DE60106281T2 - Verfahren zur Behandlung eines Östrogenrezeptor-positiven Karzinoms - Google Patents
Verfahren zur Behandlung eines Östrogenrezeptor-positiven Karzinoms Download PDFInfo
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- DE60106281T2 DE60106281T2 DE60106281T DE60106281T DE60106281T2 DE 60106281 T2 DE60106281 T2 DE 60106281T2 DE 60106281 T DE60106281 T DE 60106281T DE 60106281 T DE60106281 T DE 60106281T DE 60106281 T2 DE60106281 T2 DE 60106281T2
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- Prior art keywords
- rapamycin
- carbon atoms
- antiestrogen
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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| PCT/US2001/024615 WO2002013802A2 (en) | 2000-08-11 | 2001-08-06 | Method of treating estrogen receptor positive carcinoma |
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| US20030215445A1 (en) | 1997-05-23 | 2003-11-20 | Ginette Serrero | Methods and compositions for inhibiting the growth of hematopoietic malignant cells |
| US8512960B2 (en) * | 1997-05-23 | 2013-08-20 | A&G Pharmaceutical, Inc. | 88kDa tumorigenic growth factor and antagonists |
| US7091047B2 (en) * | 1997-05-23 | 2006-08-15 | A&G Pharmaceutical, Inc. | Methods and kits for diagnosing tumorigenicity |
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| US6309826B1 (en) * | 1997-05-23 | 2001-10-30 | Ginette Serrero | 88kDa tumorigenic growth factor and antagonists |
| US7617145B1 (en) * | 2000-10-24 | 2009-11-10 | Worldwide Farm Equipment Auctions.Com Ltd. | Adaptive bidding increments in an online auction system |
| TWI286074B (en) | 2000-11-15 | 2007-09-01 | Wyeth Corp | Pharmaceutical composition containing CCI-779 as an antineoplastic agent |
| AU2016206379B2 (en) * | 2001-02-19 | 2017-09-14 | Novartis Ag | Cancer Treatment |
| CA2438504C (en) * | 2001-02-19 | 2016-02-16 | Novartis Ag | Treatment of solid tumours with rapamycin derivatives |
| AU2011226833B9 (en) * | 2001-02-19 | 2014-07-03 | Novartis Ag | Cancer treatment |
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| KR100851648B1 (ko) * | 2001-07-09 | 2008-08-13 | 레프로스 쎄라피우틱스 아이엔씨. | 남성의 테스토스테론 결핍치료용 물질 |
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| CN100522967C (zh) | 2002-02-01 | 2009-08-05 | 阿里亚德基因治疗公司 | 含磷化合物及其应用 |
| EP1504010B1 (en) * | 2002-05-15 | 2009-03-25 | Endocyte, Inc. | Vitamin-mitomycin conjugates |
| US7411045B2 (en) * | 2002-11-19 | 2008-08-12 | A&G Pharmaceutical, Inc. | Autocrine growth factor receptor antibodies and methods |
| CA2512867C (en) | 2003-01-27 | 2014-08-26 | Endocyte, Inc. | Vitamin receptor binding drug delivery conjugates |
| ATE483724T1 (de) * | 2003-02-26 | 2010-10-15 | A & G Pharmaceuticals Inc | Verfahren zur erhöhung der ausbreitung von b- zellen |
| UA83484C2 (uk) * | 2003-03-05 | 2008-07-25 | Уайт | Спосіб лікування раку грудей комбінацією похідного рапаміцину і інгібітора ароматази - летрозолу, фармацевтична композиція |
| CN1777424A (zh) * | 2003-04-22 | 2006-05-24 | 惠氏公司 | 抗肿瘤联合药物 |
