DE69930552T2 - Exo-s-mecamylamin-formulierung und ihre verwendung in behandlungen - Google Patents
Exo-s-mecamylamin-formulierung und ihre verwendung in behandlungen Download PDFInfo
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- DE69930552T2 DE69930552T2 DE69930552T DE69930552T DE69930552T2 DE 69930552 T2 DE69930552 T2 DE 69930552T2 DE 69930552 T DE69930552 T DE 69930552T DE 69930552 T DE69930552 T DE 69930552T DE 69930552 T2 DE69930552 T2 DE 69930552T2
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- mecamylamine
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
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- Nutrition Science (AREA)
- Immunology (AREA)
- Pulmonology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US11253498P | 1998-12-16 | 1998-12-16 | |
| US112534P | 1998-12-16 | ||
| PCT/US1999/030153 WO2000035279A1 (en) | 1998-12-16 | 1999-12-16 | Exo-s-mecamylamine formulation and use in treatment |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DE69930552D1 DE69930552D1 (de) | 2006-05-11 |
| DE69930552T2 true DE69930552T2 (de) | 2006-11-30 |
Family
ID=22344414
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE69939498T Expired - Lifetime DE69939498D1 (de) | 1998-12-16 | 1999-12-16 | Exo-S-Mecamylamin-Formulierung |
| DE69930552T Expired - Lifetime DE69930552T2 (de) | 1998-12-16 | 1999-12-16 | Exo-s-mecamylamin-formulierung und ihre verwendung in behandlungen |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE69939498T Expired - Lifetime DE69939498D1 (de) | 1998-12-16 | 1999-12-16 | Exo-S-Mecamylamin-Formulierung |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US20020016370A1 (enExample) |
| EP (3) | EP1139744A4 (enExample) |
| JP (5) | JP2002532392A (enExample) |
| AT (2) | ATE320711T1 (enExample) |
| AU (2) | AU2368600A (enExample) |
| CA (2) | CA2393437C (enExample) |
| CY (1) | CY1108577T1 (enExample) |
| DE (2) | DE69939498D1 (enExample) |
| DK (2) | DK1139743T3 (enExample) |
| ES (2) | ES2260959T3 (enExample) |
| PT (2) | PT1139743E (enExample) |
| WO (2) | WO2000035280A1 (enExample) |
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| SE521512C2 (sv) | 2001-06-25 | 2003-11-11 | Niconovum Ab | Anordning för administrering av en substans till främre delen av en individs munhåla |
| US7045534B2 (en) | 2002-02-12 | 2006-05-16 | The Board Of Trustees Of The Leland Stanford Junior University | Methods of reducing angiogenesis |
| ES2708552T3 (es) | 2002-12-20 | 2019-04-10 | Niconovum Ab | Método para la preparación de un material particulado que contiene nicotina con una celulosa cristalina (en particular MCC) |
| CA2518385A1 (en) * | 2003-03-14 | 2004-09-23 | Agi Therapeutics Ltd. | Treatment of intestinal conditions with n-2,3,3-tetramethylbicyclo[2.2.1]heptan-2-amine |
| US20070224284A1 (en) | 2004-03-12 | 2007-09-27 | John Devane | Methods and compositions comprising at least one alpha3 beta4 nAChR antagonist or pharmaceutically acceptable salt thereof |
| DE10318714B4 (de) * | 2003-04-25 | 2006-03-23 | Hf Arzneimittelforschung Gmbh | Wirkstoff-Kombinationen und Therapien zur Bekämpfung des Alkoholmissbrauches |
| US8252321B2 (en) | 2004-09-13 | 2012-08-28 | Chrono Therapeutics, Inc. | Biosynchronous transdermal drug delivery for longevity, anti-aging, fatigue management, obesity, weight loss, weight management, delivery of nutraceuticals, and the treatment of hyperglycemia, alzheimer's disease, sleep disorders, parkinson's disease, aids, epilepsy, attention deficit disorder, nicotine addiction, cancer, headache and pain control, asthma, angina, hypertension, depression, cold, flu and the like |
