DE69200129D1 - Trisubstituierte Triazine und Pyrimidine, Verfahren zu deren Herstellung und diese enthaltende pharmazeutische Zusammenstellungen. - Google Patents
Trisubstituierte Triazine und Pyrimidine, Verfahren zu deren Herstellung und diese enthaltende pharmazeutische Zusammenstellungen.Info
- Publication number
- DE69200129D1 DE69200129D1 DE69200129T DE69200129T DE69200129D1 DE 69200129 D1 DE69200129 D1 DE 69200129D1 DE 69200129 T DE69200129 T DE 69200129T DE 69200129 T DE69200129 T DE 69200129T DE 69200129 D1 DE69200129 D1 DE 69200129D1
- Authority
- DE
- Germany
- Prior art keywords
- pyrimidines
- processes
- preparation
- pharmaceutical compositions
- compositions containing
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D251/00—Heterocyclic compounds containing 1,3,5-triazine rings
- C07D251/02—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings
- C07D251/12—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D251/26—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with only hetero atoms directly attached to ring carbon atoms
- C07D251/40—Nitrogen atoms
- C07D251/54—Three nitrogen atoms
- C07D251/70—Other substituted melamines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
- C07D407/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9102710A FR2673627B1 (fr) | 1991-03-07 | 1991-03-07 | Triazines et pyrimidines trisubstituees, leur procede de preparation et les compositions pharmaceutiques les contenant. |
Publications (2)
Publication Number | Publication Date |
---|---|
DE69200129D1 true DE69200129D1 (de) | 1994-06-16 |
DE69200129T2 DE69200129T2 (de) | 1994-12-01 |
Family
ID=9410429
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE69200129T Expired - Fee Related DE69200129T2 (de) | 1991-03-07 | 1992-03-06 | Trisubstituierte Triazine und Pyrimidine, Verfahren zu deren Herstellung und diese enthaltende pharmazeutische Zusammenstellungen. |
Country Status (13)
Country | Link |
---|---|
US (1) | US5238936A (de) |
EP (1) | EP0502788B1 (de) |
JP (1) | JPH0776216B2 (de) |
AT (1) | ATE105553T1 (de) |
AU (1) | AU643880B2 (de) |
CA (1) | CA2062378A1 (de) |
DE (1) | DE69200129T2 (de) |
DK (1) | DK0502788T3 (de) |
ES (1) | ES2056692T3 (de) |
FR (1) | FR2673627B1 (de) |
IE (1) | IE66187B1 (de) |
NZ (1) | NZ241867A (de) |
ZA (1) | ZA921702B (de) |
Families Citing this family (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2664594B1 (fr) * | 1990-07-11 | 1992-09-18 | Adir | Polymethylene-imines disubstituees, leur procede de preparation et les compositions pharmaceutiques les contenant. |
AU2599992A (en) * | 1991-11-12 | 1993-06-15 | Pfizer Inc. | Triazine derivatives for enhancing antitumor activity |
US5387685A (en) * | 1993-07-16 | 1995-02-07 | American Cyanamid Co | MDR reversal agents |
EP0916668A4 (de) * | 1996-07-29 | 2000-08-16 | Banyu Pharma Co Ltd | Chemokin-rezeptor-antagonisten |
EP1832655A3 (de) * | 1997-04-30 | 2008-06-18 | McGILL UNIVERSITY | Verfahren zum Erkennen und Rückgängigmachen von Resistenz gegen makrocyclische Laktonverbindungen |
US6403308B1 (en) * | 1997-04-30 | 2002-06-11 | Mcgill University | Methods for detecting and reversing resistance to macrocyclic lactone compounds |
PT1183245E (pt) * | 1999-04-22 | 2007-07-12 | Lundbeck & Co As H | Antagonistas selectivos de npy (y5) |
US6218408B1 (en) | 1999-06-30 | 2001-04-17 | Synaptic Pharmaceutical Corporation | Selective NPY (Y5) antagonists (bicyclics) |
US6989379B1 (en) | 1999-04-22 | 2006-01-24 | H. Lundbick A/S | Selective NPY (Y5) antagonists |
US6340683B1 (en) * | 1999-04-22 | 2002-01-22 | Synaptic Pharmaceutical Corporation | Selective NPY (Y5) antagonists (triazines) |
US6222040B1 (en) | 1999-06-30 | 2001-04-24 | Synaptic Pharmaceutical Corporation | Selective NPY (Y5) antagonists (tricyclics) |
US7273880B2 (en) * | 1999-06-30 | 2007-09-25 | H. Lunbeck A/S | Selective NPY (Y5) antagonists |
