DE60204232D1 - Antagonisten für calciumkanäle vom n-typ zur behandlung von schmerzen - Google Patents
Antagonisten für calciumkanäle vom n-typ zur behandlung von schmerzenInfo
- Publication number
- DE60204232D1 DE60204232D1 DE60204232T DE60204232T DE60204232D1 DE 60204232 D1 DE60204232 D1 DE 60204232D1 DE 60204232 T DE60204232 T DE 60204232T DE 60204232 T DE60204232 T DE 60204232T DE 60204232 D1 DE60204232 D1 DE 60204232D1
- Authority
- DE
- Germany
- Prior art keywords
- sup
- treatment
- pain
- antagonists
- type calcium
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4706—4-Aminoquinolines; 8-Aminoquinolines, e.g. chloroquine, primaquine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/38—Nitrogen atoms
- C07D215/42—Nitrogen atoms attached in position 4
- C07D215/44—Nitrogen atoms attached in position 4 with aryl radicals attached to said nitrogen atoms
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Neurosurgery (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Quinoline Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE0102858A SE0102858D0 (sv) | 2001-08-27 | 2001-08-27 | N-type calcium channel antagonists for the treatment of pain |
SE0102858 | 2001-08-27 | ||
PCT/SE2002/001521 WO2003018561A1 (en) | 2001-08-27 | 2002-08-23 | N-type calcium channel antagonists for the treatment of pain |
Publications (2)
Publication Number | Publication Date |
---|---|
DE60204232D1 true DE60204232D1 (de) | 2005-06-23 |
DE60204232T2 DE60204232T2 (de) | 2006-01-26 |
Family
ID=20285150
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE60204232T Expired - Fee Related DE60204232T2 (de) | 2001-08-27 | 2002-08-23 | Antagonisten für calciumkanäle vom n-typ zur behandlung von schmerzen |
Country Status (7)
Country | Link |
---|---|
US (1) | US7153865B2 (de) |
EP (1) | EP1430030B1 (de) |
JP (1) | JP2005508894A (de) |
AT (1) | ATE295837T1 (de) |
DE (1) | DE60204232T2 (de) |
SE (1) | SE0102858D0 (de) |
WO (1) | WO2003018561A1 (de) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2003055866A1 (en) * | 2001-12-21 | 2003-07-10 | Bayer Pharmaceuticals Corporation | Quinazoline and quinoline derivative compounds as inhibitors of prolylpeptidase, inducers of apoptosis and cancer treatment agents |
US7223754B2 (en) | 2003-03-10 | 2007-05-29 | Dynogen Pharmaceuticals, Inc. | Thiazolidinone, oxazolidinone, and imidazolone derivatives for treating lower urinary tract and related disorders |
MXPA05009722A (es) * | 2003-03-10 | 2006-03-09 | Schering Corp | Inhibidores heterociclicos de cinasa: metodos de uso y sintesis. |
US7084116B2 (en) | 2003-03-10 | 2006-08-01 | Dynogen Pharmaceuticals, Inc. | Methods for treating lower urinary tract disorders and the related disorders vulvodynia and vulvar vestibulitis using Cav2.2 subunit calcium channel modulators |
WO2005000285A2 (en) * | 2003-06-13 | 2005-01-06 | Dynogen Pharmaceuticals, Inc. | METHODS OF TREATING NON-INFLAMMATORY GASTROINTESTINAL TRACT DISORDERS USING Cav2.2 SUBUNIT CALCIUM CHANNEL MODULATORS |
US20060128702A1 (en) * | 2004-11-23 | 2006-06-15 | Manojit Pal | Heterocyclic and bicyclic compounds, compositions and methods |
SI1963280T1 (sl) | 2005-12-22 | 2016-02-29 | Newron Pharmaceuticals S.P.A. | 2-feniletilamino derivati kot modulatorji kalcijevih in/ali natrijevih kanalčkov |
EA018195B1 (ru) | 2007-06-15 | 2013-06-28 | Ньюрон Фармасьютикалс С.П.А. | Замещенные 2-[2-(фенил)этиламино]алканамидные производные и применение указанных соединений в качестве модуляторов натриевых и/или кальциевых каналов |
CA2780111A1 (en) | 2009-11-07 | 2011-05-12 | Merck Patent Gmbh | Heteroarylaminoquinolines as tgf-beta receptor kinase inhibitors |
EP2723710B1 (de) | 2011-06-27 | 2016-08-10 | Newron Pharmaceuticals S.p.A. | Fluorierte arylalkylaminocarboxamidderivate |
KR20210007046A (ko) * | 2013-02-01 | 2021-01-19 | 웰스태트 테러퓨틱스 코포레이션 | 항염증, 항진균, 항기생충, 및 항암 활성을 갖는 아민 화합물 |
EP2968360B1 (de) | 2013-03-14 | 2021-01-20 | ConverGene LLC | Chinolinon-derivate zur hemmung von bromdomänenhaltigen proteinen |
ES2918589T3 (es) * | 2015-11-25 | 2022-07-19 | Convergene Llc | Inhibidores de bromodomios BET bicíclicos y usos de los mismos |
JP6965432B2 (ja) * | 2017-08-29 | 2021-11-10 | チュラポーン ファンデーション | キノリンおよびナフチリジンの誘導体および組成物 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1573186A (en) * | 1977-09-14 | 1980-08-20 | Wyeth John & Brother Ltd | 4-aminoquinoline derivatives |
AU4802500A (en) * | 1999-04-26 | 2000-11-10 | Neurogen Corporation | 2-aminoquinolinecarboxamides: neurokinin receptor ligands |
-
2001
- 2001-08-27 SE SE0102858A patent/SE0102858D0/xx unknown
-
2002
- 2002-08-23 DE DE60204232T patent/DE60204232T2/de not_active Expired - Fee Related
- 2002-08-23 WO PCT/SE2002/001521 patent/WO2003018561A1/en active IP Right Grant
- 2002-08-23 JP JP2003523224A patent/JP2005508894A/ja active Pending
- 2002-08-23 EP EP02760975A patent/EP1430030B1/de not_active Expired - Lifetime
- 2002-08-23 AT AT02760975T patent/ATE295837T1/de not_active IP Right Cessation
- 2002-08-23 US US10/488,025 patent/US7153865B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
SE0102858D0 (sv) | 2001-08-27 |
US7153865B2 (en) | 2006-12-26 |
DE60204232T2 (de) | 2006-01-26 |
EP1430030A1 (de) | 2004-06-23 |
JP2005508894A (ja) | 2005-04-07 |
US20050131020A1 (en) | 2005-06-16 |
EP1430030B1 (de) | 2005-05-18 |
WO2003018561A1 (en) | 2003-03-06 |
ATE295837T1 (de) | 2005-06-15 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
8364 | No opposition during term of opposition | ||
8339 | Ceased/non-payment of the annual fee |