| AU2005284908B2 (en) | 2004-09-13 | 2011-12-08 | Morningside Venture Investments Limited | Biosynchronous transdermal drug delivery |
| BRPI0620080A2 (pt) * | 2005-12-19 | 2011-11-01 | Comentis Inc | formulações tópicas de mecamilamina para adminstração ocular e usos das mesma |
| WO2007104573A2 (en) | 2006-03-16 | 2007-09-20 | Niconovum Ab | Improved snuff composition |
| US20100040679A1 (en) * | 2006-10-09 | 2010-02-18 | Shing Yue Chang | Compositions for Reducing Nicotine Withdrawal Symptoms and/or Tobacco Usage |
| US20080243005A1 (en) * | 2007-03-30 | 2008-10-02 | Searete Llc, A Limited Liability Corporation Of The State Of Delaware | Computational user-health testing |
| US20080319276A1 (en) * | 2007-03-30 | 2008-12-25 | Searete Llc, A Limited Liability Corporation Of The State Of Delaware | Computational user-health testing |
| US20090005654A1 (en) * | 2007-03-30 | 2009-01-01 | Searete Llc, A Limited Liability Corporation Of The State Of Delaware | Computational user-health testing |
| US20080242947A1 (en) * | 2007-03-30 | 2008-10-02 | Searete Llc, A Limited Liability Corporation Of The State Of Delaware | Configuring software for effective health monitoring or the like |
| US20090018407A1 (en) * | 2007-03-30 | 2009-01-15 | Searete Llc, A Limited Corporation Of The State Of Delaware | Computational user-health testing |
| US20080242948A1 (en) * | 2007-03-30 | 2008-10-02 | Searete Llc, A Limited Liability Corporation Of The State Of Delaware | Effective low-profile health monitoring or the like |
| US20090119154A1 (en) * | 2007-11-07 | 2009-05-07 | Searete Llc, A Limited Liability Corporation Of The State Of Delaware | Determining a demographic characteristic based on computational user-health testing of a user interaction with advertiser-specified content |
| US20080242949A1 (en) * | 2007-03-30 | 2008-10-02 | Searete Llc, A Limited Liability Corporation Of The State Of Delaware | Computational user-health testing |
| US20080242951A1 (en) * | 2007-03-30 | 2008-10-02 | Searete Llc, A Limited Liability Corporation Of The State Of Delaware | Effective low-profile health monitoring or the like |
| US20080242952A1 (en) * | 2007-03-30 | 2008-10-02 | Searete Llc, A Limited Liablity Corporation Of The State Of Delaware | Effective response protocols for health monitoring or the like |
| US20090005653A1 (en) * | 2007-03-30 | 2009-01-01 | Searete Llc, A Limited Liability Corporation Of The State Of Delaware | Computational user-health testing |
| ES2521494T3 (es) * | 2007-04-02 | 2014-11-12 | Parkinson's Institute | Métodos y composiciones para la reducción de los efectos secundarios de tratamientos terapéuticos |
| WO2009143403A1 (en) * | 2008-05-23 | 2009-11-26 | Targacept, Inc. | Combination therapy for the management hypertension |
| AT507187B1 (de) * | 2008-10-23 | 2010-03-15 | Helmut Dr Buchberger | Inhalator |
| SG176766A1 (en) * | 2009-07-14 | 2012-01-30 | Targacept Inc | Exo-s-mecamylamine method, use, and compound for treatment |
| JO3250B1 (ar) | 2009-09-22 | 2018-09-16 | Novartis Ag | إستعمال منشطات مستقبل نيكوتينيك أسيتيل كولين ألفا 7 |
| KR101856046B1 (ko) | 2010-05-27 | 2018-06-25 | 카탈리스트 바이오사이언시즈, 인코포레이티드 | 니코틴 수용체 비-경쟁적 길항제 |
| HUE026804T2 (en) | 2011-02-11 | 2016-07-28 | Batmark Ltd | Inhaler component |
| AT510837B1 (de) | 2011-07-27 | 2012-07-15 | Helmut Dr Buchberger | Inhalatorkomponente |
