DE4131038A1 - Substituierte 3-phenylurazile - Google Patents

Substituierte 3-phenylurazile

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Publication number
DE4131038A1
DE4131038A1 DE4131038A DE4131038A DE4131038A1 DE 4131038 A1 DE4131038 A1 DE 4131038A1 DE 4131038 A DE4131038 A DE 4131038A DE 4131038 A DE4131038 A DE 4131038A DE 4131038 A1 DE4131038 A1 DE 4131038A1
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Germany
Prior art keywords
alkyl
alkoxy
group
cyano
alkenyl
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DE4131038A
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English (en)
Inventor
Ralf Dr Klintz
Peter Dr Schaefer
Gerhard Dr Hamprecht
Elisabeth Dr Heistracher
Hans-Josef Dr Wolf
Karl-Otto Dr Westphalen
Matthias Dr Gerber
Uwe Dr Kardorff
Helmut Dr Walter
Klaus Dr Grossmann
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BASF SE
Original Assignee
BASF SE
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=6440891&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DE4131038(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by BASF SE filed Critical BASF SE
Priority to DE4131038A priority Critical patent/DE4131038A1/de
Priority to KR1019940700895A priority patent/KR100260011B1/ko
Priority to JP50574593A priority patent/JP3253299B2/ja
Priority to PCT/EP1992/002088 priority patent/WO1993006090A1/de
Priority to BR9206518A priority patent/BR9206518A/pt
Priority to HU9400801A priority patent/HUT70880A/hu
Priority to US08/774,722 priority patent/US6239074B1/en
Priority to EP92919190A priority patent/EP0604491A1/de
Priority to CA002119036A priority patent/CA2119036A1/en
Priority to TW081107305A priority patent/TW225981B/zh
Priority to ZA927153A priority patent/ZA927153B/xx
Priority to MX9205306A priority patent/MX9205306A/es
Publication of DE4131038A1 publication Critical patent/DE4131038A1/de
Priority to US09/733,554 priority patent/US20010031865A1/en
Withdrawn legal-status Critical Current

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    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
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    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/541,3-Diazines; Hydrogenated 1,3-diazines
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    • C07C275/32Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms
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    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C275/00Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C275/28Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C275/38Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by doubly-bound oxygen atoms
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    • C07D405/04Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

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Description

Die vorliegende Erfindung betrifft neue substituierte 3-Phenyl­ urazile der allgemeinen Formel I
in der die Variablen folgende Bedeutung haben:
X¹, X² Sauerstoff oder Schwefel;
W eine Gruppe -C(R⁸)=X⁵, -C(R⁸)(X³R⁶)(X⁴R⁷), -C(R⁸)=C(R⁹)-CO-R¹⁰, -CH(R⁸)-CH(R⁹)-CO-R¹⁰,
-C(R⁸)=C(R⁹)-CH₂-CO-R¹⁰, -C(R⁸)=C(R⁹)-C(R¹¹)=C(R¹²)-CO-R¹⁰ oder
-C(R⁸)=C(R⁹)-CH₂-CH(R¹³)-CO-R¹⁰ mit
X³, X⁴ Sauerstoff oder Schwefel;
X⁵ Sauerstoff, Schwefel oder ein Rest -NR¹⁴, mit
R¹⁴ Wasserstoff, Hydroxyl, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, C₃-C₇-Cycloalkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alk­ oxy-C₁-C₆-alkyl, C₁-C₆-Alkoxy, C₃-C₆-Alkenyloxy, C₃-C₆-Alkinyloxy, C₅-C₇-Cycloalkoxy, C₅-C₇-Cyclo­ alkenyloxy, partiell oder vollständig halogenier­ tem C₁-C₆-Alkoxy, partiell oder vollständig halo­ geniertem C₃-C₆-Alkenyloxy, Hydroxy-C₁-C₆-alkoxy, Cyano-C₁-C₆-alkoxy, C₃-C₇-Cycloalkyl-C₁-C₆-alkoxy, C₁-C₆-Alkoxy-C₁-C₆-alkoxy, C₁-C₆-Alkoxy-C₃-C₆- alkenyloxy, C₁-C₆-Alkylcarbonyloxy, C₁-C₆-Alkoxy­ carbonyl-C₂-C₆-alkoxy, C₁-C₆-Alkylthio-C₁-C₆- alkoxy, Di-(C₁-C₆-alkyl)-amino-C₁-C₆-alkoxy, Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxy­ carbonyl, Phenyl-C₁-C₆-alkoxy, Phenyl-C₃-C₆- alkenyloxy oder Phenyl-C₃-C₆-alkinyloxy, wobei jeweils eine oder zwei Methylengruppen der Kohlen­ stoffketten durch -O-, -S- oder -N(C₁-C₆-Alkyl)- ersetzt sein können und wobei der Phenylring jeweils auch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆- Alkyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl, oder -N(R¹⁵)R¹⁶, wobei
R¹⁵, R¹⁶ Wasserstoff, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆- Alkinyl, C₃-C₆-Cycloalkyl, partiell oder voll­ ständig halogeniertes C₁-C₆-Alkyl, C₁-C₆-Alkoxy- C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxy­ carbonyl oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆- Alkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl, oder
R¹⁵ und R¹⁶ zusammen mit dem gemeinsamen Stick­ stoffatom einen gesättigten oder ungesättigten 4-7-gliedrigen Heterocyclus, wobei ein Ringglied durch -O-, -S-, -N=, -NH- oder -N(C₁-C₆-Alkyl)- ersetzt sein kann,
bedeuten;
R⁶, R⁷ C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alk­ oxy-C₁-C₆-alkyl oder
R⁶ und R⁷ zusammen eine gesättigte oder ungesättigte, zwei- bis viergliedrige Kohlenstoffkette, die einen Oxo-Substituenten tragen kann, wobei ein Glied dieser Kette durch ein den Variablen X³ und X⁴ nicht benach­ bartes Sauerstoff-, Schwefel- oder Stickstoffatom er­ setzt sein kann, und wobei die Kohlenstoffkette noch ein bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Amino, Halogen, C₁-C₆-Alkyl, C₂-C₆-Alkenyl, C₁-C₆-Alkoxy, C₃-C₆-Alk­ enyloxy, C₃-C₆-Alkinyloxy, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, Cyano-C₁-C₆-alkyl, Hydroxy-C₁-C₆-alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₃-C₆- Alkenyloxy-C₁-C₆-alkyl, C₃-C₆-Alkinyloxy-C₁-C₆-alkyl, Carboxy, C₁-C₆-Alkoxycarbonyl und C₁-C₆-Alkyl-carbonyl­ oxy-C₁-C₆-alkyl;
R⁸ Wasserstoff, Cyano, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆- Alkinyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₃-C₇-Cycloalkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl oder C₁-C₆-Alkoxycarbonyl;
R⁹, R¹² Wasserstoff, Cyano, Halogen C₁-C₆-Alkyl, C₁-C₆-Alkoxy Halogen-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl oder C₁-C₆- Alkoxycarbonyl;
R¹⁰ Wasserstoff, O-R¹⁷, S-R¹⁷, C₁-C₆-Alkyl, das noch einen oder zwei C₁-C₆-Alkoxysubstituenten tragen kann, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, partiell oder vollständig halo­ geniertes C₁-C₆-Alkyl, C₃-C₇-Cycloalkyl, C₁-C₆-Alkyl­ thio-C₁-C₆-alkyl, -N(R¹⁵)R¹⁶ oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy oder C₁-C₆- Alkoxycarbonyl,
R¹⁷ bedeutet Wasserstoff, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, C₃-C₇-Cycloalkyl, partiell oder vollständig halogeniertes C₂-C₆-Alkyl, partiell oder vollständig halogeniertes C₃-C₆-Alkenyl, Cyano-C₁-C₆-alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl oder C₁-C₆-Alkyl-oximino-C₁-C₆-alkyl, C₁-C₆-Alkyl­ carbonyl, C₁-C₆-Alkoxycarbonyl oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen C₁-C₆-Alkyl, partiell oder voll­ ständig halogeniertem C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl;
R¹¹ Wasserstoff, Cyano, Halogen, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxycarbonyl, -NR¹⁸R¹⁹, wobei R¹⁸ und R¹⁹ die Bedeutungen von R¹⁵ und R¹⁶ haben, oder Phenyl, das noch einen bis drei Substi­ tuenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl;
R¹³ Wasserstoff, Cyano, C₁-C₆-Alkyl oder C₁-C₆-Alkoxy­ carbonyl;
R¹ Halogen, die Cyano-, Nitro- oder Trifluormethylgruppe;
R² Wasserstoff oder Halogen;
R³ Wasserstoff, eine C₁-C₆-Alkylgruppe, eine C₃-C₆-Alkenylgruppe, eine C₃-C₆-Alkinylgruppe, eine C₃-C₈-Cycloalkylgruppe, eine C₃-C₈-Cycloalkylcarbonylgruppe, eine C₁-C₆-Cyanoalkylgruppe, eine partiell oder vollständig halogenierte C₁-C₆-Alkylgruppe, eine C₁-C₆-Alkoxy-C₁-C₆-alkylgruppe, die Formylgruppe, eine C₁-C₆- Alkanoylgruppe, eine C₁-C₆-Alkoxycarbonylgruppe, eine partiell oder vollständig halogenierte C₁-C₆-Alkylcarbonylgruppe,
eine Gruppe -N(R²⁰)R²¹, wobei R²⁰ und R²¹ für eine der Bedeutungen von R¹⁵ und R¹⁶ stehen,
die Phenylgruppe oder eine Phenyl-C₁-C₆-alkylgruppe, wobei der Phenylring jeweils noch einen bis drei Reste tragen kann, aus­ gewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₂-C₆-Alkenyl, partiell oder vollständig haloge­ niertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl;
R⁴ Wasserstoff, Cyano, Halogen, eine C₁-C₆-Alkylgrupe, eine C₂-C₆- Alkenylgruppe, eine C₂-C₆-Alkinylgruppe, eine C₃-C₇-Cycloalkyl­ gruppe, eine partiell oder vollständig halogenierte C₁-C₆-Alkyl­ gruppe, eine C₁-C₆-Hydroxylalkylgruppe, eine C₁-C₆-Cyanoalkyl­ gruppe, eine C₁-C₆-Alkoxy-C₁-C₆-alkylgruppe, eine C₁-C₆-Alkyl­ thio-C₁-C₆-alkylgruppe oder die Phenylgruppe, die noch einen bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₂-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl;
R⁵ Wasserstoff, Cyano, Nitro, Halogen, eine C₁-C₆-Alkylgruppe, eine C₂-C₆-Alkenylgruppe, eine C₂-C₆-Alkinylgruppe, eine C₃-C₇-Cyclo­ alkylgruppe, eine partiell oder vollständig halogenierte C₁-C₆- Alkylgruppe, eine C₁-C₆-Hydroxyalkylgruppe, eine C₁-C₆-Cyano­ alkylgruppe, eine C₁-C₆-Alkoxy-C₁-C₆-alkylgruppe, eine C₁-C₆- Alkylthio-C₁-C₆-alkylgruppe, die Formylgruppe, eine C₁-C₆-Alkyl­ carbonylgruppe, eine partiell oder vollständig halogenierte C₁-C₆-Alkylcarbonylgruppe, eine C₁-C₆-Alkoxycarbonylgruppe, eine Gruppe -N(R²²)R²³, wobei R²² und R²³ für eine der Bedeutungen von R¹⁵ und R¹⁶ stehen, die Phenylgruppe, die noch einen bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₂-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl, oder
R⁴ und R⁵ zusammen eine gesättigte oder ungesättigte 3- oder 4- gliedrige Kohlenstoffkette, die gewünschtenfalls ein bis drei Heteroatome als Glieder enthalten kann, ausgewählt aus einer Gruppe bestehend aus 1 oder 2 Sauerstoffatomen, 1 oder 2 Schwefelatomen und 1 bis 3 Stickstoffatomen, und wobei die Kette noch ein bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Amino, Halogen, C₁-C₆-Alkyl, C₂-C₆-Alkenyl, C₁-C₆-Alkoxy, C₁-C₆-Alkylthio und C₁-C₆-Alkoxy­ carbonyl;
mit der Maßgabe, daß nicht gleichzeitig R⁴ die Trifluormethyl­ gruppe R⁵ Wasserstoff sein können, wenn W eine Gruppe -CH=CH-CO-R¹⁰ mit R¹⁰ C₁-C₆-Alkoxy oder C₃-C₇-Cycloalkoxy bedeutet, sowie die Salze und Enolether derjenigen Verbindungen I, bei denen R³ Wasserstoff bedeutet.
Außerdem betrifft die Erfindung herbizid wirksame 3-Phenyl­ urazile der allgemeinen Formeln Ia und Ib
in denen R³′ eine C₁-C₆-Alkylgruppe, eine C₃-C₆-Alkenylgruppe oder eine C₃-C₆-Alkinylgruppe bedeutet.
Des weiteren betrifft die Erfindung herbizide, pestizide und das Wachstum der Pflanzen regulierende Mittel, welche diese Verbin­ dungen als wirksame Substanzen enthalten.
Aus der US 49 79 982 sind herbizid wirksame 3-Phenylurazile der Formel I′ bekannt
wobei Ra Wasserstoff oder Halogen, Rb C₁-C₁₂-Alkyl oder Cyclo­ alkyl und Rc C₁-C₁₂-Alkyl oder C₃-C₁₂-Alkenyl bedeuten.
Ferner werden in der EP-A 4 08 382 u. a. Strukturen der Formel I′′
wobei Rd für Wasserstoff, Alkyl, Hydroxymethyl oder Halogenalkyl, Re für Halogenalkyl, Rf für Wasserstoff, Alkyl, Halogenalkyl, Hydroxymethyl, Halogen oder Nitro, X¹ für Sauerstoff oder Schwefel, Rg für Wasserstoff, Alkyl, Alkoxy oder Alkoxyalkyl und Rh für Wasserstoff, Alkyl, Cycloalkyl, Halogenalkyl, Phenyl oder Benzyl und Ri für Halogen, Nitro oder Cyano stehen, beschrieben.
Außerdem lehrt die CH 4 82 402 Unkrautbekämpfungsmittel, die als Wirkstoffe u. a. substituierte Urazile und Thiourazile der Formel I′′′
enthalten, wobei Aryl einen gegebenenfalls durch Fluor, Chlor, Brom, Hydroxyl, Alkoxy, Cyano, Alkylthio, Alkyl oder Nitro sub­ stituierten Arylrest, Rk Dialkylphosphoryl, Alkyl, Alkenyl, Cyano, Wasserstoff, geg. subst. Alkyl, geg. subst. Carbamyl, geg. subst. Thiocarbamyl, geg. subst. Mercapto oder Acyl, Rl Alkyl, Alkoxy, Wasserstoff, Chlor oder Brom und Rm Alkylthio, Alkoxy, Alkylthioalkyl, Alkenyl, Cyano, Thiocyano, Nitro, Halogen, Wasserstoff oder geg. subst. Alkyl oder Rl und Rm zusammen eine Tri-, Tetra- oder Pentamethylenkette, bedeuten.
Andere 3-Arylurazile vom Typ der Verbindungen I sind beispiels­ weise den folgenden Druckschriften zu entnehmen: EP-A 1 95 346, EP-A 2 60 621, EP-A 4 38 209, WO 88/10 254, WO 89/02 891 und WO 89/03 825.
Die Selektivität dieser bekannten Herbizide bezüglich der Schad­ pflanzen vermag jedoch nur bedingt zu befriedigen, so daß der Erfindung neue herbizid wirksame Verbindungen als Aufgabe zu­ grunde lagen, mit denen sich (bei guter Verträglichkeit für die Nutzpflanzen) die Schadpflanzen besser als bisher gezielt be­ kämpfen lassen.
Demgemäß wurden die eingangs definierten substituierten 3-Phenyl­ urazile I, Ia und Ib gefunden.
Außerdem wurden herbizide Mittel gefunden, die diese Subtanzen enthalten und eine gute herbizide Wirkung besitzen. Sie sind verträglich und somit selektiv in breitblättrigen Kulturen sowie in monokotylen Gewächsen, welche nicht zu den Gramineen zählen.
Die erfindungsgemäßen Verbindungen I, Ia und Ib eignen sich des weiteren als Defoliations- bzw. Desiccationsmittel in z. B. Baum­ wolle, Kartoffel, Raps, Sonnenblume, Sojabohne oder Ackerbohnen. Einige Verbindungen I sind ferner brauchbar zur Bekämpfung von Schädlingen, insbesondere Insekten.
Die vorstehend für die Substituenten R¹ bis R¹⁷genannten Bedeu­ tungen stellen Sammelbegriffe für eine individuelle Aufzählung der einzelnen Gruppenmitglieder dar. Sämtliche Alkyl-, Alkenyl-, Alkinyl-, Halogenalkyl- und Halogenalkoxyteile können geradkettig oder verzweigt sein. Die Halogenalkyl- und Halogenalkoxyrest können gleiche oder verschiedene Halogenatome tragen.
Im einzelnen bedeuten beispielsweise:
- Halogen:
Fluor, Chlor, Brom und Jod, 99999 00070 552 001000280000000200012000285919988800040 0002004131038 00004 99880 vorzugsweise Fluor und Chlor;
- C₁-C₆-Alkyl:
Methyl, Ethyl, n-Propyl, 1-Methylethyl, n-Butyl, 1-Methyl-propyl, 2-Methylpropyl, 1,1-Dimethylethyl, n-Pentyl, 1-Methylbutyl, 2-Methylbutyl, 3-Methylbutyl, 2,2-Di-methylpropyl, 1-Ethylpropyl, 1,1-Dimethylpropyl, 1,2-Dimethylpropyl, n-Hexyl, 1-Methylpentyl, 2-Methylpentyl, 3-Methylpentyl, 4-Methylpentyl, 1,1-Dimethylbutyl, 1,2-Di­ methylbutyl, 1,3-Dimethylbutyl, 2,2-Dimethylbutyl, 2,3-Di­ methylbutyl, 3,3-Dimethylbutyl, 1-Ethylbutyl, 2-Ethylbutyl, 1,1,2-Trimethylpropyl, 1,2,2-Trimethylpropyl, 1-Ethyl-1- methylpropyl und 1-Ethyl-2-methylpropyl, vorzugsweise Methyl, Ethyl, Isopropyl, n-Butyl und tert.-Butyl;
- C₂-C₆-Alkenyl:
Vinyl und C₃-C₆-Alkenyl wie Prop-1-en-1-yl, Prop-2-en-1-yl, 1-Methylethenyl, n-Buten-1-yl, n-Buten-2-yl, n-Buten-3-yl, 1-Methyl-prop-1-en-1-yl, 2-Methyl-prop-1- en-1-yl, 1-Methyl-prop-2-en-1-yl, 2-Methyl-prop-2-en-1-yl, n-Penten-1-yl, n-Penten-2-yl, n-Penten-3-yl, n-Penten-4-yl, 1-Methyl-but-1-en-1-yl, 2-Methyl-but-1-en-1-yl, 3-Methyl- but-1-en-1-yl, 1-Methyl-but-2-en-1-yl, 2-Methyl-but-2- en-1-yl, 3-Methyl-but-2-en-1-yl, 1-Methyl-but-3-en-1-yl, 2-Methyl-but-3-en-1-yl, 3-Methyl-but-3-en-1-yl, 1,1-Di­ methyl-prop-2-en-1-yl, 1,2-Dimethyl-prop-1-en-1-yl, 1,2-Dimethyl-prop-2-en-1-yl, 1-Ethyl-prop-1-en-2-yl, 1-Ethyl-prop-2-en-1-yl, n-Hex-1-en-1-yl, n-Hex-2-en-1-yl, n-Hex-3-en-1-yl, n-Hex-4-en-1-yl, n-Hex-5-en-1-yl, 1-Methyl- pent-1-en-1-yl, 2-Methyl-pent-1-en-1-yl, 3-Methyl-pent-1- en-1-yl, 4-Methyl-pent-1-en-1-yl, 1-Methyl-pent-2-en-1-yl, 2-Methyl-pent-2-en-1-yl, 3-Methyl-pent-2-en-1-yl, 4-Methyl- pent-2-en-1-yl, 1-Methyl-pent-3-en-1-yl, 2-Methyl-pent-3- en-1-yl, 3-Methyl-pent-3-en-1-yl, 4-Methyl-pent-3-en-1-yl, 1-Methyl-pent-4-en-1-yl, 2-Methyl-pent-4-en-1-yl, 3-Methyl- pent-4-en-1-yl, 4-Methyl-pent-4-en-1-yl, 1,1-Dimethyl-but-2- en-1-yl, 1,1-Dimethyl-but-3-en-1-yl, 1,2-Dimethyl-but-1- en-1-yl, 1,2-Dimethyl-but-2-en-1-yl, 1,2-Dimethyl-but-3- en-1-yl, 1,3-Dimethyl-but-1-en-1-yl, 1,3-Dimethyl-but-2- en-1-yl, 1,3-Dimethyl-but-3-en-1-yl, 2,2-Dimethyl-but-3- en-1-yl, 2,3-Dimethyl-but-1-en-1-yl, 2,3-Dimethyl-but-2- en-1-yl, 2,3-Dimethyl-but-3-en-1-yl, 3,3-Dimethyl-but-1- en-1-yl, 3,3-Dimethyl-but-2-en-1-yl, 1-Ethyl-but-1-en-1-yl, 1-Ethyl-but-2-en-1-yl, 1-Ethyl-but-3-en-1-yl, 2-Ethyl- but-1-en-1-yl, 2-Ethyl-but-2-en-1-yl, 2-Ethyl-but-3-en-1-yl, 1,1,2-Trimethylprop-2-en-1-yl, 1-Ethyl-1-methyl-prop-2- en-1-yl, 1-Ethyl-2-methyl-prop-1-en-1-yl und 1-Ethyl-2- methyl-prop-2-en-1-yl, vorzugsweise Vinyl, Prop-2-en-1-yl und But-2-en-2-yl;
- C₂-C₆-Alkinyl:
Ethinyl und C₃-C₆-Alkinyl wie Prop-1-in-1-yl, Prop-2-in-3-yl, n-But-1-in-1-yl, n-But-1-in-4-yl, n-But-2- in-1-yl, n-Pent-1-in-1-yl, n-Pent-1-in-3-yl, n-Pent-1-in-4- yl, n-Pentin-5-yl, Pent-2-in-1-yl, Pent-2-in-4-yl, Pent-2- in-5-yl, 3-Methyl-but-1-in-1-yl, 3-Methyl-But-1-in-3-yl, 3-Methyl-but-1-in-4-yl, n-Hex-1-in-1-yl, n-Hex-1-in-3-yl, n-Hex-1-in-4-yl, n-Hex-1-in-5-yl, n-Hex-1-in-6-yl, n-Hex-2- in-1-yl, n-Hex-2-in-4-yl, n-Hex-2-in-5-yl, n-Hex-2-in-6-yl, n-Hex-3-in-1-yl, n-Hex-3-in-2-yl, 3-Methyl-pent-1-in-1-yl, 3-Methyl-pent-1-in-3-yl, 3-Methyl-pent-1-in-4-yl, 3-Methyl- pent-1-in-5-yl, 4-Methyl-pent-1-in-1-yl, 4-Methyl-pent-2-in- 4-yl und 4-Methyl-pent-2-in-5-yl, vorzugsweise Prop-2-inyl;
- C₃-C₈-Cycloalkyl:
Cyclopropyl, Cyclobutyl, Cyclopentyl, Cyclohexyl, Cycloheptyl und Cyclooctyl, vorzugsweise Cyclo­ propyl, Cyclopentyl und Cyclohexyl;
- partiell oder vollständig halogeniertes C₁-C₆-Alkyl:
Chlor­ methyl, Dichlormethyl, Trichlormethyl, Fluormethyl, Difluor­ methyl, Trifluormethyl, Chlorfluormethyl, Dichlorfluor­ methyl, Chlordifluormethyl, 1-Fluorethyl, 2-Fluorethyl, 2,2-Difluorethyl, 2,2,2-Trifluorethyl, 2-Chlor-2-fluorethyl, 2-Chlor-2,2-difluorethyl, 2,2-Dichlor-2-fluorethyl, 2,2,2- Trichlorethyl, Pentafluorethyl und 3-Chlorpropyl, vorzugs­ weise Trifluormethyl;
- Hydroxy-(C₁-C₆)-alkyl:
Hydroxymethyl, 1-Hydroxyeth-1-yl, 2-Hydroxyeth-1-yl, 1-Hydroxy-prop-1-yl, 2-Hydroxy-prop-1-yl, 3-Hydroxy-prop-1-yl, 1-Hydroxy-prop-2-yl, 2-Hydroxy-prop- 2-yl, 1-Hydroxy-but-1-yl, 2-Hydroxy-but-1-yl, 3-Hydroxy- but-1-yl, 4-Hydroxy-but-1-yl, 1-Hydroxy-but-2-yl, 2-Hydroxy- but-2-yl, 1-Hydroxy-but-3-yl, 1-Hydroxy-but-3-yl, 1-Hydroxy- 2-methyl-prop-3-yl, 2-Hydroxy-2-methyl-prop-3-yl, 3-Hydroxy- 2-methyl-prop-3-yl und 2-Hydroxymethyl-prop-2-yl, vorzugs­ weise Hydroxymethyl;
- Cyano-(C₁-C₆)-alkyl:
Cyanomethyl, 1-Cyanoeth-1-yl, 2-Cyano- eth-1-yl, 1-Cyano-prop-1-yl, 2-Cyano-prop-1-yl, 3-Cyano- prop-1-yl, 1-Cyano-prop-2-yl, 2-Cyano-prop-2-yl, 1-Cyano- but-1-yl, 2-Cyano-but-1-yl, 3-Cyano-but-1-yl, 4-Cyano-but-1- yl, 1-Cyano-but-2-yl, 2-Cyano-but-2-yl, 1-Cyano-but-3-yl, 2-Cyano-but-3-yl, 1-Cyano-2-methyl-prop-3-yl, 2-Cyano-2- methyl-prop-3-yl, 3-Cyano-2-methyl-prop-3-yl, und 2-Cyano- methyl-prop-2-yl, vorzugsweise Cyanomethyl;
- Amino-(C₁-C₆)-alkyl:
Aminomethyl, 1-Aminoethyl, 2-Amino­ ethyl, 1-Aminoprop-1-yl, 2-Aminoprop-1-yl, 3-Aminoprop-1-yl, 1-Aminobut-1-yl, 2-Aminobut-1-yl, 3-Aminobut-1-yl, 4-Amino­ but-1-yl, 1-Aminobut-2-yl, 2-Aminobut-2-yl, 3-Aminobut-2-yl, 3-Aminobut-2-yl, 4-Aminobut-2-yl, 1-(Aminomethyl)-eth-1-yl, 1-(Aminomethyl)-1-(methyl)-eth-1-yl, und 1-(Aminomethyl)- prop-1-yl, vorzugsweise Aminomethyl;
- Phenyl-C₁-C₆-alkyl:
Benzyl, 1-Phenylethyl, 2-Phenylethyl, 1-Phenylprop-1-yl, 2-Phenylprop-1-yl, 3-Phenylprop-1-yl, 1-Phenylbut-1-yl, 2-Phenylbut-1-yl, 3-Phenylbut-1-yl, 4-Phenylbut-1-yl, 1-Phenylbut-2-yl, 2-Phenylbut-2-yl, 3-Phenylbut-2-yl, 3-Phenylbut-2-yl, 4-Phenylbut-2-yl, 1-(Phenylmethyl)-eth-1-yl, 1-(Phenylmethyl)-1-(methyl)- eth-1-yl, und 1-(Phenylmethyl)-prop-1-yl, vorzugsweise Benzyl;
- C₁-C₆-Alkoxy:
Methoxy, Ethoxy, n-Propoxy, 1-Methylethoxy, n-Butoxy, 1-Methyl-propoxy, 2-Methylpropoxy, 1,1-Dimethyl­ ethoxy, n-Pentoxy, 1-Methylbutoxy, 2-Methylbutoxy, 3-Methyl­ butoxy, 1,1-Dimethylpropoxy, 1,2-Dimethylpropoxy, 2,2-Di­ methylpropoxy, 1-Ethylpropoxy, n-Hexoxy, 1-Methylpentoxy, 2-Methylpentoxy, 3-Methylpentoxy, 4-Methylpentoxy, 1,1-Di­ methylbutoxy, 1,2-Dimethylbutoxy, 1,3-Dimethylbutoxy, 2,2- Dimethylbutoxy, 2,3-Dimethylbutoxy, 3,3-Dimethylbutoxy, 1-Ethylbutoxy, 2-Ethylbutoxy, 1,1,2-Trimethylpropoxy, 1,2,2- Trimethylpropoxy, 1-Ethyl-1-methylpropoxy und 1-Ethyl-2- methylpropoxy, vorzugsweise C₁-C₄-Alkoxy wie Methoxy und Ethoxy;
- partiell oder vollständig halogeniertes C₁-C₆-Alkoxy:
2-Fluorethyloxy, 2,2-Difluorethyloxy, 2,2,2-Trifluorethyl­ oxy, 2-Chlor-2-fluorethyloxy, 2-Chlor-2,2-difluorethyloxy, 2,2-Dichlor-2-fluorethyloxy, 2,2,2-Trichlorethyloxy und 3-Brom-prop-1-yloxy;
- C₁-C₆-Alkylthio:
Methylthio, Ethylthio, n-Propylthio, 1-Methylethylthio, n-Butylthio, 1-Methyl-propylthio, 2-Methylpropylthio, 1,1-Dimethylethylthio, n-Pentylthio, 1-Methylbutylthio, 2-Methylbutylthio, 3-Methylbutylthio, 1,1-Dimethylpropylthio, 1,2-Dimethylpropylthio, 2-2-Di­ methylpropylthio, 1-Ethylpropylthio, n-Hexylthio, 1-Methyl­ pentylthio, 2-Methylpentylthio, 3-Methylpentylthio, 4-Methylpentylthio, 1,1-Dimethylbutylthio, 1,2-Dimethyl­ butylthio, 1,3-Dimethylbutylthio, 2,2-Dimethylbutylthio, 2,3-Dimethylbutylthio, 3,3-Dimethylbutylthio, 1-Ethylbutyl­ thio, 2-Ethylbutylthio, 1,1,2-Trimethylpropylthio, 1,2,2- Trimethylpropylthio, 1-Ethyl-1-methylpropylthio und 1-Ethyl- 2-methylpropylthio, vorzugsweise C₁-C₄-Alkylthio wie Methyl­ thio und Ethylthio;
- C₁-C₆-Alkoxy-C₁-C₆-alkyl:
Methoxymethyl, Ethoxymethyl, n-Propoxymethyl, (1-Methylethoxy)methyl, n-Butoxymethyl, (1-Methylpropoxy)methyl, (2-Methylpropoxy)methyl, (1,1-Di­ methylethoxy)methyl, Methoxyethyl, Ethoxyethyl, n-Propoxy­ ethyl, (1-Methylethoxy)ethyl, n-Butoxyethyl, (1-Methyl­ propoxy)ethyl, (2-Methylpropoxy)ethyl, (1,1-Dimethylethoxy)- ethyl, 3-(Methoxy)propyl, 2-(Methoxy)propyl und 2-(Ethoxy)- propyl, vorzugsweise C₁-C₄-Alkoxy-C₁-C₂-alkyl wie Methoxy­ methyl, Ethoxymethyl, 2-Methoxyethyl und 2-Ethoxyethyl;
- C₁-C₆-Alkylamino:
Methylamino, Ethylamino, n-Propylamino, 1-Methylethylamino, n-Butylamino, 1-Methylpropylamino, 2-Methylpropylamino, 1,1-Dimethylethylamino, n-Pentylamino, 1-Methylbutylamino, 2-Methylbutylamino, 3-Methylbutylamino, 2,2-Dimethylpropylamino, 1-Ethylpropylamino, n-Hexylamino, 1,1-Dimethylpropylamino, 1,2-Dimethylpropylamino, 1-Methyl­ pentylamino, 2-Methylpentylamino, 3-Methylpentylamino, 4-Methylpentylamino, 1,1-Dimethylbutylamino, 1,2-Dimethyl­ butylamino, 1,3-Dimethylbutylamino, 2,2-Dimethylbutylamino, 2,3-Dimethylbutylamino, 3,3-Dimethylbutylamino, 1-Ethyl­ butylamino, 2-Ethylbutylamino, 1,1,2-Trimethylpropylamino, 1,2,2-Trimethylpropylamino, 1-Ethyl-1-methylpropylamino und 1-Ethyl-2-methylpropylamino, vorzugsweise C₁-C₄-Alkylamino wie Methylamino und Ethylamino;
- Di-(C₁-C₆)-alkylamino:
N,N-Dimethylamino, N,N-Diethylamino, N,N-Dipropylamino, N,N-Di-(1-methylethyl)amino, N,N-Dibutyl­ amino, N,N-Di-(1-methylpropyl)amino, N,N-Di-(2-methyl­ propyl)amino, N,N-Di-(1,1-dimethylethyl)amino, N-Ethyl-N- methylamino, N-Methyl-N-propylamino, N-Methyl-N-(1-methyl­ ethyl)amino, N-Butyl-N-methylamino, N-Methyl-N-(1-methyl­ propyl)amino, N-Methyl-N-(2-methylpropyl)amino, N-(1,1-Di­ methylethyl)-N-methylamino, N-Ethyl-N-propylamino, N-Ethyl- N-(1-methyl-ethyl)amino, N-Butyl-N-ethylamino, N-Ethyl-N- (1-methyl-propyl)amino, N-Ethyl-N-(2-methylpropyl)amino, N-Ethyl-N-(1,1-dimethylethyl)amino, N-(1-Methylethyl)-N- propylamino, N-Butyl-N-propylamino, N-(1-Methylpropyl)-N- propylamino, N-(2-Methylpropyl)-N-propylamino, N-(1,1-Di­ methylethyl)-N-propylamino, N-Butyl-N-(1-methyl-ethyl)amino, N-(1-Methylethyl)-N-(1-methylpropyl)amino, N-(1-Methyl­ ethyl)-N-(2-methylpropyl)amino, N-(1,1-Dimethylethyl)-N-(1- methylethyl)amino, N-Butyl-N-(1-methylpropyl)amino, N-Butyl- N-(2-methylpropyl)amino, N-Butyl-N-(1,1-dimethylethyl)amino, N-(1-Methylpropyl)-N-(2-methylpropyl)amino, N-(1,1-Dimethyl­ ethyl)-N-(1-methylpropyl)amino und N-(1,1-Dimethylethyl)-N- (2-methylpropyl)amino, vorzugsweise Dimethylamino und Diethylamino;
- C₁-C₆-Alkylcarbonyl:
Methylcarbonyl, Ethylcarbonyl, Propyl­ carbonyl, 1-Methylethyl-carbonyl, Butylcarbonyl, 1-Methyl­ propylcarbonyl, 2-Methylpropylcarbonyl, 1,1-Dimethylethyl­ carbonyl, Pentylcarbonyl, 1-Methylbutylcarbonyl, 2-Methyl­ butylcarbonyl, 3-Methylbutylcarbonyl, 1,1-Dimethylpropyl­ carbonyl, 1,2-Dimethylpropylcarbonyl, 2,2-Dimethylpropyl­ carbonyl, 1-Ethylpropylcarbonyl, Hexylcarbonyl, 1-Methyl­ pentylcarbonyl, 2-Methylpentylcarbonyl, 3-Methylpentyl­ carbonyl, 4-Methylpentylcarbonyl, 1,1-Dimethylbutylcarbonyl, 1,2-Dimethylbutylcarbonyl, 1,3-Dimethylbutylcarbonyl, 2,2- Dimethylbutylcarbonyl, 2,3-Dimethylbutylcarbonyl, 3,3-Di­ methylbutylcarbonyl, 1-Ethylbutylcarbonyl, 2-Ethylbutyl­ carbonyl, 1,1,2-Trimethylpropylcarbonyl, 1,2,2-Trimethyl­ propylcarbonyl, 1-Ethyl-1-methylpropylcarbonyl und 1-Ethyl- 2-methylpropylcarbonyl, vorzugsweise C₁-C₄-Alkylcarbonyl wie Methylcarbonyl und Ethylcarbonyl;
- C₁-C₆-Alkylcarbonyloxy:
Methylcarbonyloxy, Ethylcarbonyloxy, n-Propylcarbonyloxy, 1-Methylethylcarbonyloxy, n-Butyl­ carbonyloxy, 1-Methylpropylcarbonyloxy, 2-Methylpropylcarb­ onyloxy, 1,1-Dimethylethylcarbonyloxy, n-Pentylcarbonyloxy, 1-Methylbutylcarbonyloxy, 2-Methylbutylcarbonyloxy, 3-Methylbutylcarbonyloxy, 1,1-Dimethylpropylcarbonyloxy, 1,2-Dimethylpropylcarbonyloxy, 2,2-Dimethylpropylcarbonyl­ oxy, 1-Ethylpropylcarbonyloxy, n-Hexylcarbonyloxy, 1-Methyl­ pentylcarbonyloxy, 2-Methylpentylcarbonyloxy, 3-Methyl­ pentylcarbonyloxy, 4-Methylpentylcarbonyloxy, 1,1-Dimethyl­ butylcarbonyloxy, 1,2-Dimethylbutylcarbonyloxy, 1,3-Di­ methylbutylcarbonyloxy, 2,2-Dimethylbutylcarbonyloxy, 2,3-Dimethylbutylcarbonyloxy, 3,3-Dimethylbutylcarbonyloxy, 1-Ethylbutylcarbonyloxy, 2-Ethylbutylcarbonyloxy, 1,1,2-Tri­ methylpropylcarbonyloxy, 1,2,2-Trimethylpropylcarbonyloxy, 1-Ethyl-1-methylpropylcarbonyloxy und 1-Ethyl-2-methyl­ propylcarbonyloxy, vorzugsweise C₁-C₄-Alkylcarbonyloxy wie Methylcarbonyloxy und Ethylcarbonyloxy;
- C₁-C₂-Halogenalkylcarbonyloxy:
Chloracetyl, Dichloracetyl, Trichloracetyl, Fluoracetyl, Difluoracetyl, Trifluoracetyl, Chlorfluoracetyl, Dichlorfluoracetyl, Chlordifluoracetyl, α-Fluorpropionyl, β-Fluorpropionyl, β,β,β-Difluorpropionyl, β,β,β-Trifluorpropionyl, β-Chlor-β-fluorpropionyl, β-Chlor- β,β-difluorpropionyl, β,β-Dichlor-β-fluorpropionyl, β,β,β- Trichlorpropionyl und Pentafluorpropionyl, vorzugsweise Trichloracetyl und Trifluoracetyl;
- C₁-C₆-Alkoxycarbonyl-C₁-C₆-alkyl:
Methoxycarbonylmethyl, Ethoxycarbonylmethyl, n-Propoxycarbonylmethyl, (1-Methyl­ ethoxycarbonyl)methyl, n-Butoxycarbonylmethyl, (1-Methyl­ propoxycarbonyl)methyl, (2-Methylpropoxycarbonyl)methyl, (1,1-Dimethylethoxycarbonyl)methyl, Methoxycarbonylethyl, Ethoxycarbonylethyl, n-Propoxycarbonylethyl, (1-Methyl­ ethoxycarbonyl)ethyl, n-Butoxycarbonylethyl, (1-Methyl­ propoxycarbonyl)ethyl, (2-Methylpropoxycarbonyl)ethyl, (1,1-Dimethylethoxycarbonyl)ethyl, 3-(Methoxycarbonyl)- propyl, 2-(Methoxycarbonyl)propyl und 2-(Ethoxycarbonyl)- propyl; vorzugsweise C₁-C₄-Alkoxycarbonyl-C₁-C₂-alkyl wie Methoxycarbonylmethyl, Ethoxycarbonylmethyl, 2-Methoxy­ carbonylethyl und 2-Ethoxycarbonylethyl;
- Di-(C₁-C₆)-alkylamino-(C₁-C₆)-alkoxy:
N,N-Dimethylamino­ ethoxy, N,N-Diethylaminoethoxy, N,N-Di(n-propyl)aminoethoxy, N,N-Di-(1-methylethyl)aminoethoxy, N,N-Dibutylaminoethoxy, N,N-Di-(1-methylpropyl)aminoethoxy, N,N-Di-(2-methylpropyl)- aminoethoxy, N,N-Di-(1,1-dimethylethyl)aminoethoxy, N-Ethyl- N-methylaminoethoxy, N-Methyl-N-propylaminoethoxy, N-Methyl- N-(1-methylethyl)aminoethoxy, N-Butyl-N-methylaminoethoxy, N-Methyl-N-(1-methylpropyl)aminoethoxy, N-Methyl-N-(2- methylpropyl)aminoethoxy, N-(1,1-Dimethylethyl)-N-methyl­ aminoethoxy, N-Ethyl-N-propylaminoethoxy, N-Ethyl-N-(1- methyl-ethyl)aminoethoxy, N-Butyl-N-ethylaminoethoxy, N-Ethyl-N-(1-methylpropyl)aminoethoxy, N-Ethyl-N-(2-methyl­ propyl)aminoethoxy, N-Ethyl-N-(1,1-dimethylethyl)amino­ ethoxy, N-(1-Methylethyl)-N-propylaminoethoxy, N-Butyl-N- propylaminoethoxy, N-(1-Methylpropyl)-N-propylaminoethoxy, N-(2-Methylpropyl)-N-propylaminoethoxy, N-(1,1-Dimethyl­ ethyl)-N-propylaminoethoxy, N-Butyl-N-(1-methylethyl)amino­ ethoxy, N-(1-Methylethyl)-N-(1-methylpropyl)aminoethoxy, N-(1-Methylethyl)-N-(2-methylpropyl)aminoethoxy, N-(1,1-Di­ methylethyl)-N-(1-methylethyl)aminoethoxy, N-Butyl-N-(1- methylpropyl)aminoethoxy, N-Butyl-N-(2-methylpropyl)amino­ ethoxy, N-Butyl-N-(1,1-dimethylethyl)aminoethoxy, N-(1-Methylpropyl)-N-(2-methyl-propyl)aminoethoxy, N-(1,1- Dimethylethyl)-N-(1-methylpropyl)aminoethoxy, N-(1,1-Di­ methylethyl)-N-(2-methylpropyl)aminoethoxy.
Die substituierten Phenylurazile I können in Form ihrer landwirt­ schaftlich brauchbaren Salze oder Enolether vorliegen, sofern R³ Wasserstoff bedeutet.
Als landwirtschaftlich brauchbare Salze kommen im allgemeinen die Salze von solchen Basen in Betracht, welche die herbizide Wirkung von I nicht beeinträchtigen.
Als basische Salze eignen sich besonders diejenigen der Alkali­ metalle, vorzugsweise die Natrium- und Kaliumsalze, die der Erd­ alkalimetalle, vorzugsweise Calcium-, Magnesium- und Bariumsalze und die der Übergangsmetalle, vorzugsweise Mangan-, Kupfer, Zink- und Eisensalze sowie die Ammoniumsalze, die ein bis drei C₁-C₄- Alkyl-, Hydroxy-C₁-C₄-alkylsubstituenten und/oder einen Phenyl- oder Benzylsubstituenten tragen können, vorzugsweise Di­ isopropylammonium-, Tetramethylammonium-, Tetrabutylammonium-, Trimethylbenzylammonium- und Trimethyl-(2-hydroxyethyl)-ammonium­ salze, die Phosphoniumsalze, die Sulfoniumsalze, vorzugsweise Tri-(C₁-C₄)alkylsulfoniumsalze, und die Sulfoxoniumsalze, vor­ zugsweise Tri-(C₁-C₄)alkylsulfoxoniumsalze.
Im Hinblick auf die Verwendung der erfindungsgemäßen 3-Phenyl­ urazile I, Ia und Ib als herbizide, das Pflanzenwachstum regu­ lierende und insektizid wirksame Verbindungen haben die Variablen vorzugsweise folgende Bedeutung:
wobei X¹ und X² unabhängig voneinander für Schwefel oder Sauer­ stoff stehen und die Variablen X, W, R¹, R², R³, R⁴, R²³, R⁵, R⁵⁶ beliebig miteinander kombiniert werden können, mit der Maß­ gabe, daß R⁴ nicht 4.27 bedeuten darf, wenn gleichzeitig R⁵ 5,01 und W -C(R⁸)=C(R⁹)-CO-R¹⁰, wobei R⁸ 8,01, R⁹ 9.01 und R¹⁰ 10.03-10.12 oder 10.20-10.23, bedeutet.
Besonders bevorzugt bedeuten
R¹ einen Rest aus der Gruppe 1.01-1.07,
R² einen Rest aus der Gruppe 2.01-2.06,
R³ einen Rest aus der Gruppe 3.01-3.97,
R³′ einen Rest aus der Gruppe 3′.01-3′.17,
R⁴ einen Rest aus der Gruppe 4.01-4.72,
R⁵ einen Rest aus der Gruppe 5.001-5.103
oder
R⁴ und R⁵ zusammen einen Rest aus der Gruppe 45.01-45.53 und
W einen der folgenden Reste W1-W6:
W1 -C(R⁸)(X³R⁶)(R⁴R⁷)
W2 -C(R⁸)=X⁵,
W3 -C(R⁸)=C(R⁹)-CO-R¹⁰,
W4 -CR⁸=CR⁹-CH₂-CO-R¹⁰,
W5 -CR⁸=CR⁹-CR¹¹=CR¹²-CO-R¹⁰,
W6 -CR⁸=CR⁹-CH₂-CHR¹³-CO-R¹⁰;
wobei
X³ und X⁴ unabhängig voneinander O oder S,
X⁵ O, S oder NR¹⁴,
R⁶ und R⁷ unabhängig voneinander einen Rest aus der Gruppe 6.01-6.17, oder
R⁶ und R⁷ zusammen einen Rest aus der Gruppe 67.01-67.60,
R⁸ einen Rest aus der Gruppe 8.01-8.22,
R⁹ und R¹² einen Rest aus der Gruppe 9.01-9.23,
R¹⁰ einen Rest aus der Gruppe 10.01-10.138,
R¹¹ einen Rest aus der Gruppe 11.01-11.25,
R¹³ einen Rest aus der Gruppe 13.01-13.08,
R¹⁴ einen Rest aus der Gruppe 14.001-14.162,
bedeuten und alle diese Reste beliebig miteinander kombiniert werden können.
Nr.
1.01
F
1.02 Cl
1.03 Br
1.04 I
1.05 CN
1.06 NO₂
1.07 CF₃
Nr.
2.01
H
2.02 F
2.03 Cl
2.04 Br
2.05 I
2.06 CN
Nr.
3.01
H
3.02 CH₃
3.03 C₂H₅
3.04 n-C₃H₇
3.05 i-C₃H₇
3.06 n-C₄H₉
3.07 i-C₄H₉
3.08 s-C₄H₉
3.09 tert.-C₄H₉
3.10 Cyclopropyl
3.11 Cyclobutyl
3.12 Cyclopentyl
3.13 Cyclohexyl
3.14 Cycloheptyl
3.15 Cyclooctyl
3.16 CH₂-CN
3.17 CH₂CH₂-CH
3.18 CH(CH₃)CH₂-CN
3.19 C(CH₃)₂-CN
3.20 C(CH₃)₂CH₂-CN
3.21 CH₂Cl
3.22 CH₂-CH₂Cl
3.23 CH(CH₃)-CH₂Cl
3.24 C(CH₃)₂Cl
3.25 CHCl₂
3.26 CF₂Cl
3.27 CF₃
3.28 C₂F₅
3.29 CF₂H
3.30 CH₂-CH=CH₂
3.31 CH(CH₃)CH=CH₂
3.32 CH₂-CH=CH-CH₃
3.34 CH₂-phenyl
3.35 CH₂-C≡CH
3.36 CH(CH₃)C≡CH
3.37 C(CH₃)₂C≡CH
3.38 Phenyl
3.39 2-F-phenyl
3.40 3-F-phenyl
3.41 4-F-phenyl
3.42 2-Cl-phenyl
3.43 3-Cl-phenyl
3.44 4-Cl-phenyl
3.45 2-CH₃-phenyl
3.46 3-CH₃-phenyl
3.47 4-CH₃-phenyl
3.48 2-CF₃-phenyl
3.49 3-CF₃-phenyl
3.50 4-CF₃-phenyl
3.51 2-OCH₃-phenyl
3.52 3-OCH₃-phenyl
3.53 4-OCH₃-phenyl
3.54 4-COOCH₃-phenyl
3.56 4-COOC₂H₅-phenyl
3.57 4-NO₂-phenyl
3.58 4-CN-phenyl
3.59 2,4-Cl₂-phenyl
3.60 2,4-(CH₃)₂-phenyl
3.61 CHO
3.62 CO-CH₃
3.63 CO-C₂H₅
3.64 CO-n-C₃H₇
3.65 CO-i-C₃H₇
3.66 CO-n-C₄H₉
3.67 CO-i-C₄H₉
3.68 CO-s-C₄H₉
3.69 CO-tert.-C₄H₉
3.70 CO-cyclopropyl
3.71 CO-cyclopentyl
3.72 CO-cyclohexyl
3.73 CO-CF₃
3.74 CO-CCl₃
3.75 CO-OCH₃
3.76 CO-OC₂H₅
3.77 COO-n-C₃H₇
3.78 COO-i-C₃H₇
3.79 COO-n-C₄H₉
3.80 COO-i-C₄H₉
3.81 COO-s-C₄H₉
3.82 COO-tert.-C₄H₉
3.83 CH₂-OCH₃
3.84 CH(CH₃)-OCH₃
3.85 CH(CH₃)-OC₂H₅
3.86 CH(CH₃)CH₂-OCH₃
3.87 CH₂OC₂H₅
3.88 NH₂
3.89 NHCH₃
3.90 NHC₂H₅
3.91 N(CH₃)₂
3.92 N(CH₃)C₂H₅
3.93 NH-CH-CH=CH₂
3.94 NH-CH₂C≡CH
3.95 NH-Cyclopropyl
3.96 NH-Cyclopentyl
3.97 NH-Cyclohexyl
Nr.
R⁴
4.01
H
4.02 F
4.03 Cl
4.04 Br
4.05 I
4.06 CH₃
4.07 C₂H₅
4.08 n-C₃H₇
4.09 i-C₃H₇
4.10 n-C₄H₉
4.11 i-C₄H₉
4.12 s-C₄H₉
4.13 tert.-C₄H₉
4.14 Cyclopropyl
4.15 Cyclobutyl
4.16 Cyclopentyl
4.17 Cyclohexyl
4.18 Cycloheptyl
4.19 Cyclooctyl
4.20 CN
4.21 CH₂Cl
4.22 CH₂CH₂Cl
4.23 CH(CH₃)CH₂Cl
4.24 CHCl₂
4.25 CCl₃
4.26 CF₂Cl
4.27 CF₃
4.28 C₂F₅
4.29 CF₂H
4.30 CH=CH₂
4.31 CH₂-CH=CH₂
4.32 CH₂-CH=CH-CH₃
4.33 C≡CH
4.34 CH₂-C≡CH
4.35 CH(CH₃)-C≡CH
4.36 Phenyl
4.37 2-F-phenyl
4.38 3-F-phenyl
4.39 4-F-phenyl
4.40 2-Cl-phenyl
4.41 3-Cl-phenyl
4.42 4-Cl-phenyl
4.43 2-CH₃-phenyl
4.44 3-CH₃-phenyl
4.45 4-CH₃-phenyl
4.46 2-CF₃-phenyl
4.47 3-CF₃-phenyl
4.48 4-CF₃-phenyl
4.49 2-OCH₃-phenyl
4.50 3-OCH₃-phenyl
4.51 4-OCH₃-phenyl
4.52 4-COOCH₃-phenyl
4.53 4-COOC₂H₅-phenyl
4.54 4-NO₂-phenyl
4.55 4-CN-phenyl
4.56 2,4-Cl₂-phenyl
4.57 2,6-Cl₂-phenyl
4.58 2,4-(CH₃)₂-phenyl
4.59 CH₂-OCH₃
4.60 CH₂-OC₂H₅
4.61 CH₂CH₂-OCH₃
4.62 CH₂CH₂-OC₂H₅
4.63 CH(CH₃)-OCH₃
4.64 CH₂-OH
4.65 CH₂CH₂-OH
4.66 CH₂CN
4.67 CH₂CH₂-CN
4.68 CH₂SCH₃
4.69 CH₂CH₂-SCH₃
4.70 CH₂CH₂-SC₂H₅
4.71 CH₂CH₂-SC₃H₇
4.72 CH₂-SC₂H₅
Nr.
R⁵
5.001
H
5.002 F
5.003 Cl
5.004 Br
5.005 I
5.006 CH₃
5.007 C₂H₅
5.008 n-C₃H₇
5.009 i-C₃H₇
5.010 n-C₄H₉
5.011 i-C₄H₉
5.012 s-C₄H₉
5.013 tert.-C₄H₉
5.014 n-C₅H₁₁
5.015 n-C₆H₁₃
5.016 Cyclopropyl
5.017 Cyclobutyl
5.018 Cyclopentyl
5.019 Cyclohexyl
5.020 Cycloheptyl
5.021 Cyclooctyl
5.022 CN
5.023 CH₂Cl
5.024 CH₂CH₂-Cl
5.025 CH(CH₃)CH₂-Cl
5.026 CHCl₂
5.027 CCl₃
5.028 CF₂Cl
5.029 CF₃
5.030 C₂F₅
5.031 CF₂H
5.032 CH=CH₂
5.033 CH₂-CH=CH₂
5.034 CH₂-CH=CH-CH₃
5.035 C≡CH
5.036 CH₂-C≡CH
5.037 CH(CH₃)-C≡CH
5.038 Phenyl
5.039 2-F-phenyl
5.040 3-F-phenyl
5.041 4-F-phenyl
5.042 2-Cl-phenyl
5.043 3-Cl-phenyl
5.044 4-Cl-phenyl
5.045 2-CH₃-phenyl
5.046 3-CH₃-phenyl
5.047 4-CH₃-phenyl
5.048 2-CF₃-phenyl
5.049 3-CF₃-phenyl
5.050 4-CF₃-phenyl
5.051 2-OCH₃-phenyl
5.052 3-OCH₃-phenyl
5.053 4-COOCH₃-phenyl
5.054 4-COOC₂H₅-phenyl
5.055 4-SCF₃-phenyl
5.056 4-NO₂-phenyl
5.057 4-CN-phenyl
5.058 2,4-Cl₂-phenyl
5.059 2,6-Cl₂-phenyl
5.060 2,4-(CH₃)₂-phenyl
5.061 CHO
5.062 CO-CH₃
5.063 CO-C₂H₅
5.064 CO-n-C₃H₇
5.065 CO-i-C₃H₇
5.066 CO-n-C₄H₉
5.067 CO-i-C₄H₉
5.068 CO-s-C₄H₉
5.069 CO-tert.-C₄H₉
5.070 CO-C₅H₁₁
5.071 CO-C₆H₁₃
5.073 CO-CF₃
5.074 CO-CCl₃
5.075 COO-CH₃
5.076 COO-C₂H₅
5.077 COO-n-C₃H₇
5.078 COO-i-C₃H₇
5.079 COO-n-C₄H₉
5.080 COO-i-C₄H₉
5.081 COO-s-C₄H₉
5.082 COO-tert.-C₄H₉
5.083 CH₂-OCH₃
5.084 CH₂-OC₂H₅
5.085 CH₂CH₂-OCH₃
5.086 CH₂CH₂-OC₂H₅
5.087 CH(CH₃)-OCH₃
5.088 CH₂OH
5.089 CH₂CH₂-OH
5.090 CH₂CN
5.091 CH₂CH₂-CN
5.092 CH₂-SCH₃
5.093 CH₂CH₂-SCH₃
5.094 CH₂CH₂-SC₂H₅
5.095 CH₂CH₂-SC₃H₇
5.096 CH₂-SC₂H₅
5.097 NO₂
5.098 NH₂
5.099 NH(CH₃)
5.100 N(CH₃)₂
5.101 NH(C₂H₅)
5.102 N(C₂H₅)
5.103 N(CH₃)(C₂H₅)
Nr.
R⁴+R⁵
45.01
-(CH₂)₃-
45.02 -(CH₂)₄-
45.03 -CH(CH₃)-(CH₂)₃-
45.04 -CH₂-CH(CH₃)-(CH₂)₂
45.05 -(CH₂)₂-CH(CH₃)-CH₂-
45.06 -(CH₂)₃-CH(CH₃)-
45.07 -CH₂-O-CH₂-
45.08 -(CH₂)₂-O-
45.09 -CH₂-O-(CH₂)₂-
45.10 -(CH₂)₂-O-CH₂-
45.11 -S-(CH₂)₂-
45.12 -CH₂-S-CH₂-
45.13 -(CH₂)₂-S-
45.14 -S-(CH₂)₃-
45.15 -CH₂-S-(CH₂)₂-
45.16 -(CH₂)₂-S-CH₂-
45.17 -(CH₂)₃-S-
45.18 -O-CH=CH-
45.19 -CH=CH-O-
45.20 -S-CH=CH-
45.21 -CH=CH-S-
45.22 -NH-CH=CH-
45.23 -NCH₃-CH=CH-
45.24 -CH=CH-NH-
45.25 -CH=CH-NCH₃-
45.26 -N=CH-CH=CH-
45.27 -CH=N-CH=CH-
45.28 -CH=CH-N=CH-
45.29 -CH=CH-CH=N-
45.30 -CH=N-O-
45.31 -O-N=CH-
45.32 -O-CH=N-
45.33 -N=CH-O-
45.34 -CH=N-S-
45.35 -S-N=CH-
45.36 -S-CH=N-
45.37 -N=CH-S-
45.38 -N=CH-NH-
45.39 -N=CH-NCH₃-
45.40 -NH-CH=N-
45.41 -N(CH₃)-CH=N-
45.42 -CH=CH-CH=CH-
45.43 -NH-CH=CH-NH-
45.44 -N=N-CH=CH-
45.45 -S-C(CH₃)=N-
45.46 -C(NO₂)=CH-S-
45.47 -C(CN)=CH-S-
45.48 -C(NO₂)=CH-O-
45.49 -C(CN)=CH-O-
45.50 -N(CH₃)-CH=CH-N(CH₃)-
45.51 -CH=CH-N=N-
45.52 -N=N-NH-
45.53 -N=N-N(CH₃)-
Nr.
R⁶, R⁷
6.01
CH₃
6.02 C₂H₅
6.03 n-C₃H₇
6.04 i-C₃H₇
6.05 n-C₄H₉
6.06 i-C₄H₉
6.07 s-C₄H₉
6.08 tert.-C₄H₉
6.09 n-C₅H₁₁
6.10 n-C₆H₁₃
6.11 CH₂CH=CH₂
6.12 CH(CH₃)-CH=CH₂
6.13 CH₂C≡CH
6.14 CH(CH₃)C≡CH
6.15 CH₂OCH₃
6.16 C₂H₅OCH₃
6.17 C₂H₅OC₂H₅
Nr.
R⁶+R⁷
67.01
-(CH₂)₂-
67.02 -CH(CH₃)-CH₂-
67.03 -CH(C₂H₅)-CH₂-
67.04 -CH(CH₃)-CH-(CH₃)-
67.05 -C(CH₃)₂-CH₂-
67.06 -CH(CH=CH₂)-CH₂-
67.07 -CH(CH₂Cl)-CH₂-
67.08 -CH(CH₂Br)-CH₂-
67.09 -CH(CH₂OH)-CH₂-
67.10 -CH(CH₂OCH₃)-CH₂-
67.11 -CH(CH₂OC₂H₅)-CH₂-
67.12 -CH(CH₂OCH₂CH=CH₂)-CH₂-
67.13 -CH(CH₂OCH₂C≡CH)-CH₂-
67.14 -CH(COOH)-CH₂-
67.15 -CH(COOCH₃)-CH₂-
67.16 -CH(COOC₂H₅)-CH₂-
67.17 -CH(COO-n-C₃H₇)-CH₂-
67.18 -CH(COO-i-C₃H₇)-CH₂-
67.19 -CH(COO-n-C₄H₉)-CH₂-
67.20 -CH(COO-n-C₅H₁₁)-CH₂-
67.21 -CH(COO-n-C₆H₁₃)-CH₂-
67.22 -(CH₂)₃-
67.23 -CH(CH₃)-(CH₂)₂-
67.24 -CH₂-CH(CH₃)-CH₂-
67.25 -CH(C₂H₅)-(CH₂)₂-
67.26 -CH₂-CH(C₂H₅)-CH₂-
67.27 -CH(CH₃)-CH₂-CH(CH₃)-
67.28 -CH₂-C(CH₃)₂-CH₂-
67.29 -CH(CH₂OH)-(CH₂)₂-
67.30 -CH₂-CH(CH₂OH)-CH₂
67.31 -CH(CH₂OCH₃)-(CH₂)₂-
67.32 -CH(CH₂OCH₂CH=CH₂)-(CH₂)₂-
67.33 -CH(CH₂O-CO-CH₃)-CH₂-
67.33 -CH(CH₂OCH₂C≡CH)-(CH₂)₂-
67.34 -CH(CH₂OC(O)CH₃)-(CH₂)₂
67.35 -CH₂-CH(CH₂OCH₃)-CH₂-
67.36 -CH₂-CH(CH₂OCH₂CH=CH₂)-CH₂-
67.37 -CH₂-CH(CH₂OCH₂C≡CH)-CH₂-
67.38 -CH₂-CH(CH₂OC(O)CH₃)-CH₂-
67.39 -CH(CH₂Cl)-(CH₂)₂
67.40 -CH₂-CH(CH₂Cl)-CH₂-
67.41 -C(CH₃)-(COOCH₃)-CH₂-
67.42 -C(CH₃)-(COOC₂H₅)-CH₂-
67.43 -C(CH₃)(COO-n-C₃H₇)-CH₂-
67.44 -C(CH₃)(COO-n-C₄H₆)-CH₂-
67.45 -CH(CH₂CN)-CH₂-
67.46 -CH(CH₂CN)-(CH₂)₂-
67.47 -CH₂-CH(CH₂CN)-CH₂-
67.48 -CH₂-O-CH₂-
67.49 -CH₂-NH-CH₂-
67.50 -CH₂-N(CH₃)-CH₂
67.51 -(CH₂)₄-
67.52 -CH₂-CH=CH-CH₂-
67.53 -CH₂-O-(CH₂)₂-
67.54 -CO-CH₂-
67.55 -CO-(CH₂)₂-
67.56 -CH₂-CO-CH₂-
67.57 -CO-C(CH₃)₂-
67.58 -CO-O-CH₂-
67.59 -CH₂-S-CH₂-
67.60 -CH(CH₂O-CO-CH₃)-CH₂-
Nr.
R⁸
8.01
H
8.02 CH₃
8.03 C₂H₅
8.04 n-C₃H₇
8.05 i-C₃H₇
8.06 n-C₄H₉
8.07 i-C₄H₉
8.08 s-C₄H₉
8.09 tert.-C₄H₉
8.10 n-C₅H₁₁
8.11 n-C₆H₁₃
8.12 CH-CH=CH₂
8.13 CH₂-C≡CH
8.14 CF₃
8.15 CCl₃
8.16 Cyclopropyl
8.17 Cyclobutyl
8.18 Cyclopentyl
8.19 Cyclohexyl
8.20 CN
8.21 CO-OCH₃
8.22 CO-OC₂H₅
Nr.
R⁹ und R¹²
9.01
H
9.02 F
9.03 Cl
9.04 Br
9.05 I
9.06 CN
9.07 CH₃
9.08 C₂H₅
9.09 n-C₃H₇
9.10 i-C₃H₇
9.11 n-C₄H₉
9.12 i-C₄H₉
9.13 s-C₄H₉
9.14 tert.-C₄H₉
9.15 n-C₅H₁₁
9.16 OCH₃
9.17 OC₂H₅
9.18 CF₃
9.19 CO-CH₃
9.20 CO-C₂H₅
9.21 COOCH₃
9.22 COOC₂H₅
9.23 COO-n-C₃H₇
Nr.
R¹⁰
10,01
H
10.02 OH
10.03 OCH₃
10.04 OC₂H₅
10.05 O-n-C₃H₇
10.06 O-i-C₃H₇
10.07 O-n-C₄H₉
10.08 O-i-C₄H₉
10.09 O-s-C₄H₉
10.10 O-tert.-C₄H₉
10.11 O-n-C₅H₁₁
10.12 O-n-C₆H₁₃
10.14 O-CH₂CH=CH₂
10.15 O-CH(CH₃)CH=CH₂
10.16 O-CH-CH=CH-CH₂
10.17 O-CH₂-C≡CH
10.18 O-CH(CH₃)-C≡CH
10.19 O-CH₂-C≡C-CH₃
10.20 O-cyclopropyl
10.21 O-cyclobutyl
10.22 O-cyclopentyl
10.23 O-cyclohexyl
10.24 O-CH₂-CF₃
10.25 O-CH₂-CCl₃
10.26 O-(CH₂)₃-Br
10.27 O-phenyl
10.28 O-2F-phenyl
10.29 O-2Cl-phenyl
10.30 O-2Br-phenyl
10.31 O-3F-phenyl
10.32 O-3Cl-phenyl
10.33 O-3-Br-phenyl
10.34 O-4-F-phenyl
10.35 O-4-Cl-phenyl
10.36 O-4-Br-phenyl
10.37 O-4-OCH₃-phenyl
10.38 O-4-CN-phenyl
10.39 O-4-COOCH₃-phenyl
10.40 O-4-CH₃-phenyl
10.41 O-2,4-Cl₂-phenyl
10.42 O-2,4-(CH₃)₂-phenyl
10.43 O-CH₂CN
10.44 O-CH₂CH=CCl₂
10.45 O-CH₂CH=CHCl
10.46 O-CH₂OCH₃
10.47 O-CH₂OC₂H₅
10.48 O-C₂H₄OCH₃
10.49 O-C₂H₄OC₂H₅
10.50 O-CH(CH₃)-OCH₃
10.51 O-CH(CH₃)-OC₂H₅
10.52 O-CH₂C=NOCH₃
10.53 O-C₂H₄C=NOCH₃
10.54 O-CH₂C=NOC₂H₅
10.55 O-C(O)CH₃
10.56 O-C(O)C₂H₅
10.57 O-C₂H₄C=NOC₂H₅
10.58 SCH₃
10.59 SC₂H₅
10.60 S-n-C₃H₇
10.61 S-i-C₃H₇
10.62 S-CH₂CH=CH₂
10.63 S-CH₂C≡CH
10.64 S-phenyl
10.65 S-CH₂CN
10.66 S-CH₂OCH₃
10.67 CH₃
10.68 C₂H₅
10.69 n-C₃H₇
10.70 i-C₃H₇
10.71 n-C₄H₉
10.72 i-C₄H₉
10.73 s-C₄H₉
10.74 tert.-C₄H₉
10.75 n-C₅H₁₁
10.76 n-C₆H₁₃
10.77 CH₂CH=CH₂
10.78 CH₂C≡CH
10.79 CH(CH₃)CH=CH₂
10.80 CH(CH₃)C≡CH
10.81 CH₂Cl
10.82 CH₂Br
10.83 CHCl₂
10.84 CF₃
10.85 Cyclopropyl
10.86 Cyclobutyl
10.87 Cyclopentyl
10.88 Cyclohexyl
10.89 Phenyl
10.90 2-F-phenyl
10.91 3-F-phenyl
10.92 4-F-phenyl
10.93 2-Cl-phenyl
10.94 4-Cl-phenyl
10.95 2,4-Cl₂-phenyl
10.96 CH₂-OCH₃
10.97 CH(OCH₃)₂
10.98 CH₂-SCH₃
10.99 NH₂
10.100 NHCH₃
10.102 NH-n-C₃H₇
10.103 NH-i-C₃H₇
10.104 NH-n-C₄H₉
10.105 N(CH₃)₂
10.106 N(C₂H₅)₂
10.107 N(CH₃)C₂H₅
10.108 N(n-C₃H₇)₂
10.109 NH-CH₂CH=CH₂
10.110 NH-CH(CH₃)-CH=CH₂
10.111 NH-CH₂-C≡CH
10.112 NH-CH(CH₃)-C≡CH
10.113 N(CH₃)-CH₂CH=CH
10.114 N(CH₃)-CH₂C≡CH
10.115 NH-cyclopropyl
10.116 NH-cyclobutyl
10.117 NH-cyclopentyl
10.118 NH-cyclohexyl
10.119 N(CH₃)-cyclohexyl
10.120 N(C₂H₅)-cyclohexyl
10.121 NH-COCH₃
10.122 NH-COC₂H₅
10.123 NH-COOCH₃
10.124 NH-CH₂OCH₃
10.125 NH-(CH₂)₂OCH₃
10.126 N-piperindinyl
10.127 N-pyrrolidinyl
10.128 N-morpholino
10.129 N-Piperazinyl
10.130 NH-phenyl
10.131 NH-2-CH₃-phenyl
10.132 NH-2-F-phenyl
10.133 NH-4-F-phenyl
10.134 NH-2-Cl-phenyl
10.135 NH-4-Cl-phenyl
10.136 NH-2,4-Cl₂-phenyl
10.137 O-CO-OCH₃
10.138 O-CO-OC₂H₅
Nr.
