DE69428536D1 - A3 -adenosin -rezeptor agonisten - Google Patents

A3 -adenosin -rezeptor agonisten

Info

Publication number
DE69428536D1
DE69428536D1 DE69428536T DE69428536T DE69428536D1 DE 69428536 D1 DE69428536 D1 DE 69428536D1 DE 69428536 T DE69428536 T DE 69428536T DE 69428536 T DE69428536 T DE 69428536T DE 69428536 D1 DE69428536 D1 DE 69428536D1
Authority
DE
Germany
Prior art keywords
receptor
adenosine receptor
mammal
uronamide
provides
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE69428536T
Other languages
English (en)
Other versions
DE69428536T2 (de
Inventor
A Jacobson
Carola Gallo-Rodriguez
Galen J Van
Lubitz K Von
Kim Jeong
- Kr Seoul
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
US Department of Health and Human Services
National Aeronautics and Space Administration NASA
Original Assignee
US Department of Health and Human Services
National Aeronautics and Space Administration NASA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by US Department of Health and Human Services, National Aeronautics and Space Administration NASA filed Critical US Department of Health and Human Services
Application granted granted Critical
Publication of DE69428536D1 publication Critical patent/DE69428536D1/de
Publication of DE69428536T2 publication Critical patent/DE69428536T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16—Purine radicals

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
DE69428536T 1993-07-13 1994-07-13 A3 -adenosin -rezeptor agonisten Expired - Lifetime DE69428536T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US9110993A 1993-07-13 1993-07-13
US16332493A 1993-12-06 1993-12-06
PCT/US1994/007835 WO1995002604A1 (en) 1993-07-13 1994-07-13 A3 adenosine receptor agonists

Publications (2)

Publication Number Publication Date
DE69428536D1 true DE69428536D1 (de) 2001-11-08
DE69428536T2 DE69428536T2 (de) 2002-06-06

Family

ID=26783598

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69428536T Expired - Lifetime DE69428536T2 (de) 1993-07-13 1994-07-13 A3 -adenosin -rezeptor agonisten

Country Status (6)

Country Link
US (1) US5773423A (de)
EP (1) EP0708781B1 (de)
AT (1) ATE206432T1 (de)
AU (1) AU7331094A (de)
DE (1) DE69428536T2 (de)
WO (1) WO1995002604A1 (de)

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CA2627319A1 (en) 2005-11-30 2007-06-07 Prakash Jagtap Purine derivatives and methods of use thereof
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WO2010014921A2 (en) * 2008-08-01 2010-02-04 The United States Of America, As Represented By The Secretary, Department Of Health And Human Services A3 adenosine receptor antagonists and partial agonists
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WO2009152353A2 (en) 2008-06-11 2009-12-17 Lasergen, Inc. Nucleotides and nucleosides and methods for their use in dna sequencing
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WO2011158904A1 (ja) * 2010-06-18 2011-12-22 株式会社林原生物化学研究所 アデノシンｎ１－オキシドを有効成分として含有する炎症性疾患治療剤
EP2669292B1 (de) * 2011-01-26 2017-03-29 Beijing KBD Pharmaceuticals Co., Ltd. Ribofuranosyl-purin-verbindungen zur behandlung von erkrankungen im zusammenhang mit thrombozytenaggregation
CN102617680B (zh) * 2011-02-01 2014-04-02 复旦大学 一种双功能抗血小板聚集药物及其用途
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KR102048274B1 (ko) 2011-09-13 2019-11-25 애질런트 테크놀로지스, 인크. 핵산 시퀀싱을 위하여 5-메톡시, 3'-oh 차단안된, 신속하게 광절단가능한 종료 뉴클레오티드 및 핵산 시퀀싱 방법
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Also Published As

Publication number Publication date
DE69428536T2 (de) 2002-06-06
ATE206432T1 (de) 2001-10-15
EP0708781B1 (de) 2001-10-04
US5773423A (en) 1998-06-30
WO1995002604A1 (en) 1995-01-26
AU7331094A (en) 1995-02-13
EP0708781A1 (de) 1996-05-01

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