DE602006014530D1 - Pharmazeutisch aktive diazepane - Google Patents

Pharmazeutisch aktive diazepane

Info

Publication number
DE602006014530D1
DE602006014530D1 DE602006014530T DE602006014530T DE602006014530D1 DE 602006014530 D1 DE602006014530 D1 DE 602006014530D1 DE 602006014530 T DE602006014530 T DE 602006014530T DE 602006014530 T DE602006014530 T DE 602006014530T DE 602006014530 D1 DE602006014530 D1 DE 602006014530D1
Authority
DE
Germany
Prior art keywords
diazepane
pharmaceutical active
lfa
activity
diazepam
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE602006014530T
Other languages
English (en)
Inventor
Berndt Oberhauser
Dieter Scholz
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Novartis AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis AG filed Critical Novartis AG
Publication of DE602006014530D1 publication Critical patent/DE602006014530D1/de
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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    • C—CHEMISTRY; METALLURGY
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    • C07D—HETEROCYCLIC COMPOUNDS
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
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    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Rheumatology (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Oncology (AREA)
  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Dermatology (AREA)
  • Communicable Diseases (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Psychology (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Transplantation (AREA)
  • Psychiatry (AREA)
  • Emergency Medicine (AREA)
  • Obesity (AREA)
DE602006014530T 2005-04-19 2006-04-19 Pharmazeutisch aktive diazepane Expired - Fee Related DE602006014530D1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0507918.1A GB0507918D0 (en) 2005-04-19 2005-04-19 Organic compounds
PCT/EP2006/003583 WO2006111371A1 (en) 2005-04-19 2006-04-19 Pharmaceutically active diazepanes

Publications (1)

Publication Number Publication Date
DE602006014530D1 true DE602006014530D1 (de) 2010-07-08

Family

ID=34630941

Family Applications (1)

Application Number Title Priority Date Filing Date
DE602006014530T Expired - Fee Related DE602006014530D1 (de) 2005-04-19 2006-04-19 Pharmazeutisch aktive diazepane

Country Status (17)

Country Link
US (1) US20080300237A1 (de)
EP (2) EP2206704A1 (de)
JP (1) JP2008538357A (de)
KR (2) KR20100017724A (de)
CN (1) CN101163685A (de)
AT (1) ATE469134T1 (de)
AU (1) AU2006237177A1 (de)
BR (1) BRPI0610856A2 (de)
CA (1) CA2600774A1 (de)
DE (1) DE602006014530D1 (de)
ES (1) ES2345628T3 (de)
GB (1) GB0507918D0 (de)
MX (1) MX2007013007A (de)
PL (1) PL1874739T3 (de)
PT (1) PT1874739E (de)
RU (1) RU2007142498A (de)
WO (1) WO2006111371A1 (de)

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JP2018524299A (ja) 2015-06-12 2018-08-30 マッカイ メディカル ファンデーション ザ プレスビュテロス チャーチ イン タイワン マッカイ メモリアル ホスピタル 免疫応答を調節するための方法およびポリペプチド
US20180193003A1 (en) 2016-12-07 2018-07-12 Progenity Inc. Gastrointestinal tract detection methods, devices and systems
KR20190095936A (ko) 2016-12-14 2019-08-16 프로제너티, 인크. 인테그린 저해제로의 위장관 질환의 치료
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JP2008538357A (ja) 2008-10-23
EP1874739B1 (de) 2010-05-26
CN101163685A (zh) 2008-04-16
ATE469134T1 (de) 2010-06-15
MX2007013007A (es) 2008-01-11
GB0507918D0 (en) 2005-05-25
CA2600774A1 (en) 2006-10-26
KR20070121768A (ko) 2007-12-27
EP1874739A1 (de) 2008-01-09
BRPI0610856A2 (pt) 2010-08-03
WO2006111371A1 (en) 2006-10-26
KR20100017724A (ko) 2010-02-16
RU2007142498A (ru) 2009-05-27
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EP2206704A1 (de) 2010-07-14
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