DE69200129D1 - Trisubstituierte Triazine und Pyrimidine, Verfahren zu deren Herstellung und diese enthaltende pharmazeutische Zusammenstellungen. - Google Patents
Trisubstituierte Triazine und Pyrimidine, Verfahren zu deren Herstellung und diese enthaltende pharmazeutische Zusammenstellungen.Info
- Publication number
- DE69200129D1 DE69200129D1 DE69200129T DE69200129T DE69200129D1 DE 69200129 D1 DE69200129 D1 DE 69200129D1 DE 69200129 T DE69200129 T DE 69200129T DE 69200129 T DE69200129 T DE 69200129T DE 69200129 D1 DE69200129 D1 DE 69200129D1
- Authority
- DE
- Germany
- Prior art keywords
- pyrimidines
- processes
- preparation
- pharmaceutical compositions
- compositions containing
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D251/00—Heterocyclic compounds containing 1,3,5-triazine rings
- C07D251/02—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings
- C07D251/12—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D251/26—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with only hetero atoms directly attached to ring carbon atoms
- C07D251/40—Nitrogen atoms
- C07D251/54—Three nitrogen atoms
- C07D251/70—Other substituted melamines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
- C07D407/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9102710A FR2673627B1 (fr) | 1991-03-07 | 1991-03-07 | Triazines et pyrimidines trisubstituees, leur procede de preparation et les compositions pharmaceutiques les contenant. |
Publications (2)
Publication Number | Publication Date |
---|---|
DE69200129D1 true DE69200129D1 (de) | 1994-06-16 |
DE69200129T2 DE69200129T2 (de) | 1994-12-01 |
Family
ID=9410429
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE69200129T Expired - Fee Related DE69200129T2 (de) | 1991-03-07 | 1992-03-06 | Trisubstituierte Triazine und Pyrimidine, Verfahren zu deren Herstellung und diese enthaltende pharmazeutische Zusammenstellungen. |
Country Status (13)
Country | Link |
---|---|
US (1) | US5238936A (de) |
EP (1) | EP0502788B1 (de) |
JP (1) | JPH0776216B2 (de) |
AT (1) | ATE105553T1 (de) |
AU (1) | AU643880B2 (de) |
CA (1) | CA2062378A1 (de) |
DE (1) | DE69200129T2 (de) |
DK (1) | DK0502788T3 (de) |
ES (1) | ES2056692T3 (de) |
FR (1) | FR2673627B1 (de) |
IE (1) | IE66187B1 (de) |
NZ (1) | NZ241867A (de) |
ZA (1) | ZA921702B (de) |
Families Citing this family (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2664594B1 (fr) * | 1990-07-11 | 1992-09-18 | Adir | Polymethylene-imines disubstituees, leur procede de preparation et les compositions pharmaceutiques les contenant. |
AU2599992A (en) * | 1991-11-12 | 1993-06-15 | Pfizer Inc. | Triazine derivatives for enhancing antitumor activity |
US5387685A (en) * | 1993-07-16 | 1995-02-07 | American Cyanamid Co | MDR reversal agents |
EP0916668A4 (de) * | 1996-07-29 | 2000-08-16 | Banyu Pharma Co Ltd | Chemokin-rezeptor-antagonisten |
EP1832655A3 (de) * | 1997-04-30 | 2008-06-18 | McGILL UNIVERSITY | Verfahren zum Erkennen und Rückgängigmachen von Resistenz gegen makrocyclische Laktonverbindungen |
US6403308B1 (en) | 1997-04-30 | 2002-06-11 | Mcgill University | Methods for detecting and reversing resistance to macrocyclic lactone compounds |
US6218408B1 (en) | 1999-06-30 | 2001-04-17 | Synaptic Pharmaceutical Corporation | Selective NPY (Y5) antagonists (bicyclics) |
US6340683B1 (en) | 1999-04-22 | 2002-01-22 | Synaptic Pharmaceutical Corporation | Selective NPY (Y5) antagonists (triazines) |
ATE361917T1 (de) * | 1999-04-22 | 2007-06-15 | Lundbeck & Co As H | Selektive npy(y5)-antagonisten |
US6989379B1 (en) | 1999-04-22 | 2006-01-24 | H. Lundbick A/S | Selective NPY (Y5) antagonists |
US7273880B2 (en) * | 1999-06-30 | 2007-09-25 | H. Lunbeck A/S | Selective NPY (Y5) antagonists |
US6222040B1 (en) | 1999-06-30 | 2001-04-24 | Synaptic Pharmaceutical Corporation | Selective NPY (Y5) antagonists (tricyclics) |
