DE602004023971D1 - Pyrroloä2,3-büpyridinderivate, die als kinaseinhibitoren wirken; verfahren zu deren herstellung und pharmazeutische zusammensetzung, die diese enthält - Google Patents

Pyrroloä2,3-büpyridinderivate, die als kinaseinhibitoren wirken; verfahren zu deren herstellung und pharmazeutische zusammensetzung, die diese enthält

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Publication number
DE602004023971D1
DE602004023971D1 DE602004023971T DE602004023971T DE602004023971D1 DE 602004023971 D1 DE602004023971 D1 DE 602004023971D1 DE 602004023971 T DE602004023971 T DE 602004023971T DE 602004023971 T DE602004023971 T DE 602004023971T DE 602004023971 D1 DE602004023971 D1 DE 602004023971D1
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Germany
Prior art keywords
compounds
preparation
pyrroloa2
büpyridine
kinaseinhibitors
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Active
Application number
DE602004023971T
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English (en)
Inventor
Barbara Salom
Anello Matteo D
Maria Gabriella Brasca
Patrizia Giordano
Katia Martina
Frederick Arthur Brookfield
William John Trigg
Edward Andrew Boyd
Jonathan Anthony Larard
Dania Tesei
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Pfizer Italia SRL
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Pfizer Italia SRL
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Publication of DE602004023971D1 publication Critical patent/DE602004023971D1/de
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
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    • A61P35/00—Antineoplastic agents
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
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DE602004023971T 2003-12-24 2004-12-23 Pyrroloä2,3-büpyridinderivate, die als kinaseinhibitoren wirken; verfahren zu deren herstellung und pharmazeutische zusammensetzung, die diese enthält Active DE602004023971D1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0330042.3A GB0330042D0 (en) 2003-12-24 2003-12-24 Pyrrolo [2,3-b] pyridine derivatives active as kinase inhibitors process for their preparation and pharmaceutical compositions them
PCT/EP2004/014676 WO2005063747A1 (en) 2003-12-24 2004-12-23 PYRROLO[2,3-b] PYRIDINE DERIVATIVES ACTIVE AS KINASE INHIBITORS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITION COMPRISING THEM

Publications (1)

Publication Number Publication Date
DE602004023971D1 true DE602004023971D1 (de) 2009-12-17

Family

ID=30776534

Family Applications (1)

Application Number Title Priority Date Filing Date
DE602004023971T Active DE602004023971D1 (de) 2003-12-24 2004-12-23 Pyrroloä2,3-büpyridinderivate, die als kinaseinhibitoren wirken; verfahren zu deren herstellung und pharmazeutische zusammensetzung, die diese enthält

Country Status (10)

Country Link
US (2) US7888508B2 (de)
EP (1) EP1704147B1 (de)
JP (2) JP5053643B2 (de)
AT (1) ATE447571T1 (de)
BR (1) BRPI0418179A (de)
CA (1) CA2550686C (de)
DE (1) DE602004023971D1 (de)
ES (1) ES2333437T3 (de)
GB (1) GB0330042D0 (de)
WO (1) WO2005063747A1 (de)

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CA2550686C (en) 2015-09-15
CA2550686A1 (en) 2005-07-14
ES2333437T3 (es) 2010-02-22
US20050209269A1 (en) 2005-09-22
BRPI0418179A (pt) 2007-04-27
WO2005063747A1 (en) 2005-07-14
JP5053643B2 (ja) 2012-10-17
GB0330042D0 (en) 2004-01-28
JP2012121892A (ja) 2012-06-28
EP1704147B1 (de) 2009-11-04
ATE447571T1 (de) 2009-11-15
EP1704147A1 (de) 2006-09-27
US8198298B2 (en) 2012-06-12
US7888508B2 (en) 2011-02-15
JP2007516997A (ja) 2007-06-28
US20110136857A1 (en) 2011-06-09

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