R¹¹
11.01
H
11.02 F
11.03 Cl
11.04 Br
11.05 I
11.06 CN
11.07 CH₃
11.08 C₂H₅
11.09 n-C₃H₇
11.10 i-C₃H₇
11.11 n-C₄H₉
11.12 i-C₄H₉
11.13 s-C₄H₉
11.14 tert.-C₄H₉
11.15 CH₂-CH=CH₂
11.16 CH₂-C≡CH
11.17 Phenyl
11.18 4-Cl-phenyl
11.19 N(CH₃)₂
11.20 COOCH₃
11.21 COOC₂H₅
11.22 COCH₃
11.23 COC₂H₅
11.24 CH₂OCH₃
11.25 (CH₂)₂-OCH₃
Nr.
R¹³
13.01
H
13.02 CN
13.03 CH₃
13.04 C₂H₅
13.05 n-C₃H₇
13.06 i-C₃H₇
13.07 COOCH₃
13.08 COOC₂H₅
Nr.
R¹⁴
14.01
H
14.02 CH₃
14.03 C₂H₅
14.04 n-C₃H₇
14.05 i-C₃H₇
14.06 n-C₄H₉
14.07 n-C₅H₁₁
14.08 n-C₆H₁₃
14.10 CH₂CH=CH₂
14.11 CH(CH₃)-CH=CH₂
14.12 CH₂-CH=CH-CH₂
14.13 CH₂-C≡CH
14.14 CH(CH₃)-C≡CH
14.15 CH₂-C≡C-CH₃
14.16 Cyclopropyl
14.17 Cyclobutyl
14.18 Cyclopentyl
14.19 Cyclohexyl
14.20 Cycloheptyl
14.22 (CH₂)₂Cl
14.23 CH₂Cl
14.25 Phenyl
14.26 2-F-phenyl
14.27 3-F-phenyl
14.28 4-F-phenyl
14.29 2-Cl-phenyl
14.30 3-Cl-phenyl
14.31 4-Cl-phenyl
14.32 2-Br-phenyl
14.33 3-Br-phenyl
14.34 4-Br-phenyl
14.35 2-CH₃-phenyl
14.36 3-CH₃-phenyl
14.37 4-CH₃-phenyl
14.38 2-CF₃-phenyl
14.39 3-CF₃-phenyl
14.40 4-CF₃-phenyl
14.41 2-OCH₃-phenyl
14.42 3-OCH₃-phenyl
14.43 4-OCH₃-phenyl
14.44 4-NO₂-phenyl
14.45 4-CN-phenyl
14.46 2,4-Cl₂-phenyl
14.47 2,4-(CH₃)₂-phenyl
14.48 CH₂-OCH₃
14.49 (CH₂)₂-OC₂H₅
14.50 OH
14.51 OCH₃
14.52 OC₂H₅
14.53 O-n-C₃H₇
14.54 O-i-C₃H₇
14.55 O-n-C₄H₉
14.56 O-i-C₄H₉
14.57 O-s-C₄H₉
14.58 O-tert.-C₄H₉
14.59 O-CH₂CH=CH₂
14.60 O-CH(CH₃)CH=CH₂
14.61 O-CH₂C≡CH
14.62 O-CH(CH₃)-C≡CH
14.63 O-CH₂-C≡C-CH₃
14.64 O-CH₂-CH=CH-CH₃
14.65 O-cyclopentyl
14.66 O-cyclohexyl
14.67 O-cyclopent-3-enyl
14.68 O-cyclohex-3-enyl
14.69 O-(CH₂)₂-Cl
14.70 O-(CH₂)₂-Cl
14.71 O-(CH₂)-F
14.72 O-CH₂-CF₃
14.73 O-(CH₂)₂-Br
14.74 O-CH₂-CH=CHCl
14.75 O-CH₂-C(Cl)=CH₂
14.76 O-CH₂-C(Br)=CH₂
14.77 O-CH₂-CH=C(Cl)-CH₃
14.78 O-CH₂-C(Cl)=CCl₂
14.79 O-CH₂-cyclopropyl
14.80 O-CH₂-cyclobutyl
14.81 O-CH₂-cyclopentyl
14.82 O-CH₂-cyclohexyl
14.83 O-CH₂-cycloheptyl
14.84 O-CO-CH₃
14.85 O-CO-C₂H₅
14.86 O-CH₂-CN
14.87 O-(CH₂)₃-CN
14.88 O-CH₂-OCH₃
14.89 O-CH₂-OC₂H₅
14.90 O-(CH₂)₂-OCH₃
14.91 O-(CH₂)₂-OC₂H₅
14.92 O-(CH₂)₃-OC₂H₅
14.93 O-(CH₂)₂-CO-OCH₃
14.94 O-(CH₂)₂-CO-OC₂H₅
14.95 O-C(CH₃)-CO-OCH₃
14.96 O-C(CH₃)-CO-OC₂H₅
14.97 O-(CH₂)₂-OH
14.98 O-CH₂-SCH₃
14.99 O-(CH₂)₂-N(CH₃)₂
14.100 O-(CH₂)₂-N(C₂H₅)₂
14.101 O-CH₂-phenyl
14.102 O-(CH₂)₂-phenyl
14.103 O-(CH₂)₃-phenyl
14.104 O-(CH₂)₄-phenyl
14.105 O-(CH₂)₄-(4-Cl-phenyl)
14.106 O-(CH₂)₄-(4-CH₃-phenyl)
14.107 O-(CH₂)₄-(4-CH₃-phenyl)
14.108 O-(CH₂)₄-(4-F-phenyl)
14.109 O-CH₂CH=CH-phenyl
14.110 O-CH₂CH=CH-(4-F-phenyl)
14.111 O-CH₂CH=CH-(4-Cl-phenyl)
14.112 O-CH₂CH=CH-(3-OCH₃-phenyl)
14.113 O-(CH₂)₂-CH=CH-(4-F-phenyl)
14.114 O-(CH₂)₂-CH=CH-(4-Cl-phenyl)
14.115 O-(CH₂)-CH=CH-(3,4-Cl₂-phenyl)
14.116 O-CH₂-CH=C(CH₃)-(4-F-phenyl)
14.117 O-CH₂-C≡C-CH₂-phenyl
14.119 O-(CH₂)₂-O-phenyl
14.120 O-(CH₂)₂-OCH₂-phenyl
14.121 O-(CH₂)₂-OCH₂-(4-F-phenyl)
14.122 O-CH₂CH=CH-CH₂-O-phenyl
14.123 O-CH₂C≡C-CH₂-O-phenyl
14.124 O-CH₂-C≡C-CH₂-O-(4-F-phenyl)
14.125 O-(CH₂)₂-SCH₂-phenyl
14.126 O-(CH₂)₂-SCH₂-(4-Cl-phenyl)
14.127 O-(CH₂)₂-N(CH₃)-CH₂-phenyl
14.128 NH₂
14.129 NHCH₃
14.130 NH-C₂H₅
14.131 NH-n-C₃H₇
14.132 NH-i-C₃H₇
14.133 NH-n-C₄H₉
14.134 NH-i-C₄H₉
14.135 NH-s-C₄H₉
14.136 NH-tert.-C₄H₉
14.137 NH-cyclopropyl
14.138 NH-cyclobutyl
14.139 NH-cyclopentyl
14.140 NH-cyclohexyl
14.141 NH-cycloheptyl
14.142 N(CH₃)₂
14.143 N(C₂H₅)₂
14.144 NH-CH₂CH=CH₂
14.145 NH-CH₂C≡CH
14.146 NH-CH₂-CF₃
14.147 NH-CO-CH₃
14.148 NH-COC₂H₅
14.149 NH-CO-OCH₃
14.150 NH-CO-OC₂H₅
14.151 NH-COO-tert.-C₄H₉
14.152 N-Pyrrolidinyl
14.153 N-Piperdinyl
14.154 N-Morpholino
14.155 N-Piperazinyl
14.156 NH-phenyl
14.157 NH-(4-Cl-phenyl)
14.158 NH-(4-F-phenyl)
14.159 NH-(4-OCH₃-phenyl)
14.160 NH-(2,4-Cl₂-phenyl)
14.161 CH₂-OCH₃
14.162 (CH₂)₂-OCH₃
Nr.
R³′
3′.01
CH₃
3′.02 C₂H₅
3′.03 n-C₃H₇
3′.04 i-C₃H₇
3′.05 n-C₄H₉
3′.06 i-C₄H₉
3′.07 s-C₄H₉
3′.08 tert.-C₄H₉
3′.09 n-C₅H₁₁
3′.10 i-C₅H₁₁
3′.11 n-C₆H₁₃
3′.12 i-C₆H₁₃
3′.13 CH₂CH=CH₂
3′.14 -CH(CH₃)-CH=CH₂
3′.15 -CH₂-CH=CH-CH₃
3′.16 -CH(CH₃)-C≡CH
3′.17 -CH₂C≡C-CH₃
Besonders bevorzugt sind die folgenden 3-Phenylurazile I-1 bis I-24:
wobei W für eine der folgenden Bedeutungen steht:
-CHO, -COCH₃, -COC₂H₅, -CO-n-C₃H₇, -CO-i-C₃H₇, -CO-n-C₄H₉, -CO-i-C₄H₉, -CO-s-C₄H₉, -CO-tert.-C₄H₉, -CO-CH₂CH=CH₂, -CO-CF₃, -COCCl₃, -COCH₂C≡CH, -CO-cyclopropyl, -CO-cyclobutyl, -CO-cyclopentyl, -CO-cyclohexyl, -CO-CN, -CO-COOCH₃, -CO-COOC₂H₅, -CH=NH, -CH=NCH₃, -CH=NC₂H₅, -CH=N-n-C₃H₅, -CH=N-i-C₃H₅, -CH=N-n-C₄H₉, -CH=NCH₂CH=CH₂, -CH=NCH₂CH=CH₂-CH₃, -CH=NCH₂≡CH, -CH=NCH₂C≡C-CH₃, -CH=N-cyclopropyl, -CH=N-cyclobutyl, -CH=N-cyclopentyl, -CH=N-cyclohexyl, -CH=N-cycloheptyl, -CH=N-CH₂-CH₂Cl, -CH=N-CH₂Cl, -CH=N-C₆H₅, -CH=N-(4-Br-C₆H₄), -CH=N-3-F-C₆H₄, -CH=N-4-F-C₆H₄, -CH=N-2-Cl-C₆H₄, -CH=N-3-Cl-C₆H₄, -CH=N-4-Cl-C₆H₄, -CH=N-2-Br-C₆H₄, -CH=N-2-F-C₆H₄, -CH=N-2-CH₃-C₆H₄, -CH=N-3-CH₃-C₆H₄, -CH=N-4-CH₃-C₆H₄, -CH=N-2-CF₃-C₆H₄, -CH=N-3-CF₃-C₆H₄, -CH=N-4-CF₃-C₆H₄, -CH=N-2-OCH₃-C₆H₄, -CH=N-3-OCH₃-C₆H₄, -CH=N-4-OCH₃-C₆H₄, -CH=N-4-NO₂-C₆H₄, -CH=N-4-CN-C₆H₄, -CH=N-2,4-(Cl,Cl)-C₆H₄, -CH=N-2,4-(CH₃,CH₃)-C₆H₄, -CH=N-CH₂OCH₃ -CH=N-CH₂OC₂H₅, -CH=N-CH₂CH₂OCH₃, -CH=N-CH₂CH₂OC₂H₅, -CH=N-OH, -CH=N-OCH₃, -CH=N-OC₂H₅, -CH=N-O-n-C₃H₇, -CH=N-O-i-C₃H₇, -CH=N-O-n-C₄H₉, -CH=N-O-i-C₄H₉, -CH=N-O-s-C₄H₉, -CH=N-O-tert.-C₄H₉, -CH=N-O-CH₂CH=CH₂, -CH=N-O-CH(CH₃)CH=CH₂, -CH=N-O-CH₂C≡CH, -CH=N-O-CH(CH₃)-C≡CH, -CH=N-O-CH₂-CH=CH-CH₃, -CH=N-O-CH₂-CH₂-Cl, -CH=N-O-CH₂-CH₂-F, -CH=N-O-CH₂-CF₃, -CH=N-O-CH₂-CH=CHCl, -CH=N-O-CH₂-CCl=CH₂, -CH=N-O-CH₂-CBr=CH₂, -CH=N-O-CH₂-CH=CCl-CH₃, -CH=N-OC(O)CH₃, -CH=N-OC(O)C₂H₅, -CH=N-O-CH₂-CN, -CH=N-O-CH₂-CH=CH-CH₂-O-CH₃, -CH=N-O-CH₂-CH=CH-CH₂-O-tert.-C₄H₉, -CH=N-O-(CH₂)₃-C₆H₅, -CH=N-O-(CH₂)₄-C₆H₅, -CH=N-O-(CH₂)₄-4-Cl-C₆H₄, -CH=N-O-(CH₂)₄-4-OCH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-CH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-C₆H₅, -CH=N-O-CH₂CH=CH-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CH-3-OCH₃-C₆H₄, -CH=N-O-(CH₂)₂CH=CH-4-F-C₆H₄, -CH=N-O-(CH₂)CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CHCH₂-4-OCH₃-C₆H₄, -CH=N-O-CH₂-CH=C(CH₃)-C₆H₅ -CH=N-O-(CH₂)₂CH=CH-3,4(Cl,Cl)-C₆H₃, -CH=N-O-(CH₂)₃C≡C-4-F-C₆H₄, -CH₂=N-OCHOCH₃, -CH=N-OC₂H₄OCH₃, -CH=N-OCH₂OC₂H₅, -CH=N-OCH(CH₃)OCH₃, -CH=N-OCH(CH₃)COOCH₃, -CH=N-OCH(CH₃)COO-n-C₄H₉, -CH=N-NH₂, -CH=N-NHCH₃, -CH=N-NHC₂H₅, -CH=N-NH-n-C₃H₇, -CH=N-NH-i-C₃H₇, -CH=N-NH-n-C₄H₉, -CH=N-NH-i-C₄H₉, -CH=N-NH-s-C₄H₉, -CH=N-NH-tert.-C₄H₉, -CH=N-NH-cyclopropyl, -CH=N-NH-cyclobutyl, -CH=N-NH-cyclopentyl, -CH=N-NH-cyclohexyl, -CH=N-NH-cycloheptyl, -CH=N-N(CH₃)₂, -CH=N-N(C₂H₅)₂, -CH=N-N(C₃H₇)₂, -CH=N-N(i-C₃H₇)(CH₃), -CH=N-NHCH₂-C=CH, -CH=N-NHCH₂-C≡CH, -CH=N-N(CH₃)-CH₂-C≡CH, -CH=N-NHCH₂CF₃, -CH=N-NH-CO-CH₃, -CH=N-NH-CO-CH₂H₅, -CH=N-NH-COOCH₃, -CH=N-NH-COOC₂H₅, -CH=N-NH-COO-tert.-C₄H₉, -CH=N-pyrrolidin-1-yl, -CH=N-piperidin-1-yl, -CH=N-morpholin-4-yl, -CH=N-NH-C₆H₅, -CH=N-NH-(4-Cl-C₆H₄), -CH=N-NH-(4-NO₂-C₆H₄), -CH=N-NH-(4-F-C₆H₄), -CH=N-NH-(4-CH₃O-C₆H₄), -CH=N-NH-(2,4-Cl₂-C₆H₃), -CH=N-NH-(2,4-(NO₂)₂-C₆H₃), -CH=N-NH-CO-NH₂, -CH=N-NH-CO-NHCH₃, -CH=N-NH-CO-NHC₂H₅, -CH=N-NH-CO-N(CH₃)₂, -CH=CH-COOH, -CH=CH-CO-OCH₃, -CH=C-CO-OC₂H₅, -CH=CH-CO-O-n-C₃H₇, -CH=CH-CO-O-i-C₃H₇, -CH=CH-CO-O-n-C₄H₉, -CH=CH-CO-O-tert.-C₄H₉, -CH=CH-CO-O-cyclopropyl, -CH=CH-CO-O-cyclobutyl, -CH=CH-CO-O-cyclopentyl, -CH=CH-CO-O-cyclohexyl, -CH=CH-CO-O-cycloheptyl, -CH=C(CH₃)-COOH, -CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CO-O-n-C₃H₇, -CH=C(CH₃)-CO-O-i-C₃H₇, -CH=C(CH₃)-CO-O-n-C₄H₉, -CH=C(CH₃)-CO-O-tert.-C₄H₉, -CH=C(CH₃)-CO-O-cyclopropyl, -CH=C(CH₃)-CO-O-cyclobutyl, -CH=C(CH₃)-CO-O-cyclopentyl, -CH=C(CH₃)-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cycloheptyl, -CH=C(C₂H₅)-COOH, -CH=C(C₂H₅)-CO-OCH₃, -CH=C(C₂H₅)-CO-OC₂H₅, -CH=C(C₂H₅)-CO-O-n-C₃H₇, -CH=C(C₂H₅)-CO-O-i-C₃H₇, -CH=C(C₂H₅)-CO-O-n-C₄H₉, -CH=C(C₂H₅)-CO-O-tert.-C₄H₉, -CH=C(C₂H₅)-CO-O-cyclopropyl, -CH=C(C₂H₅)-CO-O-cyclobutyl, -CH=C(C₂H₅)-CO-O-cyclopentyl, -CH=C(C₂H₅)-CO-O-cyclohexyl, -CH=C(C₂H₅)-CO-O-cycloheptyl, -CH=C(Cl)-COOH, -CH=C(Cl)-CO-OCH₃, -CH=C(Cl)-CO-OC₂H₅, -CH=C(Cl)-CO-O-n-C₃H₇, -CH=C(Cl)-CO-O-i-C₃H₇, -CH=C(Cl)-CO-O-n-C₄H₉, -CH=C(Cl)-CO-O-tert.-C₄H₉, -CH=C(Cl)-CO-O-cyclopropyl, -CH=C(Cl)-CO-O-cyclobutyl, -CH=C(Cl)-CO-O-cyclopentyl, -CH=C(Cl)-CO-O-cyclohexyl, -CH=C(Cl)-CO-O-cycloheptyl, -CH=C(Br)-COOH, -CH=C(Br)-CO-OCH₃, -CH=C(Br)-CO-OC₂H₅, -CH=C(Br)-CO-O-n-C₃H₇, -CH=C(Br)-CO-O-i-C₃H₇, -CH=C(Br)-CO-O-n-C₄H₉, -CH=C(Br)-CO-O-tert.-C₄H₉, -CH=C(Br)-CO-O-cyclopropyl, -CH=C(Br)-CO-O-cyclobutyl, -CH=C(Br)-CO-O-cyclopentyl, -CH=C(Br)-CO-O-cyclohexyl, -CH=C(Br)-CO-O-cycloheptyl, -CH=C(CN)-COOH, -CH=C(CN)-CO-OCH₃, -CH=C(CN)-CO-OC₂H₅, -CH=C(CN)-CO-O-n-C₃H₇, -CH=C(CN)-CO-O-i-C₃H₇, -CH=C(CN)-CO-O-n-C₄H₉, -CH=C(CN)-CO-O-tert.-C₄H₉, -CH=C(CN)-CO-O-cyclopropyl, -CH=C(CN)-CO-O-cyclobutyl, -CH=C(CN)-CO-O-cyclopentyl, -CH=C(CN)-CO-O-cyclohexyl, -CH=C(CN)-CO-O-cycloheptyl, -CH=CH-CO-OCH₂-OCH₃, -CH=CH-CO-OCH₂-OC₂H₅, -CH=CH-CO-OCH₂-O-n-C₃H₅, -CH=CH-CO-OCH₂-O-i-C₃H₅, -CH=CH-CO-OCH(CH₃)-OCH₃, -CH=CH-CO-OCH(CH₃)-OC₂H₅, -CH=CH-CO-O-CH₂CH₂-OCH₃, -CH=CH-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-OCH₃, -CH=C(CH₃)-CO-OCH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-O-n-C₃H₅, -CH=C(CH₃)-CO-OCH₂-O-i-C₃H₅, -CH=C(CH₃)-CO-OCH(CH₃)-OCH₃, -CH=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CH₃)-CO-O-CH₂CH₂-OCH₃, -CH=C(CH₃)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-OCH₃, -CH=C(C₂H₅)-CO-OCH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-O-n-C₃H₅, -CH=C(C₂H₅)-CO-OCH₂-O-i-C₃H₅, -CH=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-OCH₃, -CH=C(Cl)-CO-OCH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-O-n-C₃H₅, -CH=C(Cl)-CO-OCH₂-O-i-C₃H₅, -CH=C(Cl)-CO-OCH(CH₃)-OCH₃, -CH=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Cl)-CO-O-CH₂CH₂-OCH₃, -CH=C(Cl)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-OCH₃, -CH=C(Br)-CO-OCH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-O-n-C₃H₅, -CH=C(Br)-CO-OCH₂-O-i-C₃H₅, -CH=C(Br)-CO-OCH(CH₃)-OCH₃, -CH=C(Br)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Br)-CO-O-CH₂CH₂-OCH₃, -CH=C(Br)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-OCH₃, -CH=C(CN)-CO-OCH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-O-n-C₃H₅, -CH=C(CN)-CO-OCH₂-O-i-C₃H₅, -CH=C(CN)-CO-OCH(CH₃)-OCH₃, -CH=C(CN)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CN)-CO-O-CH₂CH₂-OCH₃, -CH=C(CN)-CO-O-CH₂CH₂-OC₂H₅, -CH=CH-CO-OCH₂-CF₃, -CH=CH-CO-OCH₂-CCl₃, -CH=CH-CO-OCH₂-oxiranyl, -CH=CH-CO-O(CH₂)₃-Br, -CH=CH-CO-OCH₂-CH=CH₂, -CH=CH-CO-OCH₂-C≡CH, -CH=CH-CO-OCH₂-CN, -CH=CH-CO-O(CH₂)₂-CN, -CH=C(CH₃)-CO-OCH₂-CF₃, -CH=C(CH₃)-CO-OCH₂-CCl₃, -CH=C(CH₃)-CO-OCH₂-oxiranyl, -CH=C(CH₃)-CO-O(CH₂)₃-Br, -CH=C(CH₃)-CO-OCH₂-CH=CH₂, -CH=C(CH₃)-CO-OCH₂-C≡CH, -CH=C(CH₃)-CO-OCH₂-CN, -CH=C(CH₃)-CO-O(CH₂)₂-CN, -CH=C(C₂H₅)-CO-OCH₂-CF₃, -CH=C(C₂H₅)-CO-OCH₂-CCl₃, -CH=C(C₂H₅)-CO-OCH₂-oxiranyl, -CH=C(C₂H₅)-CO-O(CH₂)₃-Br, -CH=C(C₂H₅)-CO-OCH₂-CH=CH₂, -CH=C(C₂H₅)-CO-OCH₂-C≡CH, -CH=C(C₂H₅)-CO-OCH₂-CN, -CH=C(C₂H₅)-CO-O(CH₂)₂-CN, -CH=C(Cl)-CO-OCH₂-CF₃, -CH=C(Cl)-CO-OCH₂-CCl₃, -CH=C(Cl)-CO-OCH₂-oxiranyl, -CH=C(Cl)-CO-O(CH₂)₃-Br, -CH=C(Cl)-CO-OCH₂-CH=CH₂, -CH=C(Cl)-CO-OCH₂-C≡CH, -CH=C(Cl)-CO-OCH₂-CN, -CH=C(Cl)-CO-O(CH₂)₂-CN, -CH=C(Br)-CO-OCH₂-CF₃, -CH=C(Br)-CO-OCH₂-CCl₃, -CH=C(Br)-CO-OCH₂-oxiranyl, -CH=C(Br)-CO-O(CH₂)₃-Br, -CH=C(Br)-CO-OCH₂-CH=CH₂, -CH=C(Br)-CO-OCH₂-C≡CH, -CH=C(Br)-CO-OCH₂-CN, -CH=C(Br)-CO-O(CH₂)₂-CN, -CH=C(CN)-CO-OCH₂-CF₃, -CH=C(CN)-CO-OCH₂-CCl₃, -CH=C(CN)-CO-OCH₂-oxiranyl, -CH=C(CN)-CO-O(CH₂)₃-Br, -CH=C(CN)-CO-OCH₂-CH-CH₂, -CH=C(CN)-CO-OCH₂-C≡CH, -CH=C(CN)-CO-OCH₂-CN, -CH=C(CN)-CO-O(CH₂)₂-CN, -CH=CH-CO-CH₃, -CH=CH-CO-C₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-i-C₃H₇, -CH=CH-CO-n-C₄H₉, -CH=CH-CO-tert.-C₄H₉, -CH=CH-CO-CH₂Cl, -CH=CH-CO-CH₂Br, -CH=CH-CO-CHCl₂, -CH=CH-CO-CH₂-OCH₃, -CH=CH-CO-CH(OCH₃)₂, -CH=CH-CO-CH₂-SCH₃, -CH=C(CH₃)-CO-CH₃, -CH=C(CH₃)-CO-C₂H₅, -CH=C(CH₃)-CO-n-C₃H₇, -CH=C(CH₃)-CO-i-C₃H₇, -CH=C(CH₃)-CO-n-C₄H₉, -CH=C(CH₃)-CO-tert.-C₄H₉, -CH=C(CH₃)-CO-CH₂Cl, -CH=C(CH₃)-CO-CH₂Br, -CH=C(CH₃)-CO-CHCl₂, -CH=C(CH₃)-CO-CH₂-OCH₃, -CH=C(CH₃)-CO-CH(OCH₃)₂, -CH=C(CH₃)-CO-CH₂-SCH₃, -CH=C(C₂H₅)-CO-CH₃, -CH=C(C₂H₅)-CO-C₂H₅, -CH=C(C₂H₅)-CO-n-C₃H₇, -CH=C(C₂H₅)-CO-i-C₃H₇, -CH=C(C₂H₅)-CO-n-C₄H₉, -CH=C(C₂H₅)-CO-tert.-C₄H₉, -CH=C(C₂H₅)-CO-CH₂Cl, -CH=C(C₂H₅)-CO-CH₂Br, -CH=C(C₂H₅)-CO-CHCl₂, -CH=C(C₂H₅)-CO-CH₂-OCH₃, -CH=C(C₂H₅)-CO-CH(OCH₃)₂, -CH=C(C₂H₅)-CO-CH₂-SCH₃, -CH=C(Cl)-CO-CH₃, -CH=C(Cl)-CO-C₂H₅, -CH=C(Cl)-CO-n-C₃H₇, -CH=C(Cl)-CO-i-C₃H₇, -CH=C(Cl)-CO-n-C₄H₉, -CH=C(Cl)-CO-tert.-C₄H₉, -CH=C(Cl)-CO-CH₂Cl, -CH=C(Cl)-CO-CH₂Br, -CH=C(Cl)-CO-CHCl₂, -CH=C(Cl)-CO-CH₂-OCH₃, -CH=C(Cl)-CO-CH(OCH₃)₂, -CH=C(Cl)-CO-CH₂-SCH₃, -CH=C(Br)-CO-CH₃, -CH=C(Br)-CO-C₂H₅, -CH=C(Br)-CO-n-C₃H₇, -CH=C(Br)-CO-i-C₃H₇, -CH=C(Br)-CO-n-C₄H₉, -CH=C(Br)-CO-tert.-C₄H₉, -CH=C(Br)-CO-CH₂Cl, -CH=C(Br)-CO-CH₂Br, -CH=C(Br)-CO-CHCl₂, -CH=C(Br)-CO-CH₂-OCH₃, -CH=C(Br)-CO-CH(OCH₃)₂, -CH=C(Br)-CO-CH₂-SCH₃, -CH=C(CN)-CO-CH₃, -CH=C(CN)-CO-C₂H₅, -CH=C(CN)-CO-n-C₃H₇, -CH=C(CN)-CO-i-C₃H₇, -CH=C(CN)-CO-n-C₄H₉, -CH=C(CN)-CO-tert.-C₄H₉, -CH=C(CN)-CO-CH₂Cl, -CH=C(CN)-CO-CH₂Br, -CH=C(CN)-CO-CHCl₂, -CH=C(CN)-CO-CH₂-OCH₃, -CH=C(CN)-CO-CH(OCH₃)₂, -CH=C(CN)-CO-CH₂-SCH₃, -CH=CH-CO-C₆H₅, -CH=CH-CO-(4-Cl-C₆H₄), -CH=C(CH₃)-CO-C₆H₅, -CH=C(CH₃)-CO-(4-Cl-C₆H₄), -CH=C(C₂H₅)-CO-C₆H₅, -CH=C(C₂H₅)-CO-(4-Cl-C₆H₄), -CH=C(Cl)-CO-C₆H₅, -CH=C(Br)-CO-C₆H₅, -CH=C(CN)-CO-C₆H₅, -CH=CH-CO-NH₂, -CH=CH-CO-NHCH₃, -CH=CH-CO-N(CH₃)₂, -CH=CH-CO-NH-C₂H₅, -CH=CH-CO-N(C₂H₅)₂, -CH=CH-CO-NH-n-C₃H₇, -CH=CH-CO-NH-i-C₃H₇, -CH=CH-CO-NH-tert.-C₄H₉, -CH=CH-CO-NH-cyclopropyl, -CH=CH-CO-NH-cyclobutyl, -CH=CH-CO-NH-cyclopentyl, -CH=CH-CO-NH-cyclohexyl, -CH=CH-CO-NH-cycloheptyl, -CH=CH-CO-NH-cyclooctyl, -CH=CH-CO-pyrrolidin-1-yl, -CH=CH-CO-piperidin-1-yl, -CH=CH-CO-morpholin-4-yl, -CH=CH-CO-NH-CH₂CH=CH₂, -CH=CH-CO-NH-CH₂C≡CH, -CH=CH-CO-N(CH₃)-CH₂C≡CH, -CH=CH-CO-NH-(CH₂)₂Cl, -CH=CH-CO-NH-C₆H₅, -CH=C(CH₃)-CO-NH₂, -CH=C(CH₃)-CO-NHCH₃, -CH=C(CH₃)-CO-N(CH₃)₂, -CH=C(CH₃)-CO-NH-C₂H₅, -CH=C(CH₃)-CO-N(C₂H₅)₂, -CH=C(CH₃)-CO-NH-n-C₃H₇, -CH=C(CH₃)-CO-NH-i-C₃H₇, -CH=C(CH₃)-CO-NH-tert.-C₄H₉, -CH=C(CH₃)-CO-NH-cyclopropyl, -CH=C(CH₃)-CO-NH-cyclobutyl, -CH=C(CH₃)-CO-NH-cyclopentyl, -CH=C(CH₃)-CO-NH-cyclohexyl, -CH=C(CH₃)-CO-NH-cycloheptyl, -CH=C(CH₃)-CO-NH-cyclooctyl, -CH=C(CH₃)-CO-pyyrolidin-1-yl, -CH=C(CH₃)-CO-piperidin-1-yl, -CH=C(CH₃)-CO-morpholin-4-yl, -CH=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -CH=C(CH₃)-CO-NH-CH₂C≡CH, -CH=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CH₃)-CO-NH-(CH₂)₂Cl, -CH=C(CH₃)-CO-NH-C₆H₅, -CH=C(C₂H₅)-CO-NH₂, -CH=C(C₂H₅)-CO-NHCH₃, -CH=C(C₂H₅)-CO-N(CH₃)₂, -CH=C(C₂H₅)-CO-NH-C₂H₅, -CH=C(C₂H₅)-CO-N(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-n-C₃H₇, -CH=C(C₂H₅)-CO-NH-i-C₃H₇, -CH=C(C₂H₅)-CO-NH-tert.-C₄H₉, -CH=C(C₂H₅)-CO-NH-cyclopropyl, -CH=C(C₂H₅)-CO-NH-cyclobutyl, -CH=C(C₂H₅)-CO-NH-cyclopentyl, -CH=C(C₂H₅)-CO-NH-cyclohexyl, -CH=C(C₂H₅)-CO-NH-cycloheptyl, -CH=C(C₂H₅)-CO-NH-cyclooctyl, -CH=C(C₂H₅)-CO-pyrrolidin-1-yl, -CH=C(C₂H₅)-CO-piperidin-1-yl, -CH=C(C₂H₅)-CO-morpholin-4-yl, -CH=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-CH₂C≡CH, -CH=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -CH=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -CH=C(C₂H₅)-CO-NH-C₆H₅, -CH=C(Cl)-CO-NH₂, -CH=C(Cl)-CO-NHCH₃, -CH=C(Cl)-CO-N(CH₃)₂, -CH=C(Cl)-CO-NH-C₂H₅, -CH=C(Cl)-CO-N(C₂H₅)₂, -CH=C(Cl)-CO-NH-n-C₃H₇, -CH=C(Cl)-CO-NH-i-C₃H₇, -CH=C(Cl)-CO-NH-tert.-C₄H₉, -CH=C(Cl)-CO-NH-cyclopropyl, -CH=C(Cl)-CO-NH-cyclobutyl, -CH=C(Cl)-CO-NH-cyclopentyl, -CH=C(Cl)-CO-NH-cyclohexyl, -CH=C(Cl)-CO-NH-cycloheptyl, -CH=C(Cl)-CO-NH-cyclooctyl, -CH=C(Cl)-CO-pyrrolidin-1-yl, -CH=C(Cl)-CO-piperidin-1-yl, -CH=C(Cl)-CO-morpholin-4-yl, -CH=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -CH=C(Cl)-CO-NH-CH₂C≡CH, -CH=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Cl)-CO-NH-(CH₂)₂Cl, -CH=C(Cl)-CO-NH-C₆H₅, -CH=C(Br)-CO-NH₂, -CH=C(Br)-CO-NHCH₃, -CH=C(Br)-CO-N(CH₃)₂, -CH=C(Br)-CO-NH-C₂H₅, -CH=C(Br)-CO-N(C₂H₅)₂, -CH=C(Br)-CO-NH-n-C₃H₇, -CH=C(Br)-CO-NH-i-C₃H₇, -CH=C(Br)-CO-NH-tert.-C₄H₉, -CH=C(Br)-CO-NH-cyclopropyl, -CH=C(Br)-CO-NH-cyclobutyl, -CH=C(Br)-CO-NH-cyclopentyl, -CH=C(Br)-CO-NH-cyclohexyl, -CH=C(Br)-CO-NH-cycloheptyl, -CH=C(Br)-CO-NH-cyclooctyl, -CH=C(Br)-CO-pyrrolidin-1-yl, -CH=C(Br)-CO-piperidin-1-yl, -CH=C(Br)-CO-morpholin-4-yl, -CH=C(Br)-CO-NH-CH₂CH=C(Br)₂, -CH=C(Br)-CO-NH-CH₂C≡CH, -CH=C(Br)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Br)-CO-NH-(CH₂)₂Cl, -CH=C(Br)-CO-NH-C₆H₅, -CH=C(CN)-CO-NH₂, -CH=C(CN)-CO-NHCH₃, -CH=C(CN)-CO-N(CH₃)₂, -CH=C(CN)-CO-NH-C₂H₅, -CH=C(CN)-CO-N(C₂H₅)₂, -CH=C(CN)-CO-NH-n-C₃H₇, -CH=C(CN)-CO-NH-i-C₃H₇, -CH=C(CN)-CO-NH-tert.-C₄H₉, -CH=C(CN)-CO-NH-cyclopropyl, -CH=C(CN)-CO-NH-cyclobutyl, -CH=C(CN)-CO-NH-cyclopentyl, -CH=C(CN)-CO-NH-cyclohexyl, -CH=C(CN)-CO-NH-cycloheptyl, -CH=C(CN)-CO-NH-cyclooctyl, -CH=C(CN)-CO-pyrrolidin-1-yl, -CH=C(CN)-CO-piperidin-1-yl, -CH=C(CN)-CO-morpholin-4-yl, -CH=C(CN)-CO-NH-CH₂CH=C(CN)₂, -CH=C(CN)-CO-NH-CH₂C≡CH, -CH=C(CN)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CN)-CO-NH-(CH₂)₂Cl, -CH=C(CN)-CO-NH-C₆H₅, -CH=CH-CO-SCH₃, -CH=CH-CO-SC₂H₅, -CH=CH-CO-S-n-C₃H₇, -CH=CH-CO-S-i-C₃H₇, -CH=CH-CO-S-n-C₄H₉, -CH=CH-CO-S-tert.-C₄H₉, -CH=C(CH₃)-CO-SCH₃, -CH=C(CH₃)-CO-SC₂H₅, -CH=C(CH₃)-CO-S-n-C₃H₇, -CH=C(CH₃)-CO-S-i-C₃H₇, -CH=C(CH₃)-CO-S-n-C₄H₉, -CH=C(CH₃)-CO-S-tert.-C₄H₉, -CH=C(C₂H₅)-CO-SCH₃, -CH=C(C₂H₅)-CO-SC₂H₅, -CH=C(C₂H₅)-CO-S-n-C₃H₇, -CH=C(C₂H₅)-CO-S-i-C₃H₇, -CH=C(C₂H₅)-CO-S-n-C₄H₉, -CH=C(C₂H₅)-CO-S-tert.-C₄H₉, -CH=C(Cl)-CO-SCH₃, -CH=C(Cl)-CO-SC₂H₅, -CH=C(Cl)-CO-S-n-C₃H₇, -CH=C(Cl)-CO-S-i-C₃H₇, -CH=C(Cl)-CO-S-n-C₄H₉, -CH=C(Cl)-CO-S-tert.-C₄H₉, -CH=C(Br)-CO-SCH₃, -CH=C(Br)-CO-SC₂H₅, -CH=C(Br)-CO-S-n-C₃H₇, -CH=C(Br)-CO-S-i-C₃H₇, -CH=C(Br)-CO-S-n-C₄H₉, -CH=C(Br)-CO-S-tert.-C₄H₉, -CH=C(CN)-CO-SCH₃, -CH=C(CN)-CO-SC₂H₅, -CH=C(CN)-CO-S-n-C₃H₇, -CH=C(CN)-CO-S-i-C₃H₇, -CH=C(CN)-CO-S-n-C₄H₉, -CH=C(CN)-CO-S-tert.-C₄H₉, -CH=C(COCH₃)-CO-OCH₃, -CH=C(COC₂H₅)-CO-OCH₃, -CH=C(CO-n-C₃H₇)-CO-OCH₃, -CH=C(COCH₃)-CO-OC₂H₅, -CH=C(COC₂H₅)-CO-OC₂H₅, -CH=C(CO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COCH₃)-CO-O-n-C₃H₇, -CH=C(COC₂H₅)-CO-O-n-C₃H₇, -CH=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-OCH₃, -CH=C(CF₃)-CO-OC₂H₅, -CH=C(CF₃)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-O-i-C₃H₇, -CH=C(CF₃)-CO-O-n-C₄H₉, -CH=C(CF₃)-CO-O-tert.-C₄H₉, -CH=C(COOCH₃)₂, -CH=C(COOC₂H₅)₂, -CH=C(COOCH₃)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)-CO-OCH₃, -CH=C(COO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)₂, -CH=CH-CH=CH-COOH, -CH=CH-CH=CH-CO-OCH₃, -CH=CH-CH=CH-CO-OC₂H₅, -CH=CH-CH=C(COOCH₃)₂, -CH=CH-CH=C(CN)-CO-OCH₃, -CH=CH-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-OCH₃, -CH=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CH=C(Cl)-CO-OCH₃, -CH=C(CH₃)-CH=C(Br)-CO-OCH₃, -CH=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-NH₂, -CH=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -CH=CH-(CH₂)₂-COOH, -CH=CH-(CH₂)₂-CO-OCH₃, -CH=CH-(CH₂)₂-CO-OC₂H₅, -CH=CH-CH₂-CH(COOCH₃)₂, -CH=CH-CH₂-CH(COOC₂H₅)₂, -CH=CH-CH₂-CH(CN)-CO-OCH₃, -CH=CH-CH₂-CH(CN)-CO-OC₂H₅, -CH=CH-CH₂-CH(CH₃)-CO-OCH₃, -CH=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -CH=CH-(CH₂)₂-CO-NH₂, -CH=CH-(CH₂)₂-CO-NH-CH₃, -CH=CH-CH₂-COOH, -CH=CH-CH₂-CO-OCH₃, -CH=CH-CH₂-CO-OC₂H₅, -CH=C(COOCH₃)-CH₂-CO-OCH₃, -CH=C(COOCH₃)-CH₂-CO-OC₂H₅, -CH=CH-CH₂-CO-NH₂, -CH=CH-CH₂-CO-NH-CH₃, -CH=CH-CH₂-CO-N(CH₃)₂, -CH(OCH₃)₂, -CH(SCH₃)₂, -CH(OC₂H₅)₂, -CH(SC₂H₅)₂, -CH(O-n-C₃H₇)₂, -CH(O-i-C₃H₇)₂, -CH(S-n-C₃H₇)₂, -CH(S-i-C₃H₇)₂, -CH(O-n-C₄H₉)₂, -CH(O-i-C₄H₉)₂, -CH(O-s-C₄H₉)₂, -CH(O-tert.-C₄H₉)₂, -CH(S-n-C₄H₉)₂, -CH(S-i-C₄H₉)₂, -CH(S-s-C₄H₉)₂, -CH(S-tert.-C₄H₉)₂, -CH(OC₅H₁₁)₂, 1,3-Dioxolan-2-yl, 1,3-Dithio­ lan-2-yl, 1,3-Oxathiolan-2-yl, 4-Methyl-1,3-dioxolan-2-yl, 4-Methyl-1,3-dithiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 5-Methyl-1,3-oxathiolan-2-yl, 4-Ethyl-1,3-dioxolan-2-yl, 4-Ethyl- 1,4-dithiolan-2-yl, 4-Ethyl-1,3-oxathiolan-2-yl, 5-Ethyl-1,3-oxa­ thiolan-2-yl, 4,5-Dimethyl-1,3-dioxolan-2-yl, 4,4-Dimethyl-1,3- dioxolan-2-yl, 4,5-Dimethyl-1,3-dithiolan-2-yl, 5,5-Dimethyl-1,3- dithiolan-2-yl, 4,5-Dimethyl-1,3-oxathiolan-2-yl, 5,5-Dimethyl- 1,3-oxathiolan-2-yl, 4,4-Dimethyl-1,3-oxathiolan-2-yl, 4-Vinyl- 1,3-dioxolan-2-yl, 4-Vinyl-1,3-dithiolan-2-yl, 4-Vinyl-1,3-oxa­ thiolan-2-yl, 5-Vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3- dioxolan-2-yl, 4-Chlormethyl-1,3-dithiolan-2-yl, 4-Chlormethyl- 1,3-oxathiolan-2-yl, 5-Chlormethyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-1,3-dithio­ lan-2-yl, 4-Hydroxymethyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl- 1,3-oxathiolan-2-yl, 4-Methoxymethyl-1,3-dioxolan-2-yl, 4-Allyl­ oxymethyl-1,3-dioxolan-2-yl, 4-Propargyloxymethyl-1,3-dioxolan- 2-yl, 4-Acetoxymethyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-1,3-dithiolan-2-yl, 4-Propargyl­ oxymethyl-1,3-dithiolan-2-yl, 4-Acetoxymethyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl-1,3-oxathiolan-2-yl, 5-Allyloxy- methyl-1,3-oxathiolan-2-yl, 4-Propargyloxymethyl-1,3-oxathiolan-2-yl, 5-Propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxymethyl- 1,3-oxathiolan-2-yl, 5-Acetoxymethyl-1,3-oxathiolan-2-yl, 4-Methylthiomethyl-1,3-dioxolan-2-yl, 4-Methylthiomethyl-1,3- dithiolan-2-yl, 4-Carboxy-1,3-dioxolan-2-yl, 4-Carboxy-1,3- dithiolan-2-yl, 4-Methoxycarbonyl-1,3-dioxolan-2-yl, 4-Ethoxy- carbonyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-1,3-dithiolan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-4-methyl- 1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-di­ thiolan-2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-1,3- dithiolan-2-yl, 1,3-Dioxan-2-yl, 1,3-Dithian-2-yl, 1,3-Oxathian- 2-yl, 5-Methyl-1,3-dioxan-2-yl, 5-Methyl-1,3-dithian-2-yl, 5-Methyl-1,3-oxathian-2-yl, 5,5-Dimethyl-1,3-dioxan-2-yl, 4,6-Dimethyl- 1,3-dioxan-2-yl, 4,4-Dimethyl-1,3-dioxan-2-yl, 5,5-Dimethyl- 1,3-dithian-2-yl, 4,6-Dimethyl-1,3-dithian-2-yl, 4,4-Dimethyl- 1,3-dithian-2-yl, 5,5-Dimethyl-1,3-oxathian-2-yl, 4,4-Dimethyl- 1,3-oxathian-2-yl, 6,6-Dimethyl-1,3-oxathian-2-yl, 4-Hydroxymethyl-1,3-dioxan-2-yl, 4-Methoxymethyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-1,3-dithian-2-yl, 4-Methoxymethyl-1,3-dithian-2-yl, 4-Allyloxymethyl-1,3-dithian-2-yl, 4-Acetoxymethyl- 1,3-dithian-2-yl, 4-Chlormethyl-1,3-dioxan-2-yl, 4-Chlormethyl- 1,3-dithian-2-yl, 1,3-Dioxepan-2-yl, 1,3-Dithiepan-2-yl, 1,3-Dioxep-5-en-2-yl, 4-Methoxycarbonyl-1,3-dioxan-2-yl, 4-Ethoxy- carbonyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-1,3-dithian-2-yl, 4-n-Butoxycarbonyl-1,3-dithian-2-yl, 4-Methoxycarbonyl-4- methyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-Methoxy- carbonyl-4-methyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-4-methyl- 1,3-dithian-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithian-2-yl, -C(CH₃)(OCH₃)₂, -C(CH₃)(SCH₃)₂, -C(CH₃)(OC₂H₅)₂, -C(CH₃)(SC₂H₅)₂, -C(CH₃)(O-n-C₃H₇)₂, -C(CH₃)(O-i-C₃H₇)₂, -C(CH₃)(S-n-C₃H₇)₂, -C(CH₃)(S-i-C₃H₇)₂, -C(CH₃)(O-n-C₄H₉)₂, -C(CH₃)(O-i-C₄H₉)₂, -C(CH₃)(O-s-C₄H₉)₂, -C(CH₃)(O-tert.-C₄H₉)₂, -C(CH₃)(S-n-C₄H₉)₂, -C(CH₃)(S-i-C₄H₉)₂, -C(CH₃)(S-s-C₄H₉)₂, -C(CH₃)(S-tert.-C₄H₉)₂, -C(CH₃)(O-n-C₅H₁₁)′′, 2-Methyl-1,3-dioxolan-2-yl, 2-Methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-oxathiolan-2-yl, 2,4-Dimethyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-1,3- oxathiolan-2-yl, 2,5-Dimethyl-1,3-oxathiolan-2-yl, 4-Ethyl-2- methyl-1,3-dioxolan-2-yl, 4-Ethyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Ethyl-2-methyl-1,3- oxathiolan-2-yl, 2,4,5-Trimethyl-1,3-dioxolan-2-yl, 2,4,4-Trimethyl- 1,3-dioxolan-2-yl, 2,4,5-Trimethyl-1,3-dithiolan-2-yl, 2,4,4-Trimethyl-1,3-dithiolan-2-yl, 2,4,5-Trimethyl-1,3-oxathiolan-2-yl, 2,4,4-Trimethyl-1,3-oxathiolan-2-yl, 2-Methyl-4-vinyl- 1,3-dioxolan-2-yl, 2-Methyl-4-vinyl-1,3-dithiolan-2-yl, 2-Methyl- 4-vinyl-1,3-oxathiolan-2-yl, 2-Methyl-5-vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-dioxolan-2-yl, 4-Chlormethyl-2- methyl-1,3-dithiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl- 2-methyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dioxolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxy- 2-methyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dithiolan-2-yl, 4-Acetoxy-2- methyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl- 2-methyl-1,3-oxathiolan-2-yl, 5-Allyloxymethyl-2-methyl-1,3-oxathiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3- oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxy-2-methyl-1,3-oxathiolan-2-yl, 5-Acetoxy-2-methyl- 1,3-oxathiolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dioxolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-2- methyl-1,3-dioxolan-2-yl, 4-Carboxy-2-methyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-2- methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl- 2-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-2- methyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-ethoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4- ethoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-n-butoxy- carbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl-1,3- dithiolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-dioxan-2-yl, 2-Methyl-1,3-dithian-2-yl, 2-Methyl-1,3-oxathian-2-yl, 2,5- Dimethyl-1,3-dioxan-2-yl, 2,5-Dimethyl-1,3-dithian-2-yl, 2,5-Dimethyl- 1,3-oxathian-2-yl, 2,5,5-Trimethyl-1,3-dioxan-2-yl, 2,4,6- Trimethyl-1,3-dioxan-2-yl, 2,4,4-Trimethyl-1,3-dioxan-2-yl, 2,5,5-Trimethyl-1,3-dithian-2-yl, 2,4,6-Trimethyl-1,3-dithian-2-yl, 2,4,4-Trimethyl-1,3-dithian-2-yl, 2,5,5-Trimethyl-1,3-oxathian-2-yl, 2,4,4-Trimethyl-1,3-oxathian-2-yl, 2,6,6-Trimethyl- 1,3-oxathian-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-2- methyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dithian-2-yl, 4-Methoxymethyl-2- methyl-1,3-dithian-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithian-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dithian-2-yl, 4-Chlormethyl-2- methyl-1,3-dioxan-2-yl, 4-Chlormethyl-2-methyl-1,3-dithian-2-yl, -C(CH₃)=NH, -C(CH₃)=N-CH₃, -C(CH₃)=N-C₂H₅, -C(CH₃)=N-n-C₃H₇, -(CH₃)=N-i-C₃H₇, -C(CH₃)=N-n-C₄H₉, -C(CH₃)=N-CH₂CH=CH₂, -C(CH₃)=N-CH₂CH=CH₂-CH₃, -C(CH₃)=N-CH₂C≡CH, -C(CH₃)=N-CH₂C≡C-CH₃, -C(CH₃)=N-cyclopropyl, -C(CH₃)=N-cyclobutyl, -C(CH₃)=N-cyclopentyl, -C(CH₃)=N-cyclohexyl, -C(CH₃)=N-cycloheptyl, -C(CH₃)=N-CH₂-CH₂Cl, -C(CH₃)=N-CH₂Cl, -C(CH₃)=N-C₆H₅, -C(CH₃)=N-(2-F-C₆H₄), -C(CH₃)=N-(3-F-C₆H₄), -C(CH₃)=N-(4-F-C₆H₄), -C(CH₃)=N-(2-Cl-C₆H₄), -C(CH₃)=N-(3-Cl-C₆H₄), -C(CH₃)=N-(4-Cl-C₆H₄), -C(CH₃)=N-(2-CH₃-C₆H₄), -C(CH₃)=N-(3-CH₃-C₆H₄), -C(CH₃)=N-(4-CH₃-C₆H₄), -C(CH₃)=N-(2-CF₃-C₆H₄), -C(CH₃)=N-(3-CF₃-C₆H₄), -C(CH₃)=N-(4-CF₃-C₆H₄), -C(CH₃)=N-(2-OCH₃-C₆H₄), -C(CH₃)=N-(3-OCH₃-C₆H₄), -C(CH₃)=N-(4-OCH₃-C₆H₄), -C(CH₃)=N-(4-NO₂-C₆H₄), -C(CH₃)=N-(4-CN-C₆H₄), -C(CH₃)=N-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-(2,4-(CH₃)₂-C₆H₃), -C(CH₃)=N-CH₂-OCH₃, -C(CH₃)=N-CH₂-OC₂H₅, -C(CH₃)=N-CH₂CH₂-OCH₃, -C(CH₃)=N-CH₂CH-OC₂H₅, -C(CH₃)=N-OH, -C(CH₃)=N-OCH₃, -C(CH₃)=N-OC₂H₅, -C(CH₃)=N-O-n-C₃H₇, -C(CH₃)=N-O-i-C₃H₇, -C(CH₃)=N-O-n-C₄H₉, -C(CH₃)=N-O-i-C₄H₉, -C(CH₃)=N-O-s-C₄H₉, -C(CH₃)=N-O-tert.-C₄H₉, -C(CH₃)=N-OCH₂-CH=CH₂, -C(CH₃)=N-OCH(CH₃)-CH=CH₂, -C(CH₃)=N-OCH₂-C≡CH, -C(CH₃)=N-CH(CH₃)-C≡CH, -C(CH₃)=N-OCH₂-CH=C-CH₃, -C(CH₃)=N-OCH₂CH₂-Cl, -C(CH₃)=N-OCH₂CH₂-F, -C(CH₃)=N-OCH₂-CF₃, -C(CH₃)=N-OCH₂-CH=CHCl, -C(CH₃)=N-OCH₂-C(Cl)=CH₂, -C(CH₃)=N-OCH₂-C(Br)=CH₂, -C(CH₃)=N-OCH₂-CH=C(Cl)-CH₃, -C(CH₃)=N-O-CO-CH₃, -C(CH₃)=N-O-CO-C₂H₅, -C(CH₃)=N-OCH₂-CN, -C(CH₃)=N-OCH₂-CH=CH-CH₂-OCH₃, -C(CH₃)=N-OCH₂-CH=CH-CH₂-O-tert.-C₄H₉, -C(CH₃)=N-O-(CH₂)₃-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-(4-Cl-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-C₆H₅, -C(CH₃)=N-OCH₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(3-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-CH₂-(4-CH₃O-C₆H₄), -C(CH₃)=N-OCH₂-CH=C(CH₃)-C₆H₅, -C(CH₃)=N-O-(CH₂)₂-CH=CH-(3,4-Cl₂-C₆H₃), -C(CH₃)=N-O-(CH₂)₃-C≡C-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-OCH₃, -C(CH₃)=N-OCH₂CH₂-OCH₃, -C(CH₃)=N-OCH₂-OC₂H₅, -C(CH₃)=N-OCH(CH₃)-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=N-NH₂, -C(CH₃)=N-NH-CH₃, -C(CH₃)=N-NH-C₂H₅, -C(CH₃)=N-NH-n-C₃H₇, -C(CH₃)=N-NH-i-C₃H₇, -C(CH₃)=N-NH-n-C₄H₉, -C(CH₃)=N-NH-i-C₄H₉, -C(CH₃)=N-NH-s-C₄H₉, -C(CH₃)=N-NH-tert.-C₄H₉, -C(CH₃)=N-NH-cyclopropyl, -C(CH₃)=N-NH-cyclobutyl, -C(CH₃)=N-NH-cyclopentyl, -C(CH₃)=N-NH-cyclohexyl, -C(CH₃)=N-NH-cycloheptyl, -C(CH₃)=N-N(CH₃)₂, -C(CH₃)=N-N(C₂H₅)₂, -C(CH₃)=N-N(n-C₃H₇)₂, -C(CH₃)=N-N(i-C₃H₇)₂, -C(CH₃)=N-NH-CH₂-C=CH, -C(CH₃)=N-NH-CH₂-C≡CH, -C(CH₃)=N-N(CH₃)-CH₂-C≡CH, -C(CH₃)=N-NH-CH₂CF₃, -C(CH₃)=N-NH-CO-CH₃, -C(CH₃)=N-NH-CO-C₂H₅, -C(CH₃)=N-NH-CO-OCH₃, -C(CH₃)=N-NH-CO-OC₂H₅, -C(CH₃)=N-NH-CO-O-tert.-C₄H₉, -C(CH₃)=N-pyrrolidin-1-yl, -C(CH₃)=N-piperidin-1-yl, -C(CH₃)=N-morpholin-4-yl, -C(CH₃)=N-NH-C₆H₅, -C(CH₃)=N-NH-(4-Cl-C₆H₄), -C(CH₃)=N-NH-(4-NO₂-C₆H₄), -C(CH₃)=N-NH-(4-F-C₆H₄), -C(CH₃)=N-NH-(4-CH₃O-C₆H₄), -C(CH₃)=N-NH-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-NH-(2,4-(NO₂)₂-C₆H₃), -C(CH₃)=N-NH-CO-NH₂, -C(CH₃)=N-NH-CO-NHCH₃, -C(CH₃)=N-NH-CO-NHC₂H₅, -C(CH₃)=N-NH-CO-N(CH₃)₂, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=CH-CO-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -(CH₃)=CH-CO-O-n-C₄H₉, -C(CH₃)=CH-CO-O-tert.-C₄H₉, -C(CH₃)=CH-CO-O-cyclopropyl, -C(CH₃)=CH-CO-O-cyclobutyl, -C(CH₃)=CH-CO-O-cyclopentyl, -C(CH₃)=CH-CO-O-cyclohexyl, -C(CH₃)=CH-CO-O-cycloheptyl, -C(CH₃)=C(CH₃)-COOH, -C(CH₃)=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-cyclopropyl, -C(CH₃)=C(CH₃)-CO-O-cyclobutyl, -C(CH₃)=C(CH₃)-CO-O-cyclopentyl, -C(CH₃)=C(CH₃)-CO-O-cyclohexyl, -C(CH₃)=C(CH₃)- ⁹⁹⁹⁹⁹ ⁰⁰⁰⁷⁰ ⁵⁵² ⁰⁰¹⁰⁰⁰²⁸⁰⁰⁰⁰⁰00200012000285919988800040 0002004131038 00004 99880CO-O-cycloheptyl, -C(CH₃)=C(C₂H₅)-COOH, -C(CH₃)=C(C₂H₅)-CO-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-cyclo­ propyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-O- cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-O-cycloheptyl, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-O-O-n-C₄H₉, -C(CH₃)=C(Cl)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-O-cyclopropyl, -C(CH₃)=C(Cl)-CO-O-cyclobutyl, -C(CH₃)=C(Cl)-CO-O-cyclopentyl, -C(CH₃)=C(Cl)-CO-O-cyclohexyl, -C(CH₃)=C(Cl)-CO-O-cycloheptyl, -C(CH₃)=C(Br)-COOH, -C(CH₃)=C(Br)-CO-OCH₃, -C(CH₃)=C(Br)-CO-OC₂H₅, -C(CH₃)=C(Br)-CO-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-O-n-C₄H₉, -C(CH₃)=C(Br)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-O-cyclopropyl, -C(CH₃)=C(Br)-CO-O-cyclobutyl, -C(CH₃)=C(Br)-CO-O-cyclopentyl, -C(CH₃)=C(Br)-CO-O-cyclohexyl, -C(CH₃)=C(Br)-CO-O-cycloheptyl, -C(CH₃)=C(CN)-COOH, -C(CH₃)=C(CN)-CO-OCH₃, -C(CH₃)=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CN)-CO-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-O-n-C₄H₉, -C(CH₃)=C(CN)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-O-cyclopropyl, -C(CH₃)=C(CN)-CO-O-cyclobutyl, -C(CH₃)=C(CN)-CO-O-cyclopentyl, -C(CH₃)=C(CN)-CO-O-cyclohexyl, -C(CH₃)=C(CN)-CO-O-cycloheptyl, -C(CH₃)=CH-CO-OCH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-OCH(CH₃)-OCH₃, -C(CH₃)=CH-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=CH-CO-OCH₂CH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=(C₂H₅)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-O-i-C₃H₇, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-O-i-C₃H₇, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-O-i-C₃H₇, -C(CH₃)=C(CN)-CO-OCH(CH₃)OCH₃, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-CF₃, -C(CH₃)=CH-CO-OCH₂-CCl₃, -C(CH₃)=CH-CO-OCH₂-oxiranyl, -C(CH₃)=CH-CO-(CH₂)₃-Br,-C(CH₃)=CH-CO-OCH₂-CH=CH₂, -C(CH₃)=CH-CO-OCH₂-C≡CH, -C(CH₃)=CH-CO-OCH₂-CN, -C(CH₃)=CH-CO-OCH₂CH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CF₃, -C(CH₃)=C(CH₃)-CO-OCH₂-CCl3, -C(CH₃)=C(CH₃)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CH₃)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CH₃)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CH₃)-CO-OCH₂-C≡CH, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CF₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CCl₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-oxiranyl, -C(CH₃)=C(C₂H₅)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(C₂H₅)CO-OCH₂-C≡CH, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-C₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂-CF₃, -C(CH₃)=C(Cl)-CO-OCH₂-CCl₃, -C(CH₃)=C(Cl)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Cl)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(CL)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Cl)-CO-OCH₂-C≡CH, -C(CH₃)=C(Cl)-CO-OCH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂-CF₃, -C(CH₃)=C(Br)-CO-OCH₂-CCl₃, -C(CH₃)=C(Br)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Br)-CO-O(CH₂)₃-Br, -C(CH₃)=C(Br)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Br)-CO-OCH₂-C≡CH, -C(CH₃)=C(Br)-CO-OCH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂CH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂-CF₃, -C(CH₃)=C(CN)-CO-OCH₂-CCl₃, -C(CH₃)=C(CN)-OCH₂-oxiranyl, -C(CH₃)=C(CN)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CN)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CN)-CO-OCH₂-C≡CH, -C(CH₃)=C(CN)-CO-OCH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂CH₂-CN, -C(CH₃)=CH-CO-CH₃, -C(CH₃)=CH-CO-C₂H₅, -C(CH₃)=CH-CO-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-n-C₄H₉, -C(CH₃)=CH-CO-tert.-C₄H₉, -C(CH₃)=CH-CO-CH₂Cl, -C(CH₃)=CH-CO-CH₂Br, -C(CH₃)=CH-CO-CHCl₂, -C(CH₃)=CH-CO-CH₂-OCH₃, -C(CH₃)=CH-CO-CH(OCH₃)₂, -C(CH₃)=CH-CO-CH₂-SCH₃, -C(CH₃)=C(CH₃)-CO-CH₃, -C(CH₃)=C(CH₃)-CO-C₂H₅, -C(CH₃)=C(CH₃)-CO-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-CH₂Cl, -C(CH₃)=C(CH₃)-CO-CH₂Br, -C(CH₃)=C(CH₃)-CO-CHCl₂, -C(CH₃)=C(CH₃)-CO-CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-CH(OCH₃)₂, -C(CH₃)=C(CH₃)-CO-CH₂-SCH₃, -C(CH₃)=C(C₂H₅)-CO-CH₃, -C(CH₃)=C(C₂H₅)-CO-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-CH₂Cl, -C(CH₃)=C(C₂H₅)-CO-CH₂Br, -C(CH₃)=C(C₂H₅)-CO-CHCl₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-CH(OCH₃)₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-SCH₃, -C(CH₃)=C(Cl)-CO-CH₃, -C(CH₃)=C(Cl)-CO-C₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-n-C₄H₉, -C(CH₃)=C(Cl)-CO-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-CH₂Cl, -C(CH₃)=C(Cl)-CO-CHCl₂, -C(CH₃)=C(Cl(-CO-CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-CH(OCH₃)₂, -C(CH₃)=C(Cl)-CO-CH₂-SCH₃, -C(CH₃)=C(Br)-CO-CH₃, -C(CH₃)=C(Br)-CO-C₂H₅, -C(CH₃)=C(Br)-CO-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-n-C₄H₉, -C(CH₃)=C(Br)-CO-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-CH₂Cl, -C(CH₃)=C(Br)-CO-CH₂Br, -C(CH₃)=C(Br)-CO-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-CH(OCH₃)₂, -C(CH₃)=C(Br)-CO-CH₂-SCH₃, -C(CH₃)=C(CN)-CO-CH₃, -C(CH₃)=C(CN)-CO-C₂H₅, -C(CH₃)=C(CN)-CO-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-n-C₄H₉, -C(CH₃)=C(CN)-CO-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-CH₂Cl, -C(CH₃)=C(CN)-CO-CH₂Br, -C(CH₃)=C(CN)-CO-CHCl₂, -C(CH₃)=C(CN)-CO-CH₂-OCH₃, -C(CH₃)=C(CN)-CO-CH(OCH₃)₂, -C(CH₃)=C(CN)-CO-CH₂-SCH₃, -C(CH₃)=CH-CO-C₆H₅, -C(CH₃)=CH-CO-(4-Cl-C₆H₄), -C(CH₃)=C(CH₃)-CO-C₆H₅, -C(CH₃)=C(CH₃)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(C₂H₅)-CO-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(Cl)-CO-C₆H₅, -C(CH₃)=C(Br)-CO-C₆H₅, -C(CH₃)=C(CN)-CO-C₆H₅, -C(CH₃)=CH-CO-NH₂, -C(CH₃)=CH-CO-NHCH₃, -C(CH₃)=CH-CO-N(CH₃)₂, -C(CH₃)=CH-CO-NH-C₂H₅, -C(CH₃)=CH-CO-N(C₂H₅)₂, -C(CH₃)=CH-CO-NH-n-C₃H₇, -C(CH₃)=CH-CO-NH-i-C₃H₇, -C(CH₃)=CH-CO-NH-tert.-C₄H₉, -C(CH₃)=CH-CO-NH-cyclopropyl, -C(CH₃)=CH-CO-NH-cyclobutyl, -C(CH₃)=CH-CO-NH-cyclopentyl, -C(CH₃)=CH-CO-NH-cylohexyl, -C(CH₃)=CH-CO-NH-cycloheptyl, -C(CH₃)=CH-CO-NH-cyclooctyl, -C(CH₃)=CH-CO-pyrrolidin-1-yl, -C(CH₃)=CH-CO-piperidin-1-yl, -C(CH₃)=CH-CO-morpholin-4-yl, -C(CH₃)=CH-CO-NH-CH₂CH=CH₂, -C(CH₃)=CH-CO-NH-CH₂C≡CH, -C(CH₃)=CH-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=CH-CO-NH-(CH₂)₂Cl, -C(CH₃)=CH-CO-NH-C₆H₅, -C(CH₃)=C(CH₃)-CO-NH₂, -C(CH₃)=C(CH₃)-CO-NHCH₃, -C(CH₃)=C(CH₃)-CO-N(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-C₂H₅, -C(CH₃)=C(CH₃)-CO-N(C₂H₅)₂, -C(CH₃)=C(CH₃)-CO-NH-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-NH- cyclopropyl, -C(CH₃)=C(CH₃)-CO-NH-cyclobutyl, -C(CH₃)=C(CH₃)-CO-NH-cyclopentyl, -C(CH₃)=C(CH₃)-CO-NH- cyclohexyl, -C(CH₃)=C(CH₃)-CO-NH-cycloheptyl, -C(CH₃)=C(CH₃)-CO-NH-cyclooctyl, -C(CH₃)=C(CH₃)-CO- pyrrolidin-1-yl, -C(CH₃)=C(CH₃)-CO-piperidin-1-yl, -C(CH₃)=C(CH₃)-CO-morpholin-4-yl, -C(CH₃)=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-NH(CH₂)₂Cl, -C(CH₃)=C(CH₃)-CO-NH-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-NH₂, -C(CH₃)=C(C₂H₅)-CO-NHCH₃, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)₂, -C(CH₃)=C(C₂H₅)-CO-NH-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-N(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-NH- cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclo­ hexyl, -C(CH₃)=C(C₂H₅)-CO-NH-cycloheptyl, -C(CH₃)=C(C₂H₅)-CO-NH- cyclooctyl, -C(CH₃)=C(C₂H₅)-CO-pyrrolidin-1-yl, -C(CH₃)=C(C₂H₅)-CO-piperidin-1-yl, -C(CH₃)=C(C₂H₅)-CO- morpholin-4-yl, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(C₂H₅)-CO-NH-C₆H₅, -C(CH₃)=C(Cl)-CO-NH₂, -C(CH₃)=C(CH₃)=C(Cl)-CO-NHCH₃, -C(CH₃)=C(Cl)-CO-N(CH₃)₂, -C(CH₃)=C(Cl)-CO-NH-C₂H₅, -C(CH₃)=C(Cl)-CO-N(C₂H₅)₂, -C(CH₃)=C(Cl)-CO-NH-n-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-i-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-NH-cyclopropyl, -C(CH₃)=C(Cl)-CO-NH-cyclobutyl, -C(CH₃)=C(Cl)-CO-NH-cyclopentyl, -C(CH₃)=C(Cl)-CO-NH-cyclohexyl, -C(CH₃)=C(Cl)-CO-NH-cycloheptyl, -C(CH₃)=C(Cl)-CO-NH-cyclooctyl, -C(CH₃)=C(Cl)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Cl)-CO-piperidin-1- yl, -C(CH₃)=C(Cl)-CO-morpholin-4-yl, -C(CH₃)=C(Cl)-CO-NH-CH₂CH=C(Cl)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-N(CH₃)-CH₂≡CH, -C(CH₃)=C(Cl)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Cl)-NO-NH-C₆H₅, -C(CH₃)=C(Br)-CO-NH₂, -C(CH₃)=C(Br)-CO-NHCH₃, -C(CH₃)=C(Br)-CO-N(CH₃)₂, -C(CH₃)=C(Br)-CO-NH-C₂H₅, -C(CH₃)=C(Br)-CO-N(C₂H₅)₂, -C(CH₃)=C(Br)-CO-NH-n-C₃H₇, -C(CH₃)=C(Br)-CO-NH-i-C₃H₇, -C(CH₃)=C(Br)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-NH-cyclopropyl, -C(CH₃)=C(Br)-CO-NH-cyclobutyl, -C(CH₃)=C(Br)-CO-NH-cyclopentyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cycloheptyl, -C(CH₃)=C(Br)-CO-NH-cyclooctyl, -C(CH₃)=C(Br)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Br)-CO-piperidin-1-yl, -C(CH₃)=C(Br)-CO-morpholin-4-yl, -C(CH₃)=C(Br)-CO-NH-CH₂CH=C(CH₃)=C(Br)-CO-NH-CH₂C≡CH, -C(CH₃)=C(BR)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Br)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Br)-CO-NH-C₆H₅, -C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CN)-CO-NHCH₃, -C(CH₃)=C(CN)-CO-N(CH₃)₂, -C(CH₃)=C(CN)-CO-NH-C₂H₅, -C(CH₃)=C(CN)-CO-N(C₂H₅)₂, -C(CH₃)=C(CN)-CO-NH-n-C₃H₇, -C(CH₃)=C(CN)-CO-NH-i-C₃H₇, -C(CH₃)=C(CN)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-NH-cyclopropyl, -C(CH₃)=C(CN)-CO-NH-cyclobutyl, -C(CH₃)=C(CN)-CO-NH-cyclopentyl, -C(CH₃)=C(CN)-CO-NH-cyclohexyl, -C(CH₃)=C(CN)-CO-NH-cycloheptyl, -C(CH₃)=C(CN)-CO-NH-cyclooctyl, -C(CH₃)=C(CN)-CO-pyrrolidin-1-yl, -C(CH₃)=C(CN)-CO-piperidin-1-yl, -C(CH₃)=C(CN)-CO-morpholin-4-yl, -C(CH₃)=C(CN)-CO-NH-CH₂CH=C(CN)₂, -C(CH₃)=C(CN)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CN)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)=(CN)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CN)-CO-NH-C₆H₅, -C(CH₃)=CH-SO-SCH₃, -C(CH₃)=CH-CO-SC₂H₅, -C(CH₃)=CH-CO-S-n-C₃H₇, -C(CH₃)=CH-CO-S-i-C₃H₇, -C(CH₃)=CH-CO-S-n-C₄H₉, -C(CH₃)=CH-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-SCH₃, -C(CH₃)=C(CH₃)-CO-SC₂H₅, -C(CH₃)=C(CH₃)CO-S-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-S-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-SCH₃, -C(CH₃)=C(C₂H₅)-CO-SC₂H₅, -C(CH₃)=C(C₂H₅)-CO-S-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-SCH₃, -C(CH₃)=C(Cl)-CO-SC₂H₅, -C(CH₃)=C(Cl)-CO-S-n-C₃H₇, -C(CH₃)=C(Cl)-CO-S-i-C₃H₇, -C(CH₃)=C(Cl)-CO-S-n-C₄H₉, -C(CH₃)=C(Cl)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-SCH₃, -C(CH₃)=C(Br)-CO-SC₂H₅, -C(CH₃)=C(Br)-CO-S-n-C₃H₇, -C(CH₃)=C(Br)-CO-S-i-C₃H₇, -C(CH₃)=C(Br)-CO-S-n-C₄H₉, -C(CH₃)=C(Br)-CO-S-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-SCH₃, -C(CH₃)=C(CN)-CO-SC₂H₅, -C(CH₃)=C(CN)-CO-S-n-C₃H₇, -C(CH₃)=C(CN)-CO-S-i-C₃H₇, -C(CH₃)=C(CN)-CO-S-N-C₄H₉, -C(CH₃)=C(CN)-CO-S-tert.-C₄H₉, -C(CH₃)=C(COCH₃)-CO-OCH₃, -C(CH₃)=C(COC₂H₅)-CO-OCH₃, -C(CH₃)=C(CO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COCH₃)-CO-OC₂H₅, -C(CH₃)=C(COC₂H₅)-CO-OC₂H₅, -C(CH₃)=C(CO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COCH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(COC₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-OCH₃, -C(CH₃)=C(CF₃)-CO-OC₂H₅, -C(CH₃)=C(CF₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CF₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(COOCH₃)₂, -C(CH₃)=C(COOC₂H₅)₂, -C(CH₃)=C(COOCH₃)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)₂, -C(CH₃)=CH-CH=CH-COOH, -C(CH₃)=CH-CH=CH-CO-OCH₃, -C(CH₃)=CH-CH=CH-CO-OC₂H₅, -C(CH₃)=CH-CH=C(COOCH₃)₂, -C(CH₃)=CH-CH=C(CN)-CO-OCH₃, -C(CH₃)=CH-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CN)CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH₂, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -C(CH₃)=CH-(CH₂)₂-COOH, -C(CH₃)=CH-(CH₂)₂-CO-OCH₃, -C(CH₃)=CH-(CH₂)₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(COOCH₃)₂, -C(CH₃)=CH-CH₂-CH(COOC₂H₅)₂, -C(CH₃)=CH-CH₂-CH(CN)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CN)-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -C(CH₃)=CH-(CH₂)₂-CO-NH₂, -C(CH₃)=CH-(CH₂)₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-COOH, -C(CH₃)=CH-CH₂-CO-OCH₃, -C(CH₃)=CH-CH₂-CO-OC₂H₅, -C(CH₃)=C(COOCH₃)-CH₂-CO-OCH₃, -C(CH₃)=C(COOCH₃)-CH₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CO-NH₂, -C(CH₃)=CH-CH₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-CO-N(CH₃)₂.