US6225330B1 (en) | 1999-06-30 | 2001-05-01 | Synaptic Pharmaceutical Corporation | Selective NPY (Y5) antagonists (tricyclics) |
US6214853B1 (en) | 1999-06-30 | 2001-04-10 | Synaptic Pharmaceutical Corporation | Selective NPY (Y5) antagonists (bicyclics) |
US6635633B2 (en) | 2000-08-14 | 2003-10-21 | Ortho-Pharmaceutical, Inc. | Substituted pyrazoles |
US6693099B2 (en) | 2000-10-17 | 2004-02-17 | The Procter & Gamble Company | Substituted piperazine compounds optionally containing a quinolyl moiety for treating multidrug resistance |
US6376514B1 (en) | 2000-10-17 | 2002-04-23 | The Procter & Gamble Co. | Substituted six-membered heterocyclic compounds useful for treating multidrug resistance and compositions and methods thereof |
US7223759B2 (en) * | 2003-09-15 | 2007-05-29 | Anadys Pharmaceuticals, Inc. | Antibacterial 3,5-diaminopiperidine-substituted aromatic and heteroaromatic compounds |
JP6557674B2 (ja) * | 2014-03-12 | 2019-08-07 | ザ・トラスティーズ・オブ・コランビア・ユニバーシティー・イン・ザ・シティー・オブ・ニューヨーク | 新規クラスのミュー−オピオイド受容体アゴニスト |
JP6674542B2 (ja) * | 2015-07-30 | 2020-04-01 | 四川知本快車創新科技研究院有限公司Sichuan Knowledge Express Institute For Innovative Technologies Co, Ltd. | 供与体と受容体との間に2つの非共役ブリッジを有する光電変換デバイス用の熱活性化遅延蛍光有機分子 |
US10844027B2 (en) | 2015-09-16 | 2020-11-24 | The Trustees Of Columbia University In The City Of New York | Carboxylic diarylthiazepineamines as mu-opioid receptor agonists |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2524467A1 (fr) * | 1982-03-30 | 1983-10-07 | Adir | Polymethylene-imines disubstituees, leurs procedes de preparation et les compositions pharmaceutiques les renfermant |
FR2525597B1 (fr) * | 1982-04-21 | 1985-06-07 | Adir | Polymethylene diamines n,n'-substituees, leurs procedes de preparation et les compositions pharmaceutiques les renfermant |
FR2544315B1 (fr) * | 1983-04-12 | 1985-07-05 | Adir | Polymethylene imines disubstituees, leurs procedes de preparation, et les compositions pharmaceutiques les renfermant |
CA2004211A1 (en) * | 1988-11-30 | 1990-05-31 | Masataka Syoji | Piperidine derivatives and hyportensives containing the same |
FR2664594B1 (fr) * | 1990-07-11 | 1992-09-18 | Adir | Polymethylene-imines disubstituees, leur procede de preparation et les compositions pharmaceutiques les contenant. |
-
1991
- 1991-03-07 FR FR9102710A patent/FR2673627B1/fr not_active Expired - Fee Related
-
1992
- 1992-03-06 NZ NZ241867A patent/NZ241867A/en unknown
- 1992-03-06 AT AT9292400578T patent/ATE105553T1/de not_active IP Right Cessation
- 1992-03-06 AU AU11468/92A patent/AU643880B2/en not_active Ceased
- 1992-03-06 ES ES92400578T patent/ES2056692T3/es not_active Expired - Lifetime
- 1992-03-06 CA CA002062378A patent/CA2062378A1/fr not_active Abandoned
- 1992-03-06 US US07/847,916 patent/US5238936A/en not_active Expired - Fee Related
- 1992-03-06 DK DK92400578.8T patent/DK0502788T3/da active
- 1992-03-06 EP EP92400578A patent/EP0502788B1/de not_active Expired - Lifetime
- 1992-03-06 DE DE69200129T patent/DE69200129T2/de not_active Expired - Fee Related
- 1992-03-06 ZA ZA921702A patent/ZA921702B/xx unknown
- 1992-03-06 JP JP4098998A patent/JPH0776216B2/ja not_active Expired - Fee Related
- 1992-03-06 IE IE920717A patent/IE66187B1/en not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
JPH05125062A (ja) | 1993-05-21 |
EP0502788B1 (de) | 1994-05-11 |
ATE105553T1 (de) | 1994-05-15 |
ZA921702B (en) | 1992-11-25 |
DE69200129T2 (de) | 1994-12-01 |
IE66187B1 (en) | 1995-12-13 |
JPH0776216B2 (ja) | 1995-08-16 |
CA2062378A1 (fr) | 1992-09-08 |
IE920717A1 (en) | 1992-09-09 |
NZ241867A (en) | 1993-02-25 |
FR2673627A1 (fr) | 1992-09-11 |
AU643880B2 (en) | 1993-11-25 |
FR2673627B1 (fr) | 1993-05-07 |
US5238936A (en) | 1993-08-24 |
DK0502788T3 (da) | 1994-09-12 |
AU1146892A (en) | 1992-09-10 |
ES2056692T3 (es) | 1994-10-01 |
EP0502788A1 (de) | 1992-09-09 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
8364 | No opposition during term of opposition | ||
8339 | Ceased/non-payment of the annual fee |