FR2679137B1 - Nouvelles compositions pharmaceutiques a base d'un derive pregnenique et leur procede de preparation. - Google Patents

Nouvelles compositions pharmaceutiques a base d'un derive pregnenique et leur procede de preparation.

Info

Publication number
FR2679137B1
FR2679137B1 FR9109015A FR9109015A FR2679137B1 FR 2679137 B1 FR2679137 B1 FR 2679137B1 FR 9109015 A FR9109015 A FR 9109015A FR 9109015 A FR9109015 A FR 9109015A FR 2679137 B1 FR2679137 B1 FR 2679137B1
Authority
FR
France
Prior art keywords
pregnenic
derivative
preparation
pharmaceutical compositions
compositions based
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR9109015A
Other languages
English (en)
Other versions
FR2679137A1 (fr
Inventor
Gerard Schwadrohn
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Laboratoire Theramex SAM
Original Assignee
Laboratoire Theramex SAM
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to FR9109015A priority Critical patent/FR2679137B1/fr
Application filed by Laboratoire Theramex SAM filed Critical Laboratoire Theramex SAM
Priority to DK92912769T priority patent/DK0593520T3/da
Priority to JP50077393A priority patent/JP3328729B2/ja
Priority to DE69230069T priority patent/DE69230069T2/de
Priority to CA002111699A priority patent/CA2111699A1/fr
Priority to ES92912769T priority patent/ES2139602T3/es
Priority to PCT/FR1992/000549 priority patent/WO1992022300A1/fr
Priority to EP92912769A priority patent/EP0593520B1/fr
Priority to US08/170,179 priority patent/US5506220A/en
Priority to KR1019930703965A priority patent/KR100249555B1/ko
Priority to AT92912769T priority patent/ATE185071T1/de
Priority to IE922252A priority patent/IE922252A1/en
Priority to DZ920090A priority patent/DZ1600A1/fr
Priority to MA22876A priority patent/MA22592A1/fr
Priority to TNSN92063 priority patent/TNSN92063A1/fr
Priority to ZA925373A priority patent/ZA925373B/xx
Publication of FR2679137A1 publication Critical patent/FR2679137A1/fr
Application granted granted Critical
Publication of FR2679137B1 publication Critical patent/FR2679137B1/fr
Priority to GR990403060T priority patent/GR3031967T3/el
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J71/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005Oxygen-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/575Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of three or more carbon atoms, e.g. cholane, cholestane, ergosterol, sitosterol
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J9/00Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR9109015A 1991-06-18 1991-07-17 Nouvelles compositions pharmaceutiques a base d'un derive pregnenique et leur procede de preparation. Expired - Fee Related FR2679137B1 (fr)

Priority Applications (17)

Application Number Priority Date Filing Date Title
FR9109015A FR2679137B1 (fr) 1991-07-17 1991-07-17 Nouvelles compositions pharmaceutiques a base d'un derive pregnenique et leur procede de preparation.
KR1019930703965A KR100249555B1 (ko) 1991-06-18 1992-06-18 스테로이드를 함유하는 안구용 조성물, 및 녹내장 치료에 이들 조성물을 사용하는 방법
DE69230069T DE69230069T2 (de) 1991-06-18 1992-06-18 Steroide enthaltende zusammensetzungen zur anwendung am auge und ihre verwendung zur behandlung des glaukoms
CA002111699A CA2111699A1 (fr) 1991-06-18 1992-06-18 Compositions pharmaceutiques anti-glaucomateuses et leur procede d'obtention
ES92912769T ES2139602T3 (es) 1991-06-18 1992-06-18 Composiciones oculares que contienen esteroides y su utilizacion para el tratamiento del glaucoma.
PCT/FR1992/000549 WO1992022300A1 (fr) 1991-06-18 1992-06-18 Compositions oculaires contenant des steroïdes et leur utilisation pour le traitement du glaucome
EP92912769A EP0593520B1 (fr) 1991-06-18 1992-06-18 Compositions oculaires contenant des steroides et leur utilisation pour le traitement du glaucome
US08/170,179 US5506220A (en) 1991-06-18 1992-06-18 Anti-glaucomatous pharmaceutical composition and the process for obtaining them
DK92912769T DK0593520T3 (da) 1991-06-18 1992-06-18 Forbindelser med indhold af steroider og deres anvendelse til behandling af glaucom
AT92912769T ATE185071T1 (de) 1991-06-18 1992-06-18 Steroide enthaltende zusammensetzungen zur anwendung am auge und ihre verwendung zur behandlung des glaukoms
JP50077393A JP3328729B2 (ja) 1991-06-18 1992-06-18 抗緑内障薬剤組成物
IE922252A IE922252A1 (en) 1991-07-17 1992-07-10 Anti-glaucomatous pharmaceutical compositions and the¹process for obtaining them
DZ920090A DZ1600A1 (fr) 1991-07-17 1992-07-12 Compositions pharmaceutiques anti-glaucomateurses et leur procédé d'obtention.
MA22876A MA22592A1 (fr) 1991-07-17 1992-07-13 Nouveau procede d'obtention d'une composition anti-glaucomateuse et son procede d'obtention .
TNSN92063 TNSN92063A1 (fr) 1991-07-17 1992-07-16 Nouveau procede d'obtention d'une composition anti- glaucomateuse et son procede d'obtention
ZA925373A ZA925373B (en) 1991-07-17 1992-07-17 Anti-glaucomatous pharmaceutical compositions and the process for obtaining them.
GR990403060T GR3031967T3 (en) 1991-06-18 1999-11-26 Ocular compositions containing steroids and their use in treating glaucoma

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9109015A FR2679137B1 (fr) 1991-07-17 1991-07-17 Nouvelles compositions pharmaceutiques a base d'un derive pregnenique et leur procede de preparation.

Publications (2)

Publication Number Publication Date
FR2679137A1 FR2679137A1 (fr) 1993-01-22
FR2679137B1 true FR2679137B1 (fr) 1995-03-17

Family

ID=9415211

Family Applications (1)

Application Number Title Priority Date Filing Date
FR9109015A Expired - Fee Related FR2679137B1 (fr) 1991-06-18 1991-07-17 Nouvelles compositions pharmaceutiques a base d'un derive pregnenique et leur procede de preparation.

Country Status (2)

Country Link
FR (1) FR2679137B1 (fr)
ZA (1) ZA925373B (fr)

Also Published As

Publication number Publication date
ZA925373B (en) 1993-05-10
FR2679137A1 (fr) 1993-01-22

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Legal Events

Date Code Title Description
ST Notification of lapse