wobei w für eine der folgenden Bedeutungen steht:
-CHO, -COCH₃, -COC₂H₅, -CO-n-C₃H₇, -CO-i-C₃H₇, -CO-n-C₄H₉, -CO-i-C₄H₉, -CO-s-C₄H₉, -CO-tert.-C₄H₉, -CO-CH₂CH=CH₂, -CO-CF₃, -COCCl₃, -COCH₂≡CH, -CO-cyclopropyl, -CO-cyclobutyl, -CO-cyclo­ pentyl, -CO-cyclohexyl, -CO-CN, -CO-COOCH₃, -CO-COOC₂H₅, CH=NH, -CH=NCH₃, -CH=NC₂H₅, -CH=N-n-C₃H₅, -CH=N-i-C₃H₅, -CH=N-n-C₄H₉, -CH=NCH₂CH=CH₂, -CH=NCH₂CH=CH₂-CH₃, -CH=NCH₂C≡CH, -CH=NCH₂C≡C-CH₃, -CH=N-cyclopropyl, -CH=N-cyclobutyl, -CH=N-cyclopentyl, -CH=N-cyclohexyl, -CH=N-cycloheptyl, -CH=N-CH₂-CH₂Cl, -CH=N-CH₂Cl, -CH=N-C₆H₅, -CH=N-(4-Br-C₆H₄), -CH=N-3-F-C₆H₄, -CH=N-4-F-C₆H₄, -CH=N-2-Cl-C₆H₄, -CH=N-3-Cl-C₆H₄, -CH=N-4-Cl-C₆H₄, -CH=N-2-Br-C₆H₄, -CH=N-2-F-C₆H₄, -CH=N-2-CH₃-C₆H₄, -CH=N-3-CH₃-C₆H₄, -CH=N-4-CH₃-C₆H₄, -CH=N-2-CF₃-C₆H₄, -CH-N-3-CF₃-C₆H₄, -CH=N-4-CF₃-C₆H₄, -CH=N-2-OCH₃-C₆H₄, -CH=N-3-OCH₃-C₆H₄, -CH=N-4-OCH₃-C₆H₄, -CH=N-4-NO₂-C₆H₄, -CH=N-4-CN-C₆H₄, -CH=N-2,4-(Cl,Cl)-C₆H₄, -CH=N-2,4-(CH₃,CH₃)-C₆H₄, -CH=N-CH₂OCH₃, -CH=N-CH₂OC₂H₅, -CH=N-CH₂CH₂OCH₃, -CH=N-CH₂CH₂OC₂H₅, -CH=N-OH, -CH=N-OCH₃, -CH=N-OC₂H₅, -CH=N-O-n-C₃H₇, -CH=N-O-i-C₃H₇, -CH=N-O-n-C₄H₉, -CH=N-O-i-C₄H₉, -CH=N-O-s-C₄H₉, -CH=N-O-tert.-C₄H₉, -CH=N-O-CH₂CH=CH₂, -CH=N-O-CH(CH₃)CH=CH₂, -CH=N-O-CH₂C≡CH, -CH=N-O-CH(CH₃)-C≡CH, -CH=N-O-CH₂-CH=CH-CH₃, -CH=N-O-CH₂-CH₂-Cl, -CH=N-O-CH₂-CH₂-F, -CH=N-O-CH₂-CF₃, -CH=N-O-CH₂-CH=CHCl, -CH=N-O-CH₂-CCl=CH₂, -CH=N-O-CH₂-CBr=CH₂, -CH=N-O-CH₂-CH=CCl-CH₃, -CH=N-OC(O)CH₃, -CH=N-OC(O)C₂H₅, -CH=N-O-CH₂-CN, -CH=N-O-CH₂-CH=CH-CH₂-O-CH₃, -CH=N-O-CH₂-CH=CH-CH₂-O-tert.-C₄H₉, -CH=N-O-(CH₂)₃-C₆H₅, -CH=N-O-(CH₂)₄-C₆H₅, -CH=N-O-(CH₂)₄-4-Cl-C₆H₄, -CH=N-O-(CH₂)₄-4-OCH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-CH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-C₆H₅, -CH=N-O-CH₂CH=CH-4-C₆H₄, -CH=N-O-CH₂CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CH-3-OCH₃-C₆H₄, -CH=N-O-(CH₂)₂CH=CH-4-F-C₆H₄, -CH=N-O-(CH₂)CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CHCH₂-4-OCH₃-C₆H₄, -CH=N-O-CH₂-CH=C(CH₃)-C₆H₅, -CH=N-O-(CH₂)₂CH=CH-3,4(Cl,Cl)-C₆H₃, -CH=N-O-(CH₂)₃C≡C-4-F-C₆H₄, -CH₂=N-OCHOCH₃, -CH=N-OC₂H₄OCH₃, -CH=N-OCH₂OC₂H₅, -CH=N-OCH(CH₃)OCH₃, -CH=N-OCH(CH₃)COOCH₃, -CH=N-OCH(CH₃)COO-n-C₄H₉, -CH=N-NH₂, -CH=N-NHCH₃, -CH=N-NHC₂H₅, -CH=N-NH-n-C₃H₇, -CH=N-NH-i-C₃H₇, -CH=N-NH-n-C₄H₉, -CH=N-NH-i-C₄H₉, -CH=N-NH-s-C₄H₉, -CH=N-NH-tert.-C₄H₉, -CH=N-NH-cyclopropyl, -CH=N-NH-cyclobutyl, -CH=N-NH-cyclopentyl, -CH=N-NH-cyclohexyl, -CH=N-NH-cycloheptyl, -CH=N-N(CH₃)₂, -CH=N-N(C₂H₅)₂, -CH=N-N(C₃H₇)₂, -CH=N-N(i-C₃H₇)(CH₃), -CH=N-NHCH₂-C=CH, -CH=N-NHCH₂-C≡CH, -CH=N-N(CH₃)-CH₂-C≡CH, -CH=N-NHCH₂CF₃, -CH=N-NH-CO-CH₃, -CH=N-CO-CH₂H₅, -CH=N-NH-COOCH₃, -CH=N-NH-COOC₂H₅, -CH=N-NH-COO-tert.-C₄H₉, -CH=N-pyrrolidin-1-yl, -CH=N-piperidin-1-yl, -CH=N-morpholin-4-yl, -CH=N-NH-C₆H₅, -CH=N-NH-(4-Cl-C₆H₄), -CH=N-NH-4-NO₂-C₆H₄), -CH=N-NH-(4-F-C₆H₄), -CH=N-NH-(4-CH₃O-C₆H₄), -CH=N-NH-(2,4-Cl₂-C₆H₃), -CH=N-NH-(2,4-(NO₂)₂-C₆H₃), -CH=N-NH-CO-NH₂, -CH=N-NH-CO-NHCH₃, -CH=N-NH-CO-NHC₂H₅, -CH=N-NH-CO-N(CH₃)₂, -CH=CH-COOH, -CH=CH-CO-OCH₃, -CH=CH-CO-OC₂H₂, -CH=CH-CO-O-n-C₃H₇, -CH=CH-CO-O-i-C₃H₇, -CH=CH-CO-O-n-C₄H₉, -CH=CH-CO-O-tert.-C₄H₉, -CH=CH-CO-O-cyclopropyl, -CH=CH-CO-O-cyclobutyl, -CH=CH-CO-O-cyclopentyl, -CH=CH-CO-O-cyclohexyl, -CH=CH-CO-O-cycloheptyl, -CH=C(CH₃)-COOH, -CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CO-O-n-C₃H₇, -CH=C(CH₃)-CO-O-i-C₃H₇, -CH=C(CH₃)-CO-O-n-C₄H₉, -CH=C(CH₃)-CO-O-tert.-C₄H₉, -CH=C(CH₃)-CO-O-cyclopropyl, -CH=C(CH₃)-CO-O-cyclobutyl, -CH=C(CH₃)-CO-O-cyclopentyl, -CH=C(CH₃)-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cycloheptyl, -CH=C(C₂H₅)-COOH, -CH=C(C₂H₅)-CO-OCH₃, -CH=C(C₂H₅)-CO-OC₂H₅, -CH=C(C₂H₅)-CO-O-n-C₃H₇, -CH=C(C₂H₅)-CO-O-i-C₃H₇, -CH=C(C₂H₅)-CO-O-n-C₄H₉, -CH=C(C₂H₅)-CO-O-tert.-C₄H₉, -CH=C(C₂H₅)-CO-O-cyclopropyl, -CH=C(C₂H₅)-CO-O-cyclobutyl, -CH=C(C₂H₅)-CO-O-cyclopentyl, -CH=C(C₂H₅)-CO-O-cyclohexyl, -CH=C(C₂H₅)-CO-O-cycloheptyl, -CH=C(Cl)-COOH, -CH=C(Cl)-CO-OCH₃, -CH=C(Cl)-CO-OC₂H₅, -CH=C(Cl)-CO-O-n-C₃H₇, -CH=C(Cl)-CO-O-i-C₃H₇, -CH=C(Cl)-CO-O-n-C₄H₉, -CH=C(Cl)-CO-O-tert.-C₄H₉, -CH=C(Cl)-CO-O-cyclopropyl, -CH=C(Cl)-CO-O-cyclobutyl, -CH=C(Cl)-CO-O-cyclopentyl, -CH=C(Cl)-CO-O-cyclohexyl, -CH=C(Cl)-CO-O-cycloheptyl, -CH=C(Br)-COOH, -CH=C(Br)-CO-OCH₃, -CH=C(Br)-CO-OC₂H₅, -CH=C(Br)-CO-O-n-C₃H₇, -CH=C(Br)-CO-O-i-C₃H₇, -CH=C(Br)-CO-O-n-C₄H₉, -CH=C(Br)-CO-O-tert.-C₄H₉, -CH=C(Br)-CO-O-cyclopropyl, -CH=C(Br)-CO-O-cyclobutyl, -CH=C(Br)-CO-O-cyclopentyl, -CH=C(Br)-CO-O-cyclohexyl, -CH=C(Br)-CO-O-cycloheptyl, -CH=C(CN)-COOH, -CH=C(CN)-CO-OCH₃, -CH=C(CN)-CO-OC₂H₅, -CH=C(CN)-CO-O-n-C₃H₇, -CH=C(CN)-CO-O-i-C₃H₇, -CH=C(CN)-CO-O-n-C₄H₉, -CH=C(CN)-CO-O-tert.-C₄H₉, -CH=C(CN)-CO-O-cyclopropyl, -CH=C(CN)-CO-O-cyclobutyl, -CH=C(CN)-CO-O-cyclopentyl, -CH=C(CN)-CO-O-cyclohexyl, -CH=C(CN)-CO-O-cycloheptyl, -CH=CH-CO-OCH₂-OCH₃, -CH=CH-CO-OCH₂-OC₂H₅, -CH=CH-CO-OCH₂-O-n-C₃H₅, -CH=CH-CO-OCH₂-O-i-C₃H₅, -CH=CH-CO-OCH-(CH₃)-OCH₃, -CH=CH-CO-OCH(CH₃)-OC₂H₅, -CH=CH-CO-O-CH₂-CH₂-OCH₃, -CH=CH-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-OCH₃, -CH=C(CH₃)-CO-OCH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-O-n-C₃H₅, -CH=C(CH₃)-CO-OCH₂-O-i-C₃H₅, -CH=C(CH₃)-CO-OCH(CH₃)-OCH₃, -CH=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CH₃)-CO-O-CH₂CH₂-OCH₃, -CH=C(CH₃)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-OCH₃, -CH=C(C₂H₅)-CO-OCH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-O-n-C₃H₅, -CH=C(C₂H₅)-CO-OCH₂-O-i-C₃H₅, -CH=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -CH=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OCH₃, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OC₂H₂, -CH=C(Cl)-CO-OCH₂-OCH₃, -CH=C(Cl)-CO-OCH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-O-n-C₃H₅, -CH=C(Cl)-CO-OCH₂-O-i-C₃H₅, -CH=C(Cl)-CO-OCH(CH₃)-OCH₃, -CH=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Cl)-CO-O-CH₂CH₂-OCH₃, -CH=C(Cl)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-OCH₃, -CH=C(Br)-CO-OCH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-O-n-C₃H₅, -CH=C(Br)-CO-OCH₂-O-i-C₃H₅, -CH=C(Br)-CO-OCH(CH₃)-OCH₃, -CH=C(Br)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Br)-CO-O-CH₂CH₂-OCH₃, -CH=C(Br)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-OCH₃, -CH=C(CN)-CO-OCH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-O-n-C₃H₅, -CH=C(CN)-CO-OCH₂-O-i-C₃H₅, -CH=C(CN)-CO-OCH(CH₃)-OCH₃, -CH=C(CN)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CN)-CO-O-CH₂CH₂-OCH₃, -CH=C(CN)-CO-O-CH₂CH₂-OC₂H₅, -CH=CH-CO-OCH₂-CF₃, -CH=CH-CO-OCH₂-CCl₃, -CH=CH-CO-OCH₂-oxiranyl, -CH=CH-CO-O(CH₂)₃-Br, -CH=CH-CO-OCH₂-CH=CH₂, -CH=CH-CO-OCH₂-C≡CH, -CH=CH-CO-OCH₂-CN, -CH=CH-CO-O(CH₂)₂-CN, -CH=C(CH₃)-CO-OCH₂-CF₃, -CH=C(CH₃)-CO-OCH₂-CCl₃, -CH=C(CH₃)-CO-OCH₂-oxiranyl, -CH=C(CH₃)-CO-O(CH₂)₃-Br, -CH=C(CH₃)-CO-OCH₂-CH=CH₂, -CH=C(CH₃)-CO-OCH₂-C≡CH, -CH=C(CH₃)-CO-OCH₂-CN, -CH=C(CH₃)-CO-O-(CH₂)₂-CN, -CH=C(C₂H₅)-CO-OCH₂-CF₃, -CH=C(C₂H₅)-CO-OCH₂-CCl₃, -CH=C(C₂H₅)-CO-OCH₂-oxiranyl, -CH=C(C₂H₅)-CO-O(CH₂)₃-Br, -CH=C(C₂H₅)-CO-OCH₂-CH=CH₂, -CH=C(C₂H₅)-CO-OCH₂-C≡CH, -CH=C(C₂H₅)-CO-OCH₂-CN, -CH=C(C₂H₅)-CO-O(CH₂)₂-CN, -CH=C(Cl)-CO-OCH₂-CF₃, -CH=C(Cl)-CO-OCH₂-CCl₃, -CH=C(Cl)-CO-OCH₂-oxiranyl, -CH=C(Cl)-CO-O(CH₂)₃-Br, -CH=C(Cl)-CO-OCH₂-CH=CH₂, -CH=C(Cl)-CO-OCH₂-C≡CH, -CH=C(Cl)-CO-OCH₂-CN, -CH=C(Cl)-CO-O(CH₂)₂-CN, -CH=C(Br)-CO-OCH₂-CF₃, -CH=C(Br)-CO-OCH₂-CCl₃, -CH=C(Br)-CO-OCH₂-oxiranyl, -CH=C(Br)-CO-O(CH₂)₃-Br, -CH=C(Br)-CO-OCH₂-CH=CH₂, -CH=C(Br)-CO-OCH₂-C≡CH, -CH=C(Br)-CO-OCH₂-CN, -CH=C(Br)-CO-O(CH₂)₂-CN, -CH=C(CN)-CO-OCH₂-CF₃, -CH=C(CN)-CO-OCH₂-CCl₃, -CH=C(CN)-CO-OCH₂-oxiranyl, -CH=C(CN)-CO-O(CH₂)₃-Br, -CH=C(CN)-CO-OCH₂-CH=CH₂, -CH=C(CN)-CO-OCH₂-C≡CH, -CH=C(CN)-CO-OCH₂-CN, -CH=C(CN)-CO-O(CH₂)₂-CN, -CH=CH-CO-CH₃, -CH=CH-CO-C₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-i-C₃H₇, -CH=CH-CO-n-C₄H₉, -CH=CH-CO-tert.-C₄H₉, -CH=CH-CO-CH₂Cl, -CH=CH-CO-CH₂Br, -CH=CH-CO-CHCl₂, -CH=CH-CO-CH₂-OCH₃, -CH=CH-CO-CH(OCH₃)₂, -CH=CH-CO-CH₂-SCH₃, -CH=C(CH₃)-CO-CH₃, -CH=C(CH₃)-CO-C₂H₅, -CH=C-(CH₃)-CO-n-C₃H₇, -CH=C-(CH₃)-CO-i-C₃H₇, -CH=C-(CH₃)-CO-n-C₄H₉, -CH=C-(CH₃)-CO-tert.-C₄H₉, -CH=C(CH₃)-CO-CH₂Cl, -CH=C(CH₃)-CO-CH₂Br, -CH=C(CH₃)-CO-CHCl₂, -CH=C(CH₃)-CO-CH₂-OCH₃, -CH=C-(CH₃)-CO(OCH₃)₂, -CH=C(CH₃)-CO-CH₂-SCH₃, -CH=C ä(C₂H₅)-CO-CH₃, -CH=C(C₂H₅)-CO-C₂H₅, -CH=C(C₂H₅)-CO-n-C₃H₇, -CH=C(C₂H₅)-CO-i-C₃H₇, -CH=C(C₂H₅)-CO-n-C₄H₉, -CH=C(C₂H₅)-CO-tert.-C₄H₉, -CH=C(C₂H₅)-CO-CH₂Cl, -CH=C(C₂H₅)-CO-CH₂Br, -CH=C(C₂H₅)-CO-CHCl₂, -CH=C(C₂H₅)-CO-CH₂-OCH₃, -CH=C(C₂H₅)-CO-CH(OCH₃)₂, -CH=C(C₂H₅)-CO-CH₂-SCH₃, -CH=C(Cl)-CO-CH₃, -CH=C(Cl)-CO-C₂H₅, -CH=C(Cl)-CO-n-C₃H₇, -CH=C(Cl)-CO-i-C₃H₇, -CH=C(Cl)-CO-n-C₄H₉, -CH=C(Cl)-CO-tert.-C₄H₉, -CH=C(Cl)-CO-CH₂Cl, -CH=C(Cl)-CO-CH₂Br, -CH=C(Cl)-CO-CHCl₂, -CH=C(Cl)-CO-CH₂-OCH₃, -CH=C(Cl)-CO-CH(OCH₃)₂, -CH=C(Cl)-CO-CH₂-SCH₃, -CH=C(Br)-CO-CH₃, -CH=C(Br)-CO-C₂H₅, -CH=C(Br)-CO-n-C₃H₇, -CH=C(Br)-CO-i-C₃H₇, -CH=C(Br)-CO-n-C₄H₉, -CH=C(Br)-CO-tert.-C₄H₉, -CH=C(Br)-CO-CH₂Cl, -CH=C(Br)-CO-CH₂Br, -CH=C(Br)-CO-CHCl₂, -CH=C(Br)-CO-CH₂-OCH₃, -CH=C(Br)-CO-CH(OCH₃)₂, -CH=C(Br)-CO-CH₂-SCH₃, -CH=C(CN)-CO-CH₃, -CH=C(CN)-CO-C₂H₅, -CH=C(CN)-CO-n-C₃H₇, -CH=C(CN)-CO-i-C₃H₇, -CH=C(CN)-CO-n-C₄H₉, -CH=C(CN)-CO-tert.-C₄H₉, -CH=C(CN)-CO-CH₂Cl, -CH=C(CN)-CO-CH₂Br, -CH=C(CN)-CO-CHCl₂, -CH=C(CN)-CO-CH₂-OCH₃, -CH=C(CN)-CO-CH(OCH₃)₂, -CH=C(CN)-CO-CH₂-SCH₃, -CH=CH-CO-C₆H₅, -CH=CH-CO-(4-Cl-C₆H₄), -CH=C(CH₃)-CO-C₆H₅, -CH=C(CH₃)-CO-(4-Cl-C₆H₄), -CH=C(C₂H₅)-CO-C₆H₅, -CH=C(C₂H₅)-CO-(4-Cl-C₆H₄), -CH=C(Cl)-CO-C₆H₅, -CH=C(Br)-CO-C₆H₅, -CH=C(CN)-CO-C₆H₅, -CH=CH-CO-NH₂, -CH=CH-CO-NHCH₃, -CH=CH-CO-N(CH₃)₂, -CH=CH-CO-NH-C₂H₅, -CH=CH-CO-N(C₂H₅)₂, -CH=CH-CO-NH-n-C₃H₇, -CH=CH-CO-NH-i-C₃H₇, -CH=CH-CO-NH-tert.-C₄H₉, -CH=CH-CO-NH-cyclopropyl, -CH=CH-CO-NH-cyclobutyl, -CH=CH-CO-NH-cyclopentyl, -CH=CH-CO-NH-cyclohexyl, -CH=CH-CO-NH-cycloheptyl, -CH=CH-CO-NH-cyclooctyl, -CH=CH-CO-pyrrolidin-1-yl, -CH=CH-CO-piperidin-1-yl, -CH=CH-CO-morpholin-4-yl, -CH=CH-CO-NH-CH₂CH=CH₂, -CH=CH-CO-NH-CH₂C≡CH, -CH=CH-CO-N(CH₃)-CH₂C≡CH, -CH=CH-CO-NH-(CH₂)₂Cl, -CH=CH-CO-NH-C₆H₅, -CH=C(CH₃)-CO-NH₂, -CH=C(CH₃)-CO-NHCH₃, -CH=C(CH₃)-CO-N(CH₃)₂, -CH=C(CH₃)-CO-NH-C₂H₅, -CH=C(CH₃)-CO-N(C₂H₅)₂, -CH=C(CH₃)-CO-NH-n-C₃H₇, -CH=C(CH₃)-CO-NH-i-C₃H₇, -CH=C(CH₃)-CO-NH-tert.-C₄H₉, -CH=C(CH₃)-CO-NH-cyclopropyl, -CH=C(CH₃)-CO-NH-cyclobutyl, -CH=C(CH₃)-CO-NH-cyclopentyl, -CH=C(CH₃)-CO-NH-cyclohexyl, -CH=C(CH₃)-CO-NH-cycloheptyl, -CH=C(CH₃)-CO-NH-cyclooctyl, -CH=C(CH₃)-CO-pyrrolidin-1-yl, -CH=C(CH₃)-CO-piperidin-1-yl, -CH=C(CH₃)-CO-morpholin-4-yl, -CH=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -CH=C(CH₃)-CO-NH-CH₂C≡CH, -CH=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CH₃)-CO-NH-(CH₂)₂Cl, -CH=C(CH₃)-CO-NH-C₆H₅, -CH=C(C₂H₅)-CO-NH₂, -CH=C(C₂H₅)-CO-NHCH₃, -CH=C(C₂H₅)-CO-N(CH₃)₂, -CH=C(C₂H₅)-CO-NH-C₂H₅, -CH=C(C₂H₅)-CO-N(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-n-C₃H₇, -CH=C(C₂H₅)-CO-NH-i-C₃H₇, -CH=C(C₂H₅)-CO-NH-tert.-C₄H₉, -CH=C(C₂H₅)-CO-NH-cyclopropyl, -CH=C(C₂H₅)-CO-NH-cyclobutyl, -CH=C(C₂H₅)-CO-NH-cyclopentyl, -CH=C(C₂H₅)-CO-NH-cyclohexyl, -CH=C(C₂H₅)-CO-NH-cycloheptyl, -CH=C(C₂H₅)-CO-NH-cyclooctyl, -CH=C(C₂H₅)-CO-pyrrolidin-1-yl, -CH=C(C₂H₅)-CO-piperidin-1-yl, -CH=C(C₂H₅)-CO-morpholin-4-yl, -CH=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-CH₂C≡CH, -CH=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -CH=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -CH=C(C₂H₅)-CO-NH-C₆H₅, -CH=C(Cl)-CO-NH₂, -CH=C(Cl)-CO-NHCH₃, -CH=C(Cl)-CO-N(CH₃)₂, -CH=C(Cl)-CO-NH-C₂H₅, -CH=C(Cl)-CO-N(C₂H₅)₂, -CH=C(Cl)-CO-NH-n-C₃H₇, -CH=C(Cl)-CO-NH-i-C₃H₇, -CH=C(Cl)-CO-NH-tert.-C₄H₉, -CH=C(Cl)-CO-NH-cyclopropyl, -CH=C(Cl)-CO-NH-cyclobutyl, -CH=C(Cl)-CO-NH-cyclopentyl, -CH=C(Cl)-CO-NH-cyclohexyl, -CH=C(Cl)-CO-NH-cycloheptyl, -CH=C(Cl)-CO-NH-cyclooctyl, -CH=C(Cl)-CO-pyrrolidin-1-yl, -CH=C(Cl)-CO-piperidin-1-yl, -CH=C(Cl)-CO-morpholin-4-yl, -CH=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -CH=C(Cl)-CO-NH-CH₂C≡CH, -CH=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Cl)-CO-NH-(CH₂)₂Cl, -CH=C(Cl)-CO-NH-C₆H₅, -CH=C(Br)-CO-NH₂, -CH=C(Br)-CO-NHCH₃, -CH=C(Br)-CO-N(CH₃)₂, -CH=C(Br)-CO-NH-C₂H₅, -CH=C(Br)-CO-N(C₂H₅)₂, -CH=C(Br)-CO-NH-n-C₃H₇, -CH=C(Br)-CO-NH-i-C₃H₇, -CH=C(Br)-CO-NH-tert.-C₄H₉, -CH=C(Br)-CO-NH-cyclopropyl, -CH=C(Br)-CO-NH-cyclobutyl, -CH=C(Br)-CO-NH-cyclopentyl, -CH=C(Br)-CO-NH-cyclohexyl, -CH=C(Br)-CO-NH-cycloheptyl, -CH=C(Br)-CO-NH-cyclooctyl, -CH=C(Br)-CO-pyrrolidin-1-yl, -CH=C(Br)-CO-piperidin-1-yl, -CH=C(Br)-CO-morpholin-4-yl, -CH=C(Br)-CO-NH-CH₂CH=C(Br)₂, -CH=C(Br)-CO-NH-CH₂C≡CH, -CH=C(Br)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Br)-CO-NH-(CH₂)₂Cl, -CH=C(Br)-CO-NH-C₆H₅, -CH=C(CN)-CO-NH₂, -CH=C(CN)-CO-NHCH₃, -CH=C(CN)-CO-N(CH₃)₂, -CH=C(CN)-CO-NH-C₂H₅, -CH=C(CN)-CO-N(C₂H₅)₂, -CH=C(CN)-CO-NH-n-C₃H₇, -CH=C(CN)-CO-NH-i-C₃H₇, -CH=C(CN)-CO-NH-tert.-C₄H₉, -CH=C(CN)-CO-NH-cyclopropyl, -CH=C(CN)-CO-NH-cyclobutyl, -CH=C(CN)-CO-NH-cyclopentyl, -CH=C(CN)-CO-NH-cyclohexyl, -CH=C(CN)-CO-NH-cycloheptyl, -CH=C(CN)-CO-NH-cyclooctyl, -CH=C(CN)-CO-pyrrolidin-1-yl, -CH=C(CN)-CO-piperidin-1-yl, -CH=C(CN)-CO-morpholin-4-yl, -CH=C(CN)-CO-NH-CH₂CH=C(CN)₂, -CH=C(CN)-CO-NH-CH₂C≡CH, -CH=C(CN)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CN)-CO-NH-(CH₂)₂Cl, -CH=C(CN)-CO-NH-C₆H₅, -CH=CH-CO-SCH₃, -CH=CH-CO-SC₂H₅, -CH=CH-CO-S-n-C₃H₇, -CH=CH-CO-S-i-C₃H₇, -CH=CH-CO-S-n-C₄H₉, -CH=CH-CO-S-tert.-C₄H₉, -CH=C(CH₃)-CO-SCH₃, -CH=C(CH₃)-CO-SC₂H₅, -CH=C(CH₃)-CO-S-n-C₃H₇, -CH=C(CH₃)-CO-S-i-C₃H₇, -CH=C(CH₃)-CO-S-n-C₄H₉, -CH=C(CH₃)-CO-S-tert.-C₄H₉, -CH=C(C₂H₅)-CO-SCH₃, -CH=C(C₂H₅)-CO-SC₂H₅, -CH=C(C₂H₅)-CO-S-n-C₃H₇, -CH=C(C₂H₅)-CO-S-i-C₃H₇, -CH=C(C₂H₅)-CO-S-n-C₄H₉, -CH=C(C₂H₅)-CO-S-tert.-C₄H₉, -CH=C(Cl)-CO-SCH₃, -CH=C(Cl)-CO-SC₂H₅, -CH=C(Cl)-CO-S-n-C₃H₇, -CH=C(Cl)-CO-S-i-C₃H₇, -CH=C(Cl)-CO-S-n-C₄H₉, -CH=C(Cl)-CO-S-tert.-C₄H₉, -CH=C(Br)-CO-SCH₃, -CH=C(Br)-CO-SC₂H₅, -CH=C(Br)-CO-S-n-C₃H₇, -CH=C(Br)-CO-S-i-C₃H₇, -CH=C(Br)-CO-S-n-C₄H₉, -CH=C(Br)-CO-S-tert.-C₄H₉, -CH=C(CN)-CO-SCH₃, -CH=C(CN)-CO-SC₂H₅, -CH=C(CN)-CO-S-n-C₃H₇, -CH=C(CN)-CO-S-i-C₃H₇, -CH=C(CN)-CO-S-n-C₄H₉, -CH=C(CN)-CO-S-tert.-C₄H₉, -CH=C(COCH₃)-CO-OCH₃, -CH=C(COC₂H₅)-CO-OCH₃, -CH=C(CO-n-C₃H₇)-CO-OCH₃, -CH=C(COCH₃)-CO-OC₂H₅, -CH=C(COC₂H₅)-CO-OC₂H₅, -CH=C(CO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COCH₃)-CO-O-n-C₃H₇, -CH=C(COC₂H₅)-CO-O-n-C₃H₇, -CH=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-OCH₃, -CH=C(CF₃)-CO-OC₂H₅, -CH=C(CF₃)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-O-i-C₃H₇, -CH=C(CF₃)-CO-O-n-C₄H₉, -CH=C(CF₃)-CO-O-tert.-C₄H₉, -CH=C(COOCH₃)₂, -CH=C(COOC₂H₅)₂, -CH=C(COOCH₃)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)-CO-OCH₃, -CH=C(COO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)₂, -CH=CH-CH=CH-COOH, -CH=CH-CH=CH-CO-OCH₃, -CH=CH-CH=CH-CO-OC₂H₅, -CH=CH-CH=C(COOCH₃)₂, -CH=CH-CH=C(CN)-CO-OCH₃, -CH=CH-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-OCH₃, -CH=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CH=C(Cl)-CO-OCH₃, -CH=C(CH₃)-CH=C(Br)-CO-OCH₃, -CH=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-NH₂, -CH=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -CH=CH-(CH₂)₂-COOH, -CH=CH-(CH₂)₂-CO-OCH₃, -CH=CH-(CH₂)₂-CO-OC₂H₅, -CH=CH-CH₂-CH(COOCH₃)₂, -CH=CH-CH₂-CH(COOC₂H₅)₂, -CH=CH-CH₂-CH(CN)-CO-OCH₃, -CH=CH-CH₂-CH(CN)-CO-OC₂H₅, -CH=CH-CH₂-CH(CH₃)-CO-OCH₃, -CH=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -CH=CH-(CH₂)₂-CO-NH₂, -CH=CH-(CH₂)₂-CO-NH-CH₃, -CH=CH-CH₂-COOH, -CH=CH-CH₂-CO-OCH₃, -CH=CH-CH₂-CO-OC₂H₅, -CH=C(COOCH₃)-CH₂-CO-OCH₃, -CH=C(COOCH₃)-CH₂-CO-OC₂H₅, -CH=CH-CH₂-CO-NH₂, -CH=CH-CH₂-CO-NH-CH₃, -CH=CH-CH₂-CO-N(CH₃)₂, -CH(OCH₃)₂, -CH(SCH₃)₂, -CH(OC₂H₅)₂, -CH(SC₂H₅)₂, -CH(O-n-C₃H₇)₂, -CH(O-i-C₃H₇)₂, -CH(S-n-C₃H₇)₂, -CH(S-i-C₃H₇)₂, -CH(O-n-C₄H₉)₂, -CH(O-i-C₄H₉)₂, -CH(O-s-C₄H₉)₂, -CH(O-tert.-C₄H₉)₂, -CH(S-n-C₄H₉)₂, -CH(S-i-C₄H₉)₂, -CH(S-s-C₄H₉)₂, -CH(S-tert.-C₄H₉)₂, -CH(OC₅H₁₁)₂, 1,3-Dioxolan-2-yl, 1,3-Dithio­ lan-2-yl, 1,3-Oxathiolan-2-yl, 4-Methyl-1,3-dioxolan-2-yl, 4-Methyl-1,3-dithiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 5-Methyl-1,3-oxathiolan-2-yl, 4-Ethyl-1,3-dioxolan-2-yl, 4-Ethyl- 1,4-dithiolan-2-yl, 4-Ethyl-1,3-oxathiolan-2-yl, 5-Ethyl-1,3-oxa­ thiolan-2-yl, 4,5-Dimethyl-1,3-dioxolan-2-yl, 4,4-Dimethyl-1,3- dioxolan-2-yl, 4,5-Dimethyl-1,3-dithiolan-2-yl, 5,5-Dimethyl-1,3- dithiolan-2-yl, 4,5-Dimethyl-1,3-oxathiolan-2-yl, 5,5-Dimethyl- 1,3-oxathiolan-2-yl, 4,4-Dimethyl-1,3-oxathiolan-2-yl, 4-Vinyl- 1,3-dioxolan-2-yl, 4-Vinyl-1,3-dithiolan-2-yl, 4-Vinyl-1,3-oxa­ thiolan-2-yl, 5-Vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3- dioxolan-2-yl, 4-Chlormethyl-1,3-dithiolan-2-yl, 4-Chlormethyl- 1,3-oxathiolan-2-yl, 5-Chlormethyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-1,3-dithio­ lan-2-yl, 4-Hydroxymethyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl- 1,3-oxathiolan-2-yl, 4-Methoxymethyl-1,3-dioxolan-2-yl, 4-Allyl­ oxymethyl-1,3-dioxolan-2-yl, 4-Propargyloxymethyl-1,3-dioxolan- 2-yl, 4-Acetoxymethyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-1,3-dithiolan-2-yl, 4-Propargyl- oxymethyl-1,3-dithiolan-2-yl, 4-Acetoxymethyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-1,3-oxa­ thiolan-2-yl, 4-Allyloxymethyl-1,3-oxathiolan-2-yl, 5-Allyloxy- methyl-1,3-oxathiolan-2-yl, 4-Propargyloxymethyl-1,3-oxathiolan- 2-yl, 5-Propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxymethyl- 1,3-oxathiolan-2-yl, 5-Acetoxymethyl-1,3-oxathiolan-2-yl, 4-Methylthiomethyl-1,3-dioxolan-2-yl, 4-Methylthiomethyl-1,3- dithiolan-2-yl, 4-Carboxy-1,3-dioxolan-2-yl, 4-Carboxy-1,3- dithiolan-2-yl, 4-Methoxycarbonyl-1,3-dioxolan-2-yl, 4-Ethoxy- carbonyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-1,3-di­ thiolan-2-yl, 4-n-Butoxycarbonyl-1,3-dithiolan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-4-methyl- 1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-di­ thiolan-2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-1,3- dithiolan-2-yl, 1,3-Dioxan-2-yl, 1,3-Dithian-2-yl, 1,3-Oxathian- 2-yl, 5-Methyl-1,3-dioxan-2-yl, 5-Methyl-1,3-dithian-2-yl, 5-Methyl-1,3-oxathian-2-yl, 5,5-Dimethyl-1,3-dioxan-2-yl, 4,6-Di­ methyl-1,3-dioxan-2-yl, 4,4-Dimethyl-1,3-dioxan-2-yl, 5,5-Di­ methyl-1,3-dithian-2-yl, 4,6-Dimethyl-1,3-dithian-2-yl, 4,4-Di­ methyl-1,3-dithian-2-yl, 5,5-Dimethyl-1,3-oxathian-2-yl, 4,4-Di­ methyl-1,3-oxathian-2-yl, 6,6-Dimethyl-1,3-oxathian-2-yl, 4-Hydroxymethyl-1,3-dioxan-2-yl, 4-Methoxymethyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-1,3-dithian-2-yl, 4-Methoxymethyl-1,3-di­ thian-2-yl, 4-Allyloxymethyl-1,3-dithian-2-yl, 4-Acetoxymethyl- 1,3-dithian-2-yl, 4-Chlormethyl-1,3-dioxan-2-yl, 4-Chlormethyl- 1,3-dithian-2-yl, 1,3-Dioxepan-2-yl, 1,3-Dithiepan-2-yl, 1,3-Di­ oxep-5-en-2-yl, 4-Methoxycarbonyl-1,3-dioxan-2-yl, 4-Ethoxy- carbonyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-1,3-dithian-2-yl, 4-n-Butoxycarbonyl-1,3-dithian-2-yl, 4-Methoxycarbonyl-4- methyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-Methoxy- carbonyl-4-methyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-4-methyl- 1,3-dithian-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithian-2-yl, -C(CH₃)(OCH₃)₂, -C(CH₃)(SCH₃)₂, -C(CH₃)(OC₂H₅)₂, -C(CH₃)(SC₂H₅)₂, -C(CH₃)(O-n-C₃H₇)₂, -C(CH₃)(O-i-C₃H₇)₂, -C(CH₃)(S-n-C₃H₇)₂, -C(CH₃)(S-i-C₃H₇)₂, -C(CH₃)(O-n-C₄H₉)₂, -C(CH₃)(O-i-C₄H₉)₂, -C(CH₃)(O-s-C₄H₉)₂, -C(CH₃)(O-tert.-C₄H₉)₂, -C(CH₃)(S-n-C₄H₉)₂, -C(CH₃)(S-i-C₄H₉)₂, -C(CH₃)(S-s-C₄H₉)₂, -C(CH₃)(S-tert.-C₄H₉)₂, -C(CH₃)(O-n-C₅H₁₁)′′, 2-Methyl-1,3-dioxolan-2-yl, 2-Methyl-1,3-di­ thiolan-2-yl, 2-Methyl-1,3-oxathiolan-2-yl, 2,4-Dimethyl-1,3- dioxolan-2-yl, 2,4-Dimethyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-1,3- oxathiolan-2-yl, 2,5-Dimethyl-1,3-oxathiolan-2-yl, 4-Ethyl-2- methyl-1,3-dioxolan-2-yl, 4-Ethyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Ethyl-2-methyl-1,3- oxathiolan-2-yl, 2,4,5-Trimethyl-1,3-dioxolan-2-yl, 2,4,4-Tri­ methyl-1,3-dioxolan-2-yl, 2,4,5-Trimethyl-1,3-dithiolan-2-yl, 2,4,4-Trimethyl-1,3-dithiolan-2-yl, 2,4,5-Trimethyl-1,3-oxathio­ lan-2-yl, 2,4,4-Trimethyl-1,3-oxathiolan-2-yl, 2-Methyl-4-vinyl- 1,3-dioxolan-2-yl, 2-Methyl-4-vinyl-1,3-dithiolan-2-yl, 2-Methyl- 4-vinyl-1,3-oxathiolan-2-yl, 2-Methyl-5-vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-dioxolan-2-yl, 4-Chlormethyl-2- methyl-1,3-dithiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-oxathio­ lan-2-yl, 5-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Hydroxy­ methyl- 2-methyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-2- methyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dioxolan- 2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxy- 2-methyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dithiolan-2-yl, 4-Acetoxy-2- methyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-oxathio­ lan-2-yl, 5-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Allyl­ oxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Allyloxymethyl-2- methyl-1,3-oxathiolan-2-yl, 2-Methyl-4-4-propargyloxymethyl-1,3- oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxy-2-methyl-1,3-oxathiolan-2-yl, 5-Acetoxy-2-methyl- 1,3-oxathiolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dioxolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-2- methyl-1,3-dioxolan-2-yl, 4-Carboxy-2-methyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-2- methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-2-methyl-1,3-dioxo­ lan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-Eth­ oxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-2- methyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-di­ oxolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-ethoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4- ethoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-n-butoxy- carbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl-1,3- dithiolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-dioxan-2-yl, 2-Methyl-1,3-dithian-2-yl, 2-Methyl-1,3-oxathian-2-yl, 2,5- Dimethyl-1,3-dioxan-2-yl, 2,5-Dimethyl-1,3-dithian-2-yl, 2,5-Dimethyl- 1,3-oxathian-2-yl, 2,5,5-Trimethyl-1,3-dioxan-2-yl, 2,4,6- Trimethyl-1,3-dioxan-2-yl, 2,4,4-Trimethyl-1,3-dioxan-2-yl, 2,5,5-Trimethyl-1,3-dithian-2-yl, 2,4,6-Trimethyl-1,3-dithian-2- yl, 2,4,4-Trimethyl-1,3-dithian-2-yl, 2,5,5-Trimethyl-1,3-oxa­ thian-2-yl, 2,4,4-Trimethyl-1,3-oxathian-2-yl, 2,6,6-Trimethyl- 1,3-oxathian-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-2- methyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dithian-2-yl, 4-Methoxymethyl-2- methyl-1,3-dithian-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithian-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dithian-2-yl, 4-Chlormethyl-2- methyl-1,3-dioxan-2-yl, 4-Chlormethyl-2-methyl-1,3-dithian-2- yl, -C(CH₃)=NH, -C(CH₃)=N-CH₃, -C(CH₃)=N-C₂H₅, -C(CH₃)=N-n-C₃H₇, -(CH₃)=N-i-C₃H₇, -C(CH₃)=N-n-C₄H₉, -C(CH₃)=N-CH₂CH=CH₂, -C(CH₃)=N-CH₂CH=CH₂-CH₃, -C(CH₃)=N-CH₂C≡CH, -C(CH₃)=N-CH₂C≡C-CH₃, -C(CH₃)=N-cyclopropyl, -C(CH₃)=N-cyclobutyl, -C(CH₃)=N-cyclopentyl, -C(CH₃)=N-cyclohexyl, -C(CH₃)=N-cycloheptyl, -C(CH₃)=N-CH₂-CH₂Cl, -C(CH₃)=N-CH₂Cl, -C(CH₃)=N-C₆H₅, -C(CH₃)=N-(2-F-C₆H₄), -C(CH₃)=N-(3-F-C₆H₄), -C(CH₃)=N-(4-F-C₆H₄), -C(CH₃)=N-(2-Cl-C₆H₄), -C(CH₃)=N-(3-Cl-C₆H₄), -C(CH₃)=N-(4-Cl-C₆H₄), -C(CH₃)=N-(2-CH₃-C₆H₄), -C(CH₃)=N-(3-CH₃-C₆H₄), -C(CH₃)=N-(4-CH₃-C₆H₄), -C(CH₃)=N-(2-CF₃-C₆H₄), -C(CH₃)=N-(3-CF₃-C₆H₄), -C(CH₃)=N-(4-CF₃-C₆H₄), -C(CH₃)=N-(2-OCH₃-C₆H₄), -C(CH₃)=N-(3-OCH₃-C₆H₄), -C(CH₃)=N-(4-OCH₃-C₆H₄), -C(CH₃)=N-(4-NO₂-C₆H₄), -C(CH₃)=N-(4-CN-C₆H₄), -C(CH₃)=N-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-(2,4-(CH₃)₂-C₆H₃), -C(CH₃)=N-CH₂-OCH₃, -C(CH₃)=N-CH₂-OC₂H₅, -C(CH₃)=N-CH₂CH₂-OCH₃, -C(CH₃)=N-CH₂CH₂-OC₂H₅, -C(CH₃)=N-OH, -C(CH₃)=N-OCH₃, -C(CH₃)=N-OC₂H₅, -C(CH₃)=N-O-n-C₃H₇, -C(CH₃)=N-O-i-C₃H₇, -C(CH₃)=N-O-n-C₄H₉, -C(CH₃)=N-O-i-C₄H₉, -C(CH₃)=N-O-s-C₄H₉, -C(CH₃)=N-O-tert.-C₄H₉, -C(CH₃)=N-OCH₂-CH=CH₂, -C(CH₃)=N-OCH(CH₃)-CH=CH₂, -C(CH₃)=N-OCH₂-C≡CH, -C(CH₃)=N-CH(CH₃)-C≡CH, -C(CH₃)=N-OCH₂-CH=C-CH₃, -C(CH₃)=N-OCH₂CH₂-Cl, -C(CH₃)=N-OCH₂CH₂-F, -C(CH₃)=N-OCH₂-CF₃, -C(CH₃)=N-OCH₂-CH=CHCl, -C(CH₃)=N-OCH₂-C(Cl)=CH₂, -C(CH₃)=N-OCH₂-C(Br)=CH₂, -C(CH₃)=N-OCH₂-CH=C(Cl)-CH₃, -C(CH₃)=N-O-CO-CH₃, -C(CH₃)=N-O-CO-C₂H₅, -C(CH₃)=N-OCH₂-CN, -C(CH₃)=N-OCH₂-CH=CH-CH₂-OCH₃, -C(CH₃)=N-OCH₂-CH=CH-CH₂-O-tert.-C₄H₉, -C(CH₃)=N-O-(CH₂)₃-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-(4-Cl-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-C₆H₅, -C(CH₃)=N-OCH₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(3-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-CH₂-(4-CH₃O-C₆H₄), -C(CH₃)=N-OCH₂-CH=C(CH₃)-C₆H₅, -C(CH₃)=N-O-(CH₂)₂-CH=CH-(3,4-Cl₂-C₆H₃), -C(CH₃)=N-O-(CH₂)₃-C≡C-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-OCH₃, -C(CH₃)=N-OCH₂CH₂-OCH₃, -C(CH₃)=N-OCH₂-OC₂H₅, -C(CH₃)=N-OCH(CH₃)-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=N-NH₂, -C(CH₃)=N-NH-CH₃, -C(CH₃)=N-NH-C₂H₅, -C(CH₃)=N-NH-n-C₃H₇, -C(CH₃)=N-NH-i-C₃H₇, -C(CH₃)=N-NH-n-C₄H₉, -C(CH₃)=N-NH-i-C₄H₉, -C(CH₃)=N-NH-s-C₄H₉, -C(CH₃)=N-NH-tert.-C₄H₉, -C(CH₃)=N-NH-cyclopropyl, -C(CH₃)=N-NH-cyclobutyl, -C(CH₃)=N-NH-cyclopentyl, -C(CH₃)=N-NH-cyclohexyl, -C(CH₃)=N-NH-cycloheptyl, -C(CH₃)=N-N(CH₃)₂, -C(CH₃)=N-N(C₂H₅)₂, -C(CH₃)=N-N(n-C₃H₇)₂, -C(CH₃)=N-N(i-C₃H₇)₂, -C(CH₃)=N-NH-CH₂-C=CH, -C(CH₃)=N-NH-CH₂-C≡CH, -C(CH₃)=N-N(CH₃)-CH₂-C≡CH, -C(CH₃)=N-NH-CH₂CF₃, -C(CH₃)=N-NH-CO-CH₃, -C(CH₃)=N-NH-CO-C₂H₅, -C(CH₃)=N-NH-CO-OCH₃, -C(CH₃)=N-NH-CO-OC₂H₅, -C(CH₃)=N-NH-CO-O-tert.-C₄H₉, -C(CH₃)=N-pyrrolidin-1-yl, -C(CH₃)=N-piperidin-1-yl, -C(CH₃)=N-morpholin-4-yl, -C(CH₃)=N-NH-C₆H₅, -C(CH₃)=N-NH-(4-Cl-C₆H₄), -C(CH₃)=N-NH-(4-NO₂-C₆H₄), -C(CH₃)=N-NH-(4-F-C₆H₄), -C(CH₃)=N-NH-(4-CH₃O-C₆H₄), -C(CH₃)=N-NH-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-NH-(2,4-(NO₂)₂-C₆H₃), -C(CH₃)=N-NH-CO-NH₂, -C(CH₃)=N-NH-CO-NHCH₃, -C(CH₃)=N-NH-CO-NHC₂H₅, -C(CH₃)=N-NH-CO-N(CH₃)₂, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=CH-CO-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-O-n-C₄H₉, -C(CH₃)=CH-CO-O-tert.-C₄H₉, -C(CH₃)=CH-CO-O-cyclopropyl, -C(CH₃)=CH-CO-O-cyclobutyl, -C(CH₃)=CH-CO-O-cyclopentyl, -C(CH₃)=CH-CO-O-cyclohexyl, -C(CH₃)=CH-CO-O-cycloheptyl, -C(CH₃)=C(CH₃)-COOH, -C(CH₃)=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-cyclopropyl, -C(CH₃)=C(CH₃)-CO-O-cyclobutyl, -C(CH₃)=C(CH₃)-CO-O-cyclopentyl, -C(CH₃)=C(CH₃)-CO-O-cyclohexyl, -C(CH₃)=C(CH₃)-CO-O-cycloheptyl, -C(CH₃)=C(C₂H₅)-COOH, -C(CH₃)=C(C₂H₅)-CO-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-cyclo­ propyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-O- cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-O-cycloheptyl, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-O-n-C₄H₉, -C(CH₃)=C(Cl)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-O-cyclopropyl, -C(CH₃)=C(Cl)-CO-O-cyclobutyl, -C(CH₃)=C(Cl)-CO-O-cyclopentyl, -C(CH₃)=C(Cl)-CO-O-cyclohexyl, -C(CH₃)=C(Cl)-CO-O-cycloheptyl, -C(CH₃)=C(Br)-COOH, -C(CH₃)=C(Br)-CO-OCH₃, -C(CH₃)=C(Br)-CO-OC₂H₅, -C(CH₃)=C(Br)-CO-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-O-n-C₄H₉, -C(CH₃)=C(Br)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-O-cyclopropyl, -C(CH₃)=C(Br)-CO-O-cyclobutyl, -C(CH₃)=C(Br)-CO-O-cyclopentyl, -C(CH₃)=C(Br)-CO-O-cyclohexyl, -C(CH₃)=C(Br)-CO-O-cycloheptyl, -C(CH₃)=C(CN)-COOH, -C(CH₃)=C(CN)-CO-OCH₃, -C(CH₃)=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CN)-CO-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-O-n-C₄H₉, -C(CH₃)=C(CN)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-O-cyclopropyl, -C(CH₃)=C(CN)-CO-O-cyclobutyl, -C(CH₃)=C(CN)-CO-O-cyclopentyl, -C(CH₃)=C(CN)-CO-O-cyclohexyl, -C(CH₃)=C(CN)-CO-O-cycloheptyl, -C(CH₃)=CH-CO-OCH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-OCH(CH₃)-OCH₃, -C(CH₃)=CH-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=CH-CO-OCH₂CH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(C₂H5)-CO-OCH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=(C₂H₅)-CO-OCH₂CH₂-OCH₃, -(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-O-i-C₃H₇, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(cl)-CO-OCH(CH₃)-OC₂H₅, -(CH₃)=C(Cl)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-O-i-C₃H₇, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃)=C(CN)-CO-O-i-C₃H₇, -C(CH₃)=C(CN)-CO-OCH(CH₃)OCH₃, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-CF₃, -C(CH₃)=CH-CO-OCH₂-CCl₃, -C(CH₃)=CH-CO-OCH₂-oxiranyl, -C(CH₃)=CH-CO-(CH₂)₃-Br,-C(CH₃)=CH-CO-OCH₂-CH=CH₂, -C(CH₃)=CH-CO-OCH₂-C≡CH, -C(CH₃)=CH-CO-OCH₂-CN, -C(CH₃)=CH-CO-OCH₂CH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CF₃, -C(CH₃)=C(CH₃)-CO-OCH₂-CCl3, -C(CH₃)=C(CH₃)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CH₃)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CH₃)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CH₃)-CO-OCH₂-C≡CH, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CF₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CCl₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-oxiranyl, -C(CH₃)=C(C₂H₅)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(C₂H₅)CO-OCH₂-C≡CH, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂-CF₃, -C(CH₃)=C(Cl)-CO-OCH₂-CCl₃, -C(CH₃)=C(Cl)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Cl)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(CL)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Cl)-CO-OCH₂-C≡CH, -C(CH₃)=C(Cl)-CO-OCH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂-CF₃, -C(CH₃)=C(Br)-CO-OCH₂-CCl₃, -C(CH₃)=C(Br)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Br)-CO-O(CH₂)₃-Br, -C(CH₃)=C(Br)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Br)-CO-OCH₂-C≡CH, -C(CH₃)=C(Br)-CO-OCH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂CH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂-CF₃, -C(CH₃)=C(CN)-CO-OCH₂-CCl₃, -C(CH₃)=C(CN)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CN)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CN)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CN)-CO-OCH₂-C≡CH, -C(CH₃)=C(CN)-CO-OCH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂CH₂-CN, -C(CH₃)=CH-CO-CH₃, -C(CH₃)=CH-CO-C₂H₅, -C(CH₃)=CH-CO-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-n-C₄H₉, -C(CH₃)=CH-CO-tert.-C₄H₉, -C(CH₃)=CH-CO-CH₂Cl, -C(CH₃)=CH-CO-CH₂Br, -C(CH₃)=CH-CO-CHCl₂, -C(CH₃)=CH-CO-CH₂-OCH₃, -C(CH₃)=CH-CO-CH(OCH₃)₂, -C(CH₃)=CH-CO-CH₂-SCH₃, -C(CH₃)=C(CH₃)-CO-CH₃, -C(CH₃)=C(CH₃)CO-C₂H₅, -C(CH₃)=C(CH₃)-CO-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-CH₂Cl, -C(CH₃)=C(CH₃)-CO-CH₂Br, -C(CH₃)=C(CH₃)-CO-CHCl₂, -C(CH₃)=C(CH₃)-CO-CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-CH(OCH₃)₂, -C(CH₃)=C(CH₃)-CO-CH₂-SCH₃, -C(CH₃)=C(C₂H₅)-CO-CH₃, -C(CH₃)=C(C₂H₅)-CO-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-CH₂Cl, -C(CH₃)=C(C₂H₅)-CO-CH₂Br, -C(CH₃)=C(C₂H₅)-CO-CHCl₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-CH(OCH₃)₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-SCH₃, -C(CH₃)=C(Cl)-CO-CH₃, -C(CH₃)=C(Cl)-CO-C₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-n-C₄H₉, -C(CH₃)=C(Cl)-CO-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-CH₂Cl, -C(CH₃)=C(Cl)-CO-CHCl₂, -C(CH₃)=C(Cl(-CO-CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-CH(OCH₃)₂, -C(CH₃)=C(Cl)-CO-CH₂-SCH₃, -C(CH₃)=C(Br)-CO-CH₃, -C(CH₃)=C(Br)-CO-C₂H₅, -C(CH₃)=C(Br)-CO-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-n-C₄H₉, -C(CH₃)=C(Br)-CO-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-CH₂Cl, -C(CH₃)=C(Br)-CO-CH₂Br, -C(CH₃)=C(Br)-CO-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-CH(OCH₃)₂, -C(CH₃)=C(Br)-CO-CH₂-SCH₃, -C(CH₃)=C(CN)-CO-CH₃, -C(CH₃)=C(CN)-CO-C₂H₅, -C(CH₃)=C(CN)-CO-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-n-C₄H₉, -C(CH₃)=C(CN)-CO-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-CH₂Cl, -C(CH₃)=C(CN)-CO-CH₂Br, -C(CH₃)=C(CN)-CO-CHCl₂, -C(CH₃)=C(CN)-CO-CH₂-OCH₃, -C(CH₃)=C(CN)-CO-CH(OCH₃)₂, -C(CH₃)=C(CN)-CO-CH₂-SCH₃, -C(CH₃)=CH-CO-C₆H₅, -C(CH₃)=CH-CO-(4-Cl-C₆H₄), -C(CH₃)=C(CH₃)-CO-C₆H₅, -C(CH₃)=C(CH₃)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(C₂H₅)-CO-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(Cl)-CO-C₆H₅, -C(CH₃)=C(Br)-CO-C₆H₅, -C(CH₃)=C(CN)-CO-C₆H₅, -C(CH₃)=CH-CO-NH₂, -C(CH₃)=CH-CO-NHCH₃, -C(CH₃)=CH-CO-N(CH₃)₂, -C(CH₃)=CH-CO-NH-C₂H₅, -C(CH₃)=CH-CO-N(C₂H₅)₂, -C(CH₃)=CH-CO-NH-n-C₃H₇, -C(CH₃)=CH-CO-NH-i-C₃H₇, -C(CH₃)=CH-CO-NH-tert.-C₄H₉, -C(CH₃)=CH-CO-NH-cyclopropyl, -C(CH₃)=CH-CO-NH-cyclobutyl, -C(CH₃)=CH-CO-NH-cyclopentyl, -C(CH₃)=CH-CO-NH-cylohexyl, -C(CH₃)=CH-CO-NH-cycloheptyl, -C(CH₃)=CH-CO-NH-cyclooctyl, -C(CH₃)=CH-CO-pyrrolidin-1-yl, -C(CH₃)=CH-CO-piperidin-1-yl, -C(CH₃)=CH-CO-morpholin-4-yl, -C(CH₃)=CH-CO-NH-CH₂CH=CH₂, -C(CH₃)=CH-CO-NH-CH₂C≡CH, -C(CH₃)=CH-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=CH-CO-NH-(CH₂)₂Cl, -C(CH₃)=CH-CO-NH-C₆H₅, -C(CH₃)=C(CH₃)-CO-NH₂, -C(CH₃)=C(CH₃)-CO-NHCH₃, -C(CH₃)=C(CH₃)-CO-N(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-C₂H₅, -C(CH₃)=C(CH₃)-CO-N(C₂H₅)₂, -C(CH₃)=C(CH₃)-CO-NH-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-NH- cyclopropyl, -C(CH₃)=C(CH₃)-CO-NH-cyclobutyl, -C(CH₃)=C(CH₃)-CO-NH-cyclopentyl, -C(CH₃)=C(CH₃)-CO-NH- cyclohexyl, -C(CH₃)=C(CH₃)-CO-NH-cycloheptyl, -C(CH₃)=C(CH₃)-CO-NH-cyclooctyl, -C(CH₃)=C(CH₃)-CO- pyrrolidin-1-yl, -C(CH₃)=C(CH₃)-CO-piperidin-1-yl, -C(CH₃)=C(CH₃)-CO-morpholin-4-yl, -C(CH₃)=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-NH(CH₂)₂Cl, -C(CH₃)=C(CH₃)-CO-NH-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-NH₂, -C(CH₃)=C(C₂H₅)-CO-NHCH₃, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)₂, -C(CH₃)=C(C₂H₅)-CO-NH-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-N(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-NH- cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclo­ hexyl, -C(CH₃)=C(C₂H₅)-CO-NH-cycloheptyl, -C(CH₃)=C(C₂H₅)-CO-NH- cyclooctyl, -C(CH₃)=C(C₂H₅)-CO-pyrrolidin-1-yl, -C(CH₃)=C(C₂H₅)-CO-piperidin-1-yl, -C(CH₃)=C(C₂H₅)-CO- morpholin-4-yl, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(C₂H₅)-CO-NH-C₆H₅, -C(CH₃)=C(Cl)-CO-NH₂, -C(CH₃)=C(CH₃)=C(Cl)-CO-NHCH₃, -C(CH₃)=C(Cl)-CO-N(CH₃)₂, -C(CH₃)=C(Cl)-CO-NH-C₂H₅, -C(CH₃)=C(Cl)-CO-N(C₂H₅)₂, -C(CH₃)=C(Cl)-CO-NH-n-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-i-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-NH-cyclopropyl, -C(CH₃)=C(Cl)-CO-NH-cyclobutyl, -C(CH₃)=C(Cl)-CO-NH-cyclopentyl, -C(CH₃)=C(Cl)-CO-NH-cyclohexyl, -C(CH₃)=C(Cl)-CO-NH-cycloheptyl, -C(CH₃)=C(Cl)-CO-NH-cyclooctyl, -C(CH₃)=C(Cl)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Cl)-CO-piperidin-1- yl, -C(CH₃)=C(Cl)-CO-morpholin-4-yl, -C(CH₃)=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -C(CH₃)=C(Cl)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-N(CH₃)-CH₂≡CH₂C, -C(CH₃)=C(Cl)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Cl)-NO-NH-C₆H₅, -C(CH₃)=C(Br)-CO-NH₂, -C(CH₃)=C(Br)-CO-NHCH₃, -C(CH₃)=C(Br)-CO-N(CH₃)₂, -C(CH₃)=C(Br)-CO-NH-C₂H₅, -C(CH₃)=C(Br)-CO-N(C₂H₅)₂, -C(CH₃)=C(Br)-CO-NH-n-C₃H₇, -C(CH₃)=C(Br)-CO-NH-i-C₃H₇, -C(CH₃)=C(Br)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-NH-cyclopropyl, -C(CH₃)=C(Br)-CO-NH-cyclobutyl, -C(CH₃)=C(Br)-CO-NH-cyclopentyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cycloheptyl, -C(CH₃)=C(Br)-CO-NH-cyclooctyl, -C(CH₃)=C(Br)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Br)-CO-piperidin-1-yl, -C(CH₃)=C(Br)-CO-morpholin-4-yl, -C(CH₃)=C(Br)-CO-NH-CH₂CH=C(CH₃)=C(Br)-CO-NH-CH₂C≡CH, -C(CH₃)=C(BR)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Br)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Br)-CO-NH-C₆H₅, -C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CN)-CO-NHCH₃, -C(CH₃)=C(CN)-CO-N(CH₃)₂, -C(CH₃)=C(CN)-CO-NH-C₂H₅, -C(CH₃)=C(CN)-CO-N(C₂H₅)₂, -C(CH₃)=C(CN)-CO-NH-n-C₃H₇, -C(CH₃)=C(CN)-CO-NH-i-C₃H₇, -C(CH₃)=C(CN)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-NH-cyclopropyl, -C(CH₃)=C(CN)-CO-NH-cyclobutyl, -C(CH₃)=C(CN)-CO-NH-cyclopentyl, -C(CH₃)=C(CN)-CO-NH-cyclohexyl, -C(CH₃)=C(CN)-CO-NH-cycloheptyl, -C(CH₃)=C(CN)-CO-NH-cyclooctyl, -C(CH₃)=C(CN)-CO-pyrrolidin-1-yl, -C(CH₃)=C(CN)-CO-piperidin-1-yl, -C(CH₃)=C(CN)-CO-morpholin-4-yl, -C(CH₃)=C(CN)-CO-NH-CH₂CH=C(CN)₂, -C(CH₃)=C(CN)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CN)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)=(CN)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CN)-CO-NH-C₆H₅, -C(CH₃)=CH-SO-SCH₃, -C(CH₃)=CH-CO-SC₂H₅, -C(CH₃)=CH-CO-S-n-C₃H₇, -C(CH₃)=CH-CO-S-i-C₃H₇, -C(CH₃)=CH-CO-S-n-C₄H₉, -C(CH₃)=CH-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-SCH₃, -C(CH₃)=C(CH₃)-CO-SC₂H₅, -C(CH₃)=C(CH₃)CO-S-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-S-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-SCH₃, -C(CH₃)=C(C₂H₅)-CO-SC₂H₅, -C(CH₃)=C(C₂H₅)-CO-S-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-SCH₃, -C(CH₃)=C(Cl)-CO-SC₂H₅, -C(CH₃)=C(Cl)-CO-S-n-C₃H₇, -C(CH₃)=C(Cl)-CO-S-i-C₃H₇, -C(CH₃)=C(Cl)-CO-S-n-C₄H₉, -C(CH₃)=C(Cl)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-SCH₃, -C(CH₃)=C(Br)-CO-SC₂H₅, -C(CH₃)=C(Br)-CO-S-n-C₃H₇, -C(CH₃)=C(Br)-CO-S-i-C₃H₇, -C(CH₃)=C(Br)-CO-S-n-C₄H₉, -C(CH₃)=C(Br)-CO-S-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-SCH₃, -C(CH₃)=C(CN)-CO-SC₂H₅, -C(CH₃)=C(CN)-CO-S-n-C₃H₇, -C(CH₃)=Ck(CN)-CO-S-i-C₃H₇, -C(CH₃)=C(CN)-CO-S-n-C₄H₉, -C(CH₃)=C(CN)-CO-S-tert.-C₄H₉, -C(CH₃)=C(COCH₃)-CO-OCH₃, -C(CH₃)=C(COC₂H₅)-CO-OCH₃, -C(CH₃)=C(CO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COCH₃)-CO-OC₂H₅, -C(CH₃)=C(COC₂H₅)-CO-OC₂H₅, -C(CH₃)=C(CO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COCH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(COC₂H₅)-CO-O-N-C₃H₇, -C(CH₃)=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-OCH₃, -C(CH₃)=C(CF₃)-CO-OC₂H₅, -C(CH₃)=C(CF₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CF₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(COOCH₃)₂, -C(CH₃)=C(COOC₂H₅)₂, -C(CH₃)=C(COOCH₃)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)₂, -C(CH₃)=CH-CH=CH-COOH, -C(CH₃)=CH-CH=CH-CO-OCH₃, -C(CH₃)=CH-CH=CH-CO-OC₂H₅, -C(CH₃)=CH-CH=C(COOCH₃)₂, -C(CH₃)=CH-CH=C(CN)-CO-OCH₃, -C(CH₃)=CH-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CN)CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -C(CH₃)=C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -C(CH₃)=CH-(CH₂)₂-COOH, -C(CH₃)=CH-(CH₂)₂-CO-OCH₃, -C(CH₃)=CH-(CH₂)₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(COOCH₃)₂, -C(CH₃)=CH-CH₂-CH(COOH₂H₅)₂, -C(CH₃)=CH-CH₂-CN(CN)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CN)-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -C(CH₃)=CH-(CH₂)₂-CO-NH₂, -C(CH₃)=CH-(CH₂)₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-COOH, -C(CH₃)=CH-CH₂-CO-OCH₃, -C(CH₃)=CH-CH₂-CO-OC₂H₅, -C(CH₃)=C(COOCH₃)-CH₂-CO-OCH₃, -C(CH₃)=C(COOCH₃)-CH₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CO-NH₂, -C(CH₃)=CH-CH₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-CO-N(CH₃)₂.
