DE60115419D1 - Assymetrische synthese von piperazinsäure und ihre derivate - Google Patents
Assymetrische synthese von piperazinsäure und ihre derivateInfo
- Publication number
- DE60115419D1 DE60115419D1 DE60115419T DE60115419T DE60115419D1 DE 60115419 D1 DE60115419 D1 DE 60115419D1 DE 60115419 T DE60115419 T DE 60115419T DE 60115419 T DE60115419 T DE 60115419T DE 60115419 D1 DE60115419 D1 DE 60115419D1
- Authority
- DE
- Germany
- Prior art keywords
- piperazic acid
- derivatives
- piperazic
- acid
- useful
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
- C07D237/04—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having less than three double bonds between ring members or between ring members and non-ring members
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US20210400P | 2000-05-04 | 2000-05-04 | |
US202104P | 2000-05-04 | ||
PCT/US2001/013330 WO2001083458A2 (en) | 2000-05-04 | 2001-04-25 | Asymmetric synthesis of piperazic acid and derivatives thereof |
Publications (2)
Publication Number | Publication Date |
---|---|
DE60115419D1 true DE60115419D1 (de) | 2006-01-05 |
DE60115419T2 DE60115419T2 (de) | 2006-08-17 |
Family
ID=22748510
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE60115419T Expired - Lifetime DE60115419T2 (de) | 2000-05-04 | 2001-04-25 | Assymetrische synthese von piperazinsäure und ihre derivate |
Country Status (11)
Country | Link |
---|---|
US (1) | US6632942B2 (de) |
EP (1) | EP1280780B1 (de) |
AT (1) | ATE311370T1 (de) |
AU (2) | AU5725301A (de) |
CA (1) | CA2403304A1 (de) |
DE (1) | DE60115419T2 (de) |
ES (1) | ES2252224T3 (de) |
NZ (1) | NZ520998A (de) |
RU (1) | RU2002135314A (de) |
WO (1) | WO2001083458A2 (de) |
ZA (1) | ZA200206997B (de) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2853901B1 (fr) * | 2003-04-16 | 2005-06-17 | Isochem Sa | Procede de preparation de derives de l'acide hexahydropyridazine-3-carboxylique |
WO2005028449A1 (en) * | 2003-06-26 | 2005-03-31 | Honeywell Specialty Chemicals Seelze Gmbh | Improved process for the manufacture of 1,2-disubstituted hexahydropyridazine-3-carboxylic acids and esters thereof |
NZ588448A (en) * | 2004-05-15 | 2012-01-12 | Vertex Pharma | Treating seizures using interleukin-1beta converting enzyme (ICE) inhibitors |
US7531570B2 (en) * | 2004-05-27 | 2009-05-12 | Vertex Pharmaceuticals Incorporated | Treatment of diseases using ICE inhibitors |
CN102250014B (zh) * | 2010-05-18 | 2013-11-13 | 上海奥博生物医药技术有限公司 | 一种制备手性1-苄氧羰基六氢哒嗪-3-羧酸和手性1,2-二苄氧羰基六氢哒嗪-3-羧酸的方法 |
CN110343728B (zh) * | 2019-06-04 | 2021-10-08 | 浙江大学 | 一种生物转化合成六氢哒嗪-3-羧酸的方法 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4692438A (en) * | 1984-08-24 | 1987-09-08 | Hoffmann-La Roche Inc. | Pyridazo-diazepines, diazocines, and -triazepines having anti-hypertensive activity |
ATE203242T1 (de) * | 1992-05-18 | 2001-08-15 | Hoffmann La Roche | Asymmetrische hydrierung |
-
2001
- 2001-04-25 NZ NZ520998A patent/NZ520998A/en active Application Filing
- 2001-04-25 WO PCT/US2001/013330 patent/WO2001083458A2/en active IP Right Grant
- 2001-04-25 AU AU5725301A patent/AU5725301A/xx active Pending
- 2001-04-25 DE DE60115419T patent/DE60115419T2/de not_active Expired - Lifetime
- 2001-04-25 RU RU2002135314/04A patent/RU2002135314A/ru not_active Application Discontinuation
- 2001-04-25 ES ES01930747T patent/ES2252224T3/es not_active Expired - Lifetime
- 2001-04-25 AU AU2001257253A patent/AU2001257253B2/en not_active Ceased
- 2001-04-25 AT AT01930747T patent/ATE311370T1/de not_active IP Right Cessation
- 2001-04-25 EP EP01930747A patent/EP1280780B1/de not_active Expired - Lifetime
- 2001-04-25 CA CA002403304A patent/CA2403304A1/en not_active Abandoned
-
2002
- 2002-06-14 US US10/168,463 patent/US6632942B2/en not_active Expired - Fee Related
- 2002-08-30 ZA ZA200206997A patent/ZA200206997B/en unknown
Also Published As
Publication number | Publication date |
---|---|
NZ520998A (en) | 2004-11-26 |
US20030176691A1 (en) | 2003-09-18 |
AU5725301A (en) | 2001-11-12 |
US6632942B2 (en) | 2003-10-14 |
EP1280780A2 (de) | 2003-02-05 |
WO2001083458A3 (en) | 2002-05-23 |
WO2001083458A2 (en) | 2001-11-08 |
ATE311370T1 (de) | 2005-12-15 |
ES2252224T3 (es) | 2006-05-16 |
DE60115419T2 (de) | 2006-08-17 |
EP1280780B1 (de) | 2005-11-30 |
CA2403304A1 (en) | 2001-11-08 |
RU2002135314A (ru) | 2004-05-27 |
ZA200206997B (en) | 2003-11-12 |
AU2001257253B2 (en) | 2006-03-02 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
8364 | No opposition during term of opposition |