DE602005021256D1 - Verfahren zur herstellung eines 11-(4-substituierten 1-piperazinyl)dibenzoäb,füä1,4üthiazepinderivats - Google Patents

Verfahren zur herstellung eines 11-(4-substituierten 1-piperazinyl)dibenzoäb,füä1,4üthiazepinderivats

Info

Publication number
DE602005021256D1
DE602005021256D1 DE602005021256T DE602005021256T DE602005021256D1 DE 602005021256 D1 DE602005021256 D1 DE 602005021256D1 DE 602005021256 T DE602005021256 T DE 602005021256T DE 602005021256 T DE602005021256 T DE 602005021256T DE 602005021256 D1 DE602005021256 D1 DE 602005021256D1
Authority
DE
Germany
Prior art keywords
piperazinyl
preparing
derivative
fueledietiazepine
dibenzoea
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
DE602005021256T
Other languages
English (en)
Inventor
Alexander Christian Comely
Espaulella Francesc Xavier Verdaguer
Jane Llorenc Rafecas
Coto Antonio Domingo
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Union Quimico Farmaceutica SA
Original Assignee
Union Quimico Farmaceutica SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Union Quimico Farmaceutica SA filed Critical Union Quimico Farmaceutica SA
Publication of DE602005021256D1 publication Critical patent/DE602005021256D1/de
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02—Seven-membered rings
    • C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/12—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with two six-membered rings
    • C07D281/16—[b, f]-condensed

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
DE602005021256T 2005-03-07 2005-12-21 Verfahren zur herstellung eines 11-(4-substituierten 1-piperazinyl)dibenzoäb,füä1,4üthiazepinderivats Active DE602005021256D1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ES200500513A ES2234447B1 (es) 2005-03-07 2005-03-07 Procedimiento para la obtencion de un derivado de 11-(4-sustituido-1-piperazinil)dibenzo(b,f)(1,4)tiazepina.
PCT/EP2005/014055 WO2006094549A1 (en) 2005-03-07 2005-12-21 A PROCESS FOR THE PREPARATION OF AN 11-(4-SUBSTITUTED-I-PIPERAZINYL)DIBENZO[b,f][1,4]THIAZEPINE DERIVATIVE

Publications (1)

Publication Number Publication Date
DE602005021256D1 true DE602005021256D1 (de) 2010-06-24

Family

ID=34707636

Family Applications (1)

Application Number Title Priority Date Filing Date
DE602005021256T Active DE602005021256D1 (de) 2005-03-07 2005-12-21 Verfahren zur herstellung eines 11-(4-substituierten 1-piperazinyl)dibenzoäb,füä1,4üthiazepinderivats

Country Status (9)

Country Link
US (1) US7902355B2 (de)
EP (1) EP1856073B1 (de)
AT (1) ATE467624T1 (de)
DE (1) DE602005021256D1 (de)
DK (1) DK1856073T3 (de)
ES (1) ES2234447B1 (de)
NO (1) NO20075071L (de)
PT (1) PT1856073E (de)
WO (1) WO2006094549A1 (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2006113425A1 (en) 2005-04-14 2006-10-26 Teva Pharmaceutical Industries Ltd. Process for preparing quetiapine fumarate
CZ300451B6 (cs) * 2006-07-03 2009-05-20 Farmak, A. S. Zpusob prípravy solí 2-[2-(4-dibenzo[b,f][1,4]thiazepin-11-yl-1-piperazinyl)ethoxy]ethanolu (quetiapinu) a jejich cištení
CN101925587B (zh) * 2008-01-31 2013-05-01 费米有限公司 喹硫平的制备方法
US20120071649A1 (en) 2009-03-04 2012-03-22 Ranbaxy Laboratories Limited Process for the preparation of quetiapine fumarate
CN101891707B (zh) * 2010-07-29 2012-10-17 浙江海正药业股份有限公司 喹硫平或其可药用盐的制备方法
CN103664822B (zh) * 2012-09-18 2015-07-15 四川大学华西医院 一种可用作麻醉剂的化合物
CN104803947A (zh) * 2015-03-12 2015-07-29 常州康丽制药有限公司 11-(1-哌嗪基)二苯并[b,f][1,4]硫氮杂*富马酸盐的制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8607684D0 (en) * 1986-03-27 1986-04-30 Ici America Inc Thiazepine compounds
GB8705574D0 (en) * 1987-03-10 1987-04-15 Ici Plc Preparation of thiazepine compound
GB9716161D0 (en) * 1997-08-01 1997-10-08 Zeneca Ltd Process
HU227039B1 (en) * 2000-01-25 2010-05-28 Egis Gyogyszergyar Nyilvanosan New process for the production of quetiapine and intermediates therefor
US7071331B2 (en) * 2003-02-22 2006-07-04 Teva Pharmaceutical Industries Ltd. Synthesis of quetiapine and pharmaceutically acceptable salts thereof

Also Published As

Publication number Publication date
EP1856073B1 (de) 2010-05-12
ATE467624T1 (de) 2010-05-15
US20080171869A1 (en) 2008-07-17
ES2234447B1 (es) 2006-03-01
WO2006094549A1 (en) 2006-09-14
ES2234447A1 (es) 2005-06-16
NO20075071L (no) 2007-11-28
DK1856073T3 (da) 2010-08-23
EP1856073A1 (de) 2007-11-21
US7902355B2 (en) 2011-03-08
PT1856073E (pt) 2010-07-06

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