wobei W für eine der folgenden Bedeutungen steht:
-CHO, -COCH₃, -COC₂H₅, -CO-n-C₃H₇, -CO-i-C₃H₇, -CO-n-C₄H₉, -CO-i-C₄H₉, -CO-s-C₄H₉, -CO-tert.-C₄H₉, -CO-CH₂CH=CH₂, -CO-CF₃, -COCCl₃, -COCH₂C≡CH, -CO-cyclopropyl, -CO-cyclobutyl, -CO-cyclopentyl, -CO-cyclohexyl, -CO-CN, -CO-COOCH₃, -CO-COOC₂H₅, -CH=NH, -CH=NCH₃, -CH=NC₂H₅, -CH=N-n-C₃H₅, -CH=N-i-C₃H₅, -CH=N-n-C₄H₉, -CH=NCH₂CH=CH₂, -CH=NCH₂CH=CH₂-CH₃, -CH=NCH₂≡CH, -CH=NCH₂C≡C-CH₃, -CH=N-cyclopropyl, -CH=N-cyclobutyl, -CH=N-cyclopentyl, -CH=N-cyclohexyl, -CH=N-cycloheptyl, -CH=N-CH₂-CH₂Cl, -CH=N-CH₂Cl, -CH=N-C₆H₅, -CH=N-(4-Br-C₆H₄), -CH=N-3-F-C₆H₄, -CH=N-4-F-C₆H₄, -CH=N-2-Cl-C₆H₄, -CH=N-3-Cl-C₆H₄, -CH=N-4-Cl-C₆H₄, -CH=N-2-Br-C₆H₄, -CH=N-2-F-C₆H₄, -CH=N-2-CH₃-C₆H₄, -CH=N-3-CH₃-C₆H₄, -CH=N-4-CH₃-C₆H₄, -CH=N-2-CF₃-C₆H₄, -CH=N-3-CF₃-C₆H₄, -CH=N-4-CF₃-C₆H₄, -CH=N-2-OCH₃-C₆H₄, -CH=N-3-OCH₃-C₆H₄, -CH=N-4-OCH₃-C₆H₄, -CH=N-4-NO₂-C₆H₄, -CH=N-4-CN-C₆H₄, -CH=N-2,4-(Cl,Cl)-C₆H₄, -CH=N-2,4-(CH₃,CH₃)-C₆H₄, -CH=N-CH₂OCH₃ -CH=N-CH₂OC₂H₅, -CH=N-CH₂CH₂OCH₃, -CH=N-CH₂CH₂OC₂H₅, -CH=N-OH, -CH=N-OCH₃, -CH=N-OC₂H₅, -CH=N-O-n-C₃H₇, -CH=N-O-i-C₃H₇, -CH=N-O-n-C₄H₉, -CH=N-O-i-C₄H₉, -CH=N-O-s-C₄H₉, -CH=N-O-tert.-C₄H₉, -CH=N-O-CH₂CH=CH₂, -CH=N-O-CH(CH₃)CH=CH₂, -CH=N-O-CH₂C≡CH, -CH=N-O-CH(CH₃)-C≡CH, -CH=N-O-CH₂-CH=CH-CH₃, -CH=N-O-CH₂-CH₂-Cl, -CH=N-O-CH₂-CH₂-F, -CH=N-O-CH₂-CF₃, -CH=N-O-CH₂-CH=CHCl, -CH=N-O-CH₂-CCl=CH₂, -CH=N-O-CH₂-CBr=CH₂, -CH=N-O-CH₂-CH=CCl-CH₃, -CH=N-OC(O)CH₃, -CH=N-OC(O)C₂H₅, -CH=N-O-CH₂-CN, -CH=N-O-CH₂-CH=CH-CH₂-O-CH₃, -CH=N-O-CH₂-CH=CH-CH₂-O-tert.-C₄H₉, -CH=N-O-(CH₂)₃-C₆H₅, -CH=N-O-(CH₂)₄-C₆H₅, -CH=N-O-(CH₂)₄-4-Cl-C₆H₄, -CH=N-O-(CH₂)₄-4-OCH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-CH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-C₆H₅, -CH=N-O-CH₂CH=CH-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CH-3-OCH₃-C₆H₄, -CH=N-O-(CH₂)₂CH=CH-4-F-C₆H₄, -CH=N-O-(CH₂)CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CHCH₂-4-OCH₃-C₆H₄, -CH=N-O-CH₂-CH=C(CH₃)-C₆H₅ -CH=N-O-(CH₂)₂CH=CH-3,4(Cl,Cl)-C₆H₃, -CH=N-O-(CH₂)₃C≡C-4-F-C₆H₄, -CH₂=N-OCHOCH₃, -CH=N-OC₂H₄OCH₃, -CH=N-OCH₂OC₂H₅, -CH=N-OCH(CH₃)OCH₃, -CH=N-OCH(CH₃)COOCH₃, -CH=N-OCH(CH₃)COO-n-C₄H₉, -CH=N-NH₂, -CH=N-NHCH₃, -CH=N-NHC₂H₅, -CH=N-NH-n-C₃H₇, -CH=N-NH-i-C₃H₇, -CH=N-NH-n-C₄H₉, -CH=N-NH-cyclopropyl, -CH=N-NH-cyclobutyl, -CH=N-NH-cyclopentyl, -CH=N-NH-cyclohexyl, -CH=N-NH-cycloheptyl, -CH=N-N(CH₃)₂, -CH=N-N(C₂H₅)₂, -CH=N-N(C₃H₇)₂, -CH=N-N(i-C₃H₇)(CH₃), -CH=N-NHCH₂-C=CH, -CH=N-NHCH₂-C≡CH, -CH=N-N(CH₃)-CH₂-C≡CH, -CH=N-NHCH₂CF₃, -CH=N-NH-CO-CH₃, -CH=N-NH-CO-CH₂H₅, -CH=N-NH-COOCH₃, -CH=N-NH-COOC₂H₅, -CH=N-NH-COO-tert.-C₄H₉, -CH=N-pyrrolidin-1-yl, -CH=N-piperidin-1-yl, -CH=N-morpholin-4-yl, -CH=N-NH-C₆H₅, -CH=N-NH-(4-Cl-C₆H₄), -CH=N-NH-(4-NO₂-C₆H₄), -CH=N-NH-(4-F-C₆H₄), -CH=N-NH-(4-CH₃O-C₆H₄), -CH=N-NH-(2,4-Cl₂-C₆H₃), -CH=N-NH-(2,4-(NO₂)₂-C₆H₃), -CH=N-NH-CO-NH₂, -CH=N-NH-CO-NHCH₃, -CH=N-NH-CO-NHC₂H₅, -CH=N-NH-CO-N(CH₃)₂, -CH=CH-COOH, -CH=CH- CO-OCH₃, -CH=C-CO-OC₂H₅, -CH=CH-CO-O-n-C₃H₇, -CH=CH-CO-O-i-C₃H₇, -CH=CH-CO-O-n-C₄H₉, -CH=CH-CO-O-tert.-C₄H₉, -CH=CH-CO-O-cyclopropyl, -CH=CH-CO-O-cyclobutyl, -CH=CH-CO-O-cycloheptyl, -CH=C(CH₃)-COOH, -CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CO-O-n-C₃H₇, -CH=C(CH₃)-CO-O-i-C₃H₇, -CH=C(CH₃)-CO-O-n-C₄H₉, -CH=C(CH₃)-CO-O-tert.-C₄H₉, -CH=C(CH₃)-CO-O-cyclopropyl, -CH=C(CH₃)-CO-O-cyclobutyl, -CH=C(CH₃)-CO-O-cyclopentyl, -CH=C(CH₃)-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cycloheptyl, -CH=C(C₂H₅)-COOH, -CH=C(C₂H₅)-CO-OCH₃, -CH=C(C₂H₅)-CO-OC₂H₅, -CH=C(C₂H₅)-CO-O-n-C₃H₇, -CH=C(C₂H₅)-CO-O-i-C₃H₇, -CH=C(C₂H₅)-CO-O-n-C₄H₉, -CH=C(C₂H₅)-CO-O-tert.-C₄H₉, -CH=C(C₂H₅)-CO 99999 00070 552 001000280000000200012000285919988800040 0002004131038 00004 99880 äO-cyclopentyl, -CH=C(C₂H₅)-CO-O-cyclohexyl, -CH=C(C₂H₅)-CO-O-cycloheptyl, -CH=C(Cl)-COOH, -CH=C(Cl)-CO-OCH₃, -CH=C(Cl)-CO-OC₂H₅, -CH=C(Cl)-CO-O-n-C₃H₇, -CH=C(Cl)-CO-O-i-C₃H₇, -CH=C(Cl)-CO-O-n-C₄H₉, -CH=C(Cl)-CO-O-tert.-C₄H₉, -CH=C(Cl)-CO-O-cyclopropyl, -CH=C(Cl)-CO-O-cyclobutyl, -CH=C(Cl)-CO-O-cyclopentyl, -CH=C(Cl)-CO-O-cyclohexyl, -CH=C(Cl)-CO-O-cycloheptyl, -CH=C(Br)-COOH, -CH=C(Br)-CO-OCH₃, -CH=C(Br)-CO-OC₂H₅, -CH=C(Br)-CO-O-n-C₃H₇, -CH=C(Br)-CO-O-i-C₃H₇, -CH=C(Br)-CO-O-n-C₄H₉, -CH=C(Br)-CO-O-tert.-C₄H₉, -CH=C(Br)-CO-O-cyclopropyl, -CH=C(Br)-CO-O-cyclobutyl, -CH=C(Br)-CO-O-cyclopentyl, -CH=C(Br)-CO-O-cyclohexyl, -CH=C(Br)-CO-O-cycloheptyl, -CH=C(CN)-COOH, -CH=C(CN)-CO-OCH₃, -CH=C(CN)-CO-OC₂H₅, -CH=C(CN)-CO-O-n-C₃H₇, -CH=C(CN)-CO-O-i-C₃H₇, -CH=C(CN)-CO-O-n-C₄H₉, -CH=C(CN)-CO-O-tert.-C₄H₉, -CH=C(CN)-CO-O-cyclopropyl, -CH=C(CN)-CO-O-cyclobutyl, -CH=C(CN)-CO-O-cyclopentyl, -CH=C(CN)-CO-O-cyclohexyl, -CH=C(CN)-CO-O-cycloheptyl, -CH=CH-CO-OCH₂-OCH₃, -CH=CH-CO-OCH₂-OC₂H₅, -CH=CH-CO-OCH₂-O-n-C₃H₅, -CH=CH-CO-OCH₂-O-i-C₃H₅, -CH=CH-CO-OCH(CH₃)-OCH₃, -CH=CH-CO-OCH(CH₃)-OC₂H₅, -CH=CH-CO-O-CH₂CH₂-OCH₃, -CH=CH-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-OCH₃, -CH=C(CH₃)-CO-OCH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-O-n-C₃H₅, -CH=C(CH₃)-CO-OCH₂-O-i-C₃H₅, -CH=C(CH₃)-CO-OCH(CH₃)-OCH₃, -CH=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CH₃)-CO-O-CH₂CH₂-OCH₃, -CH=C(CH₃)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-OCH₃, -CH=C(C₂H₅)-CO-OCH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-O-n-C₃H₅, -CH=C(C₂H₅)-CO-OCH₂-O-i-C₃H₅, -CH=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-OCH₃, -CH=C(Cl)-CO-OCH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-O-n-C₃H₅, -CH=C(Cl)-CO-OCH₂-O-i-C₃H₅, -CH=C(Cl)-CO-OCH(CH₃)-OCH₃, -CH=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Cl)-CO-O-CH₂CH₂-OCH₃, -CH=C(Cl)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-OCH₃, -CH=C(Br)-CO-OCH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-O-n-C₃H₅, -CH=C(Br)-CO-OCH₂-O-i-C₃H₅, -CH=C(Br)-CO-OCH(CH₃)-OCH₃, -CH=C(Br)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Br)-CO-O-CH₂CH₂-OCH₃, -CH=C(Br)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-OCH₃, -CH=C(CN)-CO-OCH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-O-n-C₃H₅, -CH=C(CN)-CO-OCH₂-O-i-C₃H₅, -CH=C(CN)-CO-OCH(CH₃)-OCH₃, -CH=C(CN)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CN)-CO-O-CH₂CH₂-OCH₃, -CH=C(CN)-CO-O-CH₂CH₂-OC₂H₅, -CH=CH-CO-OCH₂-CF₃, -CH=CH-CO-OCH₂-CCl₃, -CH=CH-CO-OCH₂-oxiranyl, -CH=CH-CO-O(CH₂)₃-Br, -CH=CH-CO-OCH₂-CH=CH₂, -CH=CH-CO-OCH₂-C≡CH, -CH=CH-CO-OCH₂-CN, -CH=CH-CO-O(CH₂)₂-CN, -CH=C(CH₃)-CO-OCH₂-CF₃, -CH=C(CH₃)-CO-OCH₂-CCl₃, -CH=C(CH₃)-CO-OCH₂-oxiranyl, -CH=C(CH₃)-CO-O(CH₂)₃-Br, -CH=C(CH₃)-CO-OCH₂-CH=CH₂, -CH=C(CH₃)-CO-OCH₂-C≡CH, -CH=C(CH₃)-CO-OCH₂-CN, -CH=C(CH₃)-CO-O(CH₂)₂-CN, -CH=C(C₂H₅)-CO-OCH₂-CF₃, -CH=C(C₂H₅)-CO-OCH₂-CCl₃, -CH=C(C₂H₅)-CO-OCH₂-oxiranyl, -CH=C(C₂H₅)-CO-O(CH₂)₃-Br, -CH=C(C₂H₅)-CO-OCH₂-CH=CH₂, -CH=C(C₂H₅)-CO-OCH₂-C≡CH, -CH=C(C₂H₅)-CO-OCH₂-CN, -CH=C(C₂H₅)-CO-O(CH₂)₂-CN, -CH=C(Cl)-CO-OCH₂-CF₃, -OH=C(Cl)-CO-OCH₂-CCl₃, -CH=C(Cl)-CO-OCH₂-oxiranyl, -CH=C(Cl)-CO-O(CH₂)₃-Br, -CH=C(Cl)-CO-OCH₂-CH=CH₂, -CH=C(Cl)-CO-OCH₂-C≡CH, -CH=C(Cl)-CO-OCH₂-CN, -CH=C(Cl)-CO-O(CH₂)₂-CN, -CH=C(Br)-CO-OCH₂-CF₃, -CH=C(Br)-CO-OCH₂-CCl₃, -CH=C(Br)-CO-OCH₂-oxiranyl, -CH=C(Br)-CO-O(CH₂)₃-Br, -CH=C(Br)-CO-OCH₂-CH=CH₂, -CH=C(Br)-CO-OCH₂-C≡CH, -CH=C(Br)-CO-OCH₂-CN, -CH=C(Br)-CO-O(CH₂)₂-CN, -CH=C(CN)-CO-OCH₂-CF₃, -CH=C(CN)-CO-OCH₂-CCl₃, -CH=C(CN)-CO-OCH₂-oxiranyl, -CH=C(CN)-CO-O(CH₂)₃-Br, -CH=C(CN)-CO-OCH₂-CH=CH₂, -CH=C(CN)-CO-OCH₂-C≡CH, -CH=C(CN)-CO-OCH₂-CN, -CH=C(CN)-CO-O(CH₂)₂-CN, -CH=CH-CO-CH₃, -CH=CH=CO-C₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-i-C₃H₇, -CH=CH-CO-n-C₄H₉, -CH=CH-CO-tert.-C₄H₉, -CH=CH-CO-CH₂Cl, -CH=CH-CO-CH₂Br, -CH=CH-CO-CHCl₂, -CH=CH-CO-CH₂-OCH₃, -CH=CH-CO-CH(OCH₃)₂, -CH=CH-CO-CH₂-SCH₃, -CH=C(CH₃)-CO-CH₃, -CH=C(CH₃)-CO-C₂H₅, -CH=C(CH₃)-CO-n-C₃H₇, -CH=C(CH₃)-CO-i-C₃H₇, -CH=C(CH₃)-CO-n-C₄H₉, -CH=C(CH₃)-CO-tert.-C₄H₉, -CH=C(CH₃)-CO-CH₂Cl, -CH=C(CH₃)-CO-CH₃Br, -CH=C(CH₃)-CO-CHCl₂, -CH=C(CH₃)-CO-CH₂-OCH₃, -CH=C(CH₃)-CO-CH(OCH₃)₂, -CH=C(CH₃)-CO-CH₂-SCH₃, -CH=C(C₂H₅)-CO-CH₃, -CH=C(C₂H₅)-CO-C₂H₅, -CH=C(C₂H₅)-CO-n-C₃H₇, -CH=C(C₂H₅)-CO-i-CH₃H₇, -CH=C(C₂H₅)-CO-n-C₄H₉, -CH=C(C₂H₅)-CO-tert.-C₄H₉, -CH=C(C₂H₅)-CO-CH₂Cl, -CH=C(C₂H₅)-CO-CH₂Br, -CH=C(C₂H₅)-CO-CHCl₂, -CH=C(C₂H₅)-CO-CH₂-OCH₃, -CH=C(C₂H₅)-CO-CH(OCH₃)₂, -CH=C(C₂H₅)-CO-CH₂-SCH₃, -CH=C(Cl)-CO-CH₃, -CH=C(Cl)-CO-C₂H₅, -CH=C(Cl)-CO-n-C₃H₇, -CH=C(Cl)-CO-i-C₃H₇, -CH=C(Cl)-CO-n-C₄H₉, -CH=C(Cl)-CO-tert.-C₄H₉, -CH=C(Cl)-CO-CH₂Cl, -CH=C(Cl)-CO-CH₂Br, -CH=C(Cl)-CO-CHCl₂, -CH=C(Cl)-CO-CH₂-OCH₃, -CH=C(Cl)-CO-CH(OCH₃)₂, -CH=C(Cl)-CO-CH₂-SCH₃, -CH=C(Br)-CO-CH₃, -CH=C(Br)-CO-C₂H₅, -CH=C(Br)-CO-n-C₃H₇, -CH=C(Br)-CO-i-C₃H₇, -CH=C(Br)-CO-n-C₄H₉, -CH=C(Br)-CO-tert.-C₄H₉, -CH=C(Br)-CO-CH₂Cl, -CH=C(Br)-CO-CH₂Br, -CH=C(Br)-CO-CHCl₂, -CH=C(Br)-CO-CH₂-OCH₃, -CH=C(Br)-CO-CH(OCH₃)₂, -CH=C(Br)-CO-CH₂-SCH₃, -CH=C(CN)-CO-CH₃, -CH=C(CN)-CO-C₂H₅, -CH=C(CN)-CO-n-C₃H₇, -CH=C(CN)-CO-i-C₃H₇, -CH=C(CN)-CO-n-C₄H₉, -CH=C(CN)-CO-tert.-C₄H₉, -CH=C(CN)-CO-CH₂Cl, -CH=C(CN)-CO-CH₂Br, -CH=C(CN)-CO-CHCl₂, -CH=C(CN)-CO-CH₂-OCH₃, -CH=C(CN)-CO-CH(OCH₃)₂, -CH=C(CN)-CO-CH₂-SCH₃, -CH=CH-CO-C₆H₅, -CH=CH-CO-(4-Cl-C₆H₄), -CH=C(CH₃)-CO-C₆H₅, -CH=C(CH₃)-CO-(4-Cl-C₆H₄), -CH=C(C₂H₅)-CO-C₆H₅, -CH=C(C₂H₅-CO-(4-Cl-C₆H₄), -CH=C(Cl)-CO-C₆H₅, -CH=C(Br)-CO-C₆H₅, -CH=C(CN)-CO-C₆H₅, -CH=CH-CO-NH₂, -CH=CH-CO-NHCH₃, -CH=CH-CO-N(CH₃)₂, -CH=CO-NH-C₂H₅, -CH=CH-CO-N(C₂H₅)₂, -CH=CH-CO-NH-n-C₃H₇, -CH=CH-CO-NH-i-C₃H₇, -CH=CH-CO-NH-tert.-C₄H₉, -CH=CH-CO-NH-cyclopropyl, -CH=CH-CO-NH-cyclobutyl, -CH=CH-CO-NH-cyclopentyl, -CH=CH-CO-NH-cyclohexyl, -CH=CH-CO-NH-cycloheptyl, -CH=CH-CO-NH-cyclooctyl, -CH=CH-CO-pyrrolidin-1-yl, -CH=CH-CO-piperidin-1-yl, -CH=CH-CO-morpholin-4-yl, -CH=CH-CO-NH-CH₂CH=CH₂, -CH=CH-CO-NH-CH₂C≡CH, -CH=CH-CO-N(CH₃)-CH₂C≡CH, -CH=CH-CO-NH-(CH₂)₂Cl, -CH=CH-CO-NH-C₆H₅, -CH≡C(CH₃)-CO-NH₂, -CH=(CH₃)-CO-NHCH₃, -CH=C(CH₃)-CO-N(CH₃)₂, -CH=C(CH₃)-CO-NH-C₂H₅, -CH=C(CH₃)-CO-N(C₂H₅)₂, -CH=C(CH₃)-CO-NH-n-C₃H₇, -CH=C(CH₃)-CO-NH-i-C₃H₇, -CH=C(CH₃)-CO-NH-tert.-C₄H₉, -CH=C(CH₃)-CO-NH-cyclopropyl, -CH=C(CH₃)-CO-NH-cyclobutyl, -CH=C(CH₃)-CO-NH-cyclopentyl, -CH=C(CH₃)-CO-NH-cyclohexyl, -CH=C(CH₃)-CO-NH-cycloheptyl, -CH=C(CH₃)-CO-NH-cyclooctyl, -CH=C(CH₃)-CO-pyrrolidin-1-yl, -CH=C(CH₃)-CO-piperidin-1-yl, -CH=C(CH₃)-CO-morpholin-4-yl, -CH=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -CH=C(CH₃)-CO-NH-CH₂C≡CH, -CH=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CH₃)-CO-NH-(CH₂)₂Cl, -CH=C(CH₃)-CO-NH-C₆H₅, -CH=C(C₂H₅)-CO-NH₂, -CH=C(C₂H₅)-CO-NHCH₃, -CH=C(C₂H₅)-CO-N(CH₃)₂, -CH=C(C₂H₅)-CO-NH-C₂H₅, -CH=C(C₂H₅)-CO-N(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-n-C₃H₇, -CH=C(C₂H₅)-CO-NH-i-C₃H₇, -CH=C(C₂H₅)-CO-NH-tert.-C₄H₉, -CH=C(C₂H₅)-CO-NH-cyclopropyl, -CH=C(C₂H₅)-CO-NH-cyclobutyl, -CH=C(C₂H₅)-CO-NH-cyclopentyl, -CH=C(C₂H₅)-CO-NH-cyclohexyl, -CH=C(C₂H₅)-CO-NH-cycloheptyl, -CH=C(C₂H₅)-CO-NH-cyclooctyl, -CH=C(C₂H₅)-CO-pyrrolidin-1-yl, -CH=C(C₂H₅)-CO-piperidin-1-yl, -CH=C(C₂H₅)-CO-morpholin-4-yl, -CH=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-CH₂≡CH, -CH=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -CH=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -CH=C(C₂H₅)-CO-NH-C₆H₅, -CH=C(Cl)-CO-NH₂, -CH=C(Cl)-CO-NHCH₃, -CH=C(Cl)-CO-N(CH₃)₂, -CH=C(Cl)-CO-NH-C₂H₅, -CH=C(Cl)-CO-N(C₂H₅)₂, -CH=C(Cl)-CO-NH-n-C₃H₇, -CH=C(Cl)-CO-NH-i-C₃H₇, -CH=C(Cl)-CO-NH-tert.-C₄H₉, -CH=C(Cl)-CO-NH-cyclopropyl, -CH=C(Cl)-CO-NH-cyclobutyl, -CH=C(Cl)-CO-NH-cyclopentyl, -CH=C(Cl)-CO-NH-cyclohexyl, -CH=C(Cl)-CO-NH-cycloheptyl, -CH=C(Cl)-CO-NH-cyclooctyl, -CH=C(Cl)-CO-pyrrolidin-1-yl, -CH=C(Cl)-CO-piperidin-1-yl, -CH=C(Cl)-CO-morpholin-4-yl, -CH=C(Cl)-CO-NH-CH₂CH=(Cl)₂, -CH=C(Cl)-CO-NH-CH₂C≡CH, -CH=C(Cl)-CO-NH(CH₃)-CH₂C≡CH, -CH=C(Cl)-CO-NH-(CH₂)₂Cl, -CH=C(Cl)-CO-NH-C₆H₅, -CH=C(Br)-CO-NH₂, -CH=C(Br)-CO-NH-NHCH₃, -CH=C(Br)-CO-N(CH₃)₂, -CH=C(Br)-CO-NH-C₂H₅, -CH=C(Br)-CO-N(C₂H₅)₂, -CH=C(Br)-CO-NH-n-C₃H₇, -CH=C(Br)-CO-NH-i-C₃H₇, -CH=C(Br)-CO-NH-tert.-C₄H₉, -CH=C(Br)-CO-NH-cyclopropyl, -CH=C(Br)-CO-NH-cyclobutyl, -CH=C(Br)-CO-NH-cyclopentyl, -CH=C(Br)-CO-NH-cyclohexyl, -CH=C(Br)-CO-NH-cycloheptyl, -CH=C(Br)-CO-NH-cyclooctyl, -CH=C(Br)-CO-pyrrolidin-1-yl, -CH=C(Br)-CO-piperidin-1-yl, -CH=C(Br)-CO-morpholin-4-yl, -CH=C(Br)-CO-NH-CH₂CH=C(Br)₂, -CH=C(Br)-CO-NH-CH₂C≡CH, -CH=C(Br)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Br)-CO-NH-(CH₂)₂Cl, -CH=C(Br)-CO-NH-C₆H₅, -CH=C(CN)-CO-NH₂, -CH=C(CN)-CO-NHCH₃, -CH=C(CN)-CO-N(CH₃)₂, -CH=C(CN)-CO-NH-C₂H₅, -CH=C(CN)-CO-N(C₂H₅)₂, -CH=C(CN)-CO-NH-n-C₃H₇, -CH=C(CN)-CO-NH-i-C₃H₇, -CH=C(CN)-CO-NH-tert.-C₄H₉, -CH=C(CN)-CO-NH-cyclopropyl, -CH=C(CN)-CO-NH-cyclobutyl, -CH=C(CN)-CO-NH-cyclopentyl, -CH=C(CN)-CO-NH-cyclohexyl, -CH=C(CN)-CO-NH-cycloheptyl, -CH=C(CN)-CO-NH-cyclooctyl, -CH=C(CN)-CO-pyrrolidin-1-yl, -CH=C(CN)-CO-piperidin-1-yl, -CH=C(CN)-CO-morpholin-4-yl, -CH=C(CN)-CO-NH-CH₂CH=C(CN)₂, -CH=C(CN)-CO-NH-CH₂C≡CH, -CH=C(CN)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CN)-CO-NH-(CH₂)₂Cl, -CH=C(CN)-CO-NH-C₆H₅, -CH=CH-CO-SCH₃, -CH=CH-CO-SC₂H₅, -CH=CH-CO-S-n-C₃H₇, -CH=CH-CO-S-i-C₃H₇, -CH=CH-CO-S-n-C₄H₉, -CH=CH-CO-S-tert.-C₄H₉, -CH=C(CH₃)-CO-SCH₃, -CH=C(CH₃)-CO-SC₂H₅, -CH=C(CH₃)-CO-S-n-C₃H₇, -CH=C(CH₃)-CO-S-i-C₃H₇, -CH=C(CH₃)-CO-S-n-C₄H₉, -CH=C(CH₃)-CO-S-tert.-C₄H₉, -CH=C(C₂H₅)-CO-SCH₃, -CH=C(C₂H₅)-CO-SC₂H₅, -CH=C(C₂H₅)-CO-S-n-C₃H₇, -CH=C(C₂H₅)-CO-S-i-C₃H₇, -CH=C(C₂H₅)-CO-S-n-C₄H₉, -CH=C(C₂H₅)-CO-S-tert.-C₄H₉, -CH=C(Cl)-CO-SCH₃, -CH=C(Cl)-CO-SC₂H₅, -CH=C(Cl)-CO-S-n-C₃H₇, -CH=C(Cl)-CO-S-i-C₃H₇, -CH=C(Cl)-CO-S-n-C₄H₉, -CH=C(Cl)-CO-S-tert.-C₄H₉, -CH=C(Br)-CO-SCH₃, -CH=C(Br)-CO-SC₂H₅, -CH=C(Br)-CO-S-n-C₃H₇, -CH=C(Br)-CO-S-i-C₃H₇, -CH=C(Br)-CO-S-n-C₄H₉, -CH=C(Br)-CO-S-tert.-C₄H₉, -CH=C(CN)-CO-SCH₃, -CH=C(CN)-CO-SC₂H₅, -CH=C(CN)-CO-S-n-C₃H₇, -CH=C(CN)-CO-S-i-C₃H₇, -CH=C(CN)-CO-S-n-C₄H₉, -CH=C(CN)-CO-S-tert.-C₄H₉, -CH=C(COCH₃)-CO-OCH₃, -CH=C(COC₂H₅)-CO-OCH₃, -CH=C(CO-n-C₃H₇)-CO-OCH₃, -CH=C(COCH₃)-CO-OC₂H₅, -CH=C(COC₂H₅)-CO-OC₂H₅, -CH=C(CO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COCH₃)-CO-O-n-C₃H₇, -CH=C(COC₂H₅)-CO-O-n-C₃H₇, -CH=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-OCH₃, -CH=C(CF₃)-CO-OC₂H₅, -CH=C(CF₃)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-O-i-C₃H₇, -CH=C(CF₃)-CO-O-n-C₄H₉, -CH=C(CF₃)-CO-O-tert.-C₄H₉, -CH=C(COOCH₃)₂, -CH=C(COOC₂H₅)₂, -CH=C(COOCH₃)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)-CO-OCH₃, -CH=C(COO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)₂, -CH=CH-CH=CH-COOH, -CH=CH-CH=CH-CO-OCH₃, -CH=CH-CH=CH-CO-OC₂H₅, -CH=CH-CH=C(COOCH₃)₂, -CH=CH-CH=C(CN)-CO-OCH₃, -CH=CH-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-OCH₃, -CH=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CH=C(Cl)-CO-OCH₃, -CH=C(CH₃)-CH=C(Br)-CO-OCH₃, -CH=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-NH₂, -CH=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -CH=CH-(CH₂)₂-COOH, -CH=CH-(CH₂)₂-CO-OCH₃, -CH=CH-(CH₂)₂-CO-OC₂H₅, -CH=CH-CH₂-CH(COOCH₃)₂, -CH=CH-CH₂-CH(COOC₂H₅)₂, -CH=CH-CH₂-CH(CN)-CO-OCH₃, -CH=CH-CH₂-CH(CN)-CO-OC₂H₅, -CH=CH-CH₂-CH(CH₃)-CO-OCH₃, -CH=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -CH=CH-(CH₂)₂-CO-NH₂, -CH=CH-(CH₂)₂-CO-NH-CH₃, -CH=CH-CH₂-COOH, -CH=CH-CH₂-CO-OCH₃, -CH=CH-CH₂-CO-OC₂H₅, -CH=C(COOCH₃)-CH₂-CO-OCH₃, -CH=C(COOCH₃)-CH₂-CO-OC₂H₅, -CH=CH-CH₂-CO-NH₂, -CH=CH-CH₂-CO-NH-CH₃, -CH=CH-CH₂-CO-N(CH₃)₂, -CH(OCH₃)₂, -CH(SCH₃)₂, -CH(OC₂H₅)₂, -CH(SC₂H₅)₂, -CH(O-n-C₃H₇)₂, -CH(O-i-C₃H₇)₂, -CH(S-n-C₃H₇)₂, -CH(S-i-C₃H₇)₂, -CH(O-n-C₄H₉)₂, -CH(O-i-C₄H₉)₂, -CH(O-s-C₄H₉)₂, -CH(O-tert.-C₄H₉)₂, -CH(S-n-C₄H₉)₂, -CH(S-i-C₄H₉)₂, -CH(S-s-C₄H₉)₂, -CH(S-tert.-C₄H₉)₂, -CH(OC₅H₁₁)₂, 1,3-Dioxolan-2-yl, 1,3-Dithiolan- 2-yl, 1,3-Oxathiolan-2-yl, 4-Methyl-1,3-dioxolan-2-yl, 4-Methyl-1,3-dithiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 5-Methyl-1,3-oxathiolan-2-yl, 4-Ethyl-1,3-dioxolan-2-yl, 4-Ethyl- 1,4-dithiolan-2-yl, 4-Ethyl-1,3-oxathiolan-2-yl, 5-Ethyl-1,3-oxathiolan- 2-yl, 4,5-Dimethyl-1,3-dioxolan-2-yl, 4,4-Dimethyl-1,3- dioxolan-2-yl, 4,5-Dimethyl-1,3-dithiolan-2-yl, 5,5-Dimethyl-1,3- dithiolan-2-yl, 4,5-Dimethyl-1,3-oxathiolan-2-yl, 5,5-Dimethyl- 1,3-oxathiolan-2-yl, 4,4-Dimethyl-1,3-oxathiolan-2-yl, 4-Vinyl- 1,3-dioxolan-2-yl, 4-Vinyl-1,3-dithiolan-2-yl, 4-Vinyl-1,3-oxathiolan- 2-yl, 5-Vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3- dioxolan-2-yl, 4-Chlormethyl-1,3-dithiolan-2-yl, 4-Chlormethyl- 1,3-oxathiolan-2-yl, 5-Chlormethyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-1,3-dithiolan- 2-yl, 4-Hydroxymethyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl- 1,3-oxathiolan-2-yl, 4-Methoxymethyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl- 1,3-dioxolan-2-yl, 4-Propargyloxymethyl-1,3-dioxolan- 2-yl, 4-Acetoxymethyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-1,3-dithiolan-2-yl, 4-Propargyloxymethyl- 1,3-dithiolan-2-yl, 4-Acetoxymethyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-1,3-oxathiolan- 2-yl, 4-Allyloxymethyl-1,3-oxathiolan-2-yl, 5-Allyloxymethyl- 1,3-oxathiolan-2-yl, 4-Propargyloxymethyl-1,3-oxathiolan- 2-yl, 5-Propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxymethyl- 1,3-oxathiolan-2-yl, 5-Acetoxymethyl-1,3-oxathiolan-2-yl, 4-Methylthiomethyl-1,3-dithiolan-2-yl, 4-Methylthiomethyl-1,3- dithiolan-2-yl, 4-Carboxy-1,3-dioxolan-2-yl, 4-Carboxy-1,3- dithiolan-2-yl, 4-Methoxycarbonyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl- 1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-1,3-dithiolan- 2-yl, 4-n-Butoxycarbonyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-4-methyl- 1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithiolan- 2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-1,3- dithiolan-2-yl, 1,3-Dioxan-2-yl, 1,3-Dithian-2-yl, 1,3-Oxathian- 2-yl, 5-Methyl-1,3-dioxan-2-yl, 5-Methyl-1,3-dithian-2-yl, 5-Methyl-1,3-oxathian-2-yl, 5,5-Dimethyl-1,3-dioxan-2-yl, 4,6-Dimethyl- 1,3-dioxan-2-yl, 4,4-Dimethyl-1,3-dioxan-2-yl, 5,5-Dimethyl- 1,3-dithian-2-yl, 4,6-Dimethyl-1,3-dithian-2-yl, 4,4-Dimethyl- 1,3-dithian-2-yl, 5,5-Dimethyl-1,3-oxathian-2-yl, 4,4-Dimethyl- 1,3-oxathian-2-yl, 6,6-Dimethyl-1,3-oxathian-2-yl, 4-Hydroxymethyl-1,3-dioxan-2-yl, 4-Methoxymethyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-1,3-dioxan-2- yl, 4-Hydroxymethyl-1,3-dithian-2-yl, 4-Methoxymethyl-1,3-dithian- 2-yl, 4-Allyloxymethyl-1,3-dithian-2-yl, 4-Acetoxymethyl- 1,3-dithian-2-yl, 4-Chlormethyl-1,3-dioxan-2-yl, 4-Chlormethyl- 1,3-dithian-2-yl, 1,3-Dioxepan-2-yl, 1,3-Dithiepan-2-yl, 1,3-Dioxep- 5-en-2-yl, 4-Methoxycarbonyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl- 1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-1,3-dithian- 2-yl, 4-n-Butoxycarbonyl-1,3-dithian-2-yl, 4-Methoxycarbonyl-4- methyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxan-2- yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl- 4-methyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-4-methyl- 1,3-dithian-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithian-2-yl, -C(CH₃)(OCH₃)₂, -C(CH₃)(SCH₃)₂, -C(CH₃)(OC₂H₅)₂, -C(CH₃)(SC₂H₅)₂, -C(CH₃)(O-n-C₃H₇)₂, -C(CH₃)(O-i-C₃H₇)₂, -C(CH₃)(S-n-C₃H₇)₂, -C(CH₃)(S-i-C₃H₇)₂, -C(CH₃)(O-n-C₄H₉)₂, -C(CH₃)(O-i-C₄H₉)₂, -C(CH₃)(O-s-C₄H₉)₂, -C(CH₃)(O-tert.-C₄H₉)₂, -C(CH₃)(S-n-C₄H₉)₂, -C(CH₃)(S-i-C₄H₉)₂, -C(CH₃)(S-s-C₄H₉)₂, -C(CH₃)(S-tert.-C₄H₉)₂, -C(CH₃)(O-n-C₅H₁₁)′′, 2-Methyl-1,3-dixolan-2-yl, 2-Methyl-1,3-dithiolan- 2-yl, 2-Methyl-1,3-oxathiolan-2-yl, 2,4-Dimethyl-1,3- dixolan-2-yl, 2,4-Dimethyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-1,3- oxathiolan-2-yl, 2,5-Dimethyl-1,3-oxathiolan-2-yl, 4-Ethyl-2- methyl-1,3-dioxolan-2-yl, 4-Ethyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Ethyl-2-methyl-1,3- oxathiolan-2-yl, 2,4,5-Trimethyl-1,3-dioxolan-2-yl, 2,4,4-Trimethyl- 1,3-dioxolan-2-yl, 2,4,5-Trimethyl-1,3-dithiolan-2-yl, 2,4,4-Trimethyl-1,3-dithiolan-2-yl, 2,4,5-Trimethyl-1,3-oxathiolan- 2-yl, 2,4,4-Trimethyl-1,3-oxathiolan-2-yl, 2-Methyl-4-vinyl- 1,3-dioxothiolan-2-yl, 2-Methyl-4-vinyl-1,3-dithiolan-2-yl, 2-Methyl- 4-vinyl-1,3-oxathiolan-2-yl, 2-Methyl-5-vinyl-1,3-oxathiolan-2- yl, 4-Chlormethyl-2-methyl-1,3-dioxolan-2-yl, 4-Chlormethyl-2- methyl-1,3-dithiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-oxathiolan- 2-yl, 5-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl- 2-methyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-2- methyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dioxolan- 2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxy- 2-methyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dithiolan-2-yl, 4-Acetoxy-2- methyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-oxathiolan- 2-yl, 5-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl- 2-methyl-1,3-oxathiolan-2-yl, 5-Allyloxymethyl-2- methyl-1,3-oxathiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3- oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3-oxathiolan-2- yl, 4 Acetoxy-2-methyl-1,3-oxathiolan-2-yl, 5-Acetoxy-2-methyl- 1,3-oxathiolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dioxolan-2- yl, 2-Methyl-4-methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-2- methyl-1,3-dioxolan-2-yl, 4-Carboxy-2-methyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-2- methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-2-methyl-1,3-dioxolan- 2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl- 2-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-2- methyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dioxolan- 2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-ethoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4- ethoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl- 1,3-dioxolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl-1,3- dithiolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-dioxan-2- yl, 2-Methyl-1,3-dithian-2-yl, 2-Methyl-1,3-oxathian-2-yl, 2,5- Dimethyl-1,3-dioxan-2-yl, 2,5-Dimethyl-1,3-dithian-2-yl, 2,5-Dimethyl- 1,3-oxathian-2-yl, 2,5,5-Trimethyl-1,3-dioxan-2-yl, 2,4,6- Trimethyl-1,3-dioxan-2-yl, 2,4,4-Trimethyl-1,3-dioxan-2-yl, 2,5,5-Trimethyl-1,3-dithian-2-yl, 2,4,6-Trimethyl-1,3-dithian-2- yl, 2,4,4-Trimethyl-1,3-dithian-2-yl, 2,5,5-Trimethyl-1,3-oxathian- 2-yl, 2,4,4-Trimethyl-1,3-oxathian-2-yl, 2,6,6-Trimethyl- 1,3-oxathian-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-2- methyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dithian-2-yl, 4-Methoxymethyl-2- methyl-1,3-dithian-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithian-2- yl, 4-Acetoxymethyl-2-methyl-1,3-dithian-2-yl, 4-Chlormethyl-2- methyl-1,3-dioxan-2-yl, 4-Chlormethyl-2-methyl-1,3-dithian-2-yl, -C(CH₃)=NH, -C(CH₃)=N-CH₃, -C(CH₃)=N-C₂H₅, -C(CH₃)=N-n-C₃H₇, -(CH₃)=N-i-C₃H₇, -C(CH₃)=N-n-C₄H₉, -C(CH₃)=N-CH₂CH=CH₂, -C(CH₃)=N-CH₂CH=CH₂-CH₃, -C(CH₃)=N-CH₂C≡CH, -C(CH₃)=N-CH₂C≡C-CH₃, -C(CH₃)=N-cyclopropyl, -C(CH₃)=N-cyclobutyl, -C(CH₃)=N-cyclopentyl, -C(CH₃)=N-cyclohexyl, -C(CH₃)=N-cycloheptyl, -C(CH₃)=N-CH₂-CH₂Cl, -C(CH₃)=N-CH₂Cl, -C(CH₃)=N-C₆H₅, -C(CH₃)=N-(2-F-C₆H₄), -C(CH₃)=N-(3-F-C₆H₄), -C(CH₃)=N-(4-F-C₆H₄), -C(CH₃)=N-(2-Cl-C₆H₄), -C(CH₃)=N-(3-Cl-C₆H₄), -C(CH₃)=N-(4-Cl-C₆H₄), -C(CH₃)=N-(2-CH₃-C₆H₄), -C(CH₃)=N-(3-CH₃-C₆H₄), -C(CH₃)=N-(4-CH₃-C₆H₄), -C(CH₃)=N-(2-CF₃-C₆H₄), -C(CH₃)=N-(3-CF₃-C₆H₄), -C(CH₃)=N-(4-CF₃-C₆H₄), -C(CH₃)=N-(2-OCH₃-C₆H₄), -C(CH₃)=N-(3-OCH₃-C₆H₄), -C(CH₃)=N-(4-OCH₃-C₆H₄), -C(CH₃)=N-(4-NO₂-C₆H₄), -C(CH₃)=N-(4-CN-C₆H₄), -C(CH₃)=N-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-(2,4-(CH₃)₂-C₆H₃), -C(CH₃)=N-CH₂-OCH₃, -C(CH₃)=N-CH₂-OC₂H₅, -C(CH₃)=N-CH₂CH₂-OCH₃, -C(CH₃)=N-CH₂CH-OC₂H₅, -C(CH₃)=N-OH, -C(CH₃)=N-OCH₃, -C(CH₃)=N-OC₂H₅, -C(CH₃)=N-O-n-C₃H₇, -C(CH₃)=N-O-i-C₃H₇, -C(CH₃)=N-O-n-C₄H₉, -C(CH₃)=N-O-i-C₄H₉, -C(CH₃)=N-O-s-C₄H₉, -C(CH₃)=N-O-tert.-C₄H₉, -C(CH₃)=N-OCH₂-CH=CH₂, -C(CH₃)=N-OCH(CH₃)-CH=CH₂, -C(CH₃)=N-OCH₂-C≡CH, -C(CH₃)=N-CH(CH₃)-C≡CH, -C(CH₃)=N-OCH₂-CH=C-CH₃, -C(CH₃)=N-OCH₂CH₂-Cl, -C(CH₃)=N-OCH₂CH₂-F, -C(CH₃)=N-OCH₂-CF₃, -C(CH₃)=N-OCH₂-CH=CHCl, -C(CH₃)=N-OCH₂-C(Cl)=CH₂, -C(CH₃)=N-OCH₂-C(Br)=CH₂, -C(CH₃)=N-OCH₂-CH=C(Cl)-CH₃, -C(CH₃)=N-O-CO-CH₃, -C(CH₃)=N-O-CO-C₂H₅, -C(CH₃)=N-OCH₂-CN, -C(CH₃)=N-OCH₂-CH=CH-CH₂-OCH₃, -C(CH₃)=N-OCH₂-CH=CH-CH₂-O-tert.-C₄H₉, -C(CH₃)=N-O-(CH₂)₃-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-(4-Cl-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-C₆H₅, -C(CH₃)=N-OCH₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(3-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-CH₂-(4-CH₃O-C₆H₄), -C(CH₃)=N-OCH₂-CH=C(CH₃)-C₆H₅, -C(CH₃)=N-O-(CH₂)₂-CH=CH-(3,4-Cl₂-C₆H₃), -C(CH₃)=N-O-(CH₂)₃-C≡C-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-OCH₃, -C(CH₃)=N-OCH₂CH₂-OCH₃, -C(CH₃)=N-OCH₂-OC₂H₅, -C(CH₃)=N-OCH(CH₃)-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=N-NH₂, -C(CH₃)=N-NH-CH₃, -C(CH₃)=N-NH-C₂H₅, -C(CH₃)=N-NH-n-C₃H₇, -C(CH₃)=N-NH-i-C₃H₇, -C(CH₃)=N-NH-n-C₄H₉, -C(CH₃)=N-NH-i-C₄H₉, -C(CH₃)=N-NH-s-C₄H₉, -C(CH₃)=N-NH-tert.-C₄H₉, -C(CH₃)=N-NH-cyclopropyl, -C(CH₃)=N-NH-cyclobutyl, -C(CH₃)=N-NH-cyclopentyl, -C(CH₃)=N-NH-cyclohexyl, -C(CH₃)=N-NH-cycloheptyl, -C(CH₃)=N-N(CH₃)₂, -C(CH₃)=N-N(C₂H₅)₂, -C(CH₃)=N-N(n-C₃H₇)₂, -C(CH₃)=N-N(i-C₃H₇)₂, -C(CH₃)=N-NH-CH₂-C=CH, -C(CH₃)=N-NH-CH₂-C≡CH, -C(CH₃)=N-N(CH₃)-CH₂-C≡CH, -C(CH₃)=N-NH-CH₂CF₃, -C(CH₃)=N-NH-CO-CH₃, -C(CH₃)=N-NH-CO-C₂H₅, -C(CH₃)=N-NH-CO-OCH₃, -C(CH₃)=N-NH-CO-OC₂H₅, -C(CH₃)=N-NH-CO-O-tert.-C₄H₉, -C(CH₃)=N-pyrrolidin-1-yl, -C(CH₃)=N-piperidin-1-yl, -C(CH₃)=N-morpholin-4-yl, -C(CH₃)=N-NH-C₆H₅, -C(CH₃)=N-NH-(4-Cl-C₆H₄), -C(CH₃)=N-NH-(4-NO₂-C₆H₄), -C(CH₃)=N-NH-(4-F-C₆H₄), -C(CH₃)=N-NH-(4-CH₃O-C₆H₄), -C(CH₃)=N-NH-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-NH-(2,4-(NO₂)₂-C₆H₃), -C(CH₃)=N-NH-CO-NH₂, -C(CH₃)=N-NH-CO-NHCH₃, -C(CH₃)=N-NH-CO-NHC₂H₅, -C(CH₃)=N-NH-CO-N(CH₃)₂, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=CH-CO-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -(CH₃)=CH-CO-O-n-C₄H₉, -C(CH₃)=CH-CO-O-tert.-C₄H₉, -C(CH₃)=CH-CO-O-cyclopropyl, -C(CH₃)=CH-CO-O-cyclobutyl, -C(CH₃)=CH-CO-O-cyclopentyl, -C(CH₃)=CH-CO-O-cyclohexyl, -C(CH₃)=CH-CO-O-cycloheptyl, -C(CH₃)=C(CH₃)-COOH, -C(CH₃)=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-cyclopropyl, -C(CH₃)=C(CH₃)-CO-O-cyclobutyl, -C(CH₃)=C(CH₃)-CO-O-cyclopentyl, -C(CH₃)=C(CH₃)-CO-O-cyclohexyl, -C(CH₃)=C(CH₃)-CO-O-cycloheptyl, -C(CH₃)=C(C₂H₅)-COOH, -C(CH₃)=C(C₂H₅)-CO-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-O- cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-O-cycloheptyl, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-O-n-C₄H₉, -C(CH₃)=C(Cl)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-O-cyclopropyl, -C(CH₃)=C(Cl)-CO-O-cyclobutyl, -C(CH₃)=C(Cl)-CO-O-cyclopentyl, -C(CH₃)=C(Cl)-CO-O-cyclohexyl, -C(CH₃)=C(Cl)-CO-O-cycloheptyl, -C(CH₃)=C(Br)-COOH, -C(CH₃)=C(Br)-CO-OCH₃, -C(CH₃)=C(Br)-CO-OC₂H₅, -C(CH₃)=C(Br)-CO-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-O-n-C₄H₉, -C(CH₃)=C(Br)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-O-cyclopropyl, -C(CH₃)=C(Br)-CO-O-cyclobutyl, -C(CH₃)=C(Br)-CO-O-cyclopentyl, -C(CH₃)=C(Br)-CO-O-cyclohexyl, -C(CH₃)=C(Br)-CO-O-cycloheptyl, -C(CH₃)=C(CN)-COOH, -C(CH₃)=C(CN)-CO-OCH₃, -C(CH₃)=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CN)-CO-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-O-n-C₄H₉, -C(CH₃)=C(CN)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-O-cyclopropyl, -C(CH₃)=C(CN)-CO-O-cyclobutyl, -C(CH₃)=C(CN)-CO-O-cyclopentyl, -C(CH₃)=C(CN)-CO-O-cyclohexyl, -C(CH₃)=C(CN)-CO-O-cycloheptyl, -C(CH₃)=CH-CO-OCH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=CH-CO-O-i-C₃H₇, -C(CH₃)=CH-CO-OCH(CH₃)-OCH₃, -C(CH₃)=CH-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=CH-CO-OCH₂CH₂-OCH₃, -C(CH₃)=CH-CO äOCH₂CH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=(C₂H₅)-CO-OCH₂CH₂-OCH₃, -(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-O-i-C₃H₇, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -(CH₃)=C(Cl)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-O-i-C₃H₇, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-O-i-C₃H₇, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-CF₃, -C(CH₃)=CH-CO-OCH₂-CCl₃, -C(CH₃)=CH-CO-OCH₂-oxiranyl, -C(CH₃)=CH-CO-O-(CH₂)₃-Br,-C(CH₃)=CH-CO-OCH₂-CH=CH₂, -C(CH₃)=CH-CO-OCH₂-C≡CH, -C(CH₃)=CH-CO-OCH₂-CN, -C(CH₃)=CH-CO-OCH₂CH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CF₃, -C(CH₃)=C(CH₃)-CO-OCH₂-CCl₃, -C(CH₃)=C(CH₃)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CH₃)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(CH₃)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CH₃)-CO-OCH₂-C≡CH, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CF₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CCl₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-oxiranyl, -C(CH₃)=C(C₂H₅)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(C₂H₅)-CO-OCH₂-C≡CH, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-C₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂-CF₃, -C(CH₃)=C(Cl)-CO-OCH₂-CCl₃, -C(CH₃)=C(Cl)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Cl)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Cl)-CO-OCH₂-CH≡CH₂, -C(CH₃)=C(Cl)-CO-OCH₂-C≡CH, -C(CH₃)=C(Cl)-CO-OCH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂-CF₃, -C(CH₃)=C(Br)-CO-OCH₂-CCl₃, -C(CH₃)=C(Br)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Br)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Br)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Br)-CO-OCH₂-C≡CH, -C(CH₃)=C(Br)-CO-OCH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂CH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂-CF₃, -C(CH₃)=C(CN)-CO-OCH₂-CCl₃, -C(CH₃)=C(CN)-OCH₂-oxiranyl, -C(CH₃)=C(CN)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CN)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CN)-CO-OCH₂-C≡CH, -C(CH₃)=C(CN)-CO-OCH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂CH₂-CN, -C(CH₃)=CH-CO-CH₃, -C(CH₃)=CH-CO-C₂H₅, -C(CH₃)=CH-CO-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-n-C₄H₉, -C(CH₃)=CH-CO-tert.-C₄H₉, -C(CH₃)=CH-CO-CH₂Cl, -C(CH₃)=CH-CO-CH₂Br, -C(CH₃)=CH-CO-CHCl₂, -C(CH₃)=CH-CO-CH₂-OCH₃, -C(CH₃)=CH-CO-CH(OCH₃)₂, -C(CH₃)=CH-CO-CH₂-SCH₃, -C(CH₃)=C(CH₃)-CO-CH₃, -C(CH₃)=C(CH₃)-CO-C₂H₅, -C(CH₃)=C(CH₃)-CO-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-CH₂Cl, -C(CH₃)=C(CH₃)-CO-CH₂Br, -C(CH₃)=C(CH₃)-CO-CHCl₂, -C(CH₃)=C(CH₃)-CO-CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-CH(OCH₃)₂, -C(CH₃)=C(CH₃)-CO-CH₂-SCH₃, -C(CH₃)=C(C₂H₅)-CO-CH₃, -C(CH₃)=C(C₂H₅)-CO-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-CH₂Cl, -C(CH₃)=C(C₂H₅)-CO-CH₂Br, -C(CH₃)=C(C₂H₅)-CO-CHCl₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-CH(OCH₃)₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-SCH₃, -C(CH₃)=C(Cl)-CO-CH₃, -C(CH₃)=C(Cl)-CO-C₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-n-C₄H₉, -C(CH₃)=C(Cl)-CO-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-CH₂Cl, -C(CH₃)=C(Cl)-CO-CHCl₂, -C(CH₃)=C(Cl(-CO-CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-CH(OCH₃)₂, -C(CH₃)=C(Cl)-CO-CH₂-SCH₃, -C(CH₃)=C(Br)-CO-CH₃, -C(CH₃)=C(Br)-CO-C₂H₅, -C(CH₃)=C(Br)-CO-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-n-C₄H₉, -C(CH₃)=C(Br)-CO-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-CH₂Cl, -C(CH₃)=C(Br)-CO-CH₂Br, -C(CH₃)=C(Br)-CO-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-CH(OCH₃)₂, -C(CH₃)=C(Br)-CO-CH₂-SCH₃, -C(CH₃)=C(CN)-CO-CH₃, -C(CH₃)=C(CN)-CO-C₂H₅, -C(CH₃)=C(CN)-CO-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-n-C₄H₉, -C(CH₃)=C(CN)-CO-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-CH₂Cl, -C(CH₃)=C(CN)-CO-CH₂Br, -C(CH₃)=C(CN)-CO-CHCl₂, -C(CH₃)=C(CN)-CO-CH₂-OCH₃, -C(CH₃)=C(CN)-CO-CH(OCH₃)₂, -C(CH₃)=C(CN)-CO-CH₂-SCH₃, -C(CH₃)=CH-CO-C₆H₅, -C(CH₃)=CH-CO-(4-Cl-C₆H₄), -C(CH₃)=C(CH₃)-CO-C₆H₅, -C(CH₃)=C(CH₃)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(C₂H₅)-CO-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(Cl)-CO-C₆H₅, -C(CH₃)=C(Br)-CO-C₆H₅, -C(CH₃)=C(CN)-CO-C₆H₅, -C(CH₃)=CH-CO-NH₂, -C(CH₃)=CH-CO-NHCH₃, -C(CH₃)=CH-CO-N(CH₃)₂, -C(CH₃)=CH-CO-NH-C₂H₅, -C(CH₃)=CH-CO-N(C₂H₅)₂, -C(CH₃)=CH-CO-NH-n-C₃H₇, -C(CH₃)=CH-CO-NH-i-C₃H₇, -C(CH₃)=CH-CO-NH-tert.-C₄H₉, -C(CH₃)=CH-CO-NH-cyclopropyl, -C(CH₃)=CH-CO-NH-cyclobutyl, -C(CH₃)=CH-CO-NH-cyclopentyl, -C(CH₃)=CH-CO-NH-cylohexyl, -C(CH₃)=CH-CO-NH-cycloheptyl, -C(CH₃)=CH-CO-NH-cyclooctyl, -C(CH₃)=CH-CO-pyrrolidin-1-yl, -C(CH₃)=CH-CO-piperidin-1-yl, -C(CH₃)=CH-CO-morpholin-4-yl, -C(CH₃)=CH-CO-NH-CH₂CH=CH₂, -C(CH₃)=CH-CO-NH-CH₂C≡CH, -C(CH₃)=CH-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=CH-CO-NH-(CH₂)₂Cl, -C(CH₃)=CH-CO-NH-C₆H₅, -C(CH₃)=C(CH₃)-CO-NH₂, -C(CH₃)=C(CH₃)-CO-NHCH₃, -C(CH₃)=C(CH₃)-CO-N(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-C₂H₅, -C(CH₃)=C(CH₃)-CO-N(C₂H₅)₂, -C(CH₃)=C(CH₃)-CO-NH-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-NH- cyclopropyl, -C(CH₃)=C(CH₃)-CO-NH-cyclobutyl, -C(CH₃)=C(CH₃)-CO-NH-cyclopentyl, -C(CH₃)=C(CH₃)-CO-NH- cyclohexyl, -C(CH₃)=C(CH₃)-CO-NH-cycloheptyl, -C(CH₃)=C(CH₃)-CO-NH-cyclooctyl, -C(CH₃)=C(CH₃)-CO- pyrrolidin-1-yl, -C(CH₃)=C(CH₃)-CO-piperidin-1-yl, -C(CH₃)=C(CH₃)-CO-morpholin-4-yl, -C(CH₃)=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-NH(CH₂)₂Cl, -C(CH₃)=C(CH₃)-CO-NH-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-NH₂, -C(CH₃)=C(C₂H₅)-CO-NHCH₃, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)₂, -C(CH₃)=C(C₂H₅)-CO-NH-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-N(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-NH- cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-NH-cycloheptyl, -C(CH₃)=C(C₂H₅)-CO-NH- cyclooctyl, -C(CH₃)=C(C₂H₅)-CO-pyrrolidin-1-yl, -C(CH₃)=C(C₂H₅)-CO-piperidin-1-yl, -C(CH₃)=C(C₂H₅)-CO- morpholin-4-yl, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(C₂H₅)-CO-NH-C₆H₅, -C(CH₃)=C(Cl)-CO-NH₂, -C(CH₃)=C(CH₃)=C(Cl)-CO-NHCH₃, -C(CH₃)=C(Cl)-CO-N(CH₃)₂, -C(CH₃)=C(Cl)-CO-NH-C₂H₅, -C(CH₃)=C(Cl)-CO-N(C₂H₅)₂, -C(CH₃)=C(Cl)-CO-NH-n-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-i-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-NH-cyclopropyl, -C(CH₃)=C(Cl)-CO-NH-cyclobutyl, -C(CH₃)=C(Cl)-CO-NH-cyclopentyl, -C(CH₃)=C(Cl)-CO-NH-cyclohexyl, -C(CH₃)=C(Cl)-CO-NH-cycloheptyl, -C(CH₃)=C(Cl)-CO-NH-cyclooctyl, -C(CH₃)=C(Cl)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Cl)-CO-piperidin-1- yl, -C(CH₃)=C(Cl)-CO-morpholin-4-yl, -C(CH₃)=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -C(CH₃)=C(Cl)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Cl)-NO-NH-C₆H₅, -C(CH₃)=C(Br)-CO-NH₂, -C(CH₃)=C(Br)-CO-NHCH₃, -C(CH₃)=C(Br)-CO-N(CH₃)₂, -C(CH₃)=C(Br)-CO-NH-C₂H₅, -C(CH₃)=C(Br)-CO-N(C₂H₅)₂, -C(CH₃)=C(Br)-CO-NH-n-C₃H₇, -C(CH₃)=C(Br)-CO-NH-i-C₃H₇, -C(CH₃)=C(Br)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-NH-cyclopropyl, -C(CH₃)=C(Br)-CO-NH-cyclobutyl, -C(CH₃)=C(Br)-CO-NH-cyclopentyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cycloheptyl, -C(CH₃)=C(Br)-CO-NH-cyclooctyl, -C(CH₃)=C(Br)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Br)-CO-piperidin-1-yl, -C(CH₃)=C(Br)-CO-morpholin-4-yl, -C(CH₃)=C(Br)-CO-NH-CH₂CH=C(Br)₂, -C(CH₃)=C(Br)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Br)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Br)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Br)-CO-NH-C₆H₅, -C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CN)-CO-NHCH₃, -C(CH₃)=C(CN)-CO-N(CH₃)₂, -C(CH₃)=C(CN)-CO-NH-C₂H₅, -C(CH₃)=C(CN)-CO-N(C₂H₅)₂, -C(CH₃)=C(CN)-CO-NH-n-C₃H₇, -C(CH₃)=C(CN)-CO-NH-i-C₃H₇, -C(CH₃)=C(CN)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-NH-cyclopropyl, -C(CH₃)=C(CN)-CO-NH-cyclobutyl, -C(CH₃)=C(CN)-CO-NH-cyclopentyl, -C(CH₃)=C(CN)-CO-NH-cyclohexyl, -C(CH₃)=C(CN)-CO-NH-cycloheptyl, -C(CH₃)=C(CN)-CO-NH-cyclooctyl, -C(CH₃)=C(CN)-CO-pyrrolidin-1-yl, -C(CH₃)=C(CN)-CO-piperidin-1-yl, -C(CH₃)=C(CN)-CO-morpholin-4-yl, -C(CH₃)=C(CN)-CO-NH-CH₂CH=C(CN)₂, -C(CH₃)=C(CN)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CN)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)=(CN)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CN)-CO-NH-C₆H₅, -C(CH₃)=CH-SO-SCH₃, -C(CH₃)=CH-CO-SC₂H₅, -C(CH₃)=CH-CO-S-n-C₃H₇, -C(CH₃)=CH-CO-S-i-C₃H₇, -C(CH₃)=CH-CO-S-n-C₄H₉, -C(CH₃)=CH-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-SCH₃, -C(CH₃)=C(CH₃)-CO-SC₂H₅, -C(CH₃)=C(CH₃)CO-S-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-S-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-SCH₃, -C(CH₃)=C(C₂H₅)-CO-SC₂H₅, -C(CH₃)=C(C₂H₅)-CO-S-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-SCH₃, -C(CH₃)=C(Cl)-CO-SC₂H₅, -C(CH₃)=C(Cl)-CO-S-n-C₃H₇, -C(CH₃)=C(Cl)-CO-S-i-C₃H₇, -C(CH₃)=C(Cl)-CO-S-n-C₄H₉, -C(CH₃)=C(Cl)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-SCH₃, -C(CH₃)=C(Br)-CO-SC₂H₅, -C(CH₃)=C(Br)-CO-S-n-C₃H₇, -C(CH₃)=C(Br)-CO-S-i-C₃H₇, -C(CH₃)=C(Br)-CO-S-n-C₄H₉, -C(CH₃)=C(Br)-CO-S-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-SCH₃, -C(CH₃)=C(CN)-CO-SC₂H₅, -C(CH₃)=C(CN)-CO-S-n-C₃H₇, -C(CH₃)=C(CN)-CO-S-i-C₃H₇, -C(CH₃)=C(CN)-CO-S-n-C₄H₉, -C(CH₃)=C(CN)-CO-S-tert.-C₄H₉, -C(CH₃)=C(COCH₃)-CO-OCH₃, -C(CH₃)=C(COC₂H₅)-CO-OCH₃, -C(CH₃)=C(CO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COCH₃)-CO-OC₂H₅, -C(CH₃)=C(COC₂H₅)-CO-OC₂H₅, -C(CH₃)=C(CO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COCH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(COC₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-OCH₃, -C(CH₃)=C(CF₃)-CO-OC₂H₅, -C(CH₃)=C(CF₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CF₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(COOCH₃)₂, -C(CH₃)=C(COOC₂H₅)₂, -C(CH₃)=C(COOCH₃)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)₂, -C(CH₃)=CH-CH=CH-COOH, -C(CH₃)=CH-CH=CH-CO-OCH₃, -C(CH₃)=CH-CH=CH-CO-OC₂H₅, -C(CH₃)=CH-CH=C(COOCH₃)₂, -C(CH₃)=CH-CH=C(CN)-CO-OCH₃, -C(CH₃)=CH-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CN)CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH₂, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -C(CH₃)=CH-(CH₂)₂-COOH, -C(CH₃)=CH-(CH₂)₂-CO-OCH₃, -C(CH₃)=CH-(CH₂)₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(COOCH₃)₂, -C(CH₃)=CH-CH₂-CH(COOC₂H₅)₂, -C(CH₃)=CH-CH₂-CH(CN)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CN)-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -C(CH₃)=CH-(CH₂)₂-CO-NH₂, -C(CH₃)=CH-(CH₂)₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-COOH, -C(CH₃)=CH-CH₂-CO-OCH₃, -C(CH₃)=CH-CH₂-CO-OC₂H₅, -C(CH₃)=C(COOCH₃)-CH₂-CO-OCH₃, -C(CH₃)=C(COOCH₃)-CH₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CO-NH₂, -C(CH₃)=CH-CH₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-CO-N(CH₃)₂.