| EP2729148A4 (en) | 2011-07-06 | 2015-04-22 | Parkinson S Inst | COMPOSITIONS AND METHOD FOR THE TREATMENT OF SYMPTOMS IN PATIENTS WITH MORBUS PARKINSON |
| KR102433286B1 (ko) | 2011-09-06 | 2022-08-16 | 니코벤처스 트레이딩 리미티드 | 가열식 끽연 가능 물질 |
| CN103763953B (zh) | 2011-09-06 | 2016-08-17 | 英美烟草(投资)有限公司 | 加热可抽吸材料 |
| AT511344B1 (de) | 2011-10-21 | 2012-11-15 | Helmut Dr Buchberger | Inhalatorkomponente |
| US8901177B2 (en) * | 2012-03-23 | 2014-12-02 | Targacept, Inc. | Method of treating bladder disorders |
| GB201207039D0 (en) | 2012-04-23 | 2012-06-06 | British American Tobacco Co | Heating smokeable material |
| GB2504076A (en) | 2012-07-16 | 2014-01-22 | Nicoventures Holdings Ltd | Electronic smoking device |
| GB2504075A (en) | 2012-07-16 | 2014-01-22 | Nicoventures Holdings Ltd | Electronic smoking device |
| GB2513637A (en) | 2013-05-02 | 2014-11-05 | Nicoventures Holdings Ltd | Electronic cigarette |
| GB2513639A (en) | 2013-05-02 | 2014-11-05 | Nicoventures Holdings Ltd | Electronic cigarette |
| GB2514893B (en) | 2013-06-04 | 2017-12-06 | Nicoventures Holdings Ltd | Container |
| GB201407426D0 (en) | 2014-04-28 | 2014-06-11 | Batmark Ltd | Aerosol forming component |
| GB2528673B (en) | 2014-07-25 | 2020-07-01 | Nicoventures Holdings Ltd | Aerosol provision system |
| JP6682533B2 (ja) * | 2014-08-22 | 2020-04-15 | アタカマ セラピューティクス，インコーポレーテッド | 多汗症を治療するための方法 |
| GB2533135B (en) | 2014-12-11 | 2020-11-11 | Nicoventures Holdings Ltd | Aerosol provision systems |
| WO2016123406A1 (en) | 2015-01-28 | 2016-08-04 | Chrono Therapeutics Inc. | Drug delivery methods and systems |
| AU2016228779A1 (en) | 2015-03-12 | 2017-09-07 | Chrono Therapeutics Inc. | Craving input and support system |
| GB201505597D0 (en) | 2015-03-31 | 2015-05-13 | British American Tobacco Co | Article for use with apparatus for heating smokable material |
| GB201505595D0 (en) | 2015-03-31 | 2015-05-13 | British American Tobacco Co | Cartridge for use with apparatus for heating smokeable material |
| GB201511349D0 (en) | 2015-06-29 | 2015-08-12 | Nicoventures Holdings Ltd | Electronic aerosol provision systems |
| GB201511361D0 (en) | 2015-06-29 | 2015-08-12 | Nicoventures Holdings Ltd | Electronic vapour provision system |
| US11924930B2 (en) | 2015-08-31 | 2024-03-05 | Nicoventures Trading Limited | Article for use with apparatus for heating smokable material |
| US20170055584A1 (en) | 2015-08-31 | 2017-03-02 | British American Tobacco (Investments) Limited | Article for use with apparatus for heating smokable material |
| GB2542838B (en) | 2015-10-01 | 2022-01-12 | Nicoventures Trading Ltd | Aerosol provision system |
| US20170119046A1 (en) | 2015-10-30 | 2017-05-04 | British American Tobacco (Investments) Limited | Apparatus for Heating Smokable Material |
| US11744964B2 (en) | 2016-04-27 | 2023-09-05 | Nicoventures Trading Limited | Electronic aerosol provision system and vaporizer therefor |
| CA3049529A1 (en) | 2017-01-06 | 2018-07-12 | Chrono Therapeutics Inc. | Transdermal drug delivery devices and methods |
| CA3101966A1 (en) | 2018-05-29 | 2019-12-05 | Morningside Venture Investments Limited | Drug delivery methods and systems |
| US12397141B2 (en) | 2018-11-16 | 2025-08-26 | Morningside Venture Investments Limited | Thermally regulated transdermal drug delivery system |
| GB202203728D0 (en) * | 2022-03-17 | 2022-05-04 | Univ Oxford Innovation Ltd | Treatments and methods for increasing dopamine |