| EP1644038A2 (en) * | 2003-06-23 | 2006-04-12 | A & G Pharmaceuticals, Inc. | Compositions and methods for restoring sensitivity of tumor cells to antitumor therapy and inducing apoptosis |
| CA2532251A1 (en) * | 2003-07-25 | 2005-02-10 | Wyeth | Cci-779 lyophilized formulations |
| JP2007517763A (ja) * | 2003-08-01 | 2007-07-05 | エイアンドジー ファーマスーティカル インコーポレイテッド | Ｈｅｒ２アンタゴニストを用いた治療への感受性を回復させる組成物および方法 |
| US7781478B2 (en) | 2004-07-14 | 2010-08-24 | Ptc Therapeutics, Inc. | Methods for treating hepatitis C |
| WO2006012527A1 (en) | 2004-07-23 | 2006-02-02 | Endocyte, Inc. | Bivalent linkers and conjugates thereof |
| EP1804779A1 (en) * | 2004-10-28 | 2007-07-11 | Wyeth | Use of an mtor inhibitor in treatment of uterine leiomyoma |
| WO2006084058A2 (en) | 2005-02-03 | 2006-08-10 | The General Hospital Corporation | Method for treating gefitinib resistant cancer |
| MX2007010892A (es) | 2005-03-07 | 2007-12-05 | Wyeth Corp | Isomero de oxepano de 42-o-(2-hidroxi)etil-rapamicina. |
| EP1863816B1 (en) * | 2005-03-16 | 2014-06-25 | Endocyte, Inc. | Synthesis and purification of pteroic acid and conjugates thereof |
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-
2001
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- 2001-08-06 DE DE60106281T patent/DE60106281T2/de not_active Expired - Fee Related
- 2001-08-06 MX MXPA03001245A patent/MXPA03001245A/es active IP Right Grant
- 2001-08-06 EP EP01961914A patent/EP1318837B1/en not_active Expired - Lifetime
- 2001-08-06 AT AT01961914T patent/ATE278421T1/de not_active IP Right Cessation
- 2001-08-06 PT PT01961914T patent/PT1318837E/pt unknown
- 2001-08-06 JP JP2002518948A patent/JP2004507465A/ja not_active Withdrawn
- 2001-08-06 CN CNB018137539A patent/CN100448487C/zh not_active Expired - Fee Related
- 2001-08-06 WO PCT/US2001/024615 patent/WO2002013802A2/en not_active Ceased
- 2001-08-06 CA CA002416976A patent/CA2416976C/en not_active Expired - Fee Related
- 2001-08-06 AU AU2001283139A patent/AU2001283139A1/en not_active Abandoned
- 2001-08-06 DK DK01961914T patent/DK1318837T3/da active
- 2001-08-06 US US09/923,217 patent/US6511986B2/en not_active Expired - Fee Related
- 2001-08-10 AR ARP010103839A patent/AR033555A1/es unknown
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| ES2228932T3 (es) | 2005-04-16 |
| EP1318837B1 (en) | 2004-10-06 |
| WO2002013802A2 (en) | 2002-02-21 |
| HK1056687A1 (en) | 2004-02-27 |
| US20020045638A1 (en) | 2002-04-18 |
| WO2002013802A3 (en) | 2003-03-27 |
| US6511986B2 (en) | 2003-01-28 |
| MXPA03001245A (es) | 2003-05-27 |
| DK1318837T3 (da) | 2005-01-10 |
| AR033555A1 (es) | 2003-12-26 |
| CA2416976A1 (en) | 2002-02-21 |
| DE60106281D1 (de) | 2004-11-11 |
| ATE278421T1 (de) | 2004-10-15 |
| CN1446106A (zh) | 2003-10-01 |
| CA2416976C (en) | 2008-05-20 |
| CN100448487C (zh) | 2009-01-07 |
| PT1318837E (pt) | 2004-12-31 |
| EP1318837A2 (en) | 2003-06-18 |
| AU2001283139A1 (en) | 2002-02-25 |
| JP2004507465A (ja) | 2004-03-11 |
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