wobei W für eine der folgenden Bedeutungen steht:
-CHO, -COCH₃, -COC₂H₅, -CO-n-C₃H₇, -CO-i-C₃H₇, -CO-n-C₄H₉, -CO-i-C₄H₉, -CO-s-C₄H₉, -CO-tert.-C₄H₉, -CO-CH₂CH=CH₂, -CO-CF₃, -COCCl₃, -COCH₂C≡CH, -CO-cyclopropyl, -CO-cyclobutyl, -CO-cyclopentyl, -CO-cyclohexyl, -CO-CN, -CO-COOCH₃, -CO-COOC₂H₅, -CH=NH, -CH=NCH₃, -CH=NC₂H₅, -CH=N-n-C₃H₅, -CH=N-i-C₃H₅, -CH=N-n-C₄H₉, -CH=NCH₂CH=CH₂, -CH=NCH₂CH=CH₂-CH₃, -CH=NCH₂≡CH, -CH=NCH₂C≡C-CH₃, -CH=N-cyclopropyl, -CH=N-cyclobutyl, -CH=N-cyclopentyl, -CH=N-cyclohexyl, -CH=N-cycloheptyl, -CH=N-CH₂-CH₂Cl, -CH=N-CH₂Cl, -CH=N-C₆H₅, -CH=N-(4-Br-C₆H₄), -CH=N-3-F-C₆H₄, -CH=N-4-F-C₆H₄, -CH=N-2-Cl-C₆H₄, -CH=N-3-Cl-C₆H₄, -CH=N-4-Cl-C₆H₄, -CH=N-2-Br-C₆H₄, -CH=N-2-F-C₆H₄, -CH=N-2-CH₃-C₆H₄, -CH=N-3-CH₃-C₆H₄, -CH=N-4-CH₃-C₆H₄, -CH=N-2-CF₃-C₆H₄, -CH=N-3-CF₃-C₆H₄, -CH=N-4-CF₃-C₆H₄, -CH=N-2-OCH₃-C₆H₄, -CH=N-3-OCH₃-C₆H₄, -CH=N-4-OCH₃-C₆H₄, -CH=N-4-NO₂-C₆H₄, -CH=N-4-CN-C₆H₄, -CH=N-2,4-(Cl,Cl)-C₆H₄, -CH=N-2,4-(CH₃,CH₃)-C₆H₄, -CH=N-CH₂OCH₃ -CH=N-CH₂OC₂H₅, -CH=N-CH₂CH₂OCH₃, -CH=N-CH₂CH₂OC₂H₅, -CH=N-OH, -CH=N-OCH₃, -CH=N-OC₂H₅, -CH=N-O-n-C₃H₇, -CH=N-O-i-C₃H₇, -CH=N-O-n-C₄H₉, -CH=N-O-i-C₄H₉, -CH=N-O-s-C₄H₉, -CH=N-O-tert.-C₄H₉, -CH=N-O-CH₂CH=CH₂, -CH=N-O-CH(CH₃)CH=CH₂, -CH=N-O-CH₂C≡CH, -CH=N-O-CH(CH₃)-C≡CH, -CH=N-O-CH₂-CH=CH-CH₃, -CH=N-O-CH₂-CH₂-Cl, -CH=N-O-CH₂-CH₂-F, -CH=N-O-CH₂-CF₃, -CH=N-O-CH₂-CH=CHCl, -CH=N-O-CH₂-CCl=CH₂, -CH=N-O-CH₂-CBr=CH₂, -CH=N-O-CH₂-CH=CCl-CH₃, -CH=N-OC(O)CH₃, -CH=N-OC(O)C₂H₅, -CH=N-O-CH₂-CN, -CH=N-O-CH₂-CH=CH-CH₂-O-CH₃, -CH=N-O-CH₂-CH=CH-CH₂-O-tert.-C₄H₉, -CH=N-O-(CH₂)₃-C₆H₅, -CH=N-O-(CH₂)₄-C₆H₅, -CH=N-O-(CH₂)₄-4-Cl-C₆H₄, -CH=N-O-(CH₂)₄-4-OCH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-CH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-C₆H₅, -CH=N-O-CH₂CH=CH-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CH-3-OCH₃-C₆H₄, -CH=N-O-(CH₂)₂CH=CH-4-F-C₆H₄, -CH=N-O-(CH₂)CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CHCH₂-4-OCH₃-C₆H₄, -CH=N-O-CH₂-CH=C(CH₃)-C₆H₅ -CH=N-O-(CH₂)₂CH=CH-3,4(Cl,Cl)-C₆H₃, -CH=N-O-(CH₂)₃C≡C-4-F-C₆H₄, -CH₂=N-OCHOCH₃, -CH=N-OC₂H₄OCH₃, -CH=N-OCH₂OC₂H₅, -CH=N-OCH(CH₃)OCH₃, -CH=N-OCH(CH₃)COOCH₃, -CH=N-OCH(CH₃)COO-n-C₄H₉, -CH=N-NH₂, -CH=N-NHCH₃, -CH=N-NHC₂H₅, -CH=N-NH-n-C₃H₇, -CH=N-NH-i-C₃H₇, -CH=N-NH-n-C₄H₉, -CH=N-NH-i-C₄H₉, -CH=N-NH-s-C₄H₉, -CH=N-NH-tert.-C₄H₉, -CH=N-NH-cyclopropyl, -CH=N-NH-cyclobutyl, -CH=N-NH-cyclopentyl, -CH=N-NH-cyclohexyl, -CH=N-NH-cycloheptyl, -CH=N-N(CH₃)₂, -CH=N-N(C₂H₅)₂, -CH=N-N(C₃H₇)₂, -CH=N-N(i-C₃H₇)(CH₃), -CH=N-NHCH₂-C=CH, -CH=N-NHCH₂-C≡CH, -CH=N-N(CH₃)-CH₂-C≡CH, -CH=N-NHCH₂CF₃, -CH=N-NH-CO-CH₃, -CH=N-NH-CO-CH₂H₅, -CH=N-NH-COOCH₃, -CH=N-NH-COOC₂H₅, -CH=N-NH-COO-tert.-C₄H₉, -CH=N-pyrrolidin-1-yl, -CH=N-piperidin-1-yl, -CH=N-morpholin-4-yl, -CH=N-NH-C₆H₅, -CH=N-NH-(4-Cl-C₆H₄), -CH=N-NH-(4-NO₂-C₆H₄), -CH=N-NH-(4-F-C₆H₄), -CH=N-NH-(4-CH₃O-C₆H₄), -CH=N-NH-(2,4-Cl₂-C₆H₃), -CH=N-NH-(2,4-(NO₂)₂-C₆H₃), -CH=N-NH-CO-NH₂, -CH=N-NH-CO-NHCH₃, -CH=N-NH-CO-NHC₂H₅, -CH=N-NH-CO-N(CH₃)₂, -CH=CH-COOH, -CH=CH-CO-OCH₃, -CH=C-CO-OC₂H₅, -CH=CH-CO-O-n-C₃H₇, -CH=CH-CO-O-i-C₃H₇, -CH=CH-CO-O-n-C₄H₉, -CH=CH-CO-O-tert.-C₄H₉, -CH=CH-CO-O-cyclopropyl, -CH=CH-CO-O-cyclobutyl, -CH=CH-CO-O-cyclopentyl, -CH=CH-CO-O-cyclohexyl, -CH=CH-CO-O-cycloheptyl, -CH=C(CH₃)-COOH, -CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CO-O-n-C₃H₇, -CH=C(CH₃)-CO-O-i-C₃H₇, -CH=C(CH₃)-CO-O-n-C₄H₉, -CH=C(CH₃)-CO-O-tert.-C₄H₉, -CH=C(CH₃)-CO-O-cyclopropyl, -CH=C(CH₃)-CO-O-cyclobutyl, -CH=C(CH₃)-CO-O-cyclopentyl, -CH=C(CH₃)-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cycloheptyl, -CH=C(C₂H₅)-COOH, -CH=C(C₂H₅)-CO-OCH₃, -CH=C(C₂H₅)-CO-OC₂H₅, -CH=C(C₂H₅)-CO-O-n-C₃H₇, -CH=C(C₂H₅)-CO-O-i-C₃H₇, -CH=C(C₂H₅)-CO-O-n-C₄H₉, -CH=C(C₂H₅)-CO-O-tert.-C₄H₉, -CH=C(C₂H₅)-CO-O-cyclopropyl, -CH=C(C₂H₅)-CO-O-cyclobutyl, -CH=C(C₂H₅)-CO-O-cyclopentyl, -CH=C(C₂H₅)-CO-O-cyclohexyl, -CH=C(C₂H₅)-CO-O-cycloheptyl, -CH=C(Cl)-COOH, -CH=C(Cl)-CO-OCH₃, -CH=C(Cl)-CO-OC₂H₅, -CH=C(Cl)-CO-O-n-C₃H₇, -CH=C(Cl)-CO-O-i-C₃H₇, -CH=C(Cl)-CO-O-n-C₄H₉, -CH=C(Cl)-CO-O-tert.-C₄H₉, -CH=C(Cl)-CO-O-cyclopropyl, -CH=C(Cl)-CO-O-cyclobutyl, -CH=C(Cl)-CO-O-cyclopentyl, -CH=C(Cl)-CO-O-cyclohexyl, -CH=C(Cl)-CO-O-cycloheptyl, -CH=C(Br)-COOH, -CH=C(Br)-CO-OCH₃, -CH=C(Br)-CO-OC₂H₅, -CH=C(Br)-CO-O-n-C₃H₇, -CH=C(Br)-CO-O-i-C₃H₇, -CH=C(Br)-CO-O-n-C₄H₉, -CH=C(Br)-CO-O-tert.-C₄H₉, -CH=C(Br)-CO-O-cyclopropyl, -CH=C(Br)-CO-O-cyclobutyl, -CH=C(Br)-CO-O-cyclopentyl, -CH=C(Br)-CO-O-cyclohexyl, -CH=C(Br)-CO-O-cycloheptyl, -CH=C(CN)-COOH, -CH=C(CN)-CO-OCH₃, -CH=C(CN)-CO-OC₂H₅, -CH=C(CN)-CO-O-n-C₃H₇, -CH=C(CN)-CO-O-i-C₃H₇, -CH=C(CN)-CO-O-n-C₄H₉, -CH=C(CN)-CO-O-tert.-C₄H₉, -CH=C(CN)-CO-O-cyclopropyl, -CH=C(CN)-CO-O-cyclobutyl, -CH=C(CN)-CO-O-cyclopentyl, -CH=C(CN)-CO-O-cyclohexyl, -CH=C(CN)-CO-O-cycloheptyl, -CH=CH-CO-OCH₂-OCH₃, -CH=CH-CO-OCH₂-OC₂H₅, -CH=CH-CO-OCH₂-O-n-C₃H₅, -CH=CH-CO-OCH₂-O-i-C₃H₅, -CH=CH-CO-OCH(CH₃)-OCH₃, -CH=CH-CO-OCH(CH₃)-OC₂H₅, -CH=CH-CO-O-CH₂CH₂-OCH₃, -CH=CH-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-OCH₃, -CH=C(CH₃)-CO-OCH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-O-n-C₃H₅, -CH=C(CH₃)-CO-OCH₂-O-i-C₃H₅, -CH=C(CH₃)-CO-OCH(CH₃)-OCH₃, -CH=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CH₃)-CO-O-CH₂CH₂-OCH₃, -CH=C(CH₃)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-OCH₃, -CH=C(C₂H₅)-CO-OCH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-O-n-C₃H₅, -CH=C(C₂H₅)-CO-OCH₂-O-i-C₃H₅, -CH=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-OCH₃, -CH=C(Cl)-CO-OCH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-O-n-C₃H₅, -CH=C(Cl)-CO-OCH₂-O-i-C₃H₅, -CH=C(Cl)-CO-OCH(CH₃)-OCH₃, -CH=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Cl)-CO-O-CH₂CH₂-OCH₃, -CH=C(Cl)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-OCH₃, -CH=C(Br)-CO-OCH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-O-n-C₃H₅, -CH=C(Br)-CO-OCH₂-O-i-C₃H₅, -CH=C(Br)-CO-OCH(CH₃)-OCH₃, -CH=C(Br)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Br)-CO-O-CH₂CH₂-OCH₃, -CH=C(Br)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-OCH₃, -CH=C(CN)-CO-OCH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-O-n-C₃H₅, -CH=C(CN)-CO-OCH₂-O-i-C₃H₅, -CH=C(CN)-CO-OCH(CH₃)-OCH₃, -CH=C(CN)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CN)-CO-O-CH₂CH₂-OCH₃, -CH=C(CN)-CO-O-CH₂CH₂-OC₂H₅, -CH=CH-CO-OCH₂-CF₃, -CH=CH-CO-OCH₂-CCl₃, -CH=CH-CO-OCH₂-oxiranyl, -CH=CH-CO-O(CH₂)₃-Br, -CH=CH-CO-OCH₂-CH=CH₂, -CH=CH-CO-OCH₂-C≡CH, -CH=CH-CO-OCH₂-CN, -CH=CH-CO-O(CH₂)₂-CN, -CH=C(CH₃)-CO-OCH₂-CF₃, -CH=C(CH₃)-CO-OCH₂-CCl₃, -CH=C(CH₃)-CO-OCH₂-oxiranyl, -CH=C(CH₃)-CO-O(CH₂)₃-Br, -CH=C(CH₃)-CO-OCH₂-CH=CH₂, -CH=C(CH₃)-CO-OCH₂-C≡CH, -CH=C(CH₃)-CO-OCH₂-CN, -CH=C(CH₃)-CO-O(CH₂)₂-CN, -CH=C(C₂H₅)-CO-OCH₂-CF₃, -CH=C(C₂H₅)-CO-OCH₂-CCl₃, -CH=C(C₂H₅)-CO-OCH₂-oxiranyl, -CH=C(C₂H₅)-CO-O(CH₂)₃-Br, -CH=C(C₂H₅)-CO-OCH₂-CH=CH₂, -CH=C(C₂H₅)-CO-OCH₂-C≡CH, -CH=C(C₂H₅)-CO-OCH₂-CN, -CH=C(C₂H₅)-CO-O(CH₂)₂-CN, -CH=C(Cl)-CO-OCH₂-CF₃, -CH=C(Cl)-CO-OCH₂-CCl₃, -CH=C(Cl)-CO-OCH₂-oxiranyl, -CH=C(Cl)-CO-O(CH₂)₃-Br, -CH=C(Cl)-CO-OCH₂-CH=CH₂, -CH=C(Cl)-CO-OCH₂-C≡CH, -CH=C(Cl)-CO-OCH₂-CN, -CH=C(Cl)-CO-O(CH₂)₂-CN, -CH=C(Br)-CO-OCH₂-CF₃, -CH=C(Br)-CO-OCH₂-CCl₃, -CH=C(Br)-CO-OCH₂-oxiranyl, -CH=C(Br)-CO-O(CH₂)₃-Br, -CH=C(Br)-CO-OCH₂-CH=CH₂, -CH=C(Br)-CO-OCH₂-C≡CH, -CH=C(Br)-CO-OCH₂-CN, -CH=C(Br)-CO-O(CH₂)₂-CN, -CH=C(CN)-CO-OCH₂-CF₃, -CH=C(CN)-CO-OCH₂-CCl₃, -CH=C(CN)-CO-OCH₂-oxiranyl -CH=C(CN)-CO-O(CH₂)₃-Br, -CH=C(CN)-CO-OCH₂-CH=CH₂, -CH=C(CN)-CO-OCH₂-C≡CH, -CH=C(CN)-CO-OCH₂-CN, -CH=C(CN)-CO-O(CH₂)₂-CN, -CH=CH-CO-CH₃, -CH=CH-CO-C₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-i-C₃H₇, -CH=CH-CO-n-C₄H₉, -CH=CH-CO-tert.-C₄H₉, -CH=CH-CO-CH₂Cl, -CH=CH-CO-CH₂Br, -CH=CH-CO-CHCl₂, -CH=CH-CO-CH₂-OCH₃, -CH=CH-CO-CH(OCH₃)₂, -CH=CH-CO-CH₂-SCH₃, -CH=C(CH₃)-CO-CH₃, -CH=C(CH₃)-CO-C₂H₅, -CH=C(CH₃)-CO-n-C₃H₇, -CH=C(CH₃)-CO-i-C₃H₇, -CH=C(CH₃)-CO-n-C₄H₉, -CH=C(CH₃)-CO-tert.-C₄H₉, -CH=C(CH₃)-CO-CH₂Cl, -CH=C(CH₃)-CO-CH₂Br, -CH=C(CH₃)-CO-CHCl₂, -CH=C(CH₃)-CO-CH₂-OCH₃, -CH=C(CH₃)-CO-CH(OCH₃)₂, -CH=C(CH₃)-CO-CH₂-SCH₃, -CH=C(C₂H₅)-CO-CH₃, -CH=C(C₂H₅)-CO-C₂H₅, -CH=C(C₂H₅)-CO-n-C₃H₇, -CH=C(C₂H₅)-CO-i-C₃H₇, -CH=C(C₂H₅)-CO-n-C₄H₉, -CH=C(C₂H₅)-CO-tert.-C₄H₉, -CH=C(C₂H₅)-CO-CH₂Cl, -CH=C(C₂H₅)-CO-CH₂Br, -CH=C(C₂H₅)-CO-CHCl₂, -CH=C(C₂H₅)-CO-CH₂-OCH₃, -CH=C(C₂H₅)-CO-CH(OCH₃)₂, -CH=C(C₂H₅)-CO-CH₂-SCH₃, -CH=C(Cl)-CO-CH₃, -CH=C(Cl)-CO-C₂H₅, -CH=C(Cl)-CO-n-C₃H₇, -CH=C(Cl)-CO-i-C₃H₇, -CH=C(Cl)-CO-n-C₄H₉, -CH=C(Cl)-CO-tert.-C₄H₉, -CH=C(Cl)-CO-CH₂Cl, -CH=C(Cl)-CO-CH₂Br, -CH=C(Cl)-CO-CHCl₂, -CH=C(Cl)-CO-CH₂-OCH₃, -CH=C(Cl)-CO-CH(OCH₃)₂, -CH=C(Cl)-CO-CH₂-SCH₃, -CH=C(Br)-CO-CH₃, -CH=C(Br)-CO-C₂H₅, -CH=C(Br)-CO-n-C₃H₇, -CH=C(Br)-CO-i-C₃H₇, -CH=C(Br)-CO-n-C₄H₉, -CH=C(Br)-CO-tert.-C₄H₉, -CH=C(Br)-CO-CH₂Cl, -CH=C(Br)-CO-CH₂Br, -CH=C(Br)-CO-CHCl₂, -CH=C(Br)-CO-CH₂-OCH₃, -CH=C(Br)-CO-CH(OCH₃)₂, -CH=C(Br)-CO-CH₂-SCH₃, -CH=C(CN)-CO-CH₃, -CH=C(CN)-CO-C₂H₅, -CH=C(CN)-CO-n-C₃H₇, -CH=C(CN)-CO-i-C₃H₇, -CH=C(CN)-CO-n-C₄H₉, -CH=C(CN)-CO-tert.-C₄H₉, -CH=C(CN)-CO-CH₂Cl, -CH=C(CN)-CO-CH₂Br, -CH=C(CN)-CO-CHCl₂, -CH=C(CN)-CO-CH₂-OCH₃, -CH=C(CN)-CO-CH(OCH₃)₂, -CH=C(CN)-CO-CH₂-SCH₃, -CH=CH-CO-C₆H₅, -CH=CH-CO-(4-Cl-C₆H₄), -CH=C(CH₃)-CO-C₆H₅, -CH=C(CH₃)-CO-(4-Cl-C₆H₄), -CH=C(C₂H₅)-CO-C₆H₅, -CH=C(C₂H₅)-CO-(4-Cl-C₆H₄), -CH=C(Cl)-CO-C₆H₅, -CH=C(Br)-CO-C₆H₅, -CH=C(CN)-CO-C₆H₅, -CH=CH-CO-NH₂, -CH=CH-CO-NHCH₃, -CH=CH-CO-N(CH₃)₂, -CH=CH-CO-NH-C₂H₅, -CH=CH-CO-N(C₂H₅)₂, -CH=CH-CO-NH-n-C₃H₇, -CH=CH-CO-NH-i-C₃H₇, -CH=CH-CO-NH-tert.-C₄H₉, -CH=CH-CO-NH-cyclopropyl, -CH=CH-CO-NH-cyclobutyl, -CH=CH-CO-NH-cyclopentyl, -CH=CH-CO-NH-cyclohexyl, -CH=CH-CO-NH-cycloheptyl, -CH=CH-CO-NH-cyclooctyl, -CH=CH-CO-pyrrolidin-1-yl, -CH=CH-CO-piperidin-1-yl, -CH=CH-CO-morpholin-4-yl, -CH=CH-CO-NH-CH₂CH=CH₂, -CH=CH-CO-NH-CH₂C≡CH, -CH=CH-CO-N(CH₃)-CH₂C≡CH, -CH=CH-CO-NH-(CH₂)₂Cl, -CH=CH-CO-NH-C₆H₅, -CH=C(CH₃)-CO-NH₂, -CH=C(CH₃)-CO-NHCH₃, -CH=C(CH₃)-CO-N(CH₃)₂, -CH=C(CH₃)-CO-NH-C₂H₅, -CH=C(CH₃)-CO-N(C₂H₅)₂, -CH=C(CH₃)-CO-NH-n-C₃H₇, -CH=C(CH₃)-CO-NH-i-C₃H₇, -CH=C(CH₃)-CO-NH-tert.-C₄H₉, -CH=C(CH₃)-CO-NH-cyclopropyl, -CH=C(CH₃)-CO-NH-cyclobutyl, -CH=C(CH₃)-CO-NH-cyclopentyl, -CH=C(CH₃)-CO-NH-cyclohexyl, -CH=C(CH₃)-CO-NH-cycloheptyl, -CH=C(CH₃)-CO-NH-cyclooctyl, -CH=C(CH₃)-CO-pyyrolidin-1-yl, -CH=C(CH₃)-CO-piperidin-1-yl, -CH=C(CH₃)-CO-morpholin-4-yl, -CH=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -CH=C(CH₃)-CO-NH-CH₂C≡CH, -CH=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CH₃)-CO-NH-(CH₂)₂Cl, -CH=C(CH₃)-CO-NH-C₆H₅, -CH=C(C₂H₅)-CO-NH₂, -CH=C(C₂H₅)-CO-NHCH₃, -CH=C(C₂H₅)-CO-N(CH₃)₂, -CH=C(C₂H₅)-CO-NH-C₂H₅, -CH=C(C₂H₅)-CO-N(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-n-C₃H₇, -CH=C(C₂H₅)-CO-NH-i-C₃H₇, -CH=C(C₂H₅)-CO-NH-tert.-C₄H₉, -CH=C(C₂H₅)-CO-NH-cyclopropyl, -CH=C(C₂H₅)-CO-NH-cyclobutyl, -CH=C(C₂H₅)-CO-NH-cyclopentyl, -CH=C(C₂H₅)-CO-NH-cyclohexyl, -CH=C(C₂H₅)-CO-NH-cycloheptyl, -CH=C(C₂H₅)-CO-NH-cyclooctyl, -CH=C(C₂H₅)-CO-pyrrolidin-1-yl, -CH=C(C₂H₅)-CO-piperidin-1-yl, -CH=C(C₂H₅)-CO-morpholin-4-yl, -CH=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-CH₂C≡CH, -CH=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -CH=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -CH=C(C₂H₅)-CO-NH-C₆H₅, -CH=C(Cl)-CO-NH₂, -CH=C(Cl)-CO-NHCH₃, -CH=C(Cl)-CO-N(CH₃)₂, -CH=C(Cl)-CO-NH-C₂H₅, -CH=C(Cl)-CO-N(C₂H₅)₂, -CH=C(Cl)-CO-NH-n-C₃H₇, -CH=C(Cl)-CO-NH-i-C₃H₇, -CH=C(Cl)-CO-NH-tert.-C₄H₉, -CH=C(Cl)-CO-NH-cyclopropyl, -CH=C(Cl)-CO-NH-cyclobutyl, -CH=C(Cl)-CO-NH-cyclopentyl, -CH=C(Cl)-CO-NH-cyclohexyl, -CH=C(Cl)-CO-NH-cycloheptyl, -CH=C(Cl)-CO-NH-cyclooctyl, -CH=C(Cl)-CO-pyrrolidin-1-yl, -CH=C(Cl)-CO-piperidin-1-yl, -CH=C(Cl)-CO-morpholin-4-yl, -CH=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -CH=C(Cl)-CO-NH-CH₂C≡CH, -CH=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Cl)-CO-NH-(CH₂)₂Cl, -CH=C(Cl)-CO-NH-C₆H₅, -CH=C(Br)-CO-NH₂, -CH=C(Br)-CO-NHCH₃, -CH=C(Br)-CO-N(CH₃)₂, -CH=C(Br)-CO-NH-C₂H₅, -CH=C(Br)-CO-N(C₂H₅)₂, -CH=C(Br)-CO-NH-n-C₃H₇, -CH=C(Br)-CO-NH-i-C₃H₇, -CH=C(Br)-CO-NH-tert.-C₄H₉, -CH=C(Br)-CO-NH-cyclopropyl, -CH=C(Br)-CO-NH-cyclobutyl, -CH=C(Br)-CO-NH-cyclopentyl, -CH=C(Br)-CO-NH-cyclohexyl, -CH=C(Br)-CO-NH-cycloheptyl, -CH=C(Br)-CO-NH-cyclooctyl, -CH=C(Br)-CO-pyrrolidin-1-yl, -CH=C(Br)-CO-piperidin-1-yl, -CH=C(Br)-CO-morpholin-4-yl, -CH=C(Br)-CO-NH-CH₂CH=C(Br)₂, -CH=C(Br)-CO-NH-CH₂C≡CH, -CH=C(Br)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Br)-CO-NH-(CH₂)₂Cl, -CH=C(Br)-CO-NH-C₆H₅, -CH=C(CN)-CO-NH₂, -CH=C(CN)-CO-NHCH₃, -CH=C(CN)-CO-N(CH₃)₂, -CH=C(CN)-CO-NH-C₂H₅, -CH=C(CN)-CO-N(C₂H₅)₂, -CH=C(CN)-CO-NH-n-C₃H₇, -CH=C(CN)-CO-NH-i-C₃H₇, -CH=C(CN)-CO-NH-tert.-C₄H₉, -CH=C(CN)-CO-NH-cyclopropyl, -CH=C(CN)-CO-NH-cyclobutyl, -CH=C(CN)-CO-NH-cyclopentyl, -CH=C(CN)-CO-NH-cyclohexyl, -CH=C(CN)-CO-NH-cycloheptyl, -CH=C(CN)-CO-NH-cyclooctyl, -CH=C(CN)-CO-pyrrolidin-1-yl, -CH=C(CN)-CO-piperidin-1-yl, -CH=C(CN)-CO-morpholin-4-yl, -CH=C(CN)-CO-NH-CH₂CH=C(CN)₂, -CH=C(CN)-CO-NH-CH₂C≡CH, -CH=C(CN)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CN)-CO-NH-(CH₂)₂Cl, -CH=C(CN)-CO-NH-C₆H₅, -CH=CH-CO-SCH₃, -CH=CH-CO-SC₂H₅, -CH=CH-CO-S-n-C₃H₇, -CH=CH-CO-S-i-C₃H₇, -CH=CH-CO-S-n-C₄H₉, -CH=CH-CO-S-tert.-C₄H₉, -CH=C(CH₃)-CO-SCH₃, -CH=C(CH₃)-CO-SC₂H₅, -CH=C(CH₃)-CO-S-n-C₃H₇, -CH=C(CH₃)-CO-S-i-C₃H₇, -CH=C(CH₃)-CO-S-n-C₄H₉, -CH=C(CH₃)-CO-S-tert.-C₄H₉, -CH=C(C₂H₅)-CO-SCH₃, -CH=C(C₂H₅)-CO-SC₂H₅, -CH=C(C₂H₅)-CO-S-n-C₃H₇, -CH=C(C₂H₅)-CO-S-i-C₃H₇, -CH=C(C₂H₅)-CO-S-n-C₄H₉, -CH=C(C₂H₅)-CO-S-tert.-C₄H₉, -CH=C(Cl)-CO-SCH₃, -CH=C(Cl)-CO-SC₂H₅, -CH=C(Cl)-CO-S-n-C₃H₇, -CH=C(Cl)-CO-S-i-C₃H₇, -CH=C(Cl)-CO-S-n-C₄H₉, -CH=C(Cl)-CO-S-tert.-C₄H₉, -CH=C(Br)-CO-SCH₃, -CH=C(Br)-CO-SC₂H₅, -CH=C(Br)-CO-S-n-C₃H₇, -CH=C(Br)-CO-S-i-C₃H₇, -CH=C(Br)-CO-S-n-C₄H₉, -CH=C(Br)-CO-S-tert.-C₄H₉, -CH=C(CN)-CO-SCH₃, -CH=C(CN)-CO-SC₂H₅, -CH=C(CN)-CO-S-n-C₃H₇, -CH=C(CN)-CO-S-i-C₃H₇, -CH=C(CN)-CO-S-n-C₄H₉, -CH=C(CN)-CO-S-tert.-C₄H₉, -CH=C(COCH₃)-CO-OCH₃, -CH=C(COC₂H₅)-CO-OCH₃, -CH=C(CO-n-C₃H₇)-CO-OCH₃, -CH=C(COCH₃)-CO-OC₂H₅, -CH=C(COC₂H₅)-CO-OC₂H₅, -CH=C(CO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COCH₃)-CO-O-n-C₃H₇, -CH=C(COC₂H₅)-CO-O-n-C₃H₇, -CH=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-OCH₃, -CH=C(CF₃)-CO-OC₂H₅, -CH=C(CF₃)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-O-i-C₃H₇, -CH=C(CF₃)-CO-O-n-C₄H₉, -CH=C(CF₃)-CO-O-tert.-C₄H₉, -CH=C(COOCH₃)₂, -CH=C(COOC₂H₅)₂, -CH=C(COOCH₃)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)-CO-OCH₃, -CH=C(COO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)₂, -CH=CH-CH=CH-COOH, -CH=CH-CH=CH-CO-OCH₃, -CH=CH-CH=CH-CO-OC₂H₅, -CH=CH-CH=C(COOCH₃)₂, -CH=CH-CH=C(CN)-CO-OCH₃, -CH=CH-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-OCH₃, -CH=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CH=C(Cl)-CO-OCH₃, -CH=C(CH₃)-CH=C(Br)-CO-OCH₃, -CH=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-NH₂, -CH=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -CH=CH-(CH₂)₂-COOH, -CH=CH-(CH₂)₂-CO-OCH₃, -CH=CH-(CH₂)₂-CO-OC₂H₅, -CH=CH-CH₂-CH(COOCH₃)₂, -CH=CH-CH₂-CH(COOC₂H₅)₂, -CH=CH-CH₂-CH(CN)-CO-OCH₃, -CH=CH-CH₂-CH(CN)-CO-OC₂H₅, -CH=CH-CH₂-CH(CH₃)-CO-OCH₃, -CH=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -CH=CH-(CH₂)₂-CO-NH₂, -CH=CH-(CH₂)₂-CO-NH-CH₃, -CH=CH-CH₂-COOH, -CH=CH-CH₂-CO-OCH₃, -CH=CH-CH₂-CO-OC₂H₅, -CH=C(COOCH₃)-CH₂-CO-OCH₃, -CH=C(COOCH₃)-CH₂-CO-OC₂H₅, -CH=CH-CH₂-CO-NH₂, -CH=CH-CH₂-CO-NH-CH₃, -CH=CH-CH₂-CO-N(CH₃)₂, -CH(OCH₃)₂, -CH(SCH₃)₂, -CH(OC₂H₅)₂, -CH(SC₂H₅)₂, -CH(O-n-C₃H₇)₂, -CH(O-i-C₃H₇)₂, -CH(S-n-C₃H₇)₂, -CH(S-i-C₃H₇)₂, -CH(O-n-C₄H₉)₂, -CH(O-i-C₄H₉)₂, -CH(O-s-C₄H₉)₂, -CH(O-tert.-C₄H₉)₂, -CH(S-n-C₄H₉)₂, -CH(S-i-C₄H₉)₂, -CH(S-s-C₄H₉)₂, -CH(S-tert.-C₄H₉)₂, -CH(OC₅H₁₁)₂, 1,3-Dioxolan-2-yl, 1,3-Dithio­ lan-2-yl, 1,3-Oxathiolan-2-yl, 4-Methyl-1,3-dioxolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 5-Methyl-1,3-oxathiolan-2-yl, 4-Ethyl-1,3-dioxolan-2-yl, 4-Ethyl- 1,4-dithiolan-2-yl, 4-Ethyl-1,3-oxathiolan-2-yl, 5-Ethyl-1,3-oxa­ thiolan-2-yl, 4,5-Dimethyl-1,3-dioxolan-2-yl, 4,4-Dimethyl-1,3- dioxolan-2-yl, 4,5-Dimethyl-1,3-dithiolan-2-yl, 5,5-Dimethyl-1,3- dithiolan-2-yl, 4,5-Dimethyl-1,3-oxathiolan-2-yl, 5,5-Dimethyl- 1,3-oxathiolan-2-yl, 4,4-Dimethyl-1,3-oxathiolan-2-yl, 4-Vinyl- 1,3-dioxolan-2-yl, 4-Vinyl-1,3-dithiolan-2-yl, 4-Vinyl-1,3-oxa­ thiolan-2-yl, 5-Vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3- dioxolan-2-yl, 4-Chlormethyl-1,3-dithiolan-2-yl, 4-Chlormethyl- 1,3-oxathiolan-2-yl, 5-Chlormethyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-1,3-dithio­ lan-2-yl, 4-Hydroxymethyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl- 1,3-oxathiolan-2-yl, 4-Methoxymethyl-1,3-dioxolan-2-yl, 4-Allyl­ oxymethyl-1,3-dioxolan-2-yl, 4-Propargyloxymethyl-1,3-dioxolan- 2-yl, 4-Acetoxymethyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-1,3-dithiolan-2-yl, 4-Propargyl­ oxymethyl-1,3-dithiolan-2-yl, 4-Acetoxymethyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl-1,3-oxathiolan-2-yl, 5-Allyloxy­ methyl-1,3-oxathiolan-2-yl, 4-Propargyloxymethyl-1,3-oxathiolan-2-yl, 5-Propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxymethyl- 1,3-oxathiolan-2-yl, 5-Acetoxymethyl-1,3-oxathiolan-2-yl, 4-Methylthiomethyl-1,3-dioxolan-2-yl, 4-Methylthiomethyl-1,3- dithiolan-2-yl, 4-Carboxy-1,3-dioxolan-2-yl, 4-Carboxy-1,3- dithiolan-2-yl, 4-Methoxycarbonyl-1,3-dioxolan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-1,3-dithiolan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-4-methyl- 1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-di­ thiolan-2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-1,3- dithiolan-2-yl, 1,3-Dioxan-2-yl, 1,3-Dithian-2-yl, 1,3-Oxathian- 2-yl, 5-Methyl-1,3-dioxan-2-yl, 5-Methyl-1,3-dithian-2-yl, 5-Methyl-1,3-oxathian-2-yl, 5,5-Dimethyl-1,3-dioxan-2-yl, 4,6-Dimethyl- 1,3-dioxan-2-yl, 4,4-Dimethyl-1,3-dioxan-2-yl, 5,5-Dimethyl- 1,3-dithian-2-yl, 4,6-Dimethyl-1,3-dithian-2-yl, 4,4-Dimethyl- 1,3-dithian-2-yl, 5,5-Dimethyl-1,3-oxathian-2-yl, 4,4-Dimethyl- 1,3-oxathian-2-yl, 6,6-Dimethyl-1,3-oxathian-2-yl, 4-Hydroxymethyl-1,3-dioxan-2-yl, 4-Methoxymethyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-1,3-dithian-2-yl, 4-Methoxymethyl-1,3-dithian-2-yl, 4-Allyloxymethyl-1,3-dithian-2-yl, 4-Acetoxymethyl- 1,3-dithian-2-yl, 4-Chlormethyl-1,3-dioxan-2-yl, 4-Chlormethyl- 1,3-dithian-2-yl, 1,3-Dioxepan-2-yl, 1,3-Dithiepan-2-yl, 1,3-Dioxep-5-en-2-yl, 4-Methoxycarbonyl-1,3-dioxan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-1,3-dithian-2-yl, 4-n-Butoxycarbonyl-1,3-dithian-2-yl, 4-Methoxycarbonyl-4- methyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-4-methyl- 1,3-dithian-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithian-2-yl, -C(CH₃)(OCH₃)₂, -C(CH₃)(SCH₃)₂, -C(CH₃)(OC₂H₅)₂, -C(CH₃)(SC₂H₅)₂, -C(CH₃)(O-n-C₃H₇)₂, -C(CH₃)(O-i-C₃H₇)₂, -C(CH₃)(S-n-C₃H₇)₂, -C(CH₃)(S-i-C₃H₇)₂, -C(CH₃)(O-n-C₄H₉)₂, -C(CH₃)(O-i-C₄H₉)₂, -C(CH₃)(O-s-C₄H₉)₂, -C(CH₃)(O-tert.-C₄H₉)₂, -C(CH₃)(S-n-C₄H₉)₂, -C(CH₃)(S-i-C₄H₉)₂, -C(CH₃)(S-s-C₄H₉)₂, -C(CH₃)(S-tert.-C₄H₉)₂, -C(CH₃)(O-n-C₅H₁₁)′′, 2-Methyl-1,3-dioxolan-2-yl, 2-Methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-oxathiolan-2-yl, 2,4-Dimethyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-1,3- oxathiolan-2-yl, 2,5-Dimethyl-1,3-oxathiolan-2-yl, 4-Ethyl-2- methyl-1,3-dioxolan-2-yl, 4-Ethyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Ethyl-2-methyl-1,3- oxathiolan-2-yl, 2,4,5-Trimethyl-1,3-dioxolan-2-yl, 2,4,4-Trimethyl- 1,3-dioxolan-2-yl, 2,4,5-Trimethyl-1,3-dithiolan-2-yl, 2,4,4-Trimethyl-1,3-dithiolan-2-yl, 2,4,5-Trimethyl-1,3-oxathiolan-2-yl, 2,4,4-Trimethyl-1,3-oxathiolan-2-yl, 2-Methyl-4-vinyl- 1,3-dioxolan-2-yl, 2-Methyl-4-vinyl-1,3-dithiolan-2-yl, 2-Methyl- 4-vinyl-1,3-oxathiolan-2-yl, 2-Methyl-5-vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-dioxolan-2-yl, 4-Chlormethyl-2- methyl-1,3-dithiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl- 2-methyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-2 methyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dioxolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxy- 2-methyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dithiolan-2-yl, 4-Acetoxy-2- methyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl- 2-methyl-1,3-oxathiolan-2-yl, 5-Allyloxymethyl-2- methyl-1,3-oxathiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3- oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxy-2-methyl-1,3-oxathiolan-2-yl, 5-Acetoxy-2-methyl- 1,3-oxathiolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dioxolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-2- methyl-1,3-dioxolan-2-yl, 4-Carboxy-2-methyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-2- methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl- 2-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-2- methyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-ethoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4- ethoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-n-butoxy­ carbony-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl-1,3- dithiolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-dioxan-2-yl, 2-Methyl-1,3-dithian-2-yl, 2-Methyl-1,3-oxathian-2-yl, 2,5- Dimethyl-1,3-dioxan-2-yl, 2,5-Dimethyl-1,3-dithian-2-yl, 2,5-Dimethyl- 1,3-oxathian-2-yl, 2,5,5-Trimethyl-1,3-dioxan-2-yl, 2,4,6- Trimethyl-1,3-dioxan-2-yl, 2,4,4-Trimethyl-1,3-dioxan-2-yl, 2,5,5-Trimethyl-1,3-dithian-2-yl, 2,4,6-Trimethyl-1,3-dithian-2-yl, 2,4,4-Trimethyl-1,3-dithian-2-yl, 2,5,5-Trimethyl-1,3-oxathian-2-yl, 2,4,4-Trimethyl-1,3-oxathian-2-yl, 2,6,6-Trimethyl- 1,3-oxathian-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-2- methyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dithian-2-yl, 4-Methoxymethyl-2- methyl-1,3-dithian-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithian-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dithian-2-yl, 4-Chlormethyl-2- methyl-1,3-dioxan-2-yl, 4-Chlormethyl-2-methyl-1,3-dithian-2-yl, -C(CH₃)=NH, -C(CH₃)=N-CH₃, -C(CH₃)=N-C₂H₅, -C(CH₃)=N-n-C₃H₇, -(CH₃)=N-i-C₃H₇, -C(CH₃)=N-n-C₄H₉, -C(CH₃)=N-CH₂CH=CH₂, -C(CH₃)=N-CH₂CH=CH₂-CH₃, -C(CH₃)=N-CH₂C≡CH, -C(CH₃)=N-CH₂C≡C-CH₃, -C(CH₃)=N-cyclopropyl, -C(CH₃)=N-cyclobutyl, -C(CH₃)=N-cyclopentyl, -C(CH₃)=N-cyclohexyl, -C(CH₃)=N-cycloheptyl, -C(CH₃)=N-CH₂-CH₂Cl, -C(CH₃)=N-CH₂Cl, -C(CH₃)=N-C₆H₅, -C(CH₃)=N-(2-F-C₆H₄), -C(CH₃)=N-(3-F-C₆H₄), -C(CH₃)=N-(4-F-C₆H₄), -C(CH₃)=N-(2-Cl-C₆H₄), -C(CH₃)=N-(3-Cl-C₆H₄), -C(CH₃)=N-(4-Cl-C₆H₄), -C(CH₃)=N-(2-CH₃-C₆H₄), -C(CH₃)=N-(3-CH₃-C₆H₄), -C(CH₃)=N-(4-CH₃-C₆H₄), -C(CH₃)=N-(2-CF₃-C₆H₄), -C(CH₃)=N-(3-CF₃-C₆H₄), -C(CH₃)=N-(4-CF₃-C₆H₄), -C(CH₃)=N-(2-OCH₃-C₆H₄), -C(CH₃)=N-(3-OCH₃-C₆H₄), -C(CH₃)=N-(4-OCH₃-C₆H₄), -C(CH₃)=N-(4-NO₂-C₆H₄), -C(CH₃)=N-(4-CN-C₆H₄), -C(CH₃)=N-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-(2,4-(CH₃)₂-C₆H₃), -C(CH₃)=N-CH₂-OCH₃, -C(CH₃)=N-CH₂-OC₂H₅, -C(CH₃)=N-CH₂CH₂-OCH₃, -C(CH₃)=N-CH₂CH₂-OC₂H₅, -C(CH₃)=N-OH, -C(CH₃)=N-OCH₃, -C(CH₃)=N-OC₂H₅, -C(CH₃)=N-O-n-C₃H₇, -C(CH₃)=N-O-i-C₃H₇, -C(CH₃)=N-O-n-C₄H₉, -C(CH₃)=N-O-i-C₄H₉, -C(CH₃)=N-O-s-C₄H₉, -C(CH₃)=N-O-tert.-C₄H₉, -C(CH₃)=N-OCH₂-CH=CH₂, -C(CH₃)=N-OCH(CH₃)-CH=CH₂, -C(CH₃)=N-OCH₂-C≡CH, -C(CH₃)=N-CH(CH₃)-C≡CH, -C(CH₃)=N-OCH₂-CH=C-CH₃, -C(CH₃)=N-OCH₂CH₂-Cl, -C(CH₃)=N-OCH₂CH₂-F, -C(CH₃)=N-OCH 99999 00070 552 001000280000000200012000285919988800040 0002004131038 00004 99880 ¥äCF₃, -C(CH₃)=N-OCH₂-CH=CHCl, -C(CH₃)=N-OCH₂-C(Cl)=CH₂, -C(CH₃)=N-OCH₂-C(Br)=CH₂, -C(CH₃)=N-OCH₂-CH=C(Cl)-CH₃, -C(CH₃)=N-O-CO-CH₃, -C(CH₃)=N-O-CO-C₂H₅, -C(CH₃)=N-OCH₂-CN, -C(CH₃)=N-OCH₂-CH=CH-CH₂-OCH₃, -C(CH₃)=N-OCH₂-CH=CH-CH₂-O-tert.-C₄H₉, -C(CH₃)=N-O-(CH₂)₃-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-(4-Cl-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-C₆H₅, -C(CH₃)=N-OCH₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(3-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-CH₂-(4-CH₃O-C₆H₄), -C(CH₃)=N-OCH₂-CH=C(CH₃)-C₆H₅, -C(CH₃)=N-O-(CH₂)₂-CH=CH-(3,4-Cl₂-C₆H₃), -C(CH₃)=N-O-(CH₂)₃-C≡C-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-OCH₃, -C(CH₃)=N-OCH₂CH₂-OCH₃, -C(CH₃)=N-OCH₂-OC₂H₅, -C(CH₃)=N-OCH(CH₃)-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=N-NH₂, -C(CH₃)=N-NH-CH₃, -C(CH₃)=N-NH-C₂H₅, -C(CH₃)=N-NH-n-C₃H₇, -C(CH₃)=N-NH-i-C₃H₇, -C(CH₃)=N-NH-n-C₄H₉, -C(CH₃)=N-NH-i-C₄H₉, -C(CH₃)=N-NH-s-C₄H₉, -C(CH₃)=N-NH-tert.-C₄H₉, -C(CH₃)=N-NH-cyclopropyl, -C(CH₃)=N-NH-cyclobutyl, -C(CH₃)=N-NH-cyclopentyl, -C(CH₃)=N-NH-cyclohexyl, -C(CH₃)=N-NH-cycloheptyl, -C(CH₃)=N-N(CH₃)₂, -C(CH₃)=N-N(C₂H₅)₂, -C(CH₃)=N-N(n-C₃H₇)₂, -C(CH₃)=N-N(i-C₃H₇)₂, -C(CH₃)=N-NH-CH₂-C=CH, -C(CH₃)=N-NH-CH₂-C≡CH, -C(CH₃)=N-N(CH₃)-CH₂-C≡CH, -C(CH₃)=N-NH-CH₂CF₃, -C(CH₃)=N-NH-CO-CH₃, -C(CH₃)=N-NH-CO-C₂H₅, -C(CH₃)=N-NH-CO-OCH₃, -C(CH₃)=N-NH-CO-OC₂H₅, -C(CH₃)=N-NH-CO-O-tert.-C₄H₉, -C(CH₃)=N-pyrrolidin-1-yl, -C(CH₃)=N-piperidin-1-yl, -C(CH₃)=N-morpholin-4-yl, -C(CH₃)=N-NH-C₆H₅, -C(CH₃)=N-NH-(4-Cl-C₆H₄), -C(CH₃)=N-NH-(4-NO₂-C₆H₄), -C(CH₃)=N-NH-(4-F-C₆H₄), -C(CH₃)=N-NH-(4-CH₃O-C₆H₄), -C(CH₃)=N-NH-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-NH-(2,4-(NO₂)₂-C₆H₃), -C(CH₃)=N-NH-CO-NH₂, -C(CH₃)=N-NH-CO-NHCH₃, -C(CH₃)=N-NH-CO-NHC₂H₅, -C(CH₃)=N-NH-CO-N(CH₃)₂, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=CH-CO-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -(CH₃)=CH-CO-O-n-C₄H₉, -C(CH₃)=CH-CO-O-tert.-C₄H₉, -C(CH₃)=CH-CO-O-cyclopropyl, -C(CH₃)=CH-CO-O-cyclobutyl, -C(CH₃)=CH-CO-O-cyclopentyl, -C(CH₃)=CH-CO-O-cyclohexyl, -C(CH₃)=CH-CO-O-cycloheptyl, -C(CH₃)=C(CH₃)-COOH, -C(CH₃)=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-cyclopropyl, -C(CH₃)=C(CH₃)-CO-O-cyclobutyl, -C(CH₃)=C(CH₃)-CO-O-cyclopentyl, -C(CH₃)=C(CH₃)-CO-O-cyclohexyl, -C(CH₃)=C(CH₃)-CO-O-cycloheptyl, -C(CH₃)=C(C₂H₅)-COOH, -C(CH₃)=C(C₂H₅)-CO-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-cyclo­ propyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-O- cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-O-cycloheptyl, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-O-n-C₄H₉, -C(CH₃)=C(Cl)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-O-cyclopropyl, -C(CH₃)=C(Cl)-CO-O-cyclobutyl, -C(CH₃)=C(Cl)-CO-O-cyclopentyl, -C(CH₃)=C(Cl)-CO-O-cyclohexyl, -C(CH₃)=C(Cl)-CO-O-cycloheptyl, -C(CH₃)=C(Br)-COOH, -C(CH₃)=C(Br)-CO-OCH₃, -C(CH₃)=C(Br)-CO-OC₂H₅, -C(CH₃)=C(Br)-CO-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-O-n-C₄H₉, -C(CH₃)=C(Br)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-O-cyclopropyl, -C(CH₃)=C(Br)-CO-O-cyclobutyl, -C(CH₃)=C(Br)-CO-O-cyclopentyl, -C(CH₃)=C(Br)-CO-O-cyclohexyl, -C(CH₃)=C(Br)-CO-O-cycloheptyl, -C(CH₃)=C(CN)-COOH, -C(CH₃)=C(CN)-CO-OCH₃, -C(CH₃)=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CN)-CO-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-O-n-C₄H₉, -C(CH₃)=C(CN)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-O-cyclopropyl, -C(CH₃)=C(CN)-CO-O-cyclobutyl, -C(CH₃)=C(CN)-CO-O-cyclopentyl, -C(CH₃)=C(CN)-CO-O-cyclohexyl, -C(CH₃)=C(CN)-CO-O-cycloheptyl, -C(CH₃)=CH-CO-OCH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-OCH(CH₃)-OCH₃, -C(CH₃)=CH-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=CH-CO-OCH₂CH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=(C₂H₅)-CO-OCH₂CH₂-OCH₃, -(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-O-i-C₃H₇, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OC₂H₅, C-(CH₃)=C(Cl)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-O-i-C₃H₇, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-O-i-C₃H₇, -C(CH₃)=C(CN)-CO-OCH(CH₃)OCH₃, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-CF₃, -C(CH₃)=CH-CO-OCH₂-CCl₃, -C(CH₃)=CH-CO-OCH₂-oxiranyl, -C(CH₃)=CH-CO-O-(CH₂)₃-Br,-C(CH₃)=CH-CO-OCH₂-CH=CH₂, -C(CH₃)=CH-CO-OCH₂-C≡CH, -C(CH₃)=CH-CO-OCH₂-CN, -C(CH₃)=CH-CO-OCH₂CH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CF₃, -C(CH₃)=C(CH₃)-CO-OCH₂-CCl₃, -C(CH₃)=C(CH₃)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CH₃)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CH₃)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CH₃)-CO-OCH₂-C≡CH, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CF₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CCl₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-oxiranyl, -C(CH₃)=C(C₂H₅)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(C₂H₅)-CO-OCH₂-C≡CH, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂-CF₃, -C(CH₃)=C(Cl)-CO-OCH₂-CCl₃, -C(CH₃)=C(Cl)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Cl)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Cl)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Cl)-CO-OCH₂-C≡CH, -C(CH₃)=C(Cl)-CO-OCH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂-CF₃, -C(CH₃)=C(Br)-CO-OCH₂-CCl₃, -C(CH₃)=C(Br)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Br)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Br)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Br)-CO-OCH₂-C≡CH, -C(CH₃)=C(Br)-CO-OCH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂CH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂-CF₃, -C(CH₃)=C(CN)-CO-OCH₂-CCl₃, -C(CH₃)=C(CN)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CN)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CN)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CN)-CO-OCH₂-C≡CH, -C(CH₃)=C(CN)-CO-OCH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂CH₂-CN, -C(CH₃)=CH-CO-CH₃, -C(CH₃)=CH-CO-C₂H₅, -C(CH₃)=CH-CO-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-n-C₄H₉, -C(CH₃)=CH-CO-tert.-C₄H₉, -C(CH₃)=CH-CO-CH₂Cl, -C(CH₃)=CH-CO-CH₂Br, -C(CH₃)=CH-CO-CHCl₂, -C(CH₃)=CH-CO-CH₂-OCH₃, -C(CH₃)=CH-CO-CH(OCH₃)₂, -C(CH₃)=CH-CO-CH₂-SCH₃, -C(CH₃)=C(CH₃)-CO-CH₃, -C(CH₃)=C(CH₃)-CO-C₂H₅, -C(CH₃)=C(CH₃)-CO-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-CH₂Cl, -C(CH₃)=C(CH₃)-CO-CH₂Br, -C(CH₃)=C(CH₃)-CO-CHCl₂, -C(CH₃)=C(CH₃)-CO-CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-CH(OCH₃)₂, -C(CH₃)=C(CH₃)-CO-CH₂-SCH₃, -C(CH₃)=C(C₂H₅)-CO-CH₃, -C(CH₃)=C(C₂H₅)-CO-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-CH₂Cl, -C(CH₃)=C(C₂H₅)-CO-CH₂Br, -C(CH₃)=C(C₂H₅)-CO-CHCl₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-CH(OCH₃)₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-SCH₃, -C(CH₃)=C(Cl)-CO-CH₃, -C(CH₃)=C(Cl)-CO-C₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-n-C₄H₉, -C(CH₃)=C(Cl)-CO-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-CH₂Cl, -C(CH₃)=C(Cl)-CO-CHCl₂, -C(CH₃)=C(Cl)-CO-CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-CH(OCH₃)₂, -C(CH₃)=C(Cl)-CO-CH₂-SCH₃, -C(CH₃)=C(Br)-CO-CH₃, -C(CH₃)=C(Br)-CO-C₂H₅, -C(CH₃)=C(Br)-CO-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-n-C₄H₉, -C(CH₃)=C(Br)-CO-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-CH₂Cl, -C(CH₃)=C(Br)-CO-CH₂Br, -C(CH₃)=C(Br)-CO-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-CH(OCH₃)₂, -C(CH₃)=C(Br)-CO-CH₂-SCH₃, -C(CH₃)=C(CN)-CO-CH₃, -C(CH₃)=C(CN)-CO-C₂H₅, -C(CH₃)=C(CN)-CO-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-n-C₄H₉, -C(CH₃)=C(CN)-CO-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-CH₂Cl, -C(CH₃)=C(CN)-CO-CH₂Br, -C(CH₃)=C(CN)-CO-CHCl₂, -C(CH₃)=C(CN)-CO-CH₂-OCH₃, -C(CH₃)=C(CN)-CO-CH(OCH₃)₂, -C(CH₃)=C(CN)-CO-CH₂-SCH₃, -C(CH₃)=CH-CO-C₆H₅, -C(CH₃)=CH-CO-(4-Cl-C₆H₄), -C(CH₃)=C(CH₃)-CO-C₆H₅, -C(CH₃)=C(CH₃)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(C₂H₅)-CO-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(Cl)-CO-C₆H₅, -C(CH₃)=C(Br)-CO-C₆H₅, -C(CH₃)=C(CN)-CO-C₆H₅, -C(CH₃)=CH-CO-NH₂, -C(CH₃)=CH-CO-NHCH₃, -C(CH₃)=CH-CO-N(CH₃)₂, -C(CH₃)=CH-CO-NH-C₂H₅, -C(CH₃)=CH-CO-N(C₂H₅)₂, -C(CH₃)=CH-CO-NH-n-C₃H₇, -C(CH₃)=CH-CO-NH-i-C₃H₇, -C(CH₃)=CH-CO-NH-tert.-C₄H₉, -C(CH₃)=CH-CO-NH-cyclopropyl, -C(CH₃)=CH-CO-NH-cyclobutyl, -C(CH₃)=CH-CO-NH-cyclopentyl, -C(CH₃)=CH-CO-NH-cyclohexyl, -C(CH₃)=CH-CO-NH-cycloheptyl, -C(CH₃)=CH-CO-NH-cyclooctyl, -C(CH₃)=CH-CO-pyrrolidin-1-yl, -C(CH₃)=CH-CO-piperidin-1-yl, -C(CH₃)=CH-CO-morpholin-4-yl, -C(CH₃)=CH-CO-NH-CH₂CH=CH₂, -C(CH₃)=CH-CO-NH-CH₂C≡CH, -C(CH₃)=CH-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=CH-CO-NH-(CH₂)₂Cl, -C(CH₃)=CH-CO-NH-C₆H₅, -C(CH₃)=C(CH₃)-CO-NH₂, -C(CH₃)=C(CH₃)-CO-NHCH₃, -C(CH₃)=C(CH₃)-CO-N(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-C₂H₅, -C(CH₃)=C(CH₃)-CO-N(C₂H₅)₂, -C(CH₃)=C(CH₃)-CO-NH-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-NH- cyclopropyl, -C(CH₃)=C(CH₃)-CO-NH-cyclobutyl, -C(CH₃)=C(CH₃)-CO-NH-cyclopentyl, -C(CH₃)=C(CH₃)-CO-NH- cyclohexyl, -C(CH₃)=C(CH₃)-CO-NH-cycloheptyl, -C(CH₃)=C(CH₃)-CO-NH-cyclooctyl, -C(CH₃)=C(CH₃)-CO- pyrrolidin-1-yl, -C(CH₃)=C(CH₃)-CO-piperidin-1-yl, -C(CH₃)=C(CH₃)-CO-morpholin-4-yl, -C(CH₃)=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-NH(CH₂)₂Cl, -C(CH₃)=C(CH₃)-CO-NH-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-NH₂, -C(CH₃)=C(C₂H₅)-CO-NHCH₃, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)₂, -C(CH₃)=C(C₂H₅)-CO-NH-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-N(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-NH- cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclo­ hexyl, -C(CH₃)=C(C₂H₅)-CO-NH-cycloheptyl, -C(CH₃)=C(C₂H₅)-CO-NH- cyclooctyl, -C(CH₃)=C(C₂H₅)-CO-pyrrolidin-1-yl, -C(CH₃)=C(C₂H₅)-CO-piperidin-1-yl, -C(CH₃)=C(C₂H₅)-CO- morpholin-4-yl, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(C₂H₅)-CO-NH-C₆H₅, -C(CH₃)=C(Cl)-CO-NH₂, -C(CH₃)=C(Cl)-CO-NHCH₃, -C(CH₃)=C(Cl)-CO-N(CH₃)₂, -C(CH₃)=C(Cl)-CO-NH-C₂H₅, -C(CH₃)=C(Cl)-CO-N(C₂H₅)₂, -C(CH₃)=C(Cl)-CO-NH-n-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-i-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-NH-cyclopropyl, -C(CH₃)=C(Cl)-CO-NH-cyclobutyl, -C(CH₃)=C(Cl)-CO-NH-cyclopentyl, -C(CH₃)=C(Cl)-CO-NH-cyclohexyl, -C(CH₃)=C(Cl)-CO-NH-cycloheptyl, -C(CH₃)=C(Cl)-CO-NH-cyclooctyl, -C(CH₃)=C(Cl)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Cl)-CO-piperidin-1- yl, -C(CH₃)=C(Cl)-CO-morpholin-4-yl, -C(CH₃)=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -C(CH₃)=C(Cl)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Cl)-NO-NH-C₆H₅, -C(CH₃)=C(Br)-CO-NH₂, -C(CH₃)=C(Br)-CO-NHCH₃, -C(CH₃)=C(Br)-CO-N(CH₃)₂, -C(CH₃)=C(Br)-CO-NH-C₂H₅, -C(CH₃)=C(Br)-CO-N(C₂H₅)₂, -C(CH₃)=C(Br)-CO-NH-n-C₃H₇, -C(CH₃)=C(Br)-CO-NH-i-C₃H₇, -C(CH₃)=C(Br)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-NH-cyclopropyl, -C(CH₃)=C(Br)-CO-NH-cyclobutyl, -C(CH₃)=C(Br)-CO-NH-cyclopentyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cycloheptyl, -C(CH₃)=C(Br)-CO-NH-cyclooctyl, -C(CH₃)=C(Br)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Br)-CO-piperidin-1-yl, -C(CH₃)=C(Br)-CO-morpholin-4-yl, -C(CH₃)=C(Br)-CO-NH-CH₂CH=C(Br)₂, -C(CH₃)=C(Br)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Br)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Br)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Br)-CO-NH-C₆H₅, -C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CN)-CO-NHCH₃, -C(CH₃)=C(CN)-CO-N(CH₃)₂, -C(CH₃)=C(CN)-CO-NH-C₂H₅, -C(CH₃)=C(CN)-CO-N(C₂H₅)₂, -C(CH₃)=C(CN)-CO-NH-n-C₃H₇, -C(CH₃)=C(CN)-CO-NH-i-C₃H₇, -C(CH₃)=C(CN)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-NH-cyclopropyl, -C(CH₃)=C(CN)-CO-NH-cyclobutyl, -C(CH₃)=C(CN)-CO-NH-cyclopentyl, -C(CH₃)=C(CN)-CO-NH-cyclohexyl, -C(CH₃)=C(CN)-CO-NH-cycloheptyl, -C(CH₃)=C(CN)-CO-NH-cyclooctyl, -C(CH₃)=C(CN)-CO-pyrrolidin-1-yl, -C(CH₃)=C(CN)-CO-piperidin-1-yl, -C(CH₃)=C(CN)-CO-morpholin-4-yl, -C(CH₃)=C(CN)-CO-NH-CH₂CH=C(CN)₂, -C(CH₃)=C(CN)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CN)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CN)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CN)-CO-NH-C₆H₅, -C(CH₃)=CH-CO-SCH₃, -C(CH₃)=CH-CO-SC₂H₅, -C(CH₃)=CH-CO-S-n-C₃H₇, -C(CH₃)=CH-CO-S-i-C₃H₇, -C(CH₃)=CH-CO-S-n-C₄H₉, -C(CH₃)=CH-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-SCH₃, -C(CH₃)=C(CH₃)-CO-SC₂H₅, -C(CH₃)=C(CH₃)CO-S-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-S-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-SCH₃, -C(CH₃)=C(C₂H₅)-CO-SC₂H₅, -C(CH₃)=C(C₂H₅)-CO-S-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-SCH₃, -C(CH₃)=C(Cl)-CO-SC₂H₅, -C(CH₃)=C(Cl)-CO-S-n-C₃H₇, -C(CH₃)=C(Cl)-CO-S-i-C₃H₇, -C(CH₃)=C(Cl)-CO-S-n-C₄H₉, -C(CH₃)=C(Cl)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-SCH₃, -C(CH₃)=C(Br)-CO-SC₂H₅, -C(CH₃)=C(Br)-CO-S-n-C₃H₇, -C(CH₃)=C(Br)-CO-S-i-C₃H₇, -C(CH₃)=C(Br)-CO-S-n-C₄H₉, -C(CH₃)=C(Br)-CO-S-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-SCH₃, -C(CH₃)=C(CN)-CO-SC₂H₅, -C(CH₃)=C(CN)-CO-S-n-C₃H₇, -C(CH₃)=C(CN)-CO-S-i-C₃H₇, -C(CH₃)=C(CN)-CO-S-n-C₄H₉, -C(CH₃)=C(CN)-CO-S-tert.-C₄H₉, -C(CH₃)=C(COCH₃)-CO-OCH₃, -C(CH₃)=C(COC₂H₅)-CO-OCH₃, -C(CH₃)=C(CO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COCH₃)-CO-OC₂H₅, -C(CH₃)=C(COC₂H₅)-CO-OC₂H₅, -C(CH₃)=C(CO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COCH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(COC₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-OCH₃, -C(CH₃)=C(CF₃)-CO-OC₂H₅, -C(CH₃)=C(CF₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CF₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(COOCH₃)₂, -C(CH₃)=C(COOC₂H₅)₂, -C(CH₃)=C(COOCH₃)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇))-CO-OCH₃, -C(CH₃)=C(COO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)₂, -C(CH₃)=CH-CH=CH-COOH, -C(CH₃)=CH-CH=CH-CO-OCH₃, -C(CH₃)=CH-CH=CH-CO-OC₂H₅, -C(CH₃)=CH-CH=C(COOCH₃)₂, -C(CH₃)=CH-CH=C(CN)-CO-OCH₃, -C(CH₃)=CH-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CN)CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH₂, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -C(CH₃)=CH-(CH₂)₂-COOH, -C(CH₃)=CH-(CH₂)₂-CO-OCH₃, -C(CH₃)=CH-(CH₂)₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(COOCH₃)₂, -C(CH₃)=CH-CH₂-CH(COOC₂H₅)₂, -C(CH₃)=CH-CH₂-CH(CN)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CN)-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -C(CH₃)=CH-(CH₂)₂-CO-NH₂, -C(CH₃)=CH-(CH₂)₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-COOH, -C(CH₃)=CH-CH₂-CO-OCH₃, -C(CH₃)=CH-CH₂-CO-OC₂H₅, -C(CH₃)=C(COOCH₃)-CH₂-CO-OCH₃, -C(CH₃)=C(COOCH₃)-CH₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CO-NH₂, -C(CH₃)=CH-CH₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-CO-N(CH₃)₂.