US6225330B1 (en) | 1999-06-30 | 2001-05-01 | Synaptic Pharmaceutical Corporation | Selective NPY (Y5) antagonists (tricyclics) |
US6214853B1 (en) | 1999-06-30 | 2001-04-10 | Synaptic Pharmaceutical Corporation | Selective NPY (Y5) antagonists (bicyclics) |
NZ524192A (en) | 2000-08-14 | 2005-02-25 | Ortho Mcneil Pharm Inc | Substituted pyrazoles |
US6693099B2 (en) | 2000-10-17 | 2004-02-17 | The Procter & Gamble Company | Substituted piperazine compounds optionally containing a quinolyl moiety for treating multidrug resistance |
US6376514B1 (en) * | 2000-10-17 | 2002-04-23 | The Procter & Gamble Co. | Substituted six-membered heterocyclic compounds useful for treating multidrug resistance and compositions and methods thereof |
US7223759B2 (en) * | 2003-09-15 | 2007-05-29 | Anadys Pharmaceuticals, Inc. | Antibacterial 3,5-diaminopiperidine-substituted aromatic and heteroaromatic compounds |
EP3116509B1 (de) | 2014-03-12 | 2022-06-22 | The Trustees of Columbia University in the City of New York | Neue klasse von mu-opioidrezeptoragonisten |
CN107849443B (zh) * | 2015-07-30 | 2020-04-21 | 四川知本快车创新科技研究院有限公司 | 给体和受体之间具有两个非共轭桥的有效热激活延迟荧光有机分子及其在光电器件中的应用 |
CN108135866A (zh) | 2015-09-16 | 2018-06-08 | 哥伦比亚大学董事会 | 羧基二芳基硫氮杂胺作为μ-阿片受体激动剂 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2524467A1 (fr) * | 1982-03-30 | 1983-10-07 | Adir | Polymethylene-imines disubstituees, leurs procedes de preparation et les compositions pharmaceutiques les renfermant |
FR2525597B1 (fr) * | 1982-04-21 | 1985-06-07 | Adir | Polymethylene diamines n,n'-substituees, leurs procedes de preparation et les compositions pharmaceutiques les renfermant |
FR2544315B1 (fr) * | 1983-04-12 | 1985-07-05 | Adir | Polymethylene imines disubstituees, leurs procedes de preparation, et les compositions pharmaceutiques les renfermant |
CA2004211A1 (en) * | 1988-11-30 | 1990-05-31 | Masataka Syoji | Piperidine derivatives and hyportensives containing the same |
FR2664594B1 (fr) * | 1990-07-11 | 1992-09-18 | Adir | Polymethylene-imines disubstituees, leur procede de preparation et les compositions pharmaceutiques les contenant. |
-
1991
- 1991-03-07 FR FR9102710A patent/FR2673627B1/fr not_active Expired - Fee Related
-
1992
- 1992-03-06 AT AT9292400578T patent/ATE105553T1/de not_active IP Right Cessation
- 1992-03-06 IE IE920717A patent/IE66187B1/en not_active IP Right Cessation
- 1992-03-06 AU AU11468/92A patent/AU643880B2/en not_active Ceased
- 1992-03-06 JP JP4098998A patent/JPH0776216B2/ja not_active Expired - Fee Related
- 1992-03-06 US US07/847,916 patent/US5238936A/en not_active Expired - Fee Related
- 1992-03-06 ZA ZA921702A patent/ZA921702B/xx unknown
- 1992-03-06 ES ES92400578T patent/ES2056692T3/es not_active Expired - Lifetime
- 1992-03-06 DK DK92400578.8T patent/DK0502788T3/da active
- 1992-03-06 EP EP92400578A patent/EP0502788B1/de not_active Expired - Lifetime
- 1992-03-06 DE DE69200129T patent/DE69200129T2/de not_active Expired - Fee Related
- 1992-03-06 CA CA002062378A patent/CA2062378A1/fr not_active Abandoned
- 1992-03-06 NZ NZ241867A patent/NZ241867A/en unknown
Also Published As
Publication number | Publication date |
---|---|
AU643880B2 (en) | 1993-11-25 |
DK0502788T3 (da) | 1994-09-12 |
AU1146892A (en) | 1992-09-10 |
NZ241867A (en) | 1993-02-25 |
EP0502788A1 (de) | 1992-09-09 |
FR2673627B1 (fr) | 1993-05-07 |
DE69200129T2 (de) | 1994-12-01 |
JPH05125062A (ja) | 1993-05-21 |
EP0502788B1 (de) | 1994-05-11 |
CA2062378A1 (fr) | 1992-09-08 |
JPH0776216B2 (ja) | 1995-08-16 |
ATE105553T1 (de) | 1994-05-15 |
ZA921702B (en) | 1992-11-25 |
US5238936A (en) | 1993-08-24 |
ES2056692T3 (es) | 1994-10-01 |
IE920717A1 (en) | 1992-09-09 |
FR2673627A1 (fr) | 1992-09-11 |
IE66187B1 (en) | 1995-12-13 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
8364 | No opposition during term of opposition | ||
8339 | Ceased/non-payment of the annual fee |