022300A1 (fr) 1992-12-23
GR3031967T3 (en) 2000-03-31
KR100249555B1 (ko) 2000-04-01
EP0593520A1 (fr) 1994-04-27
JPH06508362A (ja) 1994-09-22
DE69230069D1 (de) 1999-11-04
DE69230069T2 (de) 2000-05-25
KR940701260A (ko) 1994-05-28
EP0593520B1 (fr) 1999-09-29
JP3328729B2 (ja) 2002-09-30
CA2111699A1 (fr) 1992-12-23

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