wobei W für eine der folgenden Bedeutungen steht:
-CHO, -COCH₃, -COC₂H₅, -CO-n-C₃H₇, -CO-i-C₃H₇, -CO-n-C₄H₉, -CO-i-C₄H₉, -CO-s-C₄H₉, -CO-tert.-C₄H₉, -CO-CH₂CH=CH₂, -CO-CF₃, -COCCl₃, -COCH₂C≡CH, -CO-cyclopropyl, -CO-cyclobutyl, -CO-cyclopentyl, -CO-cyclohexyl, -CO-CN, -CO-COOCH₃, -CO-COOC₂H₅, -CH=NH, -CH=NCH₃, -CH=NC₂H₅, -CH=N-n-C₃H₅, -CH=N-i-C₃H₅, -CH=N-n-C₄H₉, -CH=NCH₂CH=CH₂, -CH=NCH₂CH=CH₂-CH₃, -CH=NCH₂≡CH, -CH=NCH₂C≡C-CH₃, -CH=N-cyclopropyl, -CH=N-cyclobutyl, -CH=N-cyclopentyl, -CH=N-cyclohexyl, -CH=N-cycloheptyl, -CH=N-CH₂-CH₂Cl, -CH=N-CH₂Cl, -CH=N-C₆H₅, -CH=N-4-Br-C₆H₄, -CH=N-3-F-C₆H₄, -CH=N-4-F-C₆H₄, -CH=N-2-Cl-C₆H₄, -CH=N-3-Cl-C₆H₄, -CH=N-4-Cl-C₆H₄, -CH=N-2-Br-C₆H₄, -CH=N-2-F-C₆H₄, -CH=N-2-CH₃-C₆H₄, -CH=N-3-CH₃-C₆H₄, -CH=N-4-CH₃-C₆H₄, -CH=N-2-CF₃-C₆H₄, -CH=N-3-CF₃-C₆H₄, -CH=N-4-CF₃-C₆H₄, -CH=N-2-OCH₃-C₆H₄, -CH=N-3-OCH₃-C₆H₄, -CH=N-4-OCH₃-C₆H₄, -CH=N-4-NO₂-C₆H₄, -CH=N-4-CN-C₆H₄, -CH=N-2,4-(Cl,Cl)-C₆H₄, -CH=N-2,4-(CH₃,CH₃)-C₆H₄, -CH=N-CH₂OCH₃, -CH=N-CH₂OC₂H₅, -CH=N-CH₂CH₂OCH₃, -CH=N-CH₂CH₂OC₂H₅, -CH=N-OH, -CH=N-OCH₃, -CH=N-OC₂H₅, -CH=N-O-n-C₃H₇, -CH=N-O-i-C₃H₇, -CH=N-O-n-C₄H₉, -CH=N-O-i-C₄H₉, -CH=N-O-s-C₄H₉, -CH=N-O-tert.-C₄H₉, -CH=N-O-CH₂CH=CH₂, -CH=N-O-CH(CH₃)CH=CH₂, -CH=N-O-CH₂C≡CH, -CH=N-O-CH(CH₃)-C≡CH, -CH=N-O-CH₂-CH=CH-CH₃, -CH=N-O-CH₂-CH₂-Cl, -CH=N-O-CH₂-CH₂-F, -CH=N-O-CH₂-CF₃, -CH=N-O-CH₂-CH=CHCl, -CH=N-O-CH₂-CCl=CH₂, -CH=N-O-CH₂-CBr=CH₂, -CH=N-O-CH₂-CH=CCl-CH₃, -CH=N-OC(O)CH₃, -CH=N-OC(O)C₂H₅, -CH=N-O-CH₂-CN, -CH=N-O-CH₂-CH=CH-CH₂-O-CH₃, -CH=N-O-CH₂-CH=CH-CH₂-O-tert.-C₄H₉, -CH=N-O-(CH₂)₃-C₆H₅, -CH=N-O-(CH₂)₄-C₆H₅, -CH=N-O-(CH₂)₄-4-Cl-C₆H₄, -CH=N-O-(CH₂)₄-4-OCH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-CH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-C₆H₅, -CH=N-O-CH₂CH=CH-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CH-3-OCH₃-C₆H₄, -CH=N-O-(CH₂)₂CH=CH-4-F-C₆H₄, -CH=N-O-(CH₂)CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CHCH₂-4-OCH₃-C₆H₄, -CH=N-O-CH₂-CH=C(CH₃)-C₆H₅, -CH=N-O-(CH₂)₂CH=CH-3,4(Cl,Cl)-C₆H₃, -CH=N-O-(CH₂)₃C≡C-4-F-C₆H₄, -CH₂=N-OCHOCH₃, -CH=N-OC₂H₄OCH₃, -CH=N-OCH₂OC₂H₅, -CH=N-OCH(CH₃)OCH₃, -CH=N-OCH(CH₃)COOCH₃, -CH=N-OCH(CH₃)COO-n-C₄H₉, -CH=N-NH₂, -CH=N-NHCH₃, -CH=N-NHC₂H₅, -CH=N-NH-n-C₃H₇, -CH=N-NH-i-C₃H₇, -CH=N-NH-n-C₄H₉, -CH=N-NH-i-C₄H₉, -CH=N-NH-s-C₄H₉, -CH=N-NH-tert.-C₄H₉, -CH=N-NH-cyclopropyl, -CH=N-NH-cyclobutyl, -CH=N-NH-cyclopentyl, -CH=N-NH-cyclohexyl, -CH=N-NH-cycloheptyl, -CH=N-N(CH₃)₂, -CH=N-N(C₂H₅)₂, -CH=N-N(C₃H₇)₂, -CH=N-N(i-C₃H₇)(CH₃), -CH=N-NHCH₂-C=CH, -CH=N-NHCH₂-C≡CH, -CH=N-N(CH₃)-CH₂-C≡CH, -CH=N-NHCH₂CF₃, -CH=N-NH-CO-CH₃, -CH=N-NH-CO-CH₂H₅, -CH=N-NH-COOCH₃, -CH=N-NH-COOC₂H₅, -CH=N-NH-COO-tert.-C₄H₉, -CH=N-pyrrolidin-1-yl, -CH=N-piperidin-1-yl, -CH=N-morpholin-4-yl, -CH=N-NH-C₆H₅, -CH=N-NH-(4-Cl-C₆H₄), -CH=N-NH-(4-NO₂-C₆H₄), -CH=N-NH-(4-F-C₆H₄), -CH=N-NH-(4-CH₃O-C₆H₄), -CH=N-NH-(2,4-Cl₂-C₆H₃), -CH=N-NH-(2,4-(NO₂)₂-C₆H₃), -CH=N-NH-CO-NH₂, -CH=N-NH-CO-NHCH₃, -CH=N-NH-CO-NHC₂H₅, -CH=N-NH-CO-N(CH₃)₂, -CH=CH-COOH, -CH=CH-CO-OCH₃, -CH=C-CO-OC₂H₅, -CH=CH-CO-O-n-C₃H₇, -CH=CH-CO-O-i-C₃H₇, -CH=CH-CO-O-n-C₄H₉, -CH=CH-CO-O-tert.-C₄H₉, -CH=CH-CO-O-cyclopropyl, -CH=CH-CO-O-cyclobutyl, -CH=CH-CO-O-cyclopentyl, -CH=CH-CO-O-cyclohexyl, -CH=CH-CO-O-cycloheptyl, -CH=C(CH₃)-COOH, -CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CO-O-n-C₃H₇, -CH=C(CH₃)-CO-O-i-C₃H₇, -CH=C(CH₃)-CO-O-n-C₄H₉, -CH=C(CH₃)-CO-O-tert.-C₄H₉, -CH=C(CH₃)-CO-O-cyclopropyl, -CH=C(CH₃)-CO-O-cyclobutyl, -CH=C(CH₃)-CO-O-cyclopentyl, -CH=C(CH₃)-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cycloheptyl, -CH=C(C₂H₅)-COOH, -CH=C(C₂H₅)-CO-OCH₃, -CH=C(C₂H₅)-CO-OC₂H₅, -CH=C(C₂H₅)-CO-O-n-C₃H₇, -CH=C(C₂H₅)-CO-O-i-C₃H₇, -CH=C(C₂H₅)-CO-O-n-C₄H₉, -CH=C(C₂H₅)-CO-O-tert.-C₄H₉, -CH=C(C₂H₅)-CO-O-cyclopropyl, -CH=C(C₂H₅)-CO-O-cyclobutyl, -CH=C(C₂H₅)-CO-O-cyclopentyl, -CH=C(C₂H₅)-CO-O-cyclohexyl, -CH=C(C₂H₅)-CO-O-cycloheptyl, -CH=C(Cl)-COOH, -CH=C(Cl)-CO-OCH₃, -CH=C(Cl)-CO-OC₂H₅, -CH=C(Cl)-CO-O-n-C₃H₇, -CH=C(Cl)-CO-O-i-C₃H₇, -CH=C(Cl)-CO-O-n-C₄H₉, -CH=C(Cl)-CO-O-tert.-C₄H₉, -CH=C(Cl)-CO-O-cyclopropyl, -CH=C(Cl)-CO-O-cyclobutyl, -CH=C(Cl)-CO-O-cyclopentyl, -CH=C(Cl)-CO-O-cyclohexyl, -CH=C(Cl)-CO-O-cycloheptyl, -CH=C(Br)-COOH, -CH=C(Br)-CO-OCH₃, -CH=C(Br)-CO-OC₂H₅, -CH=C(Br)-CO-O-n-C₃H₇, -CH=C(Br)-CO-O-i-C₃H₇, -CH=C(Br)-CO-O-n-C₄H₉, -CH=C(Br)-CO-O-tert.-C₄H₉, -CH=C(Br)-CO-O-cyclopropyl, -CH=C(Br)-CO-O-cyclobutyl, -CH=C(Br)-CO-O-cyclopentyl, -CH=C(Br)-CO-O-cyclohexyl, -CH=C(Br)-CO-O-cycloheptyl, -CH=C(CN)-COOH, -CH=C(CN)-CO-OCH₃, -CH=C(CN)-CO-OC₂H₅, -CH=C(CN)-CO-O-n-C₃H₇, -CH=C(CN)-CO-O-i-C₃H₇, -CH=C(CN)-CO-O-n-C₄H₉, -CH=C(CN)-CO-O-tert.-C₄H₉, -CH=C(CN)-CO-O-cyclopropyl, -CH=C(CN)-CO-O-cyclobutyl, -CH=C(CN)-CO-O-cyclopentyl, -CH=C(CN)-CO-O-cyclohexyl, -CH=C(CN)-CO-O-cycloheptyl, -CH=CH-CO-OCH₂-OCH₃, -CH=CH-CO-OCH₂-OC₂H₅, -CH=CH-CO-OCH₂-O-n-C₃H₅, -CH=CH-CO-OCH₂-O-i-C₃H₅, -CH=CH-CO-OCH(CH₃)-OCH₃, -CH=CH-CO-OCH(CH₃)-OC₂H₅, -CH=CH-CO-O-CH₂CH₂-OCH₃, -CH=CH-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-OCH₃, -CH=C(CH₃)-CO-OCH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-O-n-C₃H₅, -CH=C(CH₃)-CO-OCH₂-O-i-C₃H₅, -CH=C(CH₃)-CO-OCH(CH₃)-OCH₃, -CH=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CH₃)-CO-O-CH₂CH₂-OCH₃, -CH=C(CH₃)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-OCH₃, -CH=C(C₂H₅)-CO-OCH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-O-n-C₃H₅, -CH=C(C₂H₅)-CO-OCH₂-O-i-C₃H₅, -CH=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -CH=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -CH=(C₂H₅)-CO-O-CH₂CH₂-OCH₃, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-OCH₃, -CH=C(Cl)-CO-OCH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-O-n-C₃H₅, -CH=C(Cl)-CO-OCH₂-O-i-C₃H₅, -CH=C(Cl)-CO-OCH(CH₃)-OCH₃, -CH=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Cl)-CO-O-CH₂CH₂-OCH₃, -CH=C(Cl)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-OCH₃, -CH=C(Br)-CO-OCH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-O-n-C₃H₅, -CH=C(Br)-CO-OCH₂-O-i-C₃H₅, -CH=C(Br)-CO-OCH(CH₃)-OCH₃, -CH=C(Br)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Br)-CO-O-CH₂CH₂-OCH₃, -CH=C(Br)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-OCH₃, -CH=C(CN)-CO-OCH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-O-n-C₃H₅, -CH=C(CN)-CO-OCH₂-O-i-C₃H₅, -CH=C(CN)-CO-OCH(CH₃)-OCH₃, -CH=C(CN)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CN)-CO-O-CH₂CH₂-OCH₃, -CH=C(CN)-CO-O-CH₂CH₂-OC₂H₅, -CH=CH-CO-OCH₂-CF₃, -CH=CH-CO-OCH₂-CCl₃, -CH=CH-CO-OCH₂-oxiranyl, -CH=CH-CO-O(CH₂)₃-Br, -CH=CH-CO-OCH₂-CH=CH₂, -CH=CH-CO-OCH₂-C≡CH, -CH=CH-CO-OCH₂-CN, -CH=CH-CO-O(CH₂)₂-CN, -CH=C(CH₃)-CO-OCH₂-CF₃, -CH=C(CH₃)-CO-OCH₂-CCl₃, -CH=C(CH₃)-CO-OCH₂-oxiranyl, -CH=C(CH₃)-CO-O(CH₂)₃-Br, -CH=C(CH₃)-CO-OCH₂-CH=CH₂, -CH=C(CH₃)-CO-OCH₂-C≡CH, -CH=C(CH₃)-CO-OCH₂-CN, -CH=C(CH₃)-CO-O(CH₂)₂-CN, -CH=C(C₂H₅)-CO-OCH₂-CF₃, -CH=C(C₂H₅)-CO-OCH₂-CCl₃, -CH=C(C₂H₅)-CO-OCH₂-oxiranyl, -CH=C(C₂H₅)-CO-O(CH₂)₃-Br, -CH=C(C₂H₅)-CO-OCH₂-CH=CH₂, -CH=C(C₂H₅)-CO-OCH₂-C≡CH, -CH=C(C₂H₅)-CO-OCH₂-CN, -CH=C(C₂H₅)-CO-O(CH₂)₂-CN, -CH=C(Cl)-CO-OCH₂-CF₃, -CH=C(Cl)-CO-OCH₂-CCl₃, -CH=C(Cl)-CO-OCH₂-oxiranyl, -CH=C(Cl)-CO-O(CH₂)₃-Br, -CH=C(Cl)-CO-OCH₂-CH=CH₂, -CH=C(Cl)-CO-OCH₂-C≡CH, -CH=C(Cl)-CO-OCH₂-CN, -CH=C(Cl)-CO-O(CH₂)₂-CN, -CH=C(Br)-CO-OCH₂-CF₃, -CH=C(Br)-CO-OCH₂-CCl₃, -CH=C(Br)-CO-OCH₂-oxiranyl, -CH=C(Br)-CO-O(CH₂)₃-Br, -CH=C(Br)-CO-OCH₂-CH=CH₂, -CH=C(Br)-CO-OCH₂-C≡CH, -CH=C(Br)-CO-OCH₂-CN, -CH=C(Br)-CO-O(CH₂)₂-CN, -CH=C(CN)-CO-OCH₂-CF₃, -CH=C(CN)-CO-OCH₂-CCl₃, -CH=C(CN)-CO-OCH₂-oxiranyl, -CH=C(CN)-CO-O(CH₂)₃-Br, -CH=C(CN)-CO-OCH₂-CH=CH₂, -CH=C(CN)-CO-OCH₂-C≡CH, -CH=C(CN)-CO-OCH₂-CN, -CH=C(CN)-CO-O(CH₂)₂-CN, -CH=CH-CO-CH₃, -CH=CH-CO-C₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-i-C₃H₇, -CH=CH-CO-n-C₄H₉, -CH=CH-CO-tert.-C₄H₉, -CH=CH-CO-CH₂Cl, -CH=CH-CO-CH₂Br, -CH=CH-CO-CHCl₂, -CH=CH-CO-CH₂-OCH₃, -CH=CH-CO-CH(OCH₃)₂, -CH=CH-CO-CH₂-SCH₃, -CH=C(CH₃)-CO-CH₃, -CH=C(CH₃)-CO-C₂H₅, -CH=C(CH₃)-CO-n-C₃H₇, -CH=C(CH₃)-CO-i-C₃H₇, -CH=C(CH₃)-CO-n-C₄H₉, -CH=C(CH₃)-CO-tert.-C₄H₉, -CH=C(CH₃)-CO-CH₂Cl, -CH=C(CH₃)-CO-CH₂Br, -CH=C(CH₃)-CO-CHCl₂, -CH=C(CH₃)-CO-CH₂-OCH₃, -CH=C(CH₃)-CO-CH(OCH₃)₂, -CH=C(CH₃)-CO-CH₂-SCH₃, -CH=C(C₂H₅)-CO-CH₃, -CH=C(C₂H₅)-CO-C₂H₅, -CH=C(C₂H₅)-CO-n-C₃H₇, -CH=C(C₂H₅)-CO-i-C₃H₇, -CH=C(C₂H₅)-CO-n-C₄H₉, -CH=C(C₂H₅)-CO-tert.-C₄H₉, -CH=C(C₂H₅)-CO-CH₂Cl, -CH=C(C₂H₅)-CO-CH₂Br, -CH=C(C₂H₅)-CO-CHCl₂, -CH=C(C₂H₅)-CO-CH₂-OCH₃, -CH=C(C₂H₅)-CO-CH(OCH₃)₂, -CH=C(C₂H₅)-CO-CH₂-SCH₃, -CH=C(Cl)-CO-CH₃, -CH=C(Cl)-CO-C₂H₅, -CH=C(Cl)-CO-n-C₃H₇, -CH=C(Cl)-CO-i-C₃H₇, -CH=C(Cl)-CO-n-C₄H₉, -CH=C(Cl)-CO-tert.-C₄H₉, -CH=C(Cl)-CO-CH₂Cl, -CH=C(Cl)-CO-CH₂Br, -CH=C(Cl)-CO-CHCl₂, -CH=C(Cl)-CO-CH₂-OCH₃, -CH=C(Cl)-CO-CH(OCH₃)₂, -CH=C(Cl)-CO-CH₂-SCH₃, -CH=C(Br)-CO-CH₃, -CH=C(Br)-CO-C₂H₅, -CH=C(Br)-CO-n-C₃H₇, -CH=C(Br)-CO-i-C₃H₇, -CH=C(Br)-CO-n-C₄H₉, -CH=C(Br)-CO-tert.-C₄H₉, -CH=C(Br)-CO-CH₂Cl, -CH=C(Br)-CO-CH₂Br, -CH=C(Br)-CO-CHCl₂, -CH=C(Br)-CO-CH₂-OCH₃, -CH=C(Br)-CO-CH(OCH₃)₂, -CH=C(Br)-CO-CH₂-SCH₃, -CH=C(CN)-CO-CH₃, -CH=C(CN)-CO-C₂H₅, -CH=C(CN)-CO-n-C₃H₇, -CH=C(CN)-CO-i-C₃H₇, -CH=C(CN)-CO-n-C₄H₉, -CH=C(CN)-CO-tert.-C₄H₉, -CH=C(CN)-CO-CH₂Cl, -CH=C(CN)-CO-CH₂Br, -CH=C(CN)-CO-CHCl₂, -CH=C(CN)-CO-CH₂-OCH₃, -CH=C(CN)-CO-CH(OCH₃)₂, -CH=C(CN)-CO-CH₂-SCH₃, -CH=CH-CO-C₆H₅, -CH=CH-CO-(4-Cl-C₆H₄), -CH=C(CH₃)-CO-C₆H₅, -CH=C(CH₃)-CO-(4-Cl-C₆H₄), -CH=C(C₂H₅)-CO-C₆H₅, -CH=C(C₂H₅)-CO-(4-Cl-C₆H₄), -CH=C(Cl)-CO-C₆H₅, -CH=C(Br)-CO-C₆H₅, -CH=C(CN)-CO-C₆H₅, -CH=CH-CO-NH₂, -CH=CH-CO-NHCH₃, -CH=CH-CO-N(CH₃)₂, -CH=CH-CO-NH-C₂H₅, -CH=CH-CO-N(C₂H₅)₂, -CH=CH-CO-NH-n-C₃H₇, -CH=CH-CO-NH-i-C₃H₇, -CH=CH-CO-NH-tert.-C₄H₉, -CH=CH-CO-NH-cyclopropyl, -CH=CH-CO-NH-cyclobutyl, -CH=CH-CO-NH-cyclopentyl, -CH=CH-CO-NH-cyclohexyl, -CH=CH-CO-NH-cycloheptyl, -CH=CH-CO-NH-cyclooctyl, -CH=CH-CO-pyrrolidin-1-yl, -CH=CH-CO-piperidin-1-yl, -CH=CH-CO-morpholin-4-yl, -CH=CH-CO-NH-CH₂CH=CH₂, -CH=CH-CO-NH-CH₂C≡CH, -CH=CH-CO-N(CH₃)-CH₂C≡CH, -CH=CH-CO-NH-(CH₂)₂Cl, -CH=CH-CO-NH-C₆H₅, -CH=C(CH₃)-CO-NH₂, -CH=C(CH₃)-CO-NHCH₃, -CH=C(CH₃)-CO-N(CH₃)₂, -CH=C(CH₃)-CO-NH-C₂H₅, -CH=C(CH₃)-CO-N(C₂H₅)₂, -CH=C(CH₃)-CO-NH-n-C₃H₇, -CH=C(CH₃)-CO-NH-i-C₃H₇, -CH=C(CH₃)-CO-NH-tert.-C₄H₉, -CH=C(CH₃)-CO-NH-cyclopropyl, -CH=C(CH₃)-CO-NH-cyclobutyl, -CH=C(CH₃)-CO-NH-cyclopentyl, -CH=C(CH₃)-CO-NH-cyclohexyl, -CH=C(CH₃)-CO-NH-cycloheptyl, -CH=C(CH₃)-CO-NH-cyclooctyl, -CH=C(CH₃)-CO-pyrrolidin-1-yl, -CH=C(CH₃)-CO-piperidin-1-yl, -CH=C(CH₃)-CO-morpholin-4-yl, -CH=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -CH=C(CH₃)-CO-NH-CH₂C≡CH, -CH=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CH₃)-CO-NH-(CH₂)₂Cl, -CH=C(CH₃)-CO-NH-C₆H₅, -CH=C(C₂H₅)-CO-NH₂, -CH=C(C₂H₅)-CO-NHCH₃, -CH=C(C₂H₅)-CO-N(CH₃)₂, -CH=C(C₂H₅)-CO-NH-C₂H₅, -CH=C(C₂H₅)-CO-N(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-n-C₃H₇, -CH=C(C₂H₅)-CO-NH-i-C₃H₇, -CH=C(C₂H₅)-CO-NH-tert.-C₄H₉, -CH=C(C₂H₅)-CO-NH-cyclopropyl, -CH=C(C₂H₅)-CO-NH-cyclobutyl, -CH=C(C₂H₅)-CO-NH-cyclopentyl, -CH=C(C₂H₅)-CO-NH-cyclohexyl, -CH=C(C₂H₅)-CO-NH-cycloheptyl, -CH=C(C₂H₅)-CO-NH-cyclooctyl, -CH=C(C₂H₅)-CO-pyrrolidin-1-yl, -CH=C(C₂H₅)-CO-piperidin-1-yl, -CH=C(C₂H₅)-CO-morpholin-4-yl, -CH=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-CH₂C≡CH, -CH=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -CH=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -CH=C(C₂H₅)-CO-NH-C₆H₅, -CH=C(Cl)-CO-NH₂, -CH=C(Cl)-CO-NHCH₃, -CH=C(Cl)-CO-N(CH₃)₂, -CH=C(Cl)-CO-NH-C₂H₅, -CH=C(Cl)-CO-N(C₂H₅)₂, -CH=C(Cl)-CO-NH-n-C₃H₇, -CH=C(Cl)-CO-NH-i-C₃H₇, -CH=C(Cl)-CO-NH-tert.-C₄H₉, -CH=C(Cl)-CO-NH-cyclopropyl, -CH=C(Cl)-CO-NH-cyclobutyl, -CH=C(Cl)-CO-NH-cyclopentyl, -CH=C(Cl)-CO-NH-cyclohexyl, -CH=C(Cl)-CO-NH-cycloheptyl, -CH=C(Cl)-CO-NH-cyclooctyl, -CH=C(Cl)-CO-pyrrolidin-1-yl, -CH=C(Cl)-CO-piperidin-1-yl, -CH=C(Cl)-CO-morpholin-4-yl, -CH=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -CH=C(Cl)-CO-NH-CH₂C≡CH, -CH=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Cl)-CO-NH-(CH₂)₂Cl, -CH=C(Cl)-CO-NH-C₆H₅, -CH=C(Br)-CO-NH₂, -CH=C(Br)-CO-NHCH₃, -CH=C(Br)-CO-N(CH₃)₂, -CH=C(Br)-CO-NH-C₂H₅, -CH=C(Br)-CO-N(C₂H₅)₂, -CH=C(Br)-CO-NH-n-C₃H₇, -CH=C(Br)-CO-NH-i-C₃H₇, -CH=C(Br)-CO-NH-tert.-C₄H₉, -CH=C(Br)-CO-NH-cyclopropyl, -CH=C(Br)-CO-NH-cyclobutyl, -CH=C(Br)-CO-NH-cyclopentyl, -CH=C(Br)-CO-NH-cyclohexyl, -CH=C(Br)-CO-NH-cycloheptyl, -CH=C(Br)-CO-NH-cyclooctyl, -CH=C(Br)-CO-pyrrolidin-1-yl, -CH=C(Br)-CO-piperidin-1-yl, -CH=C(Br)-CO-morpholin-4-yl, -CH=C(Br)-CO-NH-CH₂CH=C(Br)₂, -CH=C(Br)-CO-NH-CH₂C≡CH, -CH=C(Br)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Br)-CO-NH-(CH₂)₂Cl, -CH=C(Br)-CO-NH-C₆H₅, -CH=C(CN)-CO-NH₂, -CH=C(CN)-CO-NHCH₃, -CH=C(CN)-CO-N(CH₃)₂, -CH=C(CN)-CO-NH-C₂H₅, -CH=C(CN)-CO-N(C₂H₅)₂, -CH=C(CN)-CO-NH-n-C₃H₇, -CH=C(CN)-CO-NH-i-C₃H₇, -CH=C(CN)-CO-NH-tert.-C₄H₉, -CH=C(CN)-CO-NH-cyclopropyl, -CH=C(CN)-CO-NH-cyclobutyl, -CH=C(CN)-CO-NH-cyclopentyl, -CH=C(CN)-CO-NH-cyclohexyl, -CH=C(CN)-CO-NH-cycloheptyl, -CH=C(CN)-CO-NH-cyclooctyl, -CH=C(CN)-CO-pyrrolidin-1-yl, -CH=C(CN)-CO-piperidin-1-yl, -CH=C(CN)-CO-morpholin-4-yl, -CH=C(CN)-CO-NH-CH₂CH=C(CN)₂, -CH=C(CN)-CO-NH-CH₂C≡CH, -CH=C(CN)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CN)-CO-NH-(CH₂)₂Cl, -CH=C(CN)-CO-NH-C₆H₅, -CH=CH-CO-SCH₃, -CH=CH-CO-SC₂H₅, -CH=CH-CO-S-n-C₃H₇, -CH=CH-CO-S-i-C₃H₇, -CH=CH-CO-S-n-C₄H₉, -CH=CH-CO-S-tert.-C₄H₉, -CH=C(CH₃)-CO-SCH₃, -CH=C(CH₃)-CO-SC₂H₅, -CH=C(CH₃)-CO-S-n-C₃H₇, -CH=C(CH₃)-CO-S-i-C₃H₇, -CH=C(CH₃)-CO-S-n-C₄H₉, -CH=C(CH₃)-CO-S-tert.-C₄H₉, -CH=C(C₂H₅)-CO-SCH₃, -CH=C(C₂H₅)-CO-SC₂H₅, -CH=C(C₂H₅)-CO-S-n-C₃H₇, -CH=C(C₂H₅)-CO-S-i-C₃H₇, -CH=C(C₂H₅)-CO-S-n-C₄H₉, -CH=C(C₂H₅)-CO-S-tert.-C₄H₉, -CH=C(Cl)-CO-SCH₃, -CH=C(Cl)-CO-SC₂H₅, -CH=C(Cl)-CO-S-n-C₃H₇, -CH=C(Cl)-CO-S-i-C₃H₇, -CH=C(Cl)-CO-S-n-C₄H₉, -CH=C(Cl)-CO-S-tert.-C₄H₉, -CH=C(Br)-CO-SCH₃, -CH=C(Br)-CO-SC₂H₅, -CH=C(Br)-CO-S-n-C₃H₇, -CH=C(Br)-CO-S-i-C₃H₇, -CH=C(Br)-CO-S-n-C₄H₉, -CH=C(Br)-CO-S-tert.-C₄H₉, -CH=C(CN)-CO-SCH₃, -CH=C(CN)-CO-SC₂H₅, -CH=C(CN)-CO-S-n-C₃H₇, -CH=C(CN)-CO-S-i-C₃H₇, -CH=C(CN)-CO-S-n-C₄H₉, -CH=C(CN)-CO-S-tert.-C₄H₉, -CH=C(COCH₃)-CO-OCH₃, -CH=C(COC₂H₅)-CO-OCH₃, -CH=C(CO-n-C₃H₇)-CO-OCH₃, -CH=C(COCH₃)-CO-OC₂H₅, -CH=C(COC₂H₅)-CO-OC₂H₅, -CH=C(CO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COCH₃)-CO-O-n-C₃H₇, -CH=C(COC₂H₅)-CO-O-n-C₃H₇, -CH=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-OCH₃, -CH=C(CF₃)-CO-OC₂H₅, -CH=C(CF₃)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-O-i-C₃H₇, -CH=C(CF₃)-CO-O-n-C₄H₉, -CH=C(CF₃)-CO-O-tert.-C₄H₉, -CH=C(COOCH₃)₂, -CH=C(COOC₂H₅)₂, -CH=C(COOCH₃)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)-CO-OCH₃, -CH=C(COO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)₂, -CH=CH-CH=CH-COOH, -CH=CH-CH=CH-CO-OCH₃, -CH=CH-CH=CH-CO-OC₂H₅, -CH=CH-CH=C(COOCH₃)₂, -CH=CH-CH=C(CN)-CO-OCH₃, -CH=CH-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-OCH₃, -CH=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CH=C(Cl)-CO-OCH₃, -CH=C(CH₃)-CH=C(Br)-CO-OCH₃, -CH=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-NH₂, -CH=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -CH=CH-(CH₂)₂-COOH, -CH=CH-(CH₂)₂-CO-OCH₃, -CH=CH-(CH₂)₂-CO-OC₂H₅, -CH=CH-CH₂-CH(COOCH₃)₂, -CH=CH-CH₂-CH(COOC₂H₅)₂, -CH=CH-CH₂-CH(CN)-CO-OCH₃, -CH=CH-CH₂-CH(CN)-CO-OC₂H₅, -CH=CH-CH₂-CH(CH₃)-CO-OCH₃, -CH=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -CH=CH-(CH₂)₂-CO-NH₂, -CH=CH-(CH₂)₂-CO-NH-CH₃, -CH=CH-CH₂-COOH, -CH=CH-CH₂-CO-OCH₃, -CH=CH-CH₂-CO-OC₂H₅, -CH=C(COOCH₃)-CH₂-CO-OCH₃, -CH=C(COOCH₃)-CH₂-CO-OC₂H₅, -CH=CH-CH₂-CO-NH₂, -CH=CH-CH₂-CO-NH-CH₃, -CH=CH-CH₂-CO-N(CH₃)₂, -CH(OCH₃)₂, -CH(SCH₃)₂, -CH(OC₂H₅)₂, -CH(SC₂H₅)₂, -CH(O-n-C₃H₇)₂, -CH(O-i-C₃H₇)₂, -CH(S-n-C₃H₇)₂, -CH(S-i-C₃H₇)₂, -CH(O-n-C₄H₉)₂, -CH(O-i-C₄H₉)₂, -CH(O-s-C₄H₉)₂, -CH(O-tert.-C₄H₉)₂, -CH(S-n-C₄H₉)₂, -CH(S-i-C₄H₉)₂, -CH(S-s-C₄H₉)₂, -CH(S-tert.-C₄H₉)₂, -CH(OC₅H₁₁)₂, 1,3-Dioxolan-2-yl, 1,3-Dithio­ lan-2-yl, 1,3-Oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 4-Methyl-1,3-dithiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 5-Methyl-1,3-oxathiolan-2-yl, 4-Ethyl-1,3-dioxolan-2-yl, 4-Ethyl- 1,4-dithiolan-2-yl, 4-Ethyl-1,3-oxathiolan-2-yl, 5-Ethyl-1,3-oxa­ thiolan-2-yl, 4,5-Dimethyl-1,3-dioxolan-2-yl, 4,4-Dimethyl-1,3- dioxolan-2-yl, 4,5-Dimethyl-1,3-dithiolan-2-yl, 5,5-Dimethyl-1,3- dithiolan-2-yl, 4,5-Dimethyl-1,3-oxathiolan-2-yl, 5,5-Dimethyl- 1,3-oxathiolan-2-yl, 4,4-Dimethyl-1,3-oxathiolan-2-yl, 4-Vinyl- 1,3-dioxolan-2-yl, 4-Vinyl-1,3-dithiolan-2-yl, 4-Vinyl-1,3-oxa­ thiolan-2-yl, 5-Vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3- dioxolan-2-yl, 4-Chlormethyl-1,3-dithiolan-2-yl, 4-Chlormethyl- 1,3-oxathiolan-2-yl, 5-Chlormethyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-1,3-dithio­ lan-2-yl, 4-Hydroxymethyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl- 1,3-oxathiolan-2-yl, 4-Methoxymethyl-1,3-dioxolan-2-yl, 4-Allyl­ oxymethyl-1,3-dioxolan-2-yl, 4-Propargyloxymethyl-1,3-dioxolan- 2-yl, 4-Acetoxymethyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-1,3-dithiolan-2-yl, 4-Propargyl­ oxymethyl-1,3-dithiolan-2-yl, 4-Acetoxymethyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl-1,3-oxathiolan-2-yl, 5-Allyloxy­ methyl-1,3-oxathiolan-2-yl, 4-Propargyloxymethyl-1,3-oxathiolan-2-yl, 5-Propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxymethyl- 1,3-oxathiolan-2-yl, 5-Acetoxymethyl-1,3-oxathiolan-2-yl, 4-Methylthiomethyl-1,3-dioxolan-2-yl, 4-Methylthiomethyl-1,3- dithiolan-2-yl, 4-Carboxy-1,3-dioxolan-2-yl, 4-Carboxy-1,3- dithiolan-2-yl, 4-Methoxycarbonyl-1,3-dioxolan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-1,3-dithiolan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-4-methyl- 1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-di­ thiolan-2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-1,3- dithiolan-2-yl, 1,3-Dioxan-2-yl, 1,3-Dithian-2-yl, 1,3-Oxathian- 2-yl, 5-Methyl-1,3-dioxan-2-yl, 5-Methyl-1,3-dithian-2-yl, 5-Methyl-1,3-oxathian-2-yl, 5,5-Dimethyl-1,3-dioxan-2-yl, 4,6-Dimethyl- 1,3-dioxan-2-yl, 4,4-Dimethyl-1,3-dioxan-2-yl, 5,5-Dimethyl- 1,3-dithian-2-yl, 4,6-Dimethyl-1,3-dithian-2-yl, 4,4-Dimethyl- 1,3-dithian-2-yl, 5,5-Dimethyl-1,3-oxathian-2-yl, 4,4-Dimethyl- 1,3-oxathian-2-yl, 6,6-Dimethyl-1,3-oxathian-2-yl, 4-Hydroxymethyl-1,3-dioxan-2-yl, 4-Methoxymethyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-1,3-dithian-2-yl, 4-Methoxymethyl-1,3-dithian-2-yl, 4-Allyloxymethyl-1,3-dithian-2-yl, 4-Acetoxymethyl- 1,3-dithian-2-yl, 4-Chlormethyl-1,3-dioxan-2-yl, 4-Chlormethyl- 1,3-dithian-2-yl, 1,3-Dioxepan-2-yl, 1,3-Dithiepan-2-yl, 1,3-Dioxep-5-en-2-yl, 4-Methoxycarbonyl-1,3-dioxan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-1,3-dithian-4-yl, 4-n-Butoxycarbonyl-1,3-dithian-2-yl, 4-Methoxycarbonyl-4- methyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-4-methyl- 1,3-dithian-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithian-2-yl, -C(CH₃)(OCH₃)₂, -C(CH₃)(SCH₃)₂, -C(CH₃)(OC₂H₅)₂, -C(CH₃)(SC₂H₅)₂, -C(CH₃)(O-n-C₃H₇)₂, -C(CH₃)(O-i-C₃H₇)₂, -C(CH₃)(S-n-C₃H₇)₂, -C(CH₃)(S-i-C₃H₇)₂, -C(CH₃)(O-n-C₄H₉)₂, -C(CH₃)(O-i-C₄H₉)₂, -C(CH₃)(O-s-C₄H₉)₂, -C(CH₃)(O-tert.-C₄H₉)₂, -C(CH₃)(S-n-C₄H₉)₂, -C(CH₃)(S-i-C₄H₉)₂, -C(CH₃)(S-s-C₄H₉)₂, -C(CH₃)(S-tert.-C₄H₉)₂, -C(CH₃)(O-n-C₅H₁₁)′′, 2-Methyl-1,3-dioxolan-2-yl, 2-Methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-oxathiolan-2-yl, 2,4-Dimethyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-1,3- oxathiolan-2-yl, 2,5-Dimethyl-1,3-oxathiolan-2-yl, 4-Ethyl-2- methyl-1,3-dioxolan-2-yl, 4-Ethyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Ethyl-2-methyl-1,3- oxathiolan-2-yl, 2,4,5-Trimethyl-1,3-dioxolan-2-yl, 2,4,4-Trimethyl- 1,3-dioxolan-2-yl, 2,4,5-Trimethyl-1,3-dithiolan-2-yl, 2,4,4-Trimethyl-1,3-dithiolan-2-yl, 2,4,5-Trimethyl-1,3-oxathiolan-2-yl, 2,4,4-Trimethyl-1,3-oxathiolan-2-yl, 2-Methyl-4-vinyl- 1,3-dioxolan-2-yl, 2-Methyl-4-vinyl-1,3-dithiolan-2-yl, 2-Methyl- 4-vinyl-1,3-oxathiolan-2-yl, 2-Methyl-5-vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-dioxolan-2-yl, 4-Chlormethyl-2- methyl-1,3-dithiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl- 2-methyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-2- methyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dioxolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxy- 2-methyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dithiolan-2-yl, 4-Acetoxy-2- methyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl- 2-methyl-1,3-oxathiolan-2-yl, 5-Allyloxymethyl-2- methyl-1,3-oxathional-2-yl, 2-Methyl-4-propargyloxymethyl-1,3- oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxy-2-methyl-1,3-oxathiolan-2-yl, 5-Acetoxy-2-methyl- 1,3-oxathiolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dioxolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-2- methyl-1,3-dioxolan-2-yl, 4-Carboxy-2-methyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-2- methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl- 2-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-2- methyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-ethoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4- ethoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-n-butoxy­ carbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl-1,3- dithiolan-2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-dioxan-2- yl, 2-Methyl-1,3-dithian-2-yl, 2-Methyl-1,3-oxathian-2-yl, 2,5- Dimethyl-1,3-dioxan-2-yl, 2,5-Dimethyl-1,3-dithian-2-yl, 2,5-Di­ methyl-1,3-oxathian-2-yl, 2,5,5-Trimethyl-1,3-dioxan-2-yl, 2,4,6- Trimethyl-1,3-dioxan-2-yl, 2,4,4-Trimethyl-1,3-dioxan-2-yl, 2,5,5-Trimethyl-1,3-dithian-2-yl, 2,4,6-Trimethyl-1,3-dithian-2- yl, 2,4,4-Trimethyl-1,3-dithian-2-yl, 2,5,5-Trimethyl-1,3-oxa­ thian-2-yl, 2,4,4-Trimethyl-1,3-oxathian-2-yl, 2,6,6-Trimethyl- 1,3-oxathian-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-2- methyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dithian-2-yl, 4-Methoxymethyl-2- methyl-1,3-dithian-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithian-2- yl, 4-Acetoxymethyl-2-methyl-1,3-dithian-2-yl, 4-Chlormethyl-2- methyl-1,3-dioxan-2-yl, 4-Chlormethyl-2-methyl-1,3-dithian-2-yl, -C(CH₃)=N, -C(CH₃)=N-CH₃, -C(CH₃)=N-C₂H₅, -C(CH₃)=N-n-C₃H₇, -C(CH₃)=N-i-C₃H₇, -C(CH₃)=N-n-C₄H₉, -C(CH₃)=N-CH₂CH=CH₂, -C(CH₃)=N-CH₂CH=CH₂-CH₃, -C(CH₃)=N-CH₂C≡CH, -C(CH₃)=N-CH₂C≡C-CH₃, -C(CH₃)=N-cyclopropyl, -C(CH₃)=N-cyclobutyl, -C(CH₃)=N-cyclo­ pentyl, -C(CH₃)=N-cyclohexyl, -C(CH₃)=N-cycloheptyl, -C(CH₃)=N-CH₂-CH₂Cl, -C(CH₃)=N-CH₂Cl, -C(CH₃)=N-C₆H₅, -C(CH₃)=N-(2-F-C₆H₄), -C(CH₃)=N-(3-F-C₆H₄), -C(CH₃)=N-(4-F-C₆H₄), -C(CH₃)=N-(2-Cl-C₆H₄), -C(CH₃)=N-(3-Cl-C₆H₄), -C(CH₃)=N-(4-Cl-C₆H₄), -C(CH₃)=N-(2-CH₃-C₆H₄), -C(CH₃)=N-(3-CH₃-C₆H₄), -C(CH₃)=N-(4-CH₃-C₆H₄), -C(CH₃)=N-(2-CF₃-C₆H₄), -C(CH₃)=N-(3-CF₃-C₆H₄), -C(CH₃)=N-(4-CF₃-C₆H₄), -C(CH₃)=N-(2-OCH₃-C₆H₄), -C(CH₃)=N-(3-OCH₃-C₆H₄), -C(CH₃)=N-(4-OCH₃-C₆H₄), -C(CH₃)=N-(4-NO₂-C₆H₄), -C(CH₃)=N-(4-CN-C₆H₄), -C(CH₃)=N-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-(2,4-(CH₃)₂-C₆H₃), -C(CH₃)=N-CH₂-OCH₃, -C(CH₃)=N-CH₂-OC₂H₅, -C(CH₃)=N-CH₂CH₂-OCH₃, -C(CH₃)=N-CH₂CH₂-OC₂H₅, -C(CH₃)=N-OH, -C(CH₃)=N-OCH₃, -C(CH₃)=N-OC₂H₅, -C(CH₃)=N-O-n-C₃H₇, -C(CH₃)=N-O-i-C₃H₇, -C(CH₃)=N-O-n-C₄H₉, -C(CH₃)=N-O-i-C₄H₉, -C(CH₃)=N-O-s-C₄H₉, -C(CH₃)=N-O-tert.-C₄H₉, -C(CH₃)=N-OCH2-CH=CH₂, -C(CH₃)=N-OCH(CH₃)-CH=CH₂, -C(CH₃)=N-OCH₂-C≡CH, -C(CH₃)=N-CH(CH₃)-C≡, -C(CH₃)=N-OCH₂-CH=C-CH₃, -C(CH₃)=N-OCH₂CH₂-Cl, -C(CH₃)=N-OCH₂CH₂-F, -C(CH₃)=N-OCH₂-CF₃, -C(CH₃)=N-OCH₂-CH=CHCl, -C(CH₃)=N-OCH₂-C(Cl)=CH₂, -C(CH₃)=N-OCH₂-C(Br)=CH₂, -C(CH₃)=N-OCH₂-CH=C(Cl)-CH₃, -C(CH₃)=N-O-CO-CH₃, -C(CH₃)=N-O-CO-C₂H₅, -C(CH₃)=N-OCH₂-CN, -C(CH₃)=N-OCH₂-CH=CH-CH₂-OCH₃, -C(CH₃)=N-OCH₂-CH=CH-CH₂-O-tert.-C₄H₉, -C(CH₃)=N-O-(CH₂)₃-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-(4-Cl-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-C₆H₅, -C(CH₃)=N-OCH₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(3-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH₂-(4-CH₃O-C₆H₄), -C(CH₃)=N-OCH₂-CH=C(CH₃)-C₆H₅, -C(CH₃)=N-O-(CH₂)₂-CH=CH-(3,4-Cl₂C₆H₃), -C(CH₃)=N-O-(CH₂)₃-C≡C-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-OCH₃, -C(CH₃)=N-OCH₂CH₂-OCH₃, -C(CH₃)=N-OCH₂-OC₂H₅, -C(CH₃)=N-OCH(CH₃)-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=N-NH₂, -C(CH₃)=N-NH-CH₃, -C(CH₃)=N-NH-C₂H₅, -C(CH₃)=N-NH-n-C₃H₇, -C(CH₃)=N-NH-i-C₃H₇, -C(CH₃)=N-NH-n-C₄H₉, -C(CH₃)=N-NH-i-C₄H₉, -C(CH₃)=N-NH-s-C₄H₉, -C(CH₃)=N-NH-tert.-C₄H₉, -C(CH₃)=N-NH-cyclopropyl, -C(CH₃)=N-NH- cyclobutyl, -C(CH₃)=N-NH-cyclopentyl, -C(CH₃)=N-NH-cyclohexyl, -C(CH₃)=N-NH-cycloheptyl, -C(CH₃)=N-N(CH₃)₂, -C(CH₃)=N-N(C₂H₅)₂, -C(CH₃)=N-N(n-C₃H₇)₂, -C(CH₃)=N-N(i-C₃H₇)₂, -C(CH₃)=N-NH-CH₂-C=CH, -C(CH₃)=N-NH-CH₂≡CH, -C(CH₃)=N-N(CH₃)-CH₂-C≡CH, -C(CH₃)=N-NH-CH₂CF₃, -C(CH₃)=N-NH-CO-CH₃, -C(CH₃)=N-NH-CO-C₂H₅, -C(CH₃)=N-NH-CO-OCH₃, -C(CH₃)=N-NH-CO-OC₂H₅, -C(CH₃)=N-NH-CO-O-tert.-C₄H₉, -C(CH₃)=N- pyrrolidin-1-yl, -C(CH₃)=N-piperidin-1-yl, -C(CH₃)=N-morpholin- 4-yl, -C(CH₃)=N-NH-C₆H₅, -C(CH₃)=N-NH-(4-Cl-C₆H₄), -C(CH₃)=N-NH-(4-NO₂-C₆H₄), -C(CH₃)=N-NH-(4-F-C₆H₄), -C(CH₃)=N-NH-(4-CH₃O-C₆H₄), -C(CH₃)=N-NH-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-NH-(2,4-(NO₂)₂-C₆H₃), -C(CH₃)=N-NH-CO-NH₂, -C(CH₃)=N-NH-CO-NHCH₃, -C(CH₃)=N-NH-CO-NHC₂H₅, -C(CH₃)=N-NH-CO-N(CH₃)₂, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=CH-CO-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-O-n-C₄H₉, -C(CH₃)=CH-CO-O-tert.-C₄H₉, -C(CH₃)=CH-CO-O-cyclopropyl, -C(CH₃)=CH-CO-O-cyclobutyl, -C(CH₃)=CH-CO-O-cyclopentyl, -C(CH₃)=CH-CO-O-cyclohexyl, -C(CH₃)=CH-CO-O-cycloheptyl, -C(CH₃)=C(CH₃)-COOH, -C(CH₃)=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-cyclopropyl, -C(CH₃)=C(CH₃)-CO-O-cyclobutyl, -C(CH₃)=C(CH₃)-CO-O-cyclopentyl, -C(CH₃)=C(CH₃)-CO-O-cyclohexyl, -C(CH₃)=C(CH₃)-CO-O-cycloheptyl, -C(CH₃)=C(C₂H₅)-COOH, -C(CH₃)=C(C₂H₅)-CO-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-cyclo­ propyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-O- cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-O-cycloheptyl, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-O-n-C₄H₉, -C(CH₃)=C(Cl)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-O-cyclopropyl, -C(CH₃)=C(Cl)-CO-O-cyclobutyl, -C(CH₃)=C(Cl)-CO-O-cyclopentyl, -C(CH₃)=C(Cl)-CO-O-cyclohexyl, -C(CH₃)=C(Cl)-CO-O-cycloheptyl, -C(CH₃)=C(Br)-COOH, -C(CH₃)=C(Br)-CO-OCH₃, -C(CH₃)=C(Br)-CO-OC₂H₅, -C(CH₃)=C(Br)-CO-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-O-n-C₄H₉, -C(CH₃)=C(Br)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-O-cyclopropyl, -C(CH₃)=C(Br)-CO-O-cyclobutyl, -C(CH₃)=C(Br)-CO-O-cyclopentyl, -C(CH₃)=C(Br)-CO-O-cyclohexyl, -C(CH₃)=C(Br)-CO-O-cycloheptyl, -C(CH₃)=C(CN)-COOH, -C(CH₃)=C(CN)-CO-OCH₃, -C(CH₃)=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CN)-CO-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-O-n-C₄H₉, -C(CH₃)=C(CN)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-O-cyclopropyl, -C(CH₃)=C(CN)-CO-O-cyclobutyl, -C(CH₃)=C(CN)-CO-O-cyclopentyl, -C(CH₃)=C(CN)-CO-O-cyclohexyl, -C(CH₃)=C(CN)-CO-O-cycloheptyl, -C(CH₃)=CH-CO-OCH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-OCH(CH₃)-OCH₃, -C(CH₃)=CH-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=CH-CO-OCH₂CH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-O-i-C₃H₇, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-O-i-C₃H₇, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-O-i-C₃H₇, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃ )=C(CN)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-CH₃, -C(CH₃)=CH-CO-OCH₂-CCl₃, -C(CH₃)=CH-CO-OCH₂-oxiranyl, -C(CH₃)=CH-CO-O-(CH₂)₃-Br, -C(CH₃)=CH-CO-OCH₂-CH=CH₂, -C(CH₃)=CH-CO-OCH₂-C≡CH, -C(CH₃)=CH-CO-OCH₂-CN, -C(CH₃)=CH-CO-OCH₂CH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CF₃, -C(CH₃)=C(CH₃)-CO-OCH₂-CCl₃, -C(CH₃)=C(CH₃)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CH₃)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(CH₃)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CH₃)-CO-OCH₂-C≡CH, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CF₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CCl₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-oxiranyl, -C(CH₃)=C(C₂H₅)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(C₂H₅)-CO-OCH₂-C≡CH, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂-CF₃, -C(CH₃)=C(Cl)-CO-OCH₂-CCl₃, -C(CH₃)=C(Cl)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Cl)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Cl)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Cl)-CO-OCH₂-C≡CH, -C(CH₃)=C(Cl)-CO-OCH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂-CF₃, -C(CH₃)=C(Br)-CO-OCH₂-CCl₃, -C(CH₃)=C(Br)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Br)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Br)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Br)-CO-OCH₂-C≡CH, -C(CH₃)=C(Br)-CO-OCH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂CH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂-CF₃, -C(CH₃)=C(CN)-CO-OCH₂-CCl₃, -C(CH₃)=C(CN)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CN)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(CN)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CN)-CO-OCH₂-C≡CH, -C(CH₃)=C(CN)-CO-OCH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂CH₂-CN, -C(CH₃)=CH-CO-CH₃, -C(CH₃)=CH-CO-C₂H₅, -C(CH₃)=CH-CO-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-n-C₄H₉, -C(CH₃)=CH-CO-tert.-C₄H₉, -C(CH₃)=CH-CO-CH₂Cl, -C(CH₃)=CH-CO-CH₂Br, -C(CH₃)=CH-CO-CHCl₂, -C(CH₃)=CH-CO-CH₂-OCH₃, -C(CH₃)=CH-CO-CH(OCH₃)₂, -C(CH₃)=CH-CO-CH₂-SCH₃, -C(CH₃)=C(CH₃)-CO-CH₃, -C(CH₃)=C(CH₃)-CO-C₂H₅, -C(CH₃)=C(CH₃)-CO-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-CH₂Cl, -C(CH₃)=C(CH₃)-CO-CH₂Br, -C(CH₃)=C(CH₃)-CO-CHCl₂, -C(CH₃)=C(CH₃)-CO-CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-CH(OCH₃)₂, -C(CH₃)=C(CH₃)-CO-CH₂-SCH₃, -C(CH₃)=C(C₂H₅)-CO-CH₃, -C(CH₃)=C(C₂H₅)-CO-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-CH₂Cl, -C(CH₃)=C(C₂H₅)-CO-CH₂Br, -C(CH₃)=C(C₂H₅)-CO-CHCl₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-CH(OCH₃)₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-SCH₃, -C(CH₃)=C(Cl)-CO-CH₃, -C(CH₃)=C(Cl)-CO-C₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-n-C₄H₉, -C(CH₃)=C(Cl)-CO-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-CH₂Cl, -C(CH₃)=C(Cl)-CO-CHCl₂, -C(CH₃)=C(Cl)-CO-CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-CH(OCH₃)₂, -C(CH₃)=C(Cl)-CO-CH₂-SCH₃, -C(CH₃)=C(Br)-CO-CH₃, -C(CH₃)=C(Br)-CO-C₂H₅, -C(CH₃)=C(Br)-CO-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-n-C₄H₉, -C(CH₃)=C(Br)-CO-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-CH₂Cl, -C(CH₃)=C(Br)-CO-CH₂Br, -C(CH₃)=C(Br)-CO-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-CH(OCH₃)₂, -C(CH₃)=C(Br)-CO-CH₂-SCH₃, -C(CH₃)=C(CN)-CO-CH₃, -C(CH₃)=C(CN)-CO-C₂H₅, -C(CH₃)=C(CN)-CO-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-n-C₄H₉, -C(CH₃)=C(CN)-CO-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-CH₂Cl, -C(CH₃)=C(CN)-CO-CH₂Br, -C(CH₃)=C(CN)-CO-CHCl₂, -C(CH₃)=C(CN)-CO-CH₂-OCH₃, -C(CH₃)=C(CN)-CO-CH(OCH₃)₂, -C(CH₃)=C(CN)-CO-CH₂-SCH₃, -C(CH₃)=CH-CO-C₆H₅, -C(CH₃)=CH-CO-(4-Cl-C₆H₄), -C(CH₃)=C(CH₃)-CO-C₆H₅, -C(CH₃)=C(CH₃)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(C₂H₅)-CO-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(Cl)-CO-C₆H₅, -C(CH₃)=C(Br)-CO-C₆H₅, -C(CH₃)=C(CN)-CO-C₆H₅, -C(CH₃)=CH-CO-NH₂, -C(CH₃)=CH-CO-NHCH₃, -C(CH₃)=CH-CO-N(CH₃)₂, -C(CH₃)=CH-CO-NH-C₂H₅, -C(CH₃)=CH-CO-N(C₂H₅)₂, -C(CH₃)=CH-CO-NH-n-C₃H₇, -C(CH₃)=CH-CO-NH-i-C₃H₇, -C(CH₃)=CH-CO-NH-tert.-C₄H₉, -C(CH₃)=CH-CO-NH-cyclopropyl, -C(CH₃)=CH-CO-NH-cyclobutyl, -C(CH₃)=CH-CO-NH-cyclopentyl, -C(CH₃)=CH-CO-NH-cyclohexyl, -C(CH₃)=CH-CO-NH-cycloheptyl, -C(CH₃)=CH-CO-NH-cyclooctyl, -C(CH₃)=CH-CO-pyrrolidin-1-yl, -C(CH₃)=CH-CO-piperidin-1-yl, -C(CH₃)=CH-CO-morpholin-4-yl, -C(CH₃)=CH-CO-NH-CH₂CH=CH₂, -C(CH₃)=CH-CO-NH-CH₂C≡CH, -C(CH₃)=CH-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=CH-CO-NH-(CH₂)₂Cl, -C(CH₃)=CH-CO-NH-C₆H₅, -C(CH₃)=C(CH₃)-CO-NH₂, -C(CH₃)=C(CH₃)-CO-NHCH₃, -C(CH₃)=C(CH₃)-CO-N(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-C₂H₅, -C(CH₃)=C(CH₃)-CO-N(C₂H₅)₂, -C(CH₃)=C(CH₃)-CO-NH-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-NH- cyclopropyl, -C(CH₃)=C(CH₃)-CO-NH-cyclobutyl, -C(CH₃)=C(CH₃)-CO-NH-cyclopentyl, -C(CH₃)=C(CH₃)-CO-NH- cyclohexyl, -C(CH₃)=C(CH₃)-CO-NH-cycloheptyl, -C(CH₃)=C(CH₃)-CO-NH-cyclooctyl, -C(CH₃)=C(CH₃)-CO- pyrrolidin-1-yl, -C(CH₃)=C(CH₃)-CO-piperidin-1-yl, -C(CH₃)=C(CH₃)-CO-morpholin-4-yl, -C(CH₃)=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CH₃)-CO-NH-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-NH₂, -C(CH₃)=C(C₂H₅)-CO-NHCH₃, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)₂, -C(CH₃)=C(C₂H₅)-CO-NH-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-N(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-NH- cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclo­ hexyl, -C(CH₃)=C(C₂H₅)-CO-NH-cycloheptyl, -C(CH₃)=C(C₂H₅)-CO-NH- cyclooctyl, -C(CH₃)=C(C₂H₅)-CO-pyrrolidin-1-yl, -C(CH₃)=C(C₂H₅)-CO-piperidin-1-yl, -C(CH₃)=C(C₂H₅)-CO- morpholin-4-yl, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(C₂H₅)-CO-NH-C₆H₅, -C(CH₃)=C(Cl)-CO-NH₂, -C(CH₃)=C(Cl)-CO-NHCH₃, -C(CH₃)=C(Cl)-CO-N(CH₃)₂, -C(CH₃)=C(Cl)-CO-NH-C₂H₅, -C(CH₃)=C(Cl)-CO-N(C₂H₅)₂, -C(CH₃)=C(Cl)-CO-NH-n-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-i-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-NH-cyclopropyl, -C(CH₃)=C(Cl)-CO-NH-cyclobutyl, -C(CH₃)=C(Cl)-CO-NH-cyclopentyl, -C(CH₃)=C(Cl)-CO-NH-cyclohexyl, -C(CH₃)=C(Cl)-CO-NH-cycloheptyl, -C(CH₃)=C(Cl)-CO-NH-cyclooctyl, -C(CH₃)=C(Cl)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Cl)-CO-piperidin-1- yl, -C(CH₃)=C(Cl)-CO-morpholin-4-yl, -C(CH₃)=C(Cl)-CO-NH-CH₂CH=C(Cl)₂ -C(CH₃)=C(Cl)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-N(CH₃)-CH₂≡CH, -C(CH₃)=C(Cl)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Cl)-NO-NH-C₆H₅, -C(CH₃)=C(Br)-CO-NH₂, -C(CH₃)=C(Br)-CO-NHCH₃, -C(CH₃)=C(Br)-CO-N(CH₃)₂, -C(CH₃)=C(Br)-CO-NH-C₂H₅, -C(CH₃)=C(Br)-CO-N(C₂H₅)₂, -C(CH₃)=C(Br)-CO-NH-n-C₃H₇, -C(CH₃)=C(Br)-CO-NH-i-C₃H₇, -C(CH₃)=C(Br)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-NH-cyclopropyl, -C(CH₃)=C(Br)-CO-NH-cyclobutyl, -C(CH₃)=C(Br)-CO-NH-cyclopentyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cycloheptyl, -C(CH₃)=C(Br)-CO-NH-cyclooctyl, -C(CH₃)=C(Br)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Br)-CO-piperidin-1-yl, -C(CH₃)=C(Br)-CO-morpholin-4-yl, -C(CH₃)=C(Br)-CO-NH-CH₂CH=C(Br)₂, -C(CH₃)=C(Br)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Br)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Br)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Br)-CO-NH-C₆H₅, -C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CN)-CO-NHCH₃, -C(CH₃)=C(CN)-CO-N(CH₃)₂, -C(CH₃)=C(CN)-CO-NH-C₂H₅, -C(CH₃)=C(CN)-CO-N(C₂H₅)₂, -C(CH₃)=C(CN)-CO-NH-n-C₃H₇, -C(CH₃)=C(CN)-CO-NH-i-C₃H₇, -C(CH₃)=C(CN)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-NH-cyclopropyl, -C(CH₃)=C(CN)-CO-NH-cyclobutyl, -C(CH₃)=C(CN)-CO-NH-cyclopentyl, -C(CH₃)=C(CN)-CO-NH-cyclohexyl, -C(CH₃)=C(CN)-CO-NH-cycloheptyl, -C(CH₃)=C(CN)-CO-NH-cyclooctyl, -C(CH₃)=C(CN)-CO-pyrrolidin-1-yl, -C(CH₃)=C(CN)-CO-piperidin-1-yl, -C(CH₃)=C(CN)-CO-morpholin-4-yl, -C(CH₃)=C(CN)-CO-NH-CH₂CH=C(CN)₂, -C(CH₃)=C(CN)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CN)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=(CN)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CN)-CO-NH-C₆H₅, -C(CH₃)=CH-CO-SCH₃, -C(CH₃)=CH-CO-SC₂H₅, -C(CH₃)=CH-CO-S-n-C₃H₇, -C(CH₃)=CH-CO-S-i-C₃H₇, -C(CH₃)=CH-CO-S-n-C₄H₉, -C(CH₃)=CH-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-SCH₃, -C(CH₃)=C(CH₃)-CO-SC₂H₅, -C(CH₃)=C(CH₃)CO-S-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-S-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-SCH₃, -C(CH₃)=C(C₂H₅)-CO-SC₂H₅, -C(CH₃)=C(C₂H₅)-CO-S-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-SCH₃, -C(CH₃)=C(Cl)-CO-SC₂H₅, -C(CH₃)=C(Cl)-CO-S-n-C₃H₇, -C(CH₃)=C(Cl)-CO-S-i-C₃H₇, -C(CH₃)=C(Cl)-CO-S-n-C₄H₉, -C(CH₃)=C(Cl)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-SCH₃, -C(CH₃)=C(Br)-CO-SC₂H₅, -C(CH₃)=C(Br)-CO-S-n-C₃H₇, -C(CH₃)=C(Br)-CO-S-i-C₃H₇, -C(CH₃)=C(Br)-CO-S-n-C₄H₉, -C(CH₃)=C(Br)-CO-S-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-SCH₃, -C(CH₃)=C(CN)-CO-SC₂H₅, -C(CH₃)=C(CN)-CO-S-n-C₃H₇, -C(CH₃)=C(CN)-CO-S-i-C₃H₇, -C(CH₃)=C(CN)-CO-S-n-C₄H₉, -C(CH₃)=C(CN)-CO-S-tert.-C₄H₉, -C(CH₃)=C(COCH₃)-CO-OCH₃, -C(CH₃)=C(COC₂H₅)-CO-OCH₃, -C(CH₃)=C(CO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COCH₃)-CO-OC₂H₅, -C(CH₃)=C(COC₂H₅)-CO-OC₂H₅, -C(CH₃)=C(CO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COCH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(COC₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-OCH₃, -C(CH₃)=C(CF₃)-CO-OC₂H₅, -C(CH₃)=C(CF₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CF₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(COOCH₃)₂, -C(CH₃)=C(COOC₂H₅)₂, -C(CH₃)=C(COOCH₃)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)₂, -C(CH₃)=CH-CH=CH-COOH, -C(CH₃)=CH-CH=CH-CO-OCH₃, -C(CH₃)=CH-CH=CH-CO-OC₂H₅, -C(CH₃)=CH-CH=C(COOCH₃)₂, -C(CH₃)=CH-CH=C(CN)-CO-OCH₃, -C(CH₃)=CH-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CN)CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH₂, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -C(CH₃)=CH-(CH₂)₂-COOH, -C(CH₃)=CH-(CH₂)₂-CO-OCH₃, -C(CH₃)=CH-(CH₂)₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(COOCH₃)₂, -C(CH₃)=CH-CH₂-CH(COOC₂H₅)₂, -C(CH₃)=CH-CH₂-CH(CN)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CN)-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -C(CH₃)=CH-(CH₂)₂-CO-NH₂, -C(CH₃)=CH-(CH₂)₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-COOH, -C(CH₃)=CH-CH₂-CO-OCH₃, -C(CH₃)=CH-CH₂-CO-OC₂H₅, -C(CH₃)=C(COOCH₃)-CH₂-CO-OCH₃, -C(CH₃)=C(COOCH₃)-CH₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CO-NH₂, -C(CH₃)=CH-CH₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-CO-N(CH₃)₂.