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| US5039801A (en) * | 1985-12-20 | 1991-08-13 | The United States Of America As Represented By The Department Of Health & Human Services | Thermal fragmentation of methylbenzylurea disastereomers or secondary amines and preparation of optically active secondary amines |
| US4749686A (en) * | 1986-12-04 | 1988-06-07 | New York Medical College | Combinations of renal vasodilators and α1 -adrenergic or ganglionic blocking agents and methods for treating diseases |
| EP0302595B1 (en) * | 1987-07-07 | 1994-02-02 | Beecham Group Plc | Pinacidil for treatment of pulmonary hypertension or right heart failure |
| US5691365A (en) * | 1995-07-18 | 1997-11-25 | University Of Kentucky Research Foundation | Nicotinic receptor antagonists in the treatment of neuropharmacological disorders |
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- 1999-12-16 PT PT99967401T patent/PT1139743E/pt unknown
- 1999-12-16 DK DK99967401T patent/DK1139743T3/da active
- 1999-12-16 DE DE69939498T patent/DE69939498D1/de not_active Expired - Lifetime
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- 1999-12-16 AU AU23686/00A patent/AU2368600A/en not_active Abandoned
- 1999-12-16 WO PCT/US1999/030153 patent/WO2000035279A1/en not_active Ceased
- 1999-12-16 PT PT05024899T patent/PT1634498E/pt unknown
- 1999-12-16 JP JP2000587609A patent/JP2002532393A/ja not_active Withdrawn
- 1999-12-16 CA CA002393442A patent/CA2393442A1/en not_active Abandoned
- 1999-12-16 DK DK05024899T patent/DK1634498T3/da active
- 1999-12-16 AT AT05024899T patent/ATE406797T1/de active
- 1999-12-16 EP EP99967401A patent/EP1139743B1/en not_active Expired - Lifetime
- 1999-12-16 ES ES05024899T patent/ES2313187T3/es not_active Expired - Lifetime
- 1999-12-16 EP EP05024899A patent/EP1634498B1/en not_active Expired - Lifetime
- 1999-12-16 AU AU23682/00A patent/AU2368200A/en not_active Abandoned
-
2001
- 2001-06-15 US US09/882,934 patent/US20020016370A1/en not_active Abandoned
-
2008
- 2008-11-19 CY CY20081101333T patent/CY1108577T1/el unknown
-
2011
- 2011-03-14 JP JP2011055716A patent/JP2011126909A/ja not_active Withdrawn
-
2013
- 2013-12-13 JP JP2013258032A patent/JP2014051528A/ja active Pending
-
2016
- 2016-01-25 JP JP2016011658A patent/JP2016065108A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| EP1139743B1 (en) | 2006-03-22 |
| JP2011126909A (ja) | 2011-06-30 |
| PT1634498E (pt) | 2008-10-28 |
| DK1139743T3 (da) | 2006-07-31 |
| EP1139744A1 (en) | 2001-10-10 |
| ATE320711T1 (de) | 2006-04-15 |
| JP2016065108A (ja) | 2016-04-28 |
| EP1634498A2 (en) | 2006-03-15 |
| US20020016370A1 (en) | 2002-02-07 |
| WO2000035279A1 (en) | 2000-06-22 |
| ES2260959T3 (es) | 2006-11-01 |
| JP2014051528A (ja) | 2014-03-20 |
| CA2393437C (en) | 2009-12-15 |
| EP1634498A3 (en) | 2006-03-29 |
| AU2368600A (en) | 2000-07-03 |
| AU2368200A (en) | 2000-07-03 |
| DE69930552D1 (de) | 2006-05-11 |
| DK1634498T3 (da) | 2008-12-15 |
| ATE406797T1 (de) | 2008-09-15 |
| EP1634498B1 (en) | 2008-09-03 |
| JP2002532392A (ja) | 2002-10-02 |
| CY1108577T1 (el) | 2014-04-09 |
| ES2313187T3 (es) | 2009-03-01 |
| DE69939498D1 (de) | 2008-10-16 |
| WO2000035280A1 (en) | 2000-06-22 |
| EP1139743A1 (en) | 2001-10-10 |
| EP1139743A4 (en) | 2003-01-02 |
| EP1139744A4 (en) | 2003-01-02 |
| PT1139743E (pt) | 2006-06-30 |
| CA2393437A1 (en) | 2000-06-22 |
| CA2393442A1 (en) | 2000-06-22 |
| JP2002532393A (ja) | 2002-10-02 |
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| Date | Code | Title | Description |
|---|---|---|---|
| 8364 | No opposition during term of opposition |