wobei W für eine der folgenden Bedeutungen steht:
-CHO, -COCH₃, -COC₂H₅, -CO-n-C₃H₇, -CO-i-C₃H₇, -CO-n-C₄H₉, -CO-i-C₄H₉, -CO-s-C₄H₉, -CO-tert.-C₄H₉, -CO-CH₂CH=CH₂, -CO-CF₃, -COCCl₃, -COCH₂C≡CH, -CO-cyclopropyl, -CO-cyclobutyl, -CO-cyclo­ pentyl, -CO-cyclohexyl, -CO-CN, -CO-COOCH₃, -CO-COOC₂H₅, -CH=NH, -CH=NCH₃, -CH=NC₂H₅, -CH=N-n-C₃H₅, -CH=N-i-C₃H₅, -CH=N-n-C₄H₉, -CH=NCH₂CH=CH₂, -CH=NCH₂CH=CH₂-CH₃, -CH=NCH₂≡CH, -CH=NCH₂C≡C-CH₃, -CH=N-cyclopropyl, -CH=N-cyclobutyl, -CH=N-cyclopentyl, -CH=N-cyclohexyl, -CH=N-cycloheptyl, -CH=N-CH₂-CH₂Cl, -CH=N-CH₂Cl, -CH=N-C₆H₅, -CH=N-(4-Br-C₆H₄), -CH=N-3-F-C₆H₄, -CH=N-4-F-C₆H₄, -CH=N-2-Cl-C₆H₄, -CH=N-3-Cl-C₆H₄, -CH=N-4-Cl-C₆H₄, -CH=N-2-Br-C₆H₄, -CH=N-2-F-C₆H₄, -CH=N-2-CH₃-C₆H₄, -CH=N-3-CH₃-C₆H₄, -CH=N-4-CH₃-C₆H₄, -CH=N-2-CF₃-C₆H₄, -CH=N-3-CF₃-C₆H₄, -CH=N-4-CF₃-C₆H₄, -CH=N-2-OCH₃-C₆H₄, -CH=N-3-OCH₃-C₆H₄, -CH=N-4-OCH₃-C₆H₄, -CH=N-4-NO₂-C₆H₄, -CH=N-4-CN-C₆H₄, -CH=N-2,4-(Cl,Cl)-C₆H₄, -CH=N-2,4-(CH₃,CH₃)-C₆H 99999 00070 552 001000280000000200012000285919988800040 0002004131038 00004 99880₄, -CH=N-CH₂OCH₃ -CH=N-CH₂OC₂H₅, -CH=N-CH₂CH₂OCH₃, -CH=N-CH₂CH₂OC₂H₅, -CH=N-OH, -CH=N-OCH₃, -CH=N-OC₂H₅, -CH=N-O-n-C₃H₇, -CH=N-O-i-C₃H₇, -CH=N-O-n-C₄H₉, -CH=N-O-i-C₄H₉, -CH=N-O-s-C₄H₉, -CH=N-O-tert.-C₄H₉, -CH=N-O-CH₂CH=CH₂, -CH=N-O-CH(CH₃)CH=CH₂, -CH=N-O-CH₂C≡CH, -CH=N-O-CH(CH₃)-C≡CH, -CH=N-O-CH₂-CH=CH-CH₃, -CH=N-O-CH₂-CH₂-Cl, -CH=N-O-CH₂-CH₂-F, -CH=N-O-CH₂-CF₃, -CH=N-O-CH₂-CH=CHCl, -CH=N-O-CH₂-CCl=CH₂, -CH=N-O-CH₂-CBr=CH₂, -CH=N-O-CH₂-CH=CCl-CH₃, -CH=N-OC(O)CH₃, -CH=N-OC(O)C₂H₅, -CH=N-O-CH₂-CN, -CH=N-O-CH₂-CH=CH-CH₂-O-CH₃, -CH=N-O-CH₂-CH=CH-CH₂-O-tert.-C₄H₉, -CH=N-O-(CH₂)₃-C₆H₅, -CH=N-O-(CH₂)₄-C₆H₅, -CH=N-O-(CH₂)₄-4-Cl-C₆H₄, -CH=N-O-(CH₂)₄-4-OCH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-CH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-C₆H₅, -CH=N-O-CH₂CH=CH-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CH-3-OCH₃-C₆H₄, -CH=N-O-(CH₂)₂CH=CH-4-F-C₆H₄, -CH=N-O-(CH₂)CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CHCH₂-4-OCH₃-C₆H₄, -CH=N-O-CH₂-CH=C(CH₃)-C₆H₅, -CH=N-O-(CH₂)₂CH=CH-3,4(Cl,Cl)-C₆H₃, -CH=N-O-(CH₂)₃C≡C-4-F-C₆H₄, -CH₂=N-OCHOCH₃, -CH=N-OC₂H₄OCH₃, -CH=N-OCH₂OC₂H₅, -CH=N-OCH(CH₃)OCH₃, -CH=N-OCH(CH₃)COOCH₃, -CH=N-OCH(CH₃)COO-n-C₄H₉, -CH=N-NH₂, -CH=N-NHCH₃, -CH=N-NHC₂H₅, -CH=N-NH-n-C₃H₇, -CH=N-NH-i-C₃H₇, -CH=N-NH-n-C₄H₉, -CH=N-NH-i-C₄H₉, -CH=N-NH-s-C₄H₉, -CH=N-NH-tert.-C₄H₉, -CH=N-NH-cyclopropyl, -CH=N-NH-cyclobutyl, -CH=N-NH-cyclopentyl, -CH=N-NH-cyclohexyl, -CH=N-NH-cycloheptyl, -CH=N-N(CH₃)₂, -CH=N-N(C₂H₅)₂, -CH=N-N(C₃H₇)₂, -CH=N-N(i-C₃H₇)(CH₃), -CH=N-NHCH₂-C=CH, -CH=N-NHCH₂-C≡CH, -CH=N-N(CH₃)-CH₂-C≡CH, -CH=N-NHCH₂CF₃, -CH=N-NH-CO-CH₃, -CH=N-NH-CO-CH₂H₅, -CH=N-NH-COOCH₃, -CH=N-NH-COOC₂H₅, -CH=N-NH-COO-tert.-C₄H₉, -CH=N-pyrrolidin-1-yl, -CH=N-piperidin-1-yl, -CH=N-morpholin-4-yl, -CH=N-NH-C₆H₅, -CH=N-NH-(4-Cl-C₆H₄), -CH=N-NH-(4-NO₂-C₆H₄), -CH=N-NH-(4-F-C₆H₄), -CH=N-NH-(4-CH₃O-C₆H₄), -CH=N-NH-(2,4-Cl₂-C₆H₃), -CH=N-NH-(2,4-(NO₂)₂-C₆H₃), -CH=N-NH-CO-NH₂, -CH=N-NH-CO-NHCH₃, -CH=N-NH-CO-NHC₂H₅, -CH=N-NH-CO-N(CH₃)₂, -CH=CH-COOH, -CH=CH-CO-OCH₃, -CH=CH-C-CO-OC₂H₅, -CH=CH-CO-O-n-C₃H₇, -CH=CH-CO-O-i-C₃H₇, -CH=CH-CO-O-n-C₄H₉, -CH=CH-CO-O-tert.-C₄H₉, -CH=CH-CO-O-cyclopropyl, -CH=CH-CO-O-cyclobutyl, -CH=CH-CO-O-cyclopentyl, -CH=CH-CO-O-cyclohexyl, -CH=CH-CO-O-cycloheptyl, -CH=C(CH₃)-COOH, -CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CO-O-n-C₃H₇, -CH=C(CH₃)-CO-O-i-C₃H₇, -CH=C(CH₃)-CO-O-n-C₄H₉, -CH=C(CH₃)-CO-O-tert.-C₄H₉, -CH=C(CH₃)-CO-O-cyclopropyl, -CH=C(CH₃)-CO-O-cyclobutyl, -CH=C(CH₃)-CO-O-cyclopentyl, -CH=C(CH₃)-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cycloheptyl, -CH=C(C₂H₅)-COOH, -CH=C(C₂H₅)-CO-OCH₃, -CH=C(C₂H₅)-CO-OC₂H₅, -CH=C(C₂H₅)-CO-O-n-C₃H₇, -CH=C(C₂H₅)-CO-O-i-C₃H₇, -CH=C(C₂H₅)-CO-O-n-C₄H₉, -CH=C(C₂H₅)-CO-O-tert.-C₄H₉, -CH=C(C₂H₅)-CO-O-cyclopropyl, -CH=C(C₂H₅)-CO-O-cyclobutyl, -CH=C(C₂H₅)-CO-O-cyclopentyl, -CH=C(C₂H₅)-CO-O-cyclohexyl, -CH=C(C₂H₅)-CO-O-cycloheptyl, -CH=C(Cl)-COOH, -CH=C(Cl)-CO-OCH₃, -CH=C(Cl)-CO-OC₂H₅, -CH=C(Cl)-CO-O-n-C₃H₇, -CH=C(Cl)-CO-O-i-C₃H₇, -CH=C(Cl)-CO-O-n-C₄H₉, -CH=C(Cl)-CO-O-tert.-C₄H₉, -CH=C(Cl)-CO-O-cyclopropyl, -CH=C(Cl)-CO-O-cyclobutyl, -CH=C(Cl)-CO-O-cyclopentyl, -CH=C(Cl)-CO-O-cyclohexyl, -CH=C(Cl)-CO-O-cycloheptyl, -CH=C(Br)-COOH, -CH=C(Br)-CO-OCH₃, -CH=C(Br)-CO-OC₂H₅, -CH=C(Br)-CO-O-n-C₃H₇, -CH=C(Br)-CO-O-i-C₃H₇, -CH=C(Br)-CO-O-n-C₄H₉, -CH=C(Br)-CO-O-tert.-C₄H₉, -CH=C(Br)-CO-O-cyclopropyl, -CH=C(Br)-CO-O-cyclobutyl, -CH=C(Br)-CO-O-cyclopentyl, -CH=C(Br)-CO-O-cyclohexyl, -CH=C(Br)-CO-O-cycloheptyl, -CH=C(CN)-COOH, -CH=C(CN)-CO-OCH₃, -CH=C(CN)-CO-OC₂H₅, -CH=C(CN)-CO-O-n-C₃H₇, -CH=C(CN)-CO-O-i-C₃H₇, -CH=C(CN)-CO-O-n-C₄H₉, -CH=C(CN)-CO-O-tert.-C₄H₉, -CH=C(CN)-CO-O-cyclopropyl, -CH=C(CN)-CO-O-cyclobutyl, -CH=C(CN)-CO-O-cyclopentyl, -CH=C(CN)-CO-O-cyclohexyl, -CH=C(CN)-CO-O-cycloheptyl, -CH=CH-CO-OCH₂-OCH₃, -CH=CH-CO-OCH₂-OC₂H₅, -CH=CH-CO-OCH₂-O-n-C₃H₅, -CH=CH-CO-OCH₂-O-i-C₃H₅, -CH=CH-CO-OCH(CH₃)-OCH₃, -CH=CH-CO-OCH(CH₃)-OC₂H₅, -CH=CH-CO-O-CH₂CH₂-OCH₃, -CH=CH-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-OCH₃, -CH=C(CH₃)-CO-OCH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-O-n-C₃H₅, -CH=C(CH₃)-CO-OCH₂-O-i-C₃H₅, -CH=C(CH₃)-CO-OCH(CH₃)-OCH₃, -CH=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CH₃)-CO-O-CH₂CH₂-OCH₃, -CH=C(CH₃)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-OCH₃, -CH=C(C₂H₅)-CO-OCH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-O-n-C₃H₅, -CH=C(C₂H₅)-CO-OCH₂-O-i-C₃H₅, -CH=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -CH=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OCH₃, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-OCH₃, -CH=C(Cl)-CO-OCH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-O-n-C₃H₅, -CH=C(Cl)-CO-OCH₂-O-i-C₃H₅, -CH=C(Cl)-CO-OCH(CH₃)-OCH₃, -CH=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Cl)-CO-O-CH₂CH₂-OCH₃, -CH=C(Cl)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-OCH₃, -CH=C(Br)-CO-OCH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-O-n-C₃H₅, -CH=C(Br)-CO-OCH₂-O-i-C₃H₅, -CH=C(Br)-CO-OCH(CH₃)-OCH₃, -CH=C(Br)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Br)-CO-O-CH₂CH₂-OCH₃, -CH=C(Br)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-OCH₃, -CH=C(CN)-CO-OCH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-O-n-C₃H₅, -CH=C(CN)-CO-OCH₂-O-i-C₃H₅, -CH=C(CN)-CO-OCH(CH₃)-OCH₃, -CH=C(CN)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CN)-CO-O-CH₂CH₂-OCH₃, -CH=C(CN)-CO-O-CH₂CH₂-OC₂H₅, -CH=CH-CO-OCH₂-CF₃, -CH=CH-CO-OCH₂-CCl₃, -CH=CH-CO-OCH₂-oxiranyl, -CH=CH-CO-O(CH₂)₃-Br, -CH=CH-CO-OCH₂-CH=CH₂, -CH=CH-CO-OCH₂-C≡CH, -CH=CH-CO-OCH₂-CN, -CH=CH-CO-O(CH₂)₂-CN, -CH=C(CH₃)-CO-OCH₂-CF₃, -CH=C(CH₃)-CO-OCH₂-CCl₃, -CH=C(CH₃)-CO-OCH₂-oxiranyl, -CH=C(CH₃)-CO-O(CH₂)₃-Br, -CH=C(CH₃)-CO-OCH₂-CH=CH₂, -CH=C(CH₃)-CO-OCH₂-C≡CH, -CH=C(CH₃)-CO-OCH₂-CN, -CH=C(CH₃)-CO-O(CH₂)₂-CN, -CH=C(C₂H₅)-CO-OCH₂-CF₃, -CH=C(C₂H₅)-CO-OCH₂-CCl₃, -CH=C(C₂H₅)-CO-OCH₂-oxiranyl, -CH=C(C₂H₅)-CO-O(CH₂)₃-Br, -CH=C(C₂H₅)-CO-OCH₂-CH=CH₂, -CH=C(C₂H₅)-CO-OCH₂-C≡CH, -CH=C(C₂H₅)-CO-OCH₂-CN, -CH=C(C₂H₅)-CO-O(CH₂)₂-CN, -CH=C(Cl)-CO-OCH₂-CF₃, -CH=C(Cl)-CO-OCH₂-CCl₃, -CH=C(Cl)-CO-OCH₂-oxiranyl, -CH=C(Cl)-CO-O(CH₂)₃-Br, -CH=C(Cl)-CO-OCH₂-CH=CH₂, -CH=C(Cl)-CO-OCH₂-C≡CH, -CH=C(Cl)-CO-OCH₂-CN, -CH=C(Cl)-CO-O(CH₂)₂-CN, -CH=C(Br)-CO-OCH₂-CF₃, -CH=C(Br)-CO-OCH₂-CCl₃, -CH=C(Br)-CO-OCH₂-oxiranyl, -CH=C(Br)-CO-O(CH₂)₃-Br, -CH=C(Br)-CO-OCH₂-CH=CH₂, -CH=C(Br)-CO-OCH₂-C≡CH, -CH=C(Br)-CO-OCH₂-CN, -CH=C(Br)-CO-O(CH₂)₂-CN, -CH=C(CN)-CO-OCH₂-CF₃, -CH=C(CN)-CO-OCH₂-CCl₃, -CH=C(CN)-CO-OCH₂-oxiranyl, -CH=C(CN)-CO-O(CH₂)₃-Br, -CH=C(CN)-CO-OCH₂-CH=CH₂, -CH=C(CN)-CO-OCH₂-C≡CH, -CH=C(CN)-CO-OCH₂-CN, -CH=C(CN)-CO-O(CH₂)₂-CN, -CH=CH-CO-CH₃, -CH=CH-CO-C₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-i-C₃H₇, -CH=CH-CO-n-C₄H₉, -CH=CH-CO-tert.-C₄H₉, -CH=CH-CO-CH₂Cl, -CH=CH-CO-CH₂Br, -CH=CH-CO-CHCl₂, -CH=CH-CO-CH₂-OCH₃, -CH=CH-CO-CH(OCH₃)₂, -CH=CH-CO-CH₂-SCH₃, -CH=C(CH₃)-CO-CH₃, -CH=C(CH₃)-CO-C₂H₅, -CH=C(CH₃)-CO-n-C₃H₇, -CH=C(CH₃)-CO-i-C₃H₇, -CH=C(CH₃)-CO-n-C₄H₉, -CH=C(CH₃)-CO-tert.-C₄H₉, -CH=C(CH₃)-CO-CH₂Cl, -CH=C(CH₃)-CO-CH₂Br, -CH=C(CH₃)-CO-CHCl₂, -CH=C(CH₃)-CO-CH₂-OCH₃, -CH=C(CH₃)-CO-CH(OCH₃)₂, -CH=C(CH₃)-CO-CH₂-SCH₃, -CH=C(C₂H₅)-CO-CH₃, -CH=C(C₂H₅)-CO-C₂H₅, -CH=C(C₂H₅)-CO-n-C₃H₇, -CH=C(C₂H₅)-CO-i-C₃H₇, -CH=C(C₂H₅)-CO-n-C₄H₉, -CH=C(C₂H₅)-CO-tert.-C₄H₉, -CH=C(C₂H₅)-CO-CH₂Cl, -CH=C(C₂H₅)-CO-CH₂Br, -CH=C(C₂H₅)-CO-CHCl₂, -CH=C(C₂H₅)-CO-CH₂-OCH₃, -CH=C(C₂H₅)-CO-CH(OCH₃)₂, -CH=C(C₂H₅)-CO-CH₂-SCH₃, -CH=C(Cl)-CO-CH₃, -CH=C(Cl)-CO-C₂H₅, -CH=C(Cl)-CO-n-C₃H₇, -CH=C(Cl)-CO-i-C₃H₇, -CH=C(Cl)-CO-n-C₄H₉, -CH=C(Cl)-CO-tert.-C₄H₉, -CH=C(Cl)-CO-CH₂Cl, -CH=C(Cl)-CO-CH₂Br, -CH=C(Cl)-CO-CHCl₂, -CH=C(Cl)-CO-CH₂-OCH₃, -CH=C(Cl)-CO-CH(OCH₃)₂, -CH=C(Cl)-CO-CH₂-SCH₃, -CH=C(Br)-CO-CH₃, -CH=C(Br)-CO-C₂H₅, -CH=C(Br)-CO-n-C₃H₇, -CH=C(Br)-CO-i-C₃H₇, -CH=C(Br)-CO-n-C₄H₉, -CH=C(Br)-CO-tert.-C₄H₉, -CH=C(Br)-CO-CH₂Cl, -CH=C(Br)-CO-CH₂Br, -CH=C(Br)-CO-CHCl₂, -CH=C(Br)-CO-CH₂-OCH₃, -CH=C(Br)-CO-CH(OCH₃)₂, -CH=C(Br)-CO-CH₂-SCH₃, -CH=C(CN)-CO-CH₃, -CH=C(CN)-CO-C₂H₅, -CH=C(CN)-CO-n-C₃H₇, -CH=C(CN)-CO-i-C₃H₇, -CH=C(CN)-CO-n-C₄H₉, -CH=C(CN)-CO-tert.-C₄H₉, -CH=C(CN)-CO-CH₂Cl, -CH=C(CN)-CO-CH₂Br, -CH=C(CN)-CO-CHCl₂, -CH=C(CN)-CO-CH₂-OCH₃, -CH=C(CN)-CO-CH(OCH₃)₂, -CH=C(CN)-CO-CH₂-SCH₃, -CH=CH-CO-C₆H₅, -CH=CH-CO-(4-Cl-C₆H₄), -CH=C(CH₃)-CO-C₆H₅, -CH=C(CH₃)-CO-(4-Cl-C₆H₄), -CH=C(C₂H₅)-CO-C₆H₅, -CH=C(C₂H₅)-CO-(4-Cl-C₆H₄), -CH=C(Cl)-CO-C₆H₅, -CH=C(Br)-CO-C₆H₅, -CH=C(CN)-CO-C₆H₅, -CH=CH-CO-NH₂, -CH=CH-CO-NHCH₃, -CH=CH-CO-N(CH₃)₂, -CH=CH-CO-NH-C₂H₅, -CH=CH-CO-N(C₂H₅)₂, -CH=CH-CO-NH-n-C₃H₇, -CH=CH-CO-NH-i-C₃H₇, -CH=CH-CO-NH-tert.-C₄H₉, -CH=CH-CO-NH-cyclopropyl, -CH=CH-CO-NH-cyclobutyl, -CH=CH-CO-NH-cyclopentyl, -CH=CH-CO-NH-cyclohexyl, -CH=CH-CO-cycloheptyl, -CH=CH-CO-NH-cyclooctyl, -CH=CH-CO-pyrrolidin-1-yl, -CH=CH-CO-piperidin-1-yl, -CH=CH-CO-morpholin-4-yl, -CH=CH-CO-NH-CH₂CH=CH₂, -CH=CH-CO-NH-CH₂C≡CH, -CH=CH-CO-N(CH₃)-CH₂C≡CH, -CH=CH-CO-NH-(CH₂)₂Cl, -CH=CH-CO-NH-C₆H₅, -CH=C(CH₃)-CO-NH₂, -CH=C(CH₃)-CO-NHCH₃, -CH=C(CH₃)-CO-N(CH₃)₂, -CH=C(CH₃)-CO-NH-C₂H₅, -CH=C(CH₃)-CO-N(C₂H₅)₂, -CH=C(CH₃)-CO-NH-n-C₃H₇, -CH=C(CH₃)-CO-NH-i-C₃H₇, -CH=C(CH₃)-CO-NH-tert.-C₄H₉, -CH=C(CH₃)-CO-NH-cyclopropyl, -CH=C(CH₃)-CO-NH-cyclobutyl, -CH=C(CH₃)-CO-NH-cyclopentyl, -CH=C(CH₃)-CO-NH-cyclohexyl, -CH=C(CH₃)-CO-NH-cycloheptyl, -CH=C(CH₃)-CO-NH-cyclooctyl, -CH=C(CH₃)-CO-pyyrolidin-1-yl, -CH=C(CH₃)-CO-piperidin-1-yl, -CH=C(CH₃)-CO-morpholin-4-yl, -CH=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -CH=C(CH₃)-CO-NH-CH₂C≡CH, -CH=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CH₃)-CO-NH-(CH₂)₂Cl, -CH=C(CH₃)-CO-NH-C₆H₅, -CH=C(C₂H₅)-CO-NH₂, -CH=C(C₂H₅)-CO-NHCH₃, -CH=C(C₂H₅)-CO-N(CH₃)₂, -CH=C(C₂H₅)-CO-NH-C₂H₅, -CH=C(C₂H₅)-CO-N(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-n-C₃H₇, -CH=C(C₂H₅)-CO-NH-i-C₃H₇, -CH=C(C₂H₅)-CO-NH-tert.-C₄H₉, -CH=C(C₂H₅)-CO-NH-cyclopropyl, -CH=C(C₂H₅)-CO-NH-cyclobutyl, -CH=C(C₂H₅)-CO-NH-cyclopentyl, -CH=C(C₂H₅)-CO-NH-cyclohexyl, -CH=C(C₂H₅)-CO-NH-cycloheptyl, -CH=C(C₂H₅)-CO-NH-cyclooctyl, -CH=C(C₂H₅)-CO-pyrrolidin-1-yl, -CH=C(C₂H₅)-CO-piperidin-1-yl, -CH=C(C₂H₅)-CO-morpholin-4-yl, -CH=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-CH₂C≡CH, -CH=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -CH=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -CH=C(C₂H₅)-CO-NH-C₆H₅, -CH=C(Cl)-CO-NH₂, -CH=C(Cl)-CO-NHCH₃, -CH=C(Cl)-CO-N(CH₃)₂, -CH=C(Cl)-CO-NH-C₂H₅, -CH=C(Cl)-CO-N(C₂H₅)₂, -CH=C(Cl)-CO-NH-n-C₃H₇, -CH=C(Cl)-CO-NH-i-C₃H₇, -CH=C(Cl)-CO-NH-tert.-C₄H₉, -CH=C(Cl)-CO-NH-cyclopropyl, -CH=C(Cl)-CO-NH-cyclobutyl, -CH=C(Cl)-CO-NH-cyclopentyl, -CH=C(Cl)-CO-NH-cyclohexyl, -CH=C(Cl)-CO-NH-cycloheptyl, -CH=C(Cl)-CO-NH-cyclooctyl, -CH=C(Cl)-CO-pyrrolidin-1-yl, -CH=C(Cl)-CO-piperidin-1-yl, -CH=C(Cl)-CO-morpholin-4-yl, -CH=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -CH=C(Cl)-CO-NH-CH₂C≡CH, -CH=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Cl)-CO-NH-(CH₂)₂Cl, -CH=C(Cl)-CO-NH-C₆H₅, - CH=C(Br)-CO-NH₂, -CH=C(Br)-CO-NHCH₃, -CH=C(Br)-CO-N(CH₃)₂, -CH=C(Br)-CO-NH-C₂H₅, -CH=C(Br)-CO-N(C₂H₅)₂, -CH=C(Br)-CO-NH-n-C₃H₇, -CH=C(Br)-CO-NH-i-C₃H₇, -CH=C(Br)-CO-NH-tert.-C₄H₉, -CH=C(Br)-CO-NH-cyclopropyl, -CH=C(Br)-CO-NH-cyclobutyl, -CH=C(Br)-CO-NH-cyclopentyl, -CH=C(Br)-CO-NH-cyclohexyl, -CH=C(Br)-CO-NH-cycloheptyl, -CH=C(Br)-CO-NH-cyclooctyl, -CH=C(Br)-CO-pyrrolidin-1-yl, -CH=C(Br)-CO-piperidin-1-yl, -CH=C(Br)-CO-morpholin-4-yl, -CH=C(Br)-CO-NH-CH₂CH=C(Br)₂, -CH=C(Br)-CO-NH-CH₂C≡CH, -CH=C(Br)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Br)-CO-NH-(CH₂)₂Cl, -CH=C(Br)-CO-NH-C₆H₅, -CH=C(CN)-CO-NH₂, -CH=C(CN)-CO-NHCH₃, -CH=C(CN)-CO-N(CH₃)₂, -CH=C(CN)-CO-NH-C₂H₅, -CH=C(CN)-CO-N(C₂H₅)₂, -CH=C(CN)-CO-NH-n-C₃H₇, -CH=C(CN)-CO-NH-i-C₃H₇, -CH=C(CN)-CO-NH-tert.-C₄H₉, -CH=C(CN)-CO-NH-cyclopropyl, -CH=C(CN)-CO-NH-cyclobutyl, -CH=C(CN)-CO-NH-cyclopentyl, -CH=C(CN)-CO-NH-cyclohexyl, -CH=C(CN)-CO-NH-cycloheptyl, -CH=C(CN)-CO-NH-cyclooctyl, -CH=C(CN)-CO-pyrrolidin-1-yl, -CH=C(CN)-CO-piperidin-1-yl, -CH=C(CN)-CO-morpholin-4-yl, -CH=C(CN)-CO-NH-CH₂CH=C(CN)₂, -CH=C(CN)-CO-NH-CH₂C≡CH, -CH=C(CN)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CN)-CO-NH-(CH₂)₂Cl, -CH=C(CN)-CO-NH-C₆H₅, -CH=CH-CO-SCH₃, -CH=CH-CO-SC₂H₅, -CH=CH-CO-S-n-C₃H₇, -CH=CH-CO-S-i-C₃H₇, -CH=CH-CO-S-n-C₄H₉, -CH=CH-CO-S-tert.-C₄H₉, -CH=C(CH₃)-CO-SCH₃, -CH=C(CH₃)-CO-SC₂H₅, -CH=C(CH₃)-CO-S-n-C₃H₇, -CH=C(CH₃)-CO-S-i-C₃H₇, -CH=C(CH₃)-CO-S-n-C₄H₉, -CH=C(CH₃)-CO-S-tert.-C₄H₉, -CH=C(C₂H₅)-CO-SCH₃, -CH=C(C₂H₅)-CO-SC₂H₅, -CH=C(C₂H₅)-CO-S-n-C₃H₇, -CH=C(C₂H₅)-CO-S-i-C₃H₇, -CH=C(C₂H₅)-CO-S-n-C₄H₉, -CH=C(C₂H₅)-CO-S-tert.-C₄H₉, -CH=C(Cl)-CO-SCH₃, -CH=C(Cl)-CO-SC₂H₅, -CH=C(Cl)-CO-S-n-C₃H₇, -CH=C(Cl)-CO-S-i-C₃H₇, -CH=C(Cl)-CO-S-n-C₄H₉, -CH=C(Cl)-CO-S-tert.-C₄H₉, -CH=C(Br)-CO-SCH₃, -CH=C(Br)-CO-SC₂H₅, -CH=C(Br)-CO-S-n-C₃H₇, -CH=C(Br)-CO-S-i-C₃H₇, -CH=C(Br)-CO-S-n-C₄H₉, -CH=C(Br)-CO-S-tert.-C₄H₉, -CH=C(CN)-CO-SCH₃, -CH=C(CN)-CO-SC₂H₅, -CH=C(CN)-CO-S-n-C₃H₇, -CH=C(CN)-CO-S-i-C₃H₇, -CH=C(CN)-CO-S-n-C₄H₉, -CH=C(CN)-CO-S-tert.-C₄H₉, -CH=C(COCH₃)-CO-OCH₃, -CH=C(COC₂H₅)-CO-OCH₃, -CH=C(CO-n-C₃H₇)-CO-OCH₃, -CH=C(COCH₃)-CO-OC₂H₅, -CH=C(COC₂H₅)-CO-OC₂H₅, -CH=C(CO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COCH₃)-CO-O-n-C₃H₇, -CH=C(COC₂H₅)-CO-O-n-C₃H₇, -CH=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-OCH₃, -CH=C(CF₃)-CO-OC₂H₅, -CH=C(CF₃)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-O-i-C₃H₇, -CH=C(CF₃)-CO-O-n-C₄H₉, -CH=C(CF₃)-CO-O-tert.-C₄H₉, -CH=C(COOCH₃)₂, -CH=C(COOC₂H₅)₂, -CH=C(COOCH₃)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)-CO-OCH₃, -CH=C(COO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)₂, -CH=CH-CH=CH-COOH, -CH=CH-CH=CH-CO-OCH₃, -CH=CH-CH=CH-CO-OC₂H₅, -CH=CH-CH=C(COOCH₃)₂, -CH=CH-CH=C(CN)-CO-OCH₃, -CH=CH-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-OCH₃, -CH=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CH=C(Cl)-CO-OCH₃, -CH=C(CH₃)-CH=C(Br)-CO-OCH₃, -CH=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-NH₂, -CH=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -CH=CH-(CH₂)₂-COOH, -CH=CH-(CH₂)₂-CO-OCH₃, -CH=CH-(CH₂)₂-CO-OC₂H₅, -CH=CH-CH₂-CH(COOCH₃)₂, -CH=CH-CH₂-CH(COOC₂H₅)₂, -CH=CH-CH₂-CH(CN)-CO-OCH₃, -CH=CH-CH₂-CH(CN)-CO-OC₂H₅, -CH=CH-CH₂-CH(CH₃)-CO-OCH₃, -CH=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -CH=CH-(CH₂)₂-CO-NH₂, -CH=CH-(CH₂)₂-CO-NH-CH₃, -CH=CH-CH₂-COOH, -CH=CH-CH₂-CO-OCH₃, -CH=CH-CH₂-CO-OC₂H₅, -CH=C(COOCH₃)-CH₂-CO-OCH₃, -CH=C(COOCH₃)-CH₂-CO-OC₂H₅, -CH=CH-CH₂-CO-NH₂, -CH=CH-CH₂-CO-NH-CH₃, -CH=CH-CH₂-CO-N(CH₃)₂, -CH(OCH₃)₂, -CH(SCH₃)₂, -CH(OC₂H₅)₂, -CH(SC₂H₅)₂, -CH(O-n-C₃H₇)₂, -CH(O-i-C₃H₇)₂, -CH(S-n-C₃H₇)₂, -CH(S-i-C₃H₇)₂, -CH(O-n-C₄H₉)₂, -CH(O-i-C₄H₉)₂, -CH(O-s-C₄H₉)₂, -CH(O-tert.-C₄H₉)₂, -CH(S-n-C₄H₉)₂, -CH(S-i-C₄H₉)₂, -CH(S-s-C₄H₉)₂, -CH(S-tert.-C₄H₉)₂, -CH(OC₅H₁₁)₂, 1,3-Dioxolan-2-yl, 1,3-Dithio­ lan-2-yl, 1,3-Oxathiolan-2-yl, 4-Methyl-1,3-dioxolan-2-yl, 4-Methyl-1,3-dithiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 5-Methyl-1,3-oxathiolan-2-yl, 4-Ethyl-1,3-dioxolan-2-yl, 4-Ethyl- 1,4-dithiolan-2-yl, 4-Ethyl-1,3-oxathiolan-2-yl, 5-Ethyl-1,3-oxa­ thiolan-2-yl, 4,5-Dimethyl-1,3-dioxolan-2-yl, 4,4-Dimethyl-1,3- dioxolan-2-yl, 4,5-Dimethyl-1,3-dithiolan-2-yl, 5,5-Dimethyl-1,3- dithiolan-2-yl, 4,5-Dimethyl-1,3-oxathiolan-2-yl, 5,5-Dimethyl- 1,3-oxathiolan-2-yl, 4,4-Dimethyl-1,3-oxathiolan-2-yl, 4-Vinyl- 1,3-dioxolan-2-yl, 4-Vinyl-1,3-dithiolan-2-yl, 4-Vinyl-1,3-oxa­ thiolan-2-yl, 5-Vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3- dioxolan-2-yl, 4-Chlormethyl-1,3-dithiolan-2-yl, 4-Chlormethyl- 1,3-oxathiolan-2-yl, 5-Chlormethyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-1,3-dithio­ lan-2-yl, 4-Hydroxymethyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl- 1,3-oxathiolan-2-yl, 4-Methoxymethyl-1,3-dioxolan-2-yl, 4-Allyl­ oxymethyl-1,3-dioxolan-2-yl, 4-Propargyloxymethyl-1,3-dioxolan- 2-yl, 4-Acetoxymethyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-1,3-dithiolan-2-yl, 4-Propargyl­ oxymethyl-1,3-dithiolan-2-yl, 4-Acetoxymethyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-1,3-oxa­ thiolan-2-yl, 4-Allyloxymethyl-1,3-oxathiolan-2-yl, 5-Allyloxy­ methyl-1,3-oxathiolan-2-yl, 4-Propargyloxymethyl-1,3-oxathiolan- 2-yl, 5-Propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxymethyl- 1,3-oxathiolan-2-yl, 5-Acetoxymethyl-1,3-oxathiolan-2-yl, 4-Methylthiomethyl-1,3-dioxolan-2-yl, 4-Methylthiomethyl-1,3- dithiolan-2-yl, 4-Carboxy-1,3-dioxolan-2-yl, 4-Carboxy-1,3- dithiolan-2-yl, 4-Methoxycarbonyl-1,3-dioxolan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-1,3-di­ thiolan-2-yl, 4-n-Butoxycarbonyl-1,3-dithiolan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-4-methyl- 1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-di­ thiolan-2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-1,3- dithiolan-2-yl, 1,3-Dioxan-2-yl, 1,3-Dithian-2-yl, 1,3-Oxathian- 2-yl, 5-Methyl-1,3-dioxan-2-yl, 5-Methyl-1,3-dithian-2-yl, 5-Methyl-1,3-oxathian-2-yl, 5,5-Dimethyl-1,3-dioxan-2-yl, 4,6-Di­ methyl-1,3-dioxan-2-yl, 4,4-Dimethyl-1,3-dioxan-2-yl, 5,5-Di­ methyl-1,3-dithian-2-yl, 4,6-Dimethyl-1,3-dithian-2-yl, 4,4-Di­ methyl-1,3-dithian-2-yl, 5,5-Dimethyl-1,3-oxathian-2-yl, 4,4-Di­ methyl-1,3-oxathian-2-yl, 6,6-Dimethyl-1,3-oxathian-2-yl, 4-Hydroxymethyl-1,3-dioxan-2-yl, 4-Methoxymethyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-1,3-dioxan-2- yl, 4-Hydroxymethyl-1,3-dithian-2-yl, 4-Methoxymethyl-1,3-di­ thian-2-yl, 4-Allyloxymethyl-1,3-dithian-2-yl, 4-Acetoxymethyl- 1,3-dithian-2-yl, 4-Chlormethyl-1,3-dioxan-2-yl, 4-Chlormethyl- 1,3-dithian-2-yl, 1,3-Dioxepan-2-yl, 1,3-Dithiepan-2-yl, 1,3-Di­ oxep-5-en-2-yl, 4-Methoxycarbonyl-1,3-dioxan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-1,3-dithian- 4-yl, 4-n-Butoxycarbonyl-1,3-dithian-2-yl, 4-Methoxycarbonyl-4- methyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxan-2- yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-4-methyl- 1,3-dithian-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithian-2-yl, -C(CH₃)(OCH₃)₂, -C(CH₃)(SCH₃)₂, -C(CH₃)(OC₂H₅)₂, -C(CH₃)(SC₂H₅)₂, -C(CH₃)(O-n-C₃H₇)₂, -C(CH₃)(O-i-C₃H₇)₂, -C(CH₃)(S-n-C₃H₇)₂, -C(CH₃)(S-i-C₃H₇)₂, -C(CH₃)(O-n-C₄H₉)₂, -C(CH₃)(O-i-C₄H₉)₂, -C(CH₃)(O-s-C₄H₉)₂, -C(CH₃)(O-tert.-C₄H₉)₂, -C(CH₃)(S-n-C₄H₉)₂, -C(CH₃)(S-i-C₄H₉)₂, -C(CH₃)(S-s-C₄H₉)₂, -C(CH₃)(S-tert.-C₄H₉)₂, -C(CH₃)(O-n-C₅H₁₁)′′, 2-Methyl-1,3-dioxolan-2-yl, 2-Methyl-1,3-di­ thiolan-2-yl, 2-Methyl-1,3-oxathiolan-2-yl, 2,4-Dimethyl-1,3- dioxolan-2-yl, 2,4-Dimethyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-1,3- oxathiolan-2-yl, 2,5-Dimethyl-1,3-oxathiolan-2-yl, 4-Ethyl-2- methyl-1,3-dioxolan-2-yl, 4-Ethyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Ethyl-2-methyl-1,3- oxathiolan-2-yl, 2,4,5-Trimethyl-1,3-dioxolan-2-yl, 2,4,4-Tri­ methyl-1,3-dioxolan-2-yl, 2,4,5-Trimethyl-1,3-dithiolan-2-yl, 2,4,4-Trimethyl-1,3-dithiolan-2-yl, 2,4,5-Trimethyl-1,3-oxathio­ lan-2-yl, 2,4,4-Trimethyl-1,3-oxathiolan-2-yl, 2-Methyl-4-vinyl- 1,3-dioxolan-2-yl, 2-Methyl-4-vinyl-1,3-dithiolan-2-yl, 2-Methyl- 4-vinyl-1,3-oxathiolan-2-yl, 2-Methyl-5-vinyl-1,3-oxathiolan-2- yl, 4-Chlormethyl-2-methyl-1,3-dioxolan-2-yl, 4-Chlormethyl-2- methyl-1,3-dithiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-oxathio­ lan-2-yl, 5-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Hydroxy­ methyl-2-methyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-2- methyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dioxolan- 2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxy- 2-methyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dithiolan-2-yl, 4-Acetoxy-2- methyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-oxathio­ lan-2-yl, 5-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Allyl­ oxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Allyloxymethyl-2- methyl-1,3-oxathiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3- oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3-oxathiolan-2- yl, 4-Acetoxy-2-methyl-1,3-oxathiolan-2-yl, 5-Acetoxy-2-methyl- 1,3-oxathiolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dioxolan-2- yl, 2-Methyl-4-methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-2- methyl-1,3-dioxolan-2-yl, 4-Carboxy-2-methyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-2- methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-2-methyl-1,3-dioxo­ lan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-Eth­ oxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-2- methyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-di­ oxolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-ethoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4- ethoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-n-butoxy­ carbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl-1,3- dithiolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-dioxan-2- yl, 2-Methyl-1,3-dithian-2-yl, 2-Methyl-1,3-oxathian-2-yl, 2,5- Dimethyl-1,3-dioxan-2-yl, 2,5-Dimethyl-1,3-dithian-2-yl, 2,5-Di­ methyl-1,3-oxathian-2-yl, 2,5,5-Trimethyl-1,3-dioxan-2-yl, 2,4,6- Trimethyl-1,3-dioxan-2-yl, 2,2,4-Trimethyl-1,3-dioxan-2-yl, 2,5,5-Trimethyl-1,3-dithian-2-yl, 2,4,6-Trimethyl-1,3-dithian-2- yl, 2,4,4-Trimethyl-1,3-dithian-2-yl, 2,5,5-Trimethyl-1,3-oxa­ thian-2-yl, 2,4,4-Trimethyl-1,3-oxathian-2-yl, 2,6,6-Trimethyl- 1,3-oxathian-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-2- methyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dithian-2-yl, 4-Methoxymethyl-2- methyl-1,3-dithian-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithian-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dithian-2-yl, 4-Chlormethyl-2- methyl-1,3-dioxan-2-yl, 4-Chlormethyl-2-methyl-1,3-dithian-2-yl, -C(CH₃)=NH, -C(CH₃)=N-CH₃, -C(CH₃)=N-C₂H₅, -C(CH₃)=N-n-C₃H₇, -(CH₃)=N-i-C₃H₇, -C(CH₃)=N-n-C₄H₉, -C(CH₃)=N-CH₂CH=CH₂, -C(CH₃)=N-CH₂CH=CH₂-CH₃, -C(CH₃)=N-CH₂C≡CH, -C(CH₃)=N-CH₂C≡C-CH₃, -C(CH₃)=N-cyclopropyl, -C(CH₃)=N-cyclobutyl, -C(CH₃)=N-cyclo­ pentyl, -C(CH₃)=N-cyclohexyl, -C(CH₃)=N-cycloheptyl, -C(CH₃)=N-CH₂-CH₂Cl, -C(CH₃)=N-CH₂Cl, -C(CH₃)=N-C₆H₅, -C(CH₃)=N-(2-F-C₆H₄), -C(CH₃)=N-(3-F-C₆H₄), -C(CH₃)=N-(4-F-C₆H₄), -C(CH₃)=N-(2-Cl-C₆H₄), -C(CH₃)=N-(3-Cl-C₆H₄), -C(CH₃)=N-(4-Cl-C₆H₄), -C(CH₃)=N-(2-CH₃-C₆H₄), -C(CH₃)=N-(3-CH₃-C₆H₄), -C(CH₃)=N-(4-CH₃-C₆H₄), -C(CH₃)=N-(2-CF₃-C₆H₄), -C(CH₃)=N-(3-CF₃-C₆H₄), -C(CH₃)=N-(4-CF₃-C₆H₄), -C(CH₃)=N-(2-OCH₃-C₆H₄), -C(CH₃)=N-(3-OCH₃-C₆H₄), -C(CH₃)=N-(4-OCH₃-C₆H₄), -C(CH₃)=N-(4-NO₂-C₆H₄), -C(CH₃)=N-(4-CN-C₆H₄), -C(CH₃)=N-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-(2,4-(CH₃)₂-C₆H₃), -C(CH₃)=N-CH₂-OCH₃, -C(CH₃)=N-CH₂-OC₂H₅, -C(CH₃)=N-CH₂CH₂-OCH₃, -C(CH₃)=N-CH₂CH-OC₂H₅, -C(CH₃)=N-OH, -C(CH₃)=N-OCH₃, -C(CH₃)=N-OC₂H₅, -C(CH₃)=N-O-n-C₃H₇, -C(CH₃)=N-O-i-C₃H₇, -C(CH₃)=N-O-n-C₄H₉, -C(CH₃)=N-O-i-C₄H₉, -C(CH₃)=N-O-s-C₄H₉, -C(CH₃)=N-O-tert.-C₄H₉, -C(CH₃)=N-OCH₂-CH=CH₂, -C(CH₃)=N-OCH(CH₃)-CH=CH₂, -C(CH₃)=N-OCH₂-C≡CH, -C(CH₃)=N-CH(CH₃)-C≡CH, -C(CH₃)=N-OCH₂-CH=C-CH₃, -C(CH₃)=N-OCH₂CH₂-Cl, -C(CH₃)=N-OCH₂CH₂-F, -C(CH₃)=N-OCH₂-CF₃, -C(CH₃)=N-OCH₂-CH=CHCl, -C(CH₃)=N-OCH₂-C(Cl)=CH₂, -C(CH₃)=N-OCH₂-C(Br)=CH₂, -C(CH₃)=N-OCH₂-CH=C(Cl)-CH₃, -C(CH₃)=N-O-CO-CH₃, -C(CH₃)=N-O-CO-C₂H₅, -C(CH₃)=N-OCH₂-CN, -C(CH₃)=N-OCH₂-CH=CH-CH₂-OCH₃, -C(CH₃)=N-OCH₂-CH=CH-CH₂-O-tert.-C₄H₉, -C(CH₃)=N-O-(CH₂)₃-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-(4-Cl-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-C₆H₅, -C(CH₃)=N-OCH₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(3-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-CH₂-(4-CH₃O-C₆H₄), -C(CH₃)=N-OCH₂-CH=C(CH₃)-C₆H₅, -C(CH₃)=N-O-(CH₂)₂-CH=CH-(3,4-Cl₂-C₆H₃), -C(CH₃)=N-O-(CH₂)₃-C≡-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-OCH₃, -C(CH₃)=N-OCH₂CH₂-OCH₃, -C(CH₃)=N-OCH₂-OC₂H₅, -C(CH₃)=N-OCH(CH₃)-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=N-NH₂, -C(CH₃)=N-NH-CH₃, -C(CH₃)=N-NH-C₂H₅, -C(CH₃)=N-NH-n-C₃H₇, -C(CH₃)=N-NH-i-C₃H₇, -C(CH₃)=N-NH-n-C₄H₉, -C(CH₃)=N-NH-i-C₄H₉, -C(CH₃)=N-NH-s-C₄H₉, -C(CH₃)=N-NH- tert.-C₄H₉, -C(CH₃)=N-NH-cyclopropyl, -C(CH₃)=N-NH- cyclobutyl, -C(CH₃)=N-NH-cyclopentyl, -C(CH₃)=N-NH-cyclohexyl, -C(CH₃)=N-NH-cycloheptyl, -C(CH₃)=N-N(CH₃)₂, -C(CH₃)=N-N(C₂H₅)₂, -C(CH₃)=N-N(n-C₃H₇)₂, -C(CH₃)=N-N(i-C₃H₇)₂, -C(CH₃)=N-NH-CH₂-C=CH, -C(CH₃)=N-NH-CH₂-C≡CH, -C(CH₃)=N-N(CH₃)-CH₂-C≡CH, -C(CH₃)=N-NH-CH₂CF₃, -C(CH₃)=N-NH-CO-CH₃, -C(CH₃)=N-NH-CO-C₂H₅, -C(CH₃)=N-NH-CO-OCH₃, -C(CH₃)=N-NH-CO-OC₂H₅, -C(CH₃)=N-NH-CO-O-tert.-C₄H₉, -C(CH₃)=N- pyrrolidin-1-yl, -C(CH₃)=N-piperidin-1-yl, -C(CH₃)=N-morpholin- 4-yl, -C(CH₃)=N-NH-C₆H₅, -C(CH₃)=N-NH-(4-Cl-C₆H₄), -C(CH₃)=N-NH-(4-NO₂-C₆H₄), -C(CH₃)=N-NH-(4-F-C₆H₄), -C(CH₃)=N-NH-(4-CH₃O-C₆H₄), -C(CH₃)=N-NH-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-NH-(2,4-(NO₂)₂-C₆H₃), -C(CH₃)=N-NH-CO-NH₂, -C(CH₃)=N-NH-CO-NHCH₃, -C(CH₃)=N-NH-CO-NHC₂H₅, -C(CH₃)=N-NH-CO-N(CH₃)₂, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=CH-CO-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-O-n-C₄H₉, -C(CH₃)=CH-CO-O-tert.-C₄H₉, -C(CH₃)=CH-CO-O-cyclopropyl, -C(CH₃)=CH-CO-O-cyclobutyl, -C(CH₃)=CH-CO-O-cyclopentyl, -C(CH₃)=CH-CO-O-cyclohexyl, -C(CH₃)=CH-CO-O-cycloheptyl, -C(CH₃)=C(CH₃)-COOH, -C(CH₃)=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-cyclopropyl, -C(CH₃)=C(CH₃)-CO-O-cyclobutyl, -C(CH₃)=C(CH₃)-CO-O-cyclopentyl, -C(CH₃)=C(CH₃)-CO-O-cyclohexyl, -C(CH₃)=C(CH₃)-CO-O-cycloheptyl, -C(CH₃)=C(C₂H₅)-COOH, -C(CH₃)=C(C₂H₅)-CO-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-cyclo­ propyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-O- cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-O-cycloheptyl, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-O-n-C₄H₉, -C(CH₃)=C(Cl)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-O-cyclopropyl, -C(CH₃)=C(Cl)-CO-O-cyclobutyl, -C(CH₃)=C(Cl)-CO-O-cyclopentyl, -C(CH₃)=C(Cl)-CO-O-cyclohexyl, -C(CH₃)=C(Cl)-CO-O-cycloheptyl, -C(CH₃)=C(Br)-COOH, -C(CH₃)=C(Br)-CO-OCH₃, -C(CH₃)=C(Br)-CO-OC₂H₅, -C(CH₃)=C(Br)-CO-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-O-n-C₄H₉, -C(CH₃)=C(Br)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-O-cyclopropyl, -C(CH₃)=C(Br)-CO-O-cyclobutyl, -C(CH₃)=C(Br)-CO-O-cyclopentyl, -C(CH₃)=C(Br)-CO-O-cyclohexyl, -C(CH₃)=C(Br)-CO-O-cycloheptyl, -C(CH₃)=C(CN)-COOH, -C(CH₃)=C(CN)-CO-OCH₃, -C(CH₃)=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CN)-CO-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-O-n-C₄H₉, -C(CH₃)=C(CN)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-O-cyclopropyl, -C(CH₃)=C(CN)-CO-O-cyclobutyl, -C(CH₃)=C(CN)-CO-O-cyclopentyl, -C(CH₃)=C(CN)-CO-O-cyclohexyl, -C(CH₃)=C(CN)-CO-O-cycloheptyl, -C(CH₃)=CH-CO-OCH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-OCH(CH₃)-OCH₃, -C(CH₃)=CH-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=CH-CO-OCH₂CH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=(C₂H₅)-CO-OCH₂CH₂-OCH₃, -(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-O-i-C₃H₇, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -(CH₃)=C(Cl)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-O-i-C₃H₇, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-O-i-C₃H₇, -C(CH₃)=C(CN)-CO-OCH(CH₃)OCH₃, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-CF₃, -C(CH₃)=CH-CO-OCH₂-CCl₃, -C(CH₃)=CH-CO-OCH₂-oxiranyl, -C(CH₃)=CH-CO-(CH₂)₃-Br, -C(CH₃)=CH-CO-OCH₂-CH=CH₂, -C(CH₃)=CH-CO-OCH₂-C≡CH, -C(CH₃)=CH-CO-OCH₂-CN, -C(CH₃)=CH-CO-OCH₂CH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CF₃, -C(CH₃)=C(CH₃)-CO-OCH₂-CCl₃, -C(CH₃)=C(CH₃)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CH₃)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CH₃)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CH₃)-CO-OCH₂-C≡CH, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CF₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CCl₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-oxiranyl, -C(CH₃)=C(C₂H₅)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(C₂H₅)CO-OCH₂-C≡CH, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-C₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂-CF₃, -C(CH₃)=C(Cl)-CO-OCH₂-CCl₃, -C(CH₃)=C(Cl)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Cl)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Cl)-CO-OCH₂-CH≡CH₂, -C(CH₃)=C(Cl)-CO-OCH₂-C≡CH, -C(CH₃)=C(Cl)-CO-OCH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂-CF₃, -C(CH₃)=C(Br)-CO-OCH₂-CCl₃, -C(CH₃)=C(Br)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Br)-CO-O(CH₂)₃-Br, -C(CH₃)=C(Br)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Br)-CO-OCH₂-C≡CH, -C(CH₃)=C(Br)-CO-OCH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂CH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂-CF₃, -C(CH₃)=C(CN)-CO-OCH₂-CCl₃, -C(CH₃)=C(CN)-O-OCH₂-oxiranyl, -C(CH₃)=C(CN)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CN)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CN)-CO-OCH₂-C≡CH, -C(CH₃)=C(CN)-CO-OCH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂CH₂-CN, -C(CH₃)=CH-CO-CH₃, -C(CH₃)=CH-CO-C₂H₅, -C(CH₃)=CH-CO-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-n-C₄H₉, -C(CH₃)=CH-CO-tert.-C₄H₉, -C(CH₃)=CH-CO-CH₂Cl, -C(CH₃)=CH-CO-CH₂Br, -C(CH₃)=CH-CO-CHCl₂, -C(CH₃)=CH-CO-CH₂-OCH₃, -C(CH₃)=CH-CO-CH(OCH₃)₂, -C(CH₃)=CH-CO-CH₂-SCH₃, -C(CH₃)=C(CH₃)-CO-CH₃, -C(CH₃)=C(CH₃)-CO-C₂H₅, -C(CH₃)=C(CH₃)-CO-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-CH₂Cl, -C(CH₃)=C(CH₃)-CO-CH₂Br, -C(CH₃)=C(CH₃)-CO-CHCl₂, -C(CH₃)=C(CH₃)-CO-CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-CH(OCH₃)₂, -C(CH₃)=C(CH₃)-CO-CH₂-SCH₃, -C(CH₃)=C(C₂H₅)-CO-CH₃, -C(CH₃)=C(C₂H₅)-CO-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-CH₂Cl, -C(CH₃)=C(C₂H₅)-CO-CH₂Br, -C(CH₃)=C(C₂H₅)-CO-CHCl₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-CH(OCH₃)₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-SCH₃, -C(CH₃)=C(Cl)-CO-CH₃, -C(CH₃)=C(Cl)-CO-C₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-n-C₄H₉, -C(CH₃)=C(Cl)-CO-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-CH₂Cl, -C(CH₃)=C(Cl)-CO-CHCl₂, -C(CH₃)=C(Cl)-CO-CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-CH(OCH₃)₂, -C(CH₃)=C(Cl)-CO-CH₂-SCH₃, -C(CH₃)=C(Br)-CO-CH₃, -C(CH₃)=C(Br)-CO-C₂H₅, -C(CH₃)=C(Br)-CO-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-n-C₄H₉, -C(CH₃)=C(Br)-CO-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-CH₂Cl, -C(CH₃)=C(Br)-CO-CH₂Br, -C(CH₃)=C(Br)-CO-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-CH(OCH₃)₂, -C(CH₃)=C(Br)-CO-CH₂-SCH₃, -C(CH₃)=C(CN)-CO-CH₃, -C(CH₃)=C(CN)-CO-C₂H₅, -C(CH₃)=C(CN)-CO-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-n-C₄H₉, -C(CH₃)=C(CN)-CO-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-CH₂Cl, -C(CH₃)=C(CN)-CO-CH₂Br, -C(CH₃)=C(CN)-CO-CHCl₂, -C(CH₃)=C(CN)-CO-CH₂-OCH₃, -C(CH₃)=C(CN)-CO-CH(OCH₃)₂, -C(CH₃)=C(CN)-CO-CH₂-SCH₃, -C(CH₃)=CH-CO-C₆H₅, -C(CH₃)=CH-CO-(4-Cl-C₆H₄), -C(CH₃)=C(CH₃)-CO-C₆H₅, -C(CH₃)=C(CH₃)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(C₂H₅)-CO-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(Cl)-CO-C₆H₅, -C(CH₃)=C(Br)-CO-C₆H₅, -C(CH₃)=C(CN)-CO-C₆H₅, -C(CH₃)=CH-CO-NH₂, -C(CH₃)=CH-CO-NHCH₃, -C(CH₃)=CH-CO-N(CH₃)₂, -C(CH₃)=CH-CO-NH-C₂H₅, -C(CH₃)=CH-CO-N(C₂H₅)₂, -C(CH₃)=CH-CO-NH-n-C₃H₇, -C(CH₃)=CH-CO-NH-i-C₃H₇, -C(CH₃)=CH-CO-NH-tert.-C₄H₉, -C(CH₃)=CH-CO-NH-cyclopropyl, -C(CH₃)=CH-CO-NH-cyclobutyl, -C(CH₃)=CH-CO-NH-cyclopentyl, -C(CH₃)=CH-CO-NH-cyclohexyl, -C(CH₃)=CH-CO-NH-cycloheptyl, -C(CH₃)=CH-CO-NH-cyclooctyl, -C(CH₃)=CH-CO-pyrrolidin-1-yl, -C(CH₃)=CH-CO-piperidin-1-yl, -C(CH₃)=CH-CO-morpholin-4-yl, -C(CH₃)=CH-CO-NH-CH₂CH=CH₂, -C(CH₃)=CH-CO-NH-CH₂C≡CH, -C(CH₃)=CH-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=CCH-CO-NH-(CH₂)₂Cl, -C(CH₃)=CH-CO-NH-C₆H₅, -C(CH₃)=C(CH₃)-CO-NH₂, -C(CH₃)=C(CH₃)-CO-NHCH₃, -C(CH₃)=C(CH₃)-CO-N(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-C₂H₅, -C(CH₃)=C(CH₃)-CO-N(C₂H₅)₂, -C(CH₃)=C(CH₃)-CO-NH-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-NH- cyclopropyl, -C(CH₃)=C(CH₃)-CO-NH-cyclobutyl, -C(CH₃)=C(CH₃)-CO-NH-cyclopentyl, -C(CH₃)=C(CH₃)-CO-NH- cyclohexyl, -C(CH₃)=C(CH₃)-CO-NH-cycloheptyl, -C(CH₃)=C(CH₃)-CO-NH-cyclooctyl, -C(CH₃)=C(CH₃)-CO- pyrrolidin-1-yl, -C(CH₃)=C(CH₃)-CO-piperidin-1-yl, -C(CH₃)=C(CH₃)-CO-morpholin-4-yl, -C(CH₃)=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-NH(CH₂)₂Cl, -C(CH₃)=C(CH₃)-CO-NH-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-NH₂, -C(CH₃)=C(C₂H₅)-CO-NHCH₃, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)₂, -C(CH₃)=C(C₂H₅)-CO-NH-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-N(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-NH- cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclo­ hexyl, -C(CH₃)=C(C₂H₅)-CO-NH-cycloheptyl, -C(CH₃)=C(C₂H₅)-CO-NH- cyclooctyl, -C(CH₃)=C(C₂H₅)-CO-pyrrolidin-1-yl, -C(CH₃)=C(C₂H₅)-CO-piperidin-1-yl, -C(CH₃)=C(C₂H₅)-CO- morpholin-4-yl, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(C₂H₅)-CO-NH-C₆H₅, -C(CH₃)=C(Cl)-CO-NH₂, -C(CH₃)=C(CH₃)=C(Cl)-CO-NHCH₃, -C(CH₃)=C(Cl)-CO-N(CH₃)₂, -C(CH₃)=C(Cl)-CO-NH-C₂H₅, -C(CH₃)=C(Cl)-CO-N(C₂H₅)₂, -C(CH₃)=C(Cl)-CO-NH-n-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-i-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-NH-cyclopropyl, -C(CH₃)=C(Cl)-CO-NH-cyclobutyl, -C(CH₃)=C(Cl)-CO-NH-cyclopentyl, -C(CH₃)=C(Cl)-CO-NH-cyclohexyl, -C(CH₃)=C(Cl)-CO-NH-cycloheptyl, -C(CH₃)=C(Cl)-CO-NH-cyclooctyl, -C(CH₃)=C(Cl)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Cl)-CO-piperidin-1- yl, -C(CH₃)=C(Cl)-CO-morpholin-4-yl, -C(CH₃)=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -C(CH₃)=C(Cl)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-N(CH₃)-CH₂≡CH, -C(CH₃)=C(Cl)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Cl)-NO-NH-C₆H₅, -C(CH₃)=C(Br)-CO-NH₂, -C(CH₃)=C(Br)-CO-NHCH₃, -C(CH₃)=C(Br)-CO-N(CH₃)₂, -C(CH₃)=C(Br)-CO-NH-C₂H₅, -C(CH₃)=C(Br)-CO-N(C₂H₅)₂, -C(CH₃)=C(Br)-CO-NH-n-C₃H₇, -C(CH₃)=C(Br)-CO-NH-i-C₃H₇, -C(CH₃)=C(Br)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-NH-cyclopropyl, -C(CH₃)=C(Br)-CO-NH-cyclobutyl, -C(CH₃)=C(Br)-CO-NH-cyclopentyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cycloheptyl, -C(CH₃)=C(Br)-CO-NH-cyclooctyl, -C(CH₃)=C(Br)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Br)-CO-piperidin-1-yl, -C(CH₃)=C(Br)-CO-morpholin-4-yl, -C(CH₃)=C(Br)-CO-NH-CH₂CH=C(Br)₂, -C(CH₃)=C(Br)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Br)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Br)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Br)-CO-NH-C₆H₅, -C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CN)-CO-NHCH₃, -C(CH₃)=C(CN)-CO-N(CH₃)₂, -C(CH₃)=C(CN)-CO-NH-C₂H₅, -C(CH₃)=C(CN)-CO-N(C₂H₅)₂, -C(CH₃)=C(CN)-CO-NH-n-C₃H₇, -C(CH₃)=C(CN)-CO-NH-i-C₃H₇, -C(CH₃)=C(CN)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-NH-cyclopropyl, -C(CH₃)=C(CN)-CO-NH-cyclobutyl, -C(CH₃)=C(CN)-CO-NH-cyclopentyl, -C(CH₃)=C(CN)-CO-NH-cyclohexyl, -C(CH₃)=C(CN)-CO-NH-cycloheptyl, -C(CH₃)=C(CN)-CO-NH-cyclooctyl, -C(CH₃)=C(CN)-CO-pyrrolidin-1-yl, -C(CH₃)=C(CN)-CO-piperidin-1-yl, -C(CH₃)=C(CN)-CO-morpholin-4-yl, -C(CH₃)=C(CN)-CO-NH-CH₂CH=C(CN)₂, -C(CH₃)=C(CN)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CN)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CN)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CN)-CO-NH-C₆H₅, -C(CH₃)=CH-CO-SCH₃, -C(CH₃)=CH-CO-SC₂H₅, -C(CH₃)=CH-CO-S-n-C₃H₇, -C(CH₃)=CH-CO-S-i-C₃H₇, -C(CH₃)=CH-CO-S-n-C₄H₉, -C(CH₃)=CH-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-SCH₃, -C(CH₃)=C(CH₃)-CO-SC₂H₅, -C(CH₃)=C(CH₃)CO-S-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-S-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-SCH₃, -C(CH₃)=C(C₂H₅)-CO-SC₂H₅, -C(CH₃)=C(C₂H₅)-CO-S-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-SCH₃, -C(CH₃)=C(Cl)-CO-SC₂H₅, -C(CH₃)=C(Cl)-CO-S-n-C₃H₇, -C(CH₃)=C(Cl)-CO-S-i-C₃H₇, -C(CH₃)=C(Cl)-CO-S-n-C₄H₉, -C(CH₃)=C(Cl)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-SCH₃, -C(CH₃)=C(Br)-CO-SC₂H₅, -C(CH₃)=C(Br)-CO-S-n-C₃H₇, -C(CH₃)=C(Br)-CO-S-i-C₃H₇, -C(CH₃)=C(Br)-CO-S-n-C₄H₉, -C(CH₃)=C(Br)-CO-S-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-SCH₃, -C(CH₃)=C(CN)-CO-SC₂H₅, -C(CH₃)=C(CN)-CO-S-n-C₃H₇, -C(CH₃)=C(CN)-CO-S-i-C₃H₇, -C(CH₃)=C(CN)-CO-S-N-C₄H₉, -C(CH₃)=C(CN)-CO-S-tert.-C₄H₉, -C(CH₃)=C(COCH₃)-CO-OCH₃, -C(CH₃)=C(COC₂H₅)-CO-OCH₃, -C(CH₃)=C(CO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COCH₃)-CO-OC₂H₅, -C(CH₃)=C(COC₂H₅)-CO-OC₂H₅, -C(CH₃)=C(CO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COCH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(COC₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-OCH₃, -C(CH₃)=C(CF₃)-CO-OC₂H₅, -C(CH₃)=C(CF₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CF₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(COOCH₃)₂, -C(CH₃)=C(COOC₂H₅)₂, -C(CH₃)=C(COOCH₃)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)₂, -C(CH₃)=CH-CH=CH-COOH, -C(CH₃)=CH-CH=CH-CO-OCH₃, -C(CH₃)=CH-CH=CH-CO-OC₂H₅, -C(CH₃)=CH-CH=C(COOCH₃)₂, -C(CH₃)=CH-CH=C(CN)-CO-OCH₃, -C(CH₃)=CH-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CN)CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH₂, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -C(CH₃)=CH-(CH₂)₂-COOH, -C(CH₃)=CH-(CH₂)₂-CO-OCH₃, -C(CH₃)=CH-(CH₂)₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(COOCH₃)₂, -C(CH₃)=CH-CH₂-CH(COOC₂H₅)₂, -C(CH₃)=CH-CH₂-CH(CN)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CN)-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -C(CH₃)=CH-(CH₂)₂-CO-NH₂, -C(CH₃)=CH-(CH₂)₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-COOH, -C(CH₃)=CH-CH₂-CO-OCH₃, -C(CH₃)=CH-CH₂-CO-OC₂H₅, -C(CH₃)=C(COOCH₃)-CH₂-CO-OCH₃, -C(CH₃)=C(COOCH₃)-CH₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CO-NH₂, -C(CH₃)=CH-CH₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-CO-N(CH₃)₂.
wobei W für eine der folgenden Bedeutungen steht:
-CHO, -COCH₃, -COC₂H₅, -CO-n-C₃H₇, -CO-i-C₃H₇, -CO-n-C₄H₉, -CO-i-C₄H₉, -CO-s-C₄H₉, -CO-tert.-C₄H₉, -CO-CH₂CH=CH₂, -CO-CF₃, -COCCl₃, -COCH₂C≡CH, -CO-cyclopropyl, -CO-cyclobutyl, -CO-cyclopentyl, -CO-cyclohexyl, -CO-CN, -CO-COOCH₃, -CO-COOC₂H₅, -CH=NH, -CH=NCH₃, -CH=NC₂H₅, -CH=N-n-C₃H₅, -CH=N-i-C₃H₅, -CH=N-n-C₄H₉, -CH=NCH₂CH=CH₂, -CH=NCH₂CH=CH₂-CH₃, -CH=NCH₂C≡CH, -CH=NCH₂C≡C-CH₃, -CH=N-cyclopropyl, -CH=N-cyclobutyl, -CH=N-cyclopentyl, -CH=N-cyclohexyl, -CH=N-cycloheptyl, -CH=N-CH₂-CH₂Cl, -CH=N-CH₂Cl, -CH=N-C₆H₅, -CH=N-4-Br-C₆H₄, -CH=N-3-F-C₆H₄, -CH=N-4-F-C₆H₄, -CH=N-2-Cl-C₆H₄, -CH=N-3-Cl-C₆H₄, -CH=N-4-Cl-C₆H₄, -CH=N-2-Br-C₆H₄, -CH=N-2-F-C₆H₄, -CH=N-2-CH₃-C₆H₄, -CH=N-3-CH₃-C₆H₄, -CH=N-4-CH₃-C₆H₄, -CH=N-2-CF₃-C₆H₄, -CH=N-3-CF₃-C₆H₄, -CH=N-4-CF₃-C₆H₄, -CH=N-2-OCH₃-C₆H₄, -CH=N-3-OCH₃-C₆H₄, -CH=N-4-OCH₃-C₆H₄, -CH=N-4-NO₂-C₆H₄, -CH=N-4-CN-C₆H₄, -CH=N-2,4-(Cl,Cl)-C₆H₄, -CH=N-2,4-(CH₃,CH₃)-C₆H₄, -CH=N-CH₂OCH₃ -CH=N-CH₂OC₂H₅, -CH=N-CH₂CH₂OCH₃, -CH=N-CH₂CH₂OC₂H₅, -CH=N-OH, -CH=N-OCH₃, -CH=N-OC₂H₅, -CH=N-O-n-C₃H₇, -CH=N-O-i-C₃H₇, -CH=N-O-n-C₄H₉, -CH=N-O-i-C₄H₉, -CH=N-O-s-C₄H₉, -CH=N-O-tert.-C₄H₉, -CH=N-O-CH₂CH=CH₂, -CH=N-O-CH(CH₃)CH=CH₂, -CH=N-O-CH₂C≡CH, -CH=N-O-CH(CH₃)-C≡CH, -CH=N-O-CH₂-CH=CH-CH₃, -CH=N-O-CH₂-CH₂-Cl, -CH=N-O-CH₂-CH₂-F, -CH=N-O-CH₂-CF₃, -CH=N-O-CH₂-CH=CHCl, -CH=N-O-CH₂-CCl=CH₂, -CH=N-O-CH₂-CBr=CH₂, -CH=N-O-CH₂-CH=CCl-CH₃, -CH=N-OC(O)CH₃, -CH=N-OC(O)C₂H₅, -CH=N-O-CH₂-CN, -CH=N-O-CH₂-CH=CH-CH₂-O-CH₃, -CH=N-O-CH₂-CH=CH-CH₂-O-tert.-C₄H₉, -CH=N-O-(CH₂)₃-C₆H₅, -CH=N-O-(CH₂)₄-C₆H₅, -CH=N-O-(CH₂)₄-4-Cl-C₆H₄, -CH=N-O-(CH₂)₄-4-OCH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-CH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-C₆H₅, -CH=N-O-CH₂CH=CH-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CH-3-OCH₃-C₆H₄, -CH=N-O-(CH₂)₂CH=CH-4-F-C₆H₄, -CH=N-O-(CH₂)CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CHCH₂-4-OCH₃-C₆H₄, -CH=N-O-CH₂-CH=C(CH₃)-C₆H₅, -CH=N-O-(CH₂)₂CH=CH-3,4(Cl,Cl)-C₆H₃, -CH=N-O-(CH₂)₃C≡C-4-F-C₆H₄, -CH₂=N-OCHOCH₃, -CH=N-OC₂H₄OCH₃, -CH=N-OCH₂OC₂H₅, -CH=N-OCH(CH₃)OCH₃, -CH=N-OCH(CH₃)COOCH₃, -CH=N-OCH(CH₃)COO-n-C₄H₉, -CH=N-NH₂, -CH=N-NHCH₃, -CH=N-NHC₂H₅, -CH=N-NH-n-C₃H₇, -CH=N-NH-i-C₃H₇, -CH=N-NH-n-C₄H₉, -CH=N-NH-i-C₄H₉, -CH=N-NH-s-C₄H₉, -CH=N-NH-tert.-C₄H₉, -CH=N-NH-cyclopropyl, -CH=N-NH-cyclobutyl, -CH=N-NH-cyclopentyl, -CH=N-NH-cyclohexyl, -CH=N-NH-cycloheptyl, -CH=N-N(CH₃)₂, -CH=N-N(C₂H₅)₂, -CH=N-N(C₃H₇)₂, -CH=N-N(i-C₃H₇)(CH₃), -CH=N-NHCH₂-C=CH, -CH=N-NHCH₂-C≡CH, -CH=N-N(CH₃)-CH₂-C≡CH, -CH=N-NHCH₂CF₃, -CH=N-NH-CO-CH₃, -CH=N-NH-CO-CH₂H₅, -CH=N-NH-COOCH₃, -CH=N-NH-COOC₂H₅, -CH=N-NH-COO-tert.-C₄H₉, -CH=N-pyrrolidin-1-yl, -CH=N-piperidin-1-yl, -CH=N-morpholin-4-yl, -CH=N-NH-C₆H₅, -CH=N-NH-(4-Cl-C₆H₄), -CH=N-NH-(4-NO₂-C₆H₄), -CH=N-NH-(4-F-C₆H₄), -CH=N-NH-(4-CH₃O-C₆H₄), -CH=N-NH-(2,4-Cl₂-C₆H₃), -CH=N-NH-(2,4-(NO₂)₂-C₆H₃), -CH=N-NH-CO-NH₂, -CH=N-NH-CO-NHCH₃, -CH=N-NH-CO-NHC₂H₅, -CH=N-NH-CO-N(CH₃)₂, -CH=CH-COOH, -CH=CH-CO-OCH₃, -CH=C-CO-OC₂H₅, -CH=CH-CO-O-n-C₃H₇, -CH=CH-CO-O-i-C₃H₇, -CH=CH-CO-O-n-C₄H₉, -CH=CH-CO-O-tert.-C₄H₉, -CH=CH-CO-O-cyclopropyl, -CH=CH-CO-O-cyclobutyl, -CH=CH-CO-O-cyclopentyl, -CH=CH-CO-O-cyclohexyl, -CH=CH-CO-O-cycloheptyl, -CH=C(CH₃)-COOH, -CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CO-O-n-C₃H₇, -CH=C(CH₃)-CO-O-i-C₃H₇, -CH=C(CH₃)-CO-O-n-C₄H₉, -CH=C(CH₃)-CO-O-tert.-C₄H₉, -CH=C(CH₃)-CO-O-cyclopropyl, -CH=C(CH₃)-CO-O-cyclobutyl, -CH=C(CH₃)-CO-O-cyclopentyl, -CH=C(CH₃)-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cycloheptyl, -CH=C(C₂H₅)-COOH, -CH=C(C₂H₅)-CO-OCH₃, -CH=C(C₂H₅)-CO-OC₂H₅, -CH=C(C₂H₅)-CO-O-n-C₃H₇, -CH=C(C₂H₅)-CO-O-i-C₃H₇, -CH=C(C₂H₅)-CO-O-n-C₄H₉, -CH=C(C₂H₅)-CO-O-tert.-C₄H₉, -CH=(C₂H₅)-CO-O-cyclopropyl, -CH=C(C₂H₅)-CO-O-cyclobutyl, -CH=C(C₂H₅)-CO-O-cyclopentyl, -CH=C(C₂H₅)-CO-O-cyclohexyl, -CH=C(C₂H₅)-CO-O-cycloheptyl, -CH=C(Cl)-COOH, -CH=C(Cl)-CO-OCH₃, -CH=C(Cl)-CO-OC₂H₅, -CH=C(Cl)-CO-O-n-C₃H₇, -CH=C(Cl)-CO-O-i-C₃H₇, -CH=C(Cl)-CO-O-n-C₄H₉, -CH=C(Cl)-CO-O-tert.-C₄H₉, -CH=C(Cl)-CO-O-cyclopropyl, -CH=C(Cl)-CO-O-cyclobutyl, -CH=C(Cl)-CO-O-cyclopentyl, -CH=C(Cl)-CO-O-cyclohexyl, -CH=C(Cl)-CO-O-cycloheptyl, -CH=C(Br)-COOH, -CH=C(Br)-CO-OCH₃, -CH=C(Br)-CO-OC₂H₅, -CH=C(Br)-CO-O-n-C₃H₇, -CH=C(Br)-CO-O-i-C₃H₇, -CH=C(Br)-CO-O-n-C₄H₉, -CH=C(Br)-CO-O-tert.-C₄H₉, -CH=C(Br)-CO-O-cyclopropyl, -CH=C(Br)-CO-O-cyclobutyl, -CH=C(Br)-CO-O-cyclopentyl, -CH=C(Br)-CO-O-cyclohexyl, -CH=C(Br)-CO-O-cycloheptyl, -CH=C(CN)-COOH, -CH=C(CN)-CO-OCH₃, -CH=C(CN)-CO-OC₂H₅, -CH=C(CN)-CO-O-n-C₃H₇, -CH=C(CN)-CO-O-i-C₃H₇, -CH=C(CN)-CO-O-n-C₄H₉, -CH=C(CN)-CO-O-tert.-C₄H₉, -CH=C(CN)-CO-O-cyclopropyl, -CH=C(CN)-CO-O-cyclobutyl, -CH=C(CN)-CO-O-cyclopentyl, -CH=C(CN)-CO-O-cyclohexyl, -CH=C(CN)-CO-O-cycloheptyl, -CH=CH-CO-OCH₂-OCH₃, -CH=CH-CO-OCH₂-OC₂H₅, -CH=CH-CO-OCH₂-O-n-C₃H₅, -CH=CH-CO-OCH₂-O-i-C₃H₅, -CH=CH-CO-OCH(CH₃)-OCH₃, -CH=CH-CO-OCH(CH₃)-OC₂H₅, -CH=CH-CO-O-CH₂CH₂-OCH₃, -CH=CH-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-OCH₃, -CH=C(CH₃)-CO-OCH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-O-n-C₃H₅, -CH=C(CH₃)-CO-OCH₂-O-i-C₃H₅, -CH=C(CH₃)-CO-OCH(CH₃)-OCH₃, -CH=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CH₃)-CO-O-CH₂CH₂-OCH₃, -CH=C(CH₃)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-OCH₃, -CH=C(C₂H₅)-CO-OCH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-O-n-C₃H₅, -CH=C(C₂H₅)-CO-OCH₂-O-i-C₃H₅, -CH=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-OCH₃, -CH=C(Cl)-CO-OCH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-O-n-C₃H₅, -CH=C(Cl)-CO-OCH₂-O-i-C₃H₅, -CH=C(Cl)-CO-OCH(CH₃)-OCH₃, -CH=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Cl)-CO-O-CH₂CH₂-OCH₃, -CH=C(Cl)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-OCH₃, -CH=C(Br)-CO-OCH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-O-n-C₃H₅, -CH=C(Br)-CO-OCH₂-O-i-C₃H₅, -CH=C(Br)-CO-OCH(CH₃)-OCH₃, -CH=C(Br)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Br)-CO-O-CH₂CH₂-OCH₃, -CH=C(Br)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-OCH₃, -CH=C(CN)-CO-OCH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-O-n-C₃H₅, -CH=C(CN)-CO-OCH₂-O-i-C₃H₅, -CH=C(CN)-CO-OCH(CH₃)-OCH₃, -CH=C(CN)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CN)-CO-O-CH₂CH₂-OCH₃, -CH=C(CN)-CO-O-CH₂CH₂-OC₂H₅, -CH=CH-CO-OCH₂-CF₃, -CH=CH-CO-OCH₂-CCl₃, -CH=CH-CO-OCH₂-oxiranyl, -CH=CH-CO-O(CH₂)₃-Br, -CH=CH-CO-OCH₂-CH=CH₂, -CH=CH-CO-OCH₂-C≡CH, -CH=CH-CO-OCH₂-CN, -CH=CH-CO-O(CH₂)₂-CN, -CH=C(CH₃)-CO-OCH₂-CF₃, -CH=C(CH₃)-CO-OCH₂-CCl₃, -CH=C(CH₃)-CO-OCH₂-oxiranyl, -CH=C(CH₃)-CO-O(CH₂)₃-Br, -CH=C(CH₃)-CO-OCH₂-CH=CH₂, -CH=C(CH₃)-CO-OCH₂-C≡CH, -CH=C(CH₃)-CO-OCH₂-CN, -CH=C(CH₃)-CO-O(CH₂)₂-CN, -CH=C(C₂H₅)-CO-OCH₂-CF₃, -CH=C(C₂H₅)-CO-OCH₂-CCl₃, -CH=C(C₂H₅)-CO-OCH₂-oxiranyl, -CH=C(C₂H₅)-CO-O(CH₂)₃-Br, -CH=C(C₂H₅)-CO-OCH₂-CH=CH₂, -CH=C(C₂H₅)-CO-OCH₂-C≡CH, -CH=C(C₂H₅)-CO-OCH₂-CN, -CH=C(C₂H₅)-CO-O(CH₂)₂-CN, -CH=C(Cl)-CO-OCH₂-CF₃, -CH=C(Cl)-CO-OCH₂-CCl₃, -CH=C(Cl)-CO-OCH₂-oxiranyl, -CH=C(Cl)-CO-O(CH₂)₃-Br, -CH=C(Cl)-CO-OCH₂-CH=CH₂, -CH=C(Cl)-CO-OCH₂-C≡CH, -CH=C(Cl)-CO-OCH₂-CN, -CH=C(Cl)-CO-O(CH₂)₂-CN, -CH=C(Br)-CO-OCH₂-CF₃, -CH=C(Br)-CO-OCH₂-CCl₃, -CH=C(Br)-CO-OCH₂-oxiranyl, -CH=C(Br)-CO-O(CH₂)₃-Br, -CH=C(Br)-CO-OCH₂-CH=CH₂, -CH=C(Br)-CO-OCH₂-C≡CH, -CH=C(Br)-CO-OCH₂-CN, -CH=C(Br)-CO-O(CH₂)₂-CN, -CH=C(CN)-CO-OCH₂-CF₃, -CH=C(CN)-CO-OCH₂-CCl₃, -CH=C(CN)-CO-OCH₂-oxiranyl -CH=C(CN)-CO-O(CH₂)₃-Br, -CH=C(CN)-CO-OCH₂-CH=CH₂, -CH=C(CN)-CO-OCH₂-C≡CH, -CH=C(CN)-CO-OCH₂-CN, -CH=C(CN)-CO-O(CH₂)₂-CN, -CH=CH-CO-CH₃, -CH=CH-CO-C₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-i-C₃H₇, -CH=CH-CO-n-C₄H₉, -CH=CH-CO-tert.-C₄H₉, -CH=CH-CO-CH₂Cl, -CH=CH-CO-CH₂Br, -CH=CH-CO-CHCl₂, -CH=CH-CO-CH₂-OCH₃, -CH=CH-CO-CH(OCH₃)₂, -CH=CH-CO-CH₂-SCH₃, -CH=C(CH₃)-CO-CH₃, -CH=C(CH₃)-CO-C₂H₅, -CH=C(CH₃)-CO-n-C₃H₇, -CH=C(CH₃)-CO-i-C₃H₇, -CH=C(CH₃)-CO-n-C₄H₉, -CH=C(CH₃)-CO-tert.-C₄H₉, -CH=C(CH₃)-CO-CH₂Cl, -CH=C(CH₃)-CO-CH₂Br, -CH=C(CH₃)-CO-CHCl₂, -CH=C(CH₃)-CO-CH₂-OCH₃, -CH=C(CH₃)-CO-CH(OCH₃)₂, -CH=C(CH₃)-CO-CH₂-SCH₃, -CH=C(C₂H₅)-CO-CH₃, -CH=C(C₂H₅)-CO-C₂H₅, -CH=C(C₂H₅)-CO-n-C₃H₇, -CH=C(C₂H₅)-CO-i-C₃H₇, -CH=C(C₂H₅)-CO-n-C₄H₉, -CH=C(C₂H₅)-CO-tert.-C₄H₉, -CH=C(C₂H₅)-CO-CH₂Cl, -CH=C(C₂H₅)-CO-CH₂Br, -CH=C(C₂H₅)-CO-CHCl₂, -CH=C(C₂H₅)-CO-CH₂-OCH₃, -CH=C(C₂H₅)-CO-CH(OCH₃)₂, -CH=C(C₂H₅)-CO-CH₂-SCH₃, -CH=C(Cl)-CO-CH₃, -CH=C(Cl)-CO-C₂H₅, -CH=C(Cl)-CO-n-C₃H₇, -CH=C(Cl)-CO-i-C₃H₇, -CH=C(Cl)-CO-n-C₄H₉, -CH=C(Cl)-CO-tert.-C₄H₉, -CH=C(Cl)-CO-CH₂Cl, -CH=C(Cl)-CO-CH₂Br, -CH=C(Cl)-CO-CHCl₂, -CH=C(Cl)-CO-CH₂-OCH₃, -CH=C(Cl)-CO-CH(OCH₃)₂, -CH=C(Cl)-CO-CH₂-SCH₃, -CH=C(Br)-CO-CH₃, -CH=C(Br)-CO-C₂H₅, -CH=C(Br)-CO-n-C₃H₇, -CH=C(Br)-CO-i-C₃H₇, -CH=C(Br)-CO-n-C₄H₉, -CH=C(Br)-CO-tert.-C₄H₉, -CH=C(Br)-CO-CH₂Cl, -CH=C(Br)-CO-CH₂Br, -CH=C(Br)-CO-CHCl₂, -CH=C(Br)-CO-CH₂-OCH₃, -CH=C(Br)-CO-CH(OCH₃)₂, -CH=C(Br)-CO-CH₂-SCH₃, -CH=C(CN)-CO-CH₃, -CH=C(CN)-CO-C₂H₅, -CH=C(CN)-CO-n-C₃H₇, -CH=C(CN)-CO-i-C₃H₇, -CH=C(CN)-CO-n-C₄H₉, -CH=C(CN)-CO-tert.-C₄H₉, -CH=C(CN)-CO-CH₂Cl, -CH=C(CN)-CO-CH₂Br, -CH=C(CN)-CO-CHCl₂, -CH=C(CN)-CO-CH₂-OCH₃, -CH=C(CN)-CO-CH(OCH₃)₂, -CH=C(CN)-CO-CH₂-SCH₃, -CH=CH-CO-C₆H₅, -CH=CH-CO-(4-Cl-C₆H₄), -CH=C(CH₃)-CO-C₆H₅, -CH=C(CH₃)-CO-(4-Cl-C₆H₄), -CH=C(C₂H₅)-CO-C₆H₅, -CH=C(C₂H₅)-CO-(4-Cl-C₆H₄), -CH=C(Cl)-CO-C₆H₅, -CH=C(Br)-CO-C₆H₅, -CH=C(CN)-CO-C₆H₅, -CH=CH-CO-NH₂, -CH=CH-CO-NHCH₃, -CH=CH-CO-N(CH₃)₂, -CH=CH-CO-NH-C₂H₅, -CH=CH-CO-N(C₂H₅)₂, -CH=CH-CO-NH-n-C₃H₇, -CH=CH-CO-NH-i-C₃H₇, -CH=CH-CO-NH-tert.-C₄H₉, -CH=CH-CO-NH-cyclopropyl, -CH=CH-CO-NH-cyclobutyl, -CH=CH-CO-NH-cyclopentyl, -CH=CH-CO-NH-cyclohexyl, -CH=CH-CO-NH-cycloheptyl, -CH=CH-CO-NH-cyclooctyl, -CH=CH-CO-pyrrolidin-1-yl, -CH=CH-CO-piperidin-1-yl, -CH=CH-CO-morpholin-4-yl, -CH=CH-CO-NH-CH₂CH=CH₂, -CH=CH-CO-NH-CH₂C≡CH, -CH=CH-CO-N(CH₃)-CH₂C≡CH, -CH=CH-CO-NH-(CH₂)₂Cl, -CH=CH-CO-NH-C₆H₅, -CH=C(CH₃)-CO-NH₂, -CH=C(CH₃)-CO-NHCH₃, -CH=C(CH₃)-CO-N(CH₃)₂, -CH=C(CH₃)-CO-NH-C₂H₅, -CH=C(CH₃)-CO-N(C₂H₅)₂, -CH=C(CH₃)-CO-NH-n-C₃H₇, -CH=C(CH₃)-CO-NH-i-C₃H₇, -CH=C(CH₃)-CO-NH-tert.-C₄H₉, -CH=C(CH₃)-CO-NH-cyclopropyl, -CH=C(CH₃)-CO-NH-cyclobutyl, -CH=C(CH₃)-CO-NH-cyclopentyl, -CH=C(CH₃)-CO-NH-cyclohexyl, -CH=C(CH₃)-CO-NH-cycloheptyl, -CH=C(CH₃)-CO-NH-cyclooctyl, -CH=C(CH₃)-CO-pyyrolidin-1-yl, -CH=C(CH₃)-CO-piperidin-1-yl, -CH=C(CH₃)-CO-morpholin-4-yl, -CH=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -CH=C(CH₃)-CO-NH-CH₂C≡CH, -CH=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CH₃)-CO-NH-(CH₂)₂Cl, -CH=C(CH₃)-CO-NH-C₆H₅, -CH=C(C₂H₅)-CO-NH₂, -CH=C(C₂H₅)-CO-NHCH₃, -CH=C(C₂H₅)-CO-N(CH₃)₂, -CH=C(C₂H₅)-CO-NH-C₂H₅, -CH=C(C₂H₅)-CO-N(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-n-C₃H₇, -CH=C(C₂H₅)-CO-NH-i-C₃H₇, -CH=C(C₂H₅)-CO-NH-tert.-C₄H₉, -CH=C(C₂H₅)-CO-NH-cyclopropyl, -CH=C(C₂H₅)-CO-NH-cyclobutyl, -CH=C(C₂H₅)-CO-NH-cyclopentyl, -CH=C(C₂H₅)-CO-NH-cyclohexyl, -CH=C(C₂H₅)-CO-NH-cycloheptyl, -CH=C(C₂H₅)-CO-NH-cyclooctyl, -CH=C(C₂H₅)-CO-pyrrolidin-1-yl, -CH=C(C₂H₅)-CO-piperidin-1-yl, -CH=C(C₂H₅)-CO-morpholin-4-yl, -CH=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-CH₂C≡CH, -CH=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -CH=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -CH=C(C₂H₅)-CO-NH-C₆H₅, -CH=C(Cl)-CO-NH₂, -CH=C(Cl)-CO-NHCH₃, -CH=C(Cl)-CO-N(CH₃)₂, -CH=C(Cl)-CO-NH-C₂H₅, -CH=C(Cl)-CO-N(C₂H₅)₂, -CH=C(Cl)-CO-NH-n-C₃H₇, -CH=C(Cl)-CO-NH-i-C₃H₇, -CH=C(Cl)-CO-NH-tert.-C₄H₉, -CH=C(Cl)-CO-NH-cyclopropyl, -CH=C(Cl)-CO-NH-cyclobutyl, -CH=C(Cl)-CO-NH-cyclopentyl, -CH=C(Cl)-CO-NH-cyclohexyl, -CH=C(Cl)-CO-NH-cycloheptyl, -CH=C(Cl)-CO-NH-cyclooctyl, -CH=C(Cl)-CO-pyrrolidin-1-yl, -CH=C(Cl)-CO-piperidin-1-yl, -CH=C(Cl)-CO-morpholin-4-yl, -CH=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -CH=C(Cl)-CO-NH-CH₂C≡CH, -CH=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Cl)-CO-NH-(CH₂)₂Cl, -CH=C(Cl)-CO-NH-C₆H₅, -CH=C(Br)-CO-NH₂, -CH=C(Br)-CO-NHCH₃, -CH=C(Br)-CO-N(CH₃)₂, -CH=C(Br)-CO-NH-C₂H₅, -CH=C(Br)-CO-N(C₂H₅)₂, -CH=C(Br)-CO-NH-n-C₃H₇, -CH=C(Br)-CO-NH-i-C₃H₇, -CH=C(Br)-CO-NH-tert.-C₄H₉, -CH=C(Br)-CO-NH-cyclopropyl, -CH=C(Br)-CO-NH-cyclobutyl, -CH=C(Br)-CO-NH-cyclopentyl, -CH=C(Br)-CO-NH-cyclohexyl, -CH=C(Br)-CO-NH-cycloheptyl, -CH=C(Br)-CO-NH-cyclooctyl, -CH=C(Br)-CO-pyrrolidin-1-yl, -CH=C(Br)-CO-piperidin-1-yl, -CH=C(Br)-CO-morpholin-4-yl, -CH=C(Br)-CO-NH-CH₂CH=C(Br)₂, -CH=C(Br)-CO-NH-CH₂C≡CH, -CH=C(Br)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Br)-CO-NH-(CH₂)₂Cl, -CH=C(Br)-CO-NH-C₆H₅, -CH=C(CN)-CO-NH₂, -CH=C(CN)-CO-NHCH₃, -CH=C(CN)-CO-N(CH₃)₂, -CH=C(CN)-CO-NH-C₂H₅, -CH=C(CN)-CO-N(C₂H₅)₂, -CH=C(CN)-CO-NH-n-C₃H₇, -CH=C(CN)-CO-NH-i-C₃H₇, -CH=C(CN)-CO-NH-tert.-C₄H₉, -CH=C(CN)-CO-NH-cyclopropyl, -CH=C(CN)-CO-NH-cyclobutyl, -CH=C(CN)-CO-NH-cyclopentyl, -CH=C(CN)-CO-NH-cyclohexyl, -CH=C(CN)-CO-NH-cycloheptyl, -CH=C(CN)-CO-NH-cyclooctyl, -CH=C(CN)-CO-pyrrolidin-1-yl, -CH=C(CN)-CO-piperidin-1-yl, -CH=C(CN)-CO-morpholin-4-yl, -CH=C(CN)-CO-NH-CH₂CH=C(CN)₂, -CH=C(CN)-CO-NH-CH₂C≡CH, -CH=C(CN)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CN)-CO-NH-(CH₂)₂Cl, -CH=C(CN)-CO-NH-C₆H₅, -CH=CH-CO-SCH₃, -CH=CH-CO-SC₂H₅, -CH=CH-CO-S-n-C₃H₇, -CH=CH-CO-S-i-C₃H₇, -CH=CH-CO-S-n-C₄H₉, -CH=CH-CO-S-tert.-C₄H₉, -CH=C(CH₃)-CO-SCH₃, -CH=C(CH₃)-CO-SC₂H₅, -CH=C(CH₃)-CO-S-n-C₃H₇, -CH=C(CH₃)-CO-S-i-C₃H₇, -CH=C(CH₃)-CO-S-n-C₄H₉, -CH=C(CH₃)-CO-S-tert.-C₄H₉, -CH=C(C₂H₅)-CO-SCH₃, -CH=C(C₂H₅)-CO-SC₂H₅, -CH=C(C₂H₅)-CO-S-n-C₃H₇, -CH=C(C₂H₅)-CO-S-i-C₃H₇, -CH=C(C₂H₅)-CO-S-n-C₄H₉, -CH=C(C₂H₅)-CO-S-tert.-C₄H₉, -CH=C(Cl)-CO-SCH₃, -CH=C(Cl)-CO-SC₂H₅, -CH=C(Cl)-CO-S-n-C₃H₇, -CH=C(Cl)-CO-S-i-C₃H₇, -CH=C(Cl)-CO-S-n-C₄H₉, -CH=C(Cl)-CO-S-tert.-C₄H₉, -CH=C(Br)-CO-SCH₃, -CH=C(Br)-CO-SC₂H₅, -CH=C(Br)-CO-S-n-C₃H₇, -CH=C(Br)-CO-S-i-C₃H₇, -CH=C(Br)-CO-S-n-C₄H₉, -CH=C(Br)-CO-S-tert.-C₄H₉, -CH=C(CN)-CO-SCH₃, -CH=C(CN)-CO-SC₂H₅, -CH=C(CN)-CO-S-n-C₃H₇, -CH=C(CN)-CO-S-i-C₃H₇, -CH=C(CN)-CO-S-n-C₄H₉, -CH=C(CN)-CO-S-tert.-C₄H₉, -CH=C(COCH₃)-CO-OCH₃, -CH=C(COC₂H₅)-CO-OCH₃, -CH=C(CO-n-C₃H₇)-CO-OCH₃, -CH=C(COCH₃)-CO-OC₂H₅, -CH=C(COC₂H₅)-CO-OC₂H₅, -CH=C(CO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COCH₃)-CO-O-n-C₃H₇, -CH=C(COC₂H₅)-CO-O-n-C₃H₇, -CH=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-OCH₃, -CH=C(CF₃)-CO-OC₂H₅, -CH=C(CF₃)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-O-i-C₃H₇, -CH=C(CF₃)-CO-O-n-C₄H₉, -CH=C(CF₃)-CO-O-tert.-C₄H₉, -CH=C(COOCH₃)₂, -CH=C(COOC₂H₅)₂, -CH=C(COOCH₃)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)-CO-OCH₃, -CH=C(COO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)₂, -CH=CH-CH=CH-COOH, -CH=CH-CH=CH-CO-OCH₃, -CH=CH-CH=CH-CO-OC₂H₅, -CH=CH-CH=C(COOCH₃)₂, -CH=CH-CH=C(CN)-CO-OCH₃, -CH=CH-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-OCH₃, -CH=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CH=C(Cl)-CO-OCH₃, -CH=C(CH₃)-CH=C(Br)-CO-OCH₃, -CH=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-NH₂, -CH=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -CH=CH-(CH₂)₂-COOH, -CH=CH-(CH₂)₂-CO-OCH₃, -CH=CH-(CH₂)₂-CO-OC₂H₅, -CH=CH-CH₂-CH(COOCH₃)₂, -CH=CH-CH₂-CH(COOC₂H₅)₂, -CH=CH-CH₂-CH(CN)-CO-OCH₃, -CH=CH-CH₂-CH(CN)-CO-OC₂H₅, -CH=CH-CH₂-CH(CH₃)-CO-OCH₃, -CH=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -CH=CH-(CH₂)₂-CO-NH₂, -CH=CH-(CH₂)₂-CO-NH-CH₃, -CH=CH-CH₂-COOH, -CH=CH-CH₂-CO-OCH₃, -CH=CH-CH₂-CO-OC₂H₅, -CH=C(COOCH₃)-CH₂-CO-OCH₃, -CH=C(COOCH₃)-CH₂-CO-OC₂H₅, -CH=CH-CH₂-CO-NH₂, -CH=CH-CH₂-CO-NH-CH₃, -CH=CH-CH₂-CO-N(CH₃)₂, -CH(OCH₃)₂, -CH(SCH₃)₂, -CH(OC₂H₅)₂, -CH(SC₂H₅)₂, -CH(O-n-C₃H₇)₂, -CH(O-i-C₃H₇)₂, -CH(S-n-C₃H₇)₂, -CH(S-i-C₃H₇)₂, -CH(O-n-C₄H₉)₂, -CH(O-i-C₄H₉)₂, -CH(O-s-C₄H₉)₂, -CH(O-tert.-C₄H₉)₂, -CH(S-n-C₄H₉)₂, -CH(S-i-C₄H₉)₂, -CH(S-s-C₄H₉)₂, -CH(S-tert.-C₄H₉)₂, -CH(OC₅H₁₁)₂, 1,3-Dioxolan-2-yl, 1,3-Dithio­ lan-2-yl, 1,3-Oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 4-Methyl-1,3-dithiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 5-Methyl-1,3-oxathiolan-2-yl, 4-Ethyl-1,3-dioxolan-2-yl, 4-Ethyl- 1,4-dithiolan-2-yl, 4-Ethyl-1,3-oxathiolan-2-yl, 5-Ethyl-1,3-oxa­ thiolan-2-yl, 4,5-Dimethyl-1,3-dioxolan-2-yl, 4,4-Dimethyl-1,3- dioxolan-2-yl, 4,5-Dimethyl-1,3-dithiolan-2-yl, 5,5-Dimethyl-1,3- dithiolan-2-yl, 4,5-Dimethyl-1,3-oxathiolan-2-yl, 5,5-Dimethyl- 1,3-oxathiolan-2-yl, 4,4-Dimethyl-1,3-oxathiolan-2-yl, 4-Vinyl- 1,3-dioxolan-2-yl, 4-Vinyl-1,3-dithiolan-2-yl, 4-Vinyl-1,3-oxa­ thiolan-2-yl, 5-Vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3- dioxolan-2-yl, 4-Chlormethyl-1,3-dithiolan-2-yl, 4-Chlormethyl- 1,3-oxathiolan-2-yl, 5-Chlormethyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-1,3-dithio­ lan-2-yl, 4-Hydroxymethyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl- 1,3-oxathiolan-2-yl, 4-Methoxymethyl-1,3-dioxolan-2-yl, 4-Allyl­ oxymethyl-1,3-dioxolan-2-yl, 4-Propargyloxymethyl-1,3-dioxolan- 2-yl, 4-Acetoxymethyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-1,3-dithiolan-2-yl, 4-Propargyl­ oxymethyl-1,3-dithiolan-2-yl, 4-Acetoxymethyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-1,3-oxa­ thiolan-2-yl, 4-Allyloxymethyl-1,3-oxathiolan-2-yl, 5-Allyloxy­ methyl-1,3-oxathiolan-2-yl, 4-Propargyloxymethyl-1,3-oxathiolan- 2-yl, 5-Propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxymethyl- 1,3-oxathiolan-2-yl, 5-Acetoxymethyl-1,3-oxathiolan-2-yl, 4-Methylthiomethyl-1,3-dioxolan-2-yl, 4-Methylthiomethyl-1,3- dithiolan-2-yl, 4-Carboxy-1,3-dioxolan-2-yl, 4-Carboxy-1,3- dithiolan-2-yl, 4-Methoxycarbonyl-1,3-dioxolan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-1,3-di­ thiolan-2-yl, 4-n-Butoxycarbonyl-1,3-dithiolan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-4-methyl- 1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-di­ thiolan-2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-1,3- dithiolan-2-yl, 1,3-Dioxan-2-yl, 1,3-Dithian-2-yl, 1,3-Oxathian- 2-yl, 5-Methyl-1,3-dioxan-2-yl, 5-Methyl-1,3-dithian-2-yl, 5-Methyl-1,3-oxathian-2-yl, 5,5-Dimethyl-1,3-dioxan-2-yl, 4,6-Di­ methyl-1,3-dioxan-2-yl, 4,4-Dimethyl-1,3-dioxan-2-yl, 5,5-Di­ methyl-1,3-dithian-2-yl, 4,6-Dimethyl-1,3-dithian-2-yl, 4,4-Di­ methyl-1,3-dithian-2-yl, 5,5-Dimethyl-1,3-oxathian-2-yl, 4,4-Di­ methyl-1,3-oxathian-2-yl, 6,6-Dimethyl-1,3-oxathian-2-yl, 4-Hydroxymethyl-1,3-dioxan-2-yl, 4-Methoxymethyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-1,3-dioxan-2- yl, 4-Hydroxymethyl-1,3-dithian-2-yl, 4-Methoxymethyl-1,3-di­ thian-2-yl, 4-Allyloxymethyl-1,3-dithian-2-yl, 4-Acetoxymethyl- 1,3-dithian-2-yl, 4-Chlormethyl-1,3-dioxan-2-yl, 4-Chlormethyl- 1,3-dithian-2-yl, 1,3-Dioxepan-2-yl, 1,3-Dithiepan-2-yl, 1,3-Di­ oxep-5-en-2-yl, 4-Methoxycarbonyl-1,3-dioxan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-1,3-dithian- 2-yl, 4-n-Butoxycarbonyl-1,3-dithian-2-yl, 4-Methoxycarbonyl-4- methyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxan-2- yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-4-methyl- 1,3-dithian-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithian-2-yl, -C(CH₃)(OCH₃)₂, -C(CH₃)(SCH₃)₂, -C(CH₃)(OC₂H₅)₂, -C(CH₃)(SC₂H₅)₂, -C(CH₃)(O-n-C₃H₇)₂, -C(CH₃)(O-i-C₃H₇)₂, -C(CH₃)(S-n-C₃H₇)₂, -C(CH₃)(S-i-C₃H₇)₂, -C(CH₃)(O-n-C₄H₉)₂, -C(CH₃)(O-i-C₄H₉)₂, -C(CH₃)(O-s-C₄H₉)₂, -C(CH₃)(O-tert.-C₄H₉)₂, -C(CH₃)(S-n-C₄H₉)₂, -C(CH₃)(S-i-C₄H₉)₂, -C(CH₃)(S-s-C₄H₉)₂, -C(CH₃)(S-tert.-C₄H₉)₂, -C(CH₃)(O-n-C₅H₁₁)′′, 2-Methyl-1,3-dioxolan-2-yl, 2-Methyl-1,3-di­ thiolan-2-yl, 2-Methyl-1,3-oxathiolan-2-yl, 2,4-Dimethyl-1,3- dioxolan-2-yl, 2,4-Dimethyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-1,3- oxathiolan-2-yl, 2,5-Dimethyl-1,3-oxathiolan-2-yl, 4-Ethyl-2- methyl-1,3-dioxolan-2-yl, 4-Ethyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Ethyl-2-methyl-1,3- oxathiolan-2-yl, 2,4,5-Trimethyl-1,3-dioxolan-2-yl, 2,4,4-Tri­ methyl-1,3-dioxolan-2-yl, 2,4,5-Trimethyl-1,3-dithiolan-2-yl, 2,4,4-Trimethyl-1,3-dithiolan-2-yl, 2,4,5-Trim 99999 00070 552 001000280000000200012000285919988800040 0002004131038 00004 99880ethyl-1,3-oxathio­ lan-2-yl, 2,4,4-Trimethyl-1,3-oxathiolan-2-yl, 2-Methyl-4-vinyl- 1,3-dioxolan-2-yl, 2-Methyl-4-vinyl-1,3-dithiolan-2-yl, 2-Methyl- 4-vinyl-1,3-oxathiolan-2-yl, 2-Methyl-5-vinyl-1,3-oxathiolan-2- yl, 4-Chlormethyl-2-methyl-1,3-dioxolan-2-yl, 4-Chlormethyl-2- methyl-1,3-dithiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-oxathio­ lan-2-yl, 5-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Hydroxy­ methyl-2-methyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-2- methyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dioxolan- 2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxy- 2-methyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dithiolan-2-yl, 4-Acetoxy-2- methyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-oxathio­ lan-2-yl, 5-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Allyl­ oxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5 Allyloxymethyl-2- methyl-1,3-oxathiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3- oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3-oxathiolan- 2-yl, 4-Acetoxy-2-methyl-1,3-oxathiolan-2-yl, 5-Acetoxy-2-methyl- 1,3-oxathiolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dioxolan-2- yl, 2-Methyl-4-methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-2- methyl-1,3-dioxolan-2-yl, 4-Carboxy-2-methyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-2- methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-2-methyl-1,3-dioxo­ lan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-Eth­ oxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-2- methyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-di­ oxolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-ethoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4- ethoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-n-butoxy­ carbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl-1,3- dithiolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-dioxan-2- yl, 2-Methyl-1,3-dithian-2-yl, 2-Methyl-1,3-oxathian-2-yl, 2,5- Dimethyl-1,3-dioxan-2-yl, 2,5-Dimethyl-1,3-dithian-2-yl, 2,5-Di­ methyl-1,3-oxathian-2-yl, 2,5,5-Trimethyl-1,3-dioxan-2-yl, 2,4,6- Trimethyl-1,3-dioxan-2-yl, 2,4,4-Trimethyl-1,3-dioxan-2-yl, 2,5,5-Trimethyl-1,3-dithian-2-yl, 2,4,6-Trimethyl-1,3-dithian-2- yl, 2,4,4-Trimethyl-1,3-dithian-2-yl, 2,5,5-Trimethyl-1,3-oxa­ thian-2-yl, 2,4,4-Trimethyl-1,3-oxathian-2-yl, 2,6,6-Trimethyl- 1,3-oxathian-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-2- methyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dithian-2-yl, 4-Methoxymethyl-2- methyl-1,3-dithian-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithian-2- yl, 4-Acetoxymethyl-2-methyl-1,3-dithian-2-yl, 4-Chlormethyl-2- methyl-1,3-dioxan-2-yl, 4-Chlormethyl-2-methyl-1,3-dithian-2-yl, -C(CH₃)=NH, -C(CH₃)=N-CH₃, -C(CH₃)=N-C₂H₅, -C(CH₃)=N-n-C₃H₇, -(CH₃)=N-i-C₃H₇, -C(CH₃)=N-n-C₄H₉, -C(CH₃)=N-CH₂CH=CH₂, -C(CH₃)=N-CH₂CH=CH₂-CH₃, -C(CH₃)=N-CH₂C≡CH, -C(CH₃)=N-CH₂C≡C-CH₃, -C(CH₃)=N-cyclopropyl, -C(CH₃)=N-cyclobutyl, -C(CH₃)=N-cyclo­ pentyl, -C(CH₃)=N-cyclohexyl, -C(CH₃)=N-cycloheptyl, -C(CH₃)=N-CH₂-CH₂Cl, -C(CH₃)=N-CH₂Cl, -C(CH₃)=N-C₆H₅, -C(CH₃)=N-(2-F-C₆H₄), -C(CH₃)=N-(3-F-C₆H₄), -C(CH₃)=N-(4-F-C₆H₄), -C(CH₃)=N-(2-Cl-C₆H₄), -C(CH₃)=N-(3-Cl-C₆H₄), -C(CH₃)=N-(4-Cl-C₆H₄), -C(CH₃)=N-(2-CH₃-C₆H₄), -C(CH₃)=N-(3-CH₃-C₆H₄), -C(CH₃)=N-(4-CH₃-C₆H₄), -C(CH₃)=N-(2-CF₃-C₆H₄), -C(CH₃)=N-(3-CF₃-C₆H₄), -C(CH₃)=N-(4-CF₃-C₆H₄), -C(CH₃)=N-(2-OCH₃-C₆H₄), -C(CH₃)=N-(3-OCH₃-C₆H₄), -C(CH₃)=N-(4-OCH₃-C₆H₄), -C(CH₃)=N-(4-NO₂-C₆H₄), -C(CH₃)=N-(4-CN-C₆H₄), -C(CH₃)=N-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-(2,4-(CH₃)₂-C₆H₃), -C(CH₃)=N-CH₂-OCH₃, -C(CH₃)=N-CH₂-OC₂H₅, -C(CH₃)=N-CH₂CH₂-OCH₃, -C(CH₃)=N-CH₂CH-OC₂H₅, -C(CH₃)=N-OH, -C(CH₃)=N-OCH₃, -C(CH₃)=N-OC₂H₅, -C(CH₃)=N-O-n-C₃H₇, -C(CH₃)=N-O-i-C₃H₇, -C(CH₃)=N-O-n-C₄H₉, -C(CH₃)=N-O-i-C₄H₉, -C(CH₃)=N-O-s-C₄H₉, -C(CH₃)=N-O-tert.-C₄H₉, -C(CH₃)=N-OCH₂-CH=CH₂, -C(CH₃)=N-OCH(CH₃)-CH=CH₂, -C(CH₃)=N-OCH₂-C≡CH, -C(CH₃)=N-CH(CH₃)-C≡CH, -C(CH₃)=N-OCH₂-CH=C-CH₃, -C(CH₃)=N-OCH₂CH₂-Cl, -C(CH₃)=N-OCH₂CH₂-F, -C(CH₃)=N-OCH₂-CF₃, -C(CH₃)=N-OCH₂-CH=CHCl, -C(CH₃)=N-OCH₂-C(Cl)=CH₂, -C(CH₃)=N-OCH₂-C(Br)=CH₂, -C(CH₃)=N-OCH₂-CH=C(Cl)-CH₃, -C(CH₃)=N-O-CO-CH₃, -C(CH₃)=N-O-CO-C₂H₅, -C(CH₃)=N-OCH₂-CN, -C(CH₃)=N-OCH₂-CH=CH-CH₂-OCH₃, -C(CH₃)=N-OCH₂-CH=CH-CH₂-O-tert.-C₄H₉, -C(CH₃)=N-O-(CH₂)₃-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-(4-Cl-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-C₆H₅, -C(CH₃)=N-OCH₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(3-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-CH₂-(4-CH₃O-C₆H₄), -C(CH₃)=N-OCH₂-CH=C(CH₃)-C₆H₅, -C(CH₃)=N-O-(CH₂)₂-CH=CH-(3,4-Cl₂-C₆H₃), -C(CH₃)=N-O-(CH₂)₃-C≡C-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-OCH₃, -C(CH₃)=N-OCH₂CH₂-OCH₃, -C(CH₃)=N-OCH₂-OC₂H₅, -C(CH₃)=N-OCH(CH₃)-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=N-NH₂, -C(CH₃)=N-NH-CH₃, -C(CH₃)=N-NH-C₂H₅, -C(CH₃)=N-NH-n-C₃H₇, -C(CH₃)=N-NH-i-C₃H₇, -C(CH₃)=N-NH-n-C₄H₉, -C(CH₃)=N-NH-i-C₄H₉, -C(CH₃)=N-NH-s-C₄H₉, -C(CH₃)=N-NH-tert.-C₄H₉, -C(CH₃)=N-NH-cyclopropyl, -C(CH₃)=N-NH-cyclobutyl, -C(CH₃)=N-NH-cyclopentyl, -C(CH₃)=N-NH-cyclohexyl, -C(CH₃)=N-NH-cycloheptyl, -C(CH₃)=N-N(CH₃)₂, -C(CH₃)=N-N(C₂H₅)₂, -C(CH₃)=N-N(n-C₃H₇)₂, -C(CH₃)=N-N(i-C₃H₇)₂, -C(CH₃)=N-NH-CH₂-C=CH, -C(CH₃)=N-NH-CH₂-C≡CH, -C(CH₃)=N-N(CH₃)-CH₂-C≡CH, -C(CH₃)=N-NH-CH₂CF₃, -C(CH₃)=N-NH-CO-CH₃, -C(CH₃)=N-NH-CO-C₂H₅, -C(CH₃)=N-NH-CO-OCH₃, -C(CH₃)=N-NH-CO-OC₂H₅, -C(CH₃)=N-NH-CO-O-tert.-C₄H₉, -C(CH₃)=N-pyrrolidin-1-yl, -C(CH₃)=N-piperidin-1-yl, -C(CH₃)=N-morpholin-4-yl, -C(CH₃)=N-NH-C₆H₅, -C(CH₃)=N-NH-(4-Cl-C₆H₄), -C(CH₃)=N-NH-(4-NO₂-C₆H₄), -C(CH₃)=N-NH-(4-F-C₆H₄), -C(CH₃)=N-NH-(4-CH₃O-C₆H₄), -C(CH₃)=N-NH-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-NH-(2,4-(NO₂)₂-C₆H₃), -C(CH₃)=N-NH-CO-NH₂, -C(CH₃)=N-NH-CO-NHCH₃, -C(CH₃)=N-NH-CO-NHC₂H₅, -C(CH₃)=N-NH-CO-N(CH₃)₂, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=CH-CO-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-O-n-C₄H₉, -C(CH₃)=CH-CO-O-tert.-C₄H₉, -C(CH₃)=CH-CO-O-cyclopropyl, -C(CH₃)=CH-CO-O-cyclobutyl, -C(CH₃)=CH-CO-O-cyclopentyl, -C(CH₃)=CH-CO-O-cyclohexyl, -C(CH₃)=CH-CO-O-cycloheptyl, -C(CH₃)=C(CH₃)-COOH, -C(CH₃)=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-cyclopropyl, -C(CH₃)=C(CH₃)-CO-O-cyclobutyl, -C(CH₃)=C(CH₃)-CO-O-cyclopentyl, -C(CH₃)=C(CH₃)-CO-O-cyclohexyl, -C(CH₃)=C(CH₃)-CO-O-cycloheptyl, -C(CH₃)=C(C₂H₅)-COOH, -C(CH₃)=C(C₂H₅)-CO-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-cyclo­ propyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-O- cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-O-cycloheptyl, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=C(Cl)-CO-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-O-n-C₄H₉, -C(CH₃)=C(Cl)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-O-cyclopropyl, -C(CH₃)=C(Cl)-CO-O-cyclobutyl, -C(CH₃)=C(Cl)-CO-O-cyclopentyl, -C(CH₃)=C(Cl)-CO-O-cyclohexyl, -C(CH₃)=C(Cl)-CO-O-cycloheptyl, -C(CH₃)=C(Br)-COOH, -C(CH₃)=C(Br)-CO-OCH₃, -C(CH₃)=C(Br)-CO-OC₂H₅, -C(CH₃)=C(Br)-CO-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-O-n-C₄H₉, -C(CH₃)=C(Br)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-O-cyclopropyl, -C(CH₃)=C(Br)-CO-O-cyclobutyl, -C(CH₃)=C(Br)-CO-O-cyclopentyl, -C(CH₃)=C(Br)-CO-O-cyclohexyl, -C(CH₃)=C(Br)-CO-O-cycloheptyl, -C(CH₃)=C(CN)-COOH, -C(CH₃)=C(CN)-CO-OCH₃, -C(CH₃)=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CN)-CO-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-O-n-C₄H₉, -C(CH₃)=C(CN)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-O-cyclopropyl, -C(CH₃)=C(CN)-CO-O-cyclobutyl, -C(CH₃)=C(CN)-CO-O-cyclopentyl, -C(CH₃)=C(CN)-CO-O-cyclohexyl, -C(CH₃)=C(CN)-CO-O-cycloheptyl, -C(CH₃)=CH-CO-OCH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-OCH(CH₃)-OCH₃, -C(CH₃)=CH-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=CH-CO-OCH₂CH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=(C₂H₅)-CO-OCH₂CH₂-OCH₃, -(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-O-i-C₃H₇, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-O-i-C₃H₇, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-O-i-C₃H₇, -C(CH₃)=C(CN)-CO-OCH(CH₃)OCH₃, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-CF₃, -C(CH₃)=CH-CO-OCH₂-CCl₃, -C(CH₃)=CH-CO-OCH₂-oxiranyl, -C(CH₃)=CH-CO-(CH₂)₃-Br, -C(CH₃)=CH-CO-OCH₂-CH=CH₂, -C(CH₃)=CH-CO-OCH₂-C≡CH, -C(CH₃)=CH-CO-OCH₂-CN, -C(CH₃)=CH-CO-OCH₂CH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CF₃, -C(CH₃)=C(CH₃)-CO-OCH₂-CCl₃, -C(CH₃)=C(CH₃)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CH₃)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CH₃)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CH₃)-CO-OCH₂-C≡CH, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CF₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CCl₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-oxiranyl, -C(CH₃)=C(C₂H₅)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(C₂H₅)CO-OCH₂-C≡CH, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂-CF₃, -C(CH₃)=C(Cl)-CO-OCH₂-CCl₃, -C(CH₃)=C(Cl)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Cl)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Cl)-CO-OCH₂-CH≡CH₂, -C(CH₃)=C(Cl)-CO-OCH₂-C≡CH, -C(CH₃)=C(Cl)-CO-OCH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂-CF₃, -C(CH₃)=C(Br)-CO-OCH₂-CCl₃, -C(CH₃)=C(Br)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Br)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Br)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Br)-CO-OCH₂-C≡CH, -C(CH₃)=C(Br)-CO-OCH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂CH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂-CF₃, -C(CH₃)=C(CN)-CO-OCH₂-CCl₃, -C(CH₃)=C(CN)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CN)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(CN)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CN)-CO-OCH₂-C≡CH, -C(CH₃)=C(CN)-CO-OCH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂CH₂-CN, -C(CH₃)=CH-CO-CH₃, -C(CH₃)=CH-CO-C₂H₅, -C(CH₃)=CH-CO-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-n-C₄H₉, -C(CH₃)=CH-CO-tert.-C₄H₉, -C(CH₃)=CH-CO-CH₂Cl, -C(CH₃)=CH-CO-CH₂Br, -C(CH₃)=CH-CO-CHCl₂, -C(CH₃)=CH-CO-CH₂-OCH₃, -C(CH₃)=CH-CO-CH(OCH₃)₂, -C(CH₃)=CH-CO-CH₂-SCH₃, -C(CH₃)=C(CH₃)-CO-CH₃, -C(CH₃)=C(CH₃)-CO-C₂H₅, -C(CH₃)=C(CH₃)-CO-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-CH₂Cl, -C(CH₃)=C(CH₃)-CO-CH₂Br, äC(CH₃)=C(CH₃)-CO-CHCl₂, -C(CH₃)=C(CH₃)-CO-CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-CH(OCH₃)₂, -C(CH₃)=C(CH₃)-CO-CH₂-SCH₃, -C(CH₃)=C(C₂H₅)-CO-CH₃, -C(CH₃)=C(C₂H₅)-CO-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-CH₂Cl, -C(CH₃)=C(C₂H₅)-CO-CH₂Br, -C(CH₃)=C(C₂H₅)-CO-CHCl₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-CH(OCH₃)₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-SCH₃, -C(CH₃)=C(Cl)-CO-CH₃, -C(CH₃)=C(Cl)-CO-C₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-n-C₄H₉, -C(CH₃)=C(Cl)-CO-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-CH₂Cl, -C(CH₃)=C(Cl)-CO-CHCl₂, -C(CH₃)=C(Cl)-CO-CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-CH(OCH₃)₂, -C(CH₃)=C(Cl)-CO-CH₂-SCH₃, -C(CH₃)=C(Br)-CO-CH₃, -C(CH₃)=C(Br)-CO-C₂H₅, -C(CH₃)=C(Br)-CO-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-n-C₄H₉, -C(CH₃)=C(Br)-CO-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-CH₂Cl, -C(CH₃)=C(Br)-CO-CH₂Br, -C(CH₃)=C(Br)-CO-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-CH(OCH₃)₂, -C(CH₃)=C(Br)-CO-CH₂-SCH₃, -C(CH₃)=C(CN)-CO-CH₃, -C(CH₃)=C(CN)-CO-C₂H₅, -C(CH₃)=C(CN)-CO-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-n-C₄H₉, -C(CH₃)=C(CN)-CO-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-CH₂Cl, -C(CH₃)=C(CN)-CO-CH₂Br, -C(CH₃)=C(CN)-CO-CHCl₂, -C(CH₃)=C(CN)-CO-CH₂-OCH₃, -C(CH₃)=C(CN)-CO-CH(OCH₃)₂, -C(CH₃)=C(CN)-CO-CH₂-SCH₃, -C(CH₃)=CH-CO-C₆H₅, -C(CH₃)=CH-CO-(4-Cl-C₆H₄), -C(CH₃)=C(CH₃)-CO-C₆H₅, -C(CH₃)=C(CH₃)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(C₂H₅)-CO-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(Cl)-CO-C₆H₅, -C(CH₃)=C(Br)-CO-C₆H₅, -C(CH₃)=C(CN)-CO-C₆H₅, -C(CH₃)=CH-CO-NH₂, -C(CH₃)=CH-CO-NHCH₃, -C(CH₃)=CH-CO-N(CH₃)₂, -C(CH₃)=CH-CO-NH-C₂H₅, -C(CH₃)=CH-CO-N(C₂H₅)₂, -C(CH₃)=CH-CO-NH-n-C₃H₇, -C(CH₃)=CH-CO-NH-i-C₃H₇, -C(CH₃)=CH-CO-NH-tert.-C₄H₉, -C(CH₃)=CH-CO-NH-cyclopropyl, -C(CH₃)=CH-CO-NH-cyclobutyl, -C(CH₃)=CH-CO-NH-cyclopentyl, -C(CH₃)=CH-CO-NH-cyclohexyl, -C(CH₃)=CH-CO-NH-cycloheptyl, -C(CH₃)=CH-CO-NH-cyclooctyl, -C(CH₃)=CH-CO-pyrrolidin-1-yl, -C(CH₃)=CH-CO-piperidin-1-yl, -C(CH₃)=CH-CO-morpholin-4-yl, -C(CH₃)=CH-CO-NH-CH₂CH=CH₂, -C(CH₃)=CH-CO-NH-CH₂C≡CH, -C(CH₃)=CH-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=CH-CO-NH-(CH₂)₂Cl, -C(CH₃)=CH-CO-NH-C₆H₅, -C(CH₃)=C(CH₃)-CO-NH₂, -C(CH₃)=C(CH₃)-CO-NHCH₃, -C(CH₃)=C(CH₃)-CO-N(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-C₂H₅, -C(CH₃)=C(CH₃)-CO-N(C₂H₅)₂, -C(CH₃)=C(CH₃)-CO-NH-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-NH- cyclopropyl, -C(CH₃)=C(CH₃)-CO-NH-cyclobutyl, -C(CH₃)=C(CH₃)-CO-NH-cyclopentyl, -C(CH₃)=C(CH₃)-CO-NH- cyclohexyl, -C(CH₃)=C(CH₃)-CO-NH-cycloheptyl, -C(CH₃)=C(CH₃)-CO-NH-cyclooctyl, -C(CH₃)=C(CH₃)-CO- pyrrolidin-1-yl, -C(CH₃)=C(CH₃)-CO-piperidin-1-yl, -C(CH₃)=C(CH₃)-CO-morpholin-4-yl, -C(CH₃)=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-NH(CH₂)₂Cl, -C(CH₃)=C(CH₃)-CO-NH-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-NH₂, -C(CH₃)=C(C₂H₅)-CO-NHCH₃, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)₂, -C(CH₃)=C(C₂H₅)-CO-NH-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-N(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-NH- cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclo­ hexyl, -C(CH₃)=C(C₂H₅)-CO-NH-cycloheptyl, -C(CH₃)=C(C₂H₅)-CO-NH- cyclooctyl, -C(CH₃)=C(C₂H₅)-CO-pyrrolidin-1-yl, -C(CH₃)=C(C₂H₅)-CO-piperidin-1-yl, -C(CH₃)=C(C₂H₅)-CO- morpholin-4-yl, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(C₂H₅)-CO-NH-C₆H₅, -C(CH₃)=C(Cl)-CO-NH₂, -C(CH₃)=C(Cl)-CO-NHCH₃, -C(CH₃)=C(Cl)-CO-N(CH₃)₂, -C(CH₃)=C(Cl)-CO-NH-C₂H₅, -C(CH₃)=C(Cl)-CO-N(C₂H₅)₂, -C(CH₃)=C(Cl)-CO-NH-n-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-i-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-NH-cyclopropyl, -C(CH₃)=C(Cl)-CO-NH-cyclobutyl, -C(CH₃)=C(Cl)-CO-NH-cyclopentyl, -C(CH₃)=C(Cl)-CO-NH-cyclohexyl, -C(CH₃)=C(Cl)-CO-NH-cycloheptyl, -C(CH₃)=C(Cl)-CO-NH-cyclooctyl, -C(CH₃)=C(Cl)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Cl)-CO-piperidin-1- yl, -C(CH₃)=C(Cl)-CO-morpholin-4-yl, -C(CH₃)=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -C(CH₃)≡C(Cl)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-N(CH₃)-CH₂≡CH, -C(CH₃)=C(Cl)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Cl)-NO-NH-C₆H₅, -C(CH₃)=C(Br)-CO-NH₂, -C(CH₃)=C(Br)-CO-NHCH₃, -C(CH₃)=C(Br)-CO-N(CH₃)₂, -C(CH₃)=C(Br)-CO-NH-C₂H₅, -C(CH₃)=C(Br)-CO-N(C₂H₅)₂, -C(CH₃)=C(Br)-CO-NH-n-C₃H₇, -C(CH₃)=C(Br)-CO-NH-i-C₃H₇, -C(CH₃)=C(Br)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-NH-cyclopropyl, -C(CH₃)=C(Br)-CO-NH-cyclobutyl, -C(CH₃)=C(Br)-CO-NH-cyclopentyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cyclooctyl, -C(CH₃)=C(Br)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Br)-CO-piperidin-1-yl, -C(CH₃)=C(Br)-CO-morpholin-4-yl, -C(CH₃)=C(Br)-CO-NH-CH₂CH=C(Br)₂, -C(CH₃)=C(Br)-CO-NH-CH₂≡CH, -C(CH₃)=C(Br)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Br)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Br)-CO-NH-C₆H₅, -C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CN)-CO-NHCH₃, -C(CH₃)=C(CN)-CO-N(CH₃)₂, -C(CH₃)=C(CN)-CO-NH-C₂H₅, -C(CH₃)=C(CN)-CO-N(C₂H₅)₂, -C(CH₃)=C(CN)-CO-NH-n-C₃H₇, -C(CH₃)=C(CN)-CO-NH-i-C₃H₇, -C(CH₃)=C(CN)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-NH-cyclopropyl, -C(CH₃)=C(CN)-CO-NH-cyclobutyl, -C(CH₃)=C(CN)-CO-NH-cyclopentyl, -C(CH₃)=C(CN)-CO-NH-cyclohexyl, -C(CH₃)=C(CN)-CO-NH-cycloheptyl, -C(CH₃)=C(CN)-CO-NH-cyclooctyl, -C(CH₃)=C(CN)-CO-pyrrolidin-1-yl, -C(CH₃)=C(CN)-CO-piperidin-1-yl, -C(CH₃)=C(CN)-CO-morpholin-4-yl, -C(CH₃)=C(CN)-CO-NH-CH₂CH=C(CN)₂, -C(CH₃)=C(CN)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CN)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CN)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CN)-CO-NH-C₆H₅, -C(CH₃)=CH-CO-SCH₃, -C(CH₃)=CH-CO-SC₂H₅, -C(CH₃)=CH-CO-S-n-C₃H₇, -C(CH₃)=CH-CO-S-i-C₃H₇, -C(CH₃)=CH-CO-S-n-C₄H₉, -C(CH₃)=CH-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-SCH₃, -C(CH₃)=C(CH₃)-CO-SC₂H₅, -C(CH₃)=C(CH₃)-CO-S-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-S-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-SCH₃, -C(CH₃)=C(C₂H₅)-CO-SC₂H₅, -C(CH₃)=C(C₂H₅)-CO-S-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-SCH₃, -C(CH₃)=C(Cl)-CO-SC₂H₅, -C(CH₃)=C(Cl)-CO-S-n-C₃H₇, -C(CH₃)=C(Cl)-CO-S-i-C₃H₇, -C(CH₃)=C(Cl)-CO-S-n-C₄H₉, -C(CH₃)=C(Cl)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-SCH₃, -C(CH₃)=C(Br)-CO-SC₂H₅, -C(CH₃)=C(Br)-CO-S-n-C₃H₇, -C(CH₃)=C(Br)-CO-S-i-C₃H₇, -C(CH₃)=C(Br)-CO-S-n-C₄H₉, -C(CH₃)=C(Br)-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH)-CO-SCH₃, -C(CH₃)=C(CN)-CO-SC₂H₅, -C(CH₃)=C(CH)-CO-S-n-C₃H₇, -C(CH₃)=C(CN)-CO-S-i-C₃H₇, -C(CH₃)=C(CN)-CO-S-n-C₄H₉, -C(CH₃)=C(CN)-CO-S-tert.-C₄H₉, -C(CH₃)=C(COCH₃)-CO-OCH₃, -C(CH₃)=C(COC₂H₅)-CO-OCH₃, -C(CH₃)=C(CO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COCH₃)-CO-OC₂H₅, -C(CH₃)=C(COC₂H₅)-CO-OC₂H₅, -C(CH₃)=C(CO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COCH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(COC₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-OCH₃, -C(CH₃)=C(CF₃)-CO-OC₂H₅, -C(CH₃)=C(CF₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CF₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(COOCH₃)₂, -C(CH₃)=C(COOC₂H₅)₂, -C(CH₃)=C(COOCH₃)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)₂, -C(CH₃)=CH-CH=CH-COOH, -C(CH₃)=CH-CH=CH-CO-OCH₃, -C(CH₃)=CH-CH=CH-CO-OC₂H₅, -C(CH₃)=CH-CH=C(COOCH₃)₂, -C(CH₃)=CH-CH=C(CN)-CO-OCH₃, -C(CH₃)=CH-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH₂, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -C(CH₃)=CH-(CH₂)₂-COOH, -C(CH₃)=CH-(CH₂)₂-CO-OCH₃, -C(CH₃)=CH-(CH₂)₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(COOCH₃)₂, -C(CH₃)=CH-CH₂-CH(COOC₂H₅)₂, -C(CH₃)=CH-CH₂-CH(CN)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CN)-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -C(CH₃)=CH-(CH₂)₂-CO-NH₂, -C(CH₃)=CH-(CH₂)₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-COOH, -C(CH₃)=CH-CH₂-CO-OCH₃, -C(CH₃)=CH-CH₂-CO-OC₂H₅, -C(CH₃)=C(COOCH₃)-CH₂-CO-OCH₃, -C(CH₃)=C(COOCH₃)-CH₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CO-NH₂, -C(CH₃)=CH-CH₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-CO-N(CH₃)₂.
wobei W für eine der folgenden Bedeutungen steht:
-CHO, -COCH₃, -COC₂H₅, -CO-n-C₃H₇, -CO-i-C₃H₇, -CO-n-C₄H₉, -CO-i-C₄H₉, -CO-s-C₄H₉, -CO-tert.-C₄H₉, -CO-CH₂CH=CH₂, -CO-CF₃, -COCCl₃, -COCH₂C≡CH, -CO-cyclopropyl, -CO-cyclobutyl, -CO-cyclopentyl, -CO-cyclohexyl, -CO-CN, -CO-COOCH₃, -CO-COOC₂H₅, -CH=NH, -CH=NCH₃, -CH=NC₂H₅, -CH=N-n-C₃H₅, -CH=N-i-C₃H₅, -CH=N-n-C₄H₉, -CH=NCH₂CH=CH₂, -CH=NCH₂CH=CH₂-CH₃, -CH=NCH₂C≡CH, -CH=NCH₂C≡C-CH₃, -CH=N-cyclopropyl, -CH=N-cyclobutyl, -CH=N-cyclopentyl, -CH=N-cyclohexyl, -CH=N-cycloheptyl, -CH=N-CH₂-CH₂Cl, -CH=N-CH₂Cl, -CH=N-C₆H₅, -CH=N-4-Br-C₆H₄, -CH=N-3-F-C₆H₄, -CH=N-4-F-C₆H₄, -CH=N-2-Cl-C₆H₄, -CH=N-3-Cl-C₆H₄, -CH=N-4-Cl-C₆H₄, -CH=N-2-Br-C₆H₄, -CH=N-2-F-C₆H₄, -CH=N-2-CH₃-C₆H₄, -CH=N-3-CH₃-C₆H₄, -CH=N-4-CH₃-C₆H₄, -CH=N-2-CF₃-C₆H₄, -CH=N-3-CF₃-C₆H₄, -CH=N-4-CF₃-C₆H₄, -CH=N-2-OCH₃-C₆H₄, -CH=N-3-OCH₃-C₆H₄, -CH=N-4-OCH₃-C₆H₄, -CH=N-4-NO₂-C₆H₄, -CH=N-4-CN-C₆H₄, -CH=N-2,4-(Cl,Cl)-C₆H₄, -CH=N-2,4-(CH₃,CH₃)-C₆H₄, -CH=N-CH₂OCH₃, -CH=N-CH₂OC₂H₅, -CH=N-CH₂CH₂OCH₃, -CH=N-CH₂CH₂OC₂H₅, -CH=N-OH, -CH=N-OCH₃, -CH=N-OC₂H₅, -CH=N-O-n-C₃H₇, -CH=N-O-i-C₃H₇, -CH=N-O-n-C₄H₉, -CH=N-O-i-C₄H₉, -CH=N-O-s-C₄H₉, -CH=N-O-tert.-C₄H₉, -CH=N-O-CH₂CH=CH₂, -CH=N-O-CH(CH₃)CH=CH₂, -CH=N-O-CH₂C≡CH, -CH=N-O-CH(CH₃)-C≡CH, -CH=N-O-CH₂-CH=CH-CH₃, -CH=N-O-CH₂-CH₂-Cl, -CH=N-O-CH₂-CH₂-F, -CH=N-O-CH₂-CF₃, -CH=N-O-CH₂-CH=CHCl, -CH=N-O-CH₂-CCl=CH₂, -CH=N-O-CH₂-CBr=CH₂, -CH=N-O-CH₂-CH=CCl-CH₃, -CH=N-OC(O)CH₃, -CH=N-OC(O)C₂H₅, -CH=N-O-CH₂-CN, -CH=N-O-CH₂-CH=CH-CH₂-O-CH₃, -CH=N-O-CH₂-CH=CH-CH₂-O-tert.-C₄H₉, -CH=N-O-(CH₂)₃-C₆H₅, -CH=N-O-(CH₂)₄-C₆H₅, -CH=N-O-(CH₂)₄-4-Cl-C₆H₄, -CH=N-O-(CH₂)₄-4-OCH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-CH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-C₆H₅, -CH=N-O-CH₂CH=CH-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CH-3-OCH₃-C₆H₄, -CH=N-O-(CH₂)₂CH=CH-4-F-C₆H₄, -CH=N-O-(CH₂)CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CHCH₂-4-OCH₃-C₆H₄, -CH=N-O-CH₂-CH=C(CH₃)-C₆H₅, -CH=N-O-(CH₂)₂CH=CH-3,4(Cl,Cl)-C₆H₃, -CH=N-O-(CH₂)₃C≡C-4-F-C₆H₄, -CH₂=N-OCHOCH₃, -CH=N-OC₂H₄OCH₃, -CH=N-OCH₂OC₂H₅, -CH=N-OCH(CH₃)OCH₃, -CH=N-OCH(CH₃)COOCH₃, -CH=N-OCH(CH₃)COO-n-C₄H₉, -CH=N-NH₂, -CH=N-NHCH₃, -CH=N-NHC₂H₅, -CH=N-NH-n-C₃H₇, -CH=N-NH-i-C₃H₇, -CH=N-NH-n-C₄H₉, -CH=N-NH-i-C₄H₉, -CH=N-NH-s-C₄H₉, -CH=N-NH-tert.-C₄H₉, -CH=N-NH-cyclopropyl, -CH=N-NH-cyclobutyl, -CH=N-NH-cyclopentyl, -CH=N-NH-cyclohexyl, -CH=N-NH-cycloheptyl, -CH=N-N(CH₃)₂, -CH=N-N(C₂H₅)₂, -CH=N-N(C₃H₇)₂, -CH=N-N(i-C₃H₇)(CH₃), -CH=N-NHCH₂-C=CH, -CH=N-NHCH₂-C≡CH, -CH=N-N(CH₃)-CH₂-C≡CH, -CH=N-NHCH₂CF₃, -CH=N-NH-CO-CH₃, -CH=N-NH-CO-CH₂H₅, -CH=N-NH-COOCH₃, -CH=N-NH-COOC₂H₅, -CH=N-NH-COO-tert.-C₄H₉, -CH=N-pyrrolidin-1-yl, -CH=N-piperidin-1-yl, -CH=N-morpholin-4-yl, -CH=N-NH-C₆H₅, -CH=N-NH-(4-Cl-C₆H₄), -CH=N-NH-(4-NO₂-C₆H₄), -CH=N-NH-(4-F-C₆H₄), -CH=N-NH-(4-CH₃O-C₆H₄), -CH=N-NH-(2,4-Cl₂-C₆H₃), -CH=N-NH-(2,4-(NO₂)₂-C₆H₃), -CH=N-NH-CO-NH₂, -CH=N-NH-CO-NHCH₃, -CH=N-NH-CO-NHC₂H₅, -CH=N-NH-CO-N(CH₃)₂, -CH=CH-COOH, -CH=CH-CO-OCH₃, -CH=C-CO-OC₂H₅, -CH=CH-CO-O-n-C₃H₇, -CH=CH-CO-O-i-C₃H₇, -CH=CH-CO-O-n-C₄H₉, -CH=CH-CO-O-tert.-C₄H₉, -CH=CH-CO-O-cyclopropyl, -CH=CH-CO-O-cyclobutyl, -CH=CH-CO-O-cyclopentyl, -CH=CH-CO-O-cyclohexyl, -CH=CH-CO-O-cycloheptyl, -CH=C(CH₃)-COOH, -CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CO-O-n-C₃H₇, -CH=C(CH₃)-CO-O-i-C₃H₇, -CH=C(CH₃)-CO-O-n-C₄H₉, -CH=C(CH₃)-CO-O-tert.-C₄H₉, -CH=C(CH₃)-CO-O-cyclopropyl, -CH=C(CH₃)-CO-O-cyclobutyl, -CH=C(CH₃)-CO-O-cyclopentyl, -CH=C(CH₃)-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cycloheptyl, -CH=C(C₂H₅)-COOH, -CH=C(C₂H₅)-CO-OCH₃, -CH=C(C₂H₅)-CO-OC₂H₅, -CH=C(C₂H₅)-CO-O-n-C₃H₇, -CH=C(C₂H₅)-CO-O-i-C₃H₇, -CH=C(C₂H₅)-CO-O-n-C₄H₉, -CH=C(C₂H₅)-CO-O-tert.-C₄H₉, -CH=C(C₂H₅)-CO-O-cyclopropyl, -CH=C(C₂H₅)-CO-O-cyclobutyl, -CH=C(C₂H₅)-CO-O-cyclopentyl, -CH=C(C₂H₅)-CO-O-cyclohexyl, -CH=C(C₂H₅)-CO-O-cycloheptyl, -CH=C(Cl)-COOH, -CH=C(Cl)-CO-OCH₃, -CH=C(Cl)-CO-OC₂H₅, -CH=C(Cl)-CO-O-n-C₃H₇, -CH=C(Cl)-CO-O-i-C₃H₇, -CH=C(Cl)-CO-O-n-C₄H₉, -CH=C(Cl)-CO-O-tert.-C₄H₉, -CH=C(Cl)-CO-O-cyclopropyl, -CH=C(Cl)-CO-O-cyclobutyl, -CH=C(Cl)-CO-O-cyclopentyl, -CH=C(Cl)-CO-O-cyclohexyl, -CH=C(Cl)-CO-O-cycloheptyl, -CH=C(Br)-COOH, -CH=C(Br)-CO-OCH₃, -CH=C(Br)-CO-OC₂H₅, -CH=C(Br)-CO-O-n-C₃H₇, -CH=C(Br)-CO-O-i-C₃H₇, -CH=C(Br)-CO-O-n-C₄H₉, -CH=C(Br)-CO-O-tert.-C₄H₉, -CH=C(Br)-CO-O-cyclopropyl, -CH=C(Br)-CO-O-cyclobutyl, -CH=C(Br)-CO-O-cyclopentyl, -CH=C(Br)-CO-O-cyclohexyl, -CH=C(Br)-CO-O-cycloheptyl, -CH=C(CN)-COOH, -CH=C(CN)-CO-OCH₃, -CH=C(CN)-CO-OC₂H₅, -CH=C(CN)-CO-O-n-C₃H₇, -CH=C(CN)-CO-O-i-C₃H₇, -CH=C(CN)-CO-O-n-C₄H₉, -CH=C(CN)-CO-O-tert.-C₄H₉, -CH=C(CN)-CO-O-cyclopropyl, -CH=C(CN)-CO-O-cyclobutyl, -CH=C(CN)-CO-O-cyclopentyl, -CH=C(CN)-CO-O-cyclohexyl, -CH=C(CN)-CO-O-cycloheptyl, -CH=CH-CO-OCH₂-OCH₃, -CH=CH-CO-OCH₂-OC₂H₅, -CH=CH-CO-OCH₂-O-n-C₃H₅, -CH=CH-CO-OCH₂-O-i-C₃H₅, -CH=CH-CO-OCH(CH₃)-OCH₃, -CH=CH-CO-OCH(CH₃)-OC₂H₅, -CH=CH-CO-O-CH₂CH₂-OCH₃, -CH=CH-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-OCH₃, -CH=C(CH₃)-CO-OCH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-O-n-C₃H₅, -CH=C(CH₃)-CO-OCH₂-O-i-C₃H₅, -CH=C(CH₃)-CO-OCH(CH₃)-OCH₃, -CH=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CH₃)-CO-O-CH₂CH₂-OCH₃, -CH=C(CH₃)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-OCH₃, -CH=C(C₂H₅)-CO-OCH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-O-n-C₃H₅, -CH=C(C₂H₅)-CO-OCH₂-O-i-C₃H₅, -CH=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -CH=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OCH₃, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-OCH₃, -CH=C(Cl)-CO-OCH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-O-n-C₃H₅, -CH=C(Cl)-CO-OCH₂-O-i-C₃H₅, -CH=C(Cl)-CO-OCH(CH₃)-OCH₃, -CH=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Cl)-CO-O-CH₂CH₂-OCH₃, -CH=C(Cl)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-OCH₃, -CH=C(Br)-CO-OCH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-O-n-C₃H₅, -CH=C(Br)-CO-OCH₂-O-i-C₃H₅, -CH=C(Br)-CO-OCH(CH₃)-OCH₃, -CH=C(Br)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Br)-CO-O-CH₂CH₂-OCH₃, -CH=C(Br)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-OCH₃, -CH=C(CN)-CO-OCH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-O-n-C₃H₅, -CH=C(CN)-CO-OCH₂-O-i-C₃H₅, -CH=C(CN)-CO-OCH(CH₃)-OCH₃, -CH=C(CN)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CN)-CO-O-CH₂CH₂-OCH₃, -CH=C(CN)-CO-O-CH₂CH₂-OC₂H₅, -CH=CH-CO-OCH₂-CF₃, -CH=CH-CO-OCH₂-CCl₃, -CH=CH-CO-OCH₂-oxiranyl, -CH=CH-CO-O(CH₂)₃-Br, -CH=CH-CO-OCH₂-CH=CH₂, -CH=CH-CO-OCH₂-C≡CH, -CH=CH-CO-OCH₂-CN, -CH=CH-CO-O(CH₂)₂-CN, -CH=C(CH₃)-CO-OCH₂-CF₃, -CH=C(CH₃)-CO-OCH₂-CCl₃, -CH=C(CH₃)-CO-OCH₂-oxiranyl, -CH=C(CH₃)-CO-O(CH₂)₃-Br, -CH=C(CH₃)-CO-OCH₂-CH=CH₂, -CH=C(CH₃)-CO-OCH₂-C≡CH, -CH=C(CH₃)-CO-OCH₂-CN, -CH=C(CH₃)-CO-O(CH₂)₂-CN, -CH=C(C₂H₅)-CO-OCH₂-CF₃, -CH=C(C₂H₅)-CO-OCH₂-CCl₃, -CH=C(C₂H₅)-CO-OCH₂-oxiranyl, -CH=C(C₂H₅)-CO-O(CH₂)₃-Br, -CH=C(C₂H₅)-CO-OCH₂-CH=CH₂, -CH=C(C₂H₅)-CO-OCH₂-C≡CH, -CH=C(C₂H₅)-CO-OCH₂-CN, -CH=C(C₂H₅)-CO-O(CH₂)₂-CN, -CH=C(Cl)-CO-OCH₂-CF₃, -CH=C(Cl)-CO-OCH₂-CCl₃, -CH=C(Cl)-CO-OCH₂-oxiranyl, -CH=C(Cl)-CO-O(CH₂)₃-Br, -CH=C(Cl)-CO-OCH₂-CH=CH₂, -CH=C(Cl)-CO-OCH₂-C≡CH, -CH=C(Cl)-CO-OCH₂-CN, -CH=C(Cl)-CO-O(CH₂)₂-CN, -CH=C(Br)-CO-OCH₂-CF₃, -CH=C(Br)-CO-OCH₂-CCl₃, -CH=C(Br)-CO-OCH₂-oxiranyl, -CH=C(Br)-CO-O(CH₂)₃-Br, -CH=C(Br)-CO-OCH₂-CH=CH₂, -CH=C(Br)-CO-OCH₂-C≡CH, -CH=C(Br)-CO-OCH₂-CN, -CH=C(Br)-CO-O(CH₂)₂-CN, -CH=C(CN)-CO-OCH₂-CF₃, -CH=C(CN)-CO-OCH₂-CCl₃, -CH=C(CN)-CO-OCH₂-oxiranyl, -CH=C(CN)-CO-O(CH₂)₃-Br, -CH=C(CN)-CO-OCH₂-CH=CH₂, -CH=C(CN)-CO-OCH₂-C≡CH, -CH=C(CN)-CO-OCH₂-CN, -CH=C(CN)-CO-O(CH₂)₂-CN, -CH=CH-CO-CH₃, -CH=CH-CO-C₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-i-C₃H₇, -CH=CH-CO-n-C₄H₉, -CH=CH-CO-tert.-C₄H₉, -CH=CH-CO-CH₂Cl, -CH=CH-CO-CH₂Br, -CH=CH-CO-CHCl₂, -CH=CH-CO-CH₂-OCH₃, -CH=CH-CO-CH(OCH₃)₂, -CH=CH-CO-CH₂-SCH₃, -CH=C(CH₃)-CO-CH₃, -CH=C(CH₃)-CO-C₂H₅, -CH=C(CH₃)-CO-n-C₃H₇, -CH=C(CH₃)-CO-i-C₃H₇, -CH=C(CH₃)-CO-n-C₄H₉, -CH=C(CH₃)-CO-tert.-C₄H₉, -CH=C(CH₃)-CO-CH₂Cl, -CH=C(CH₃)-CO-CH₂Br, -CH=C(CH₃)-CO-CHCl₂, -CH=C(CH₃)-CO-CH₂-OCH₃, -CH=C(CH₃)-CO-CH(OCH₃)₂, -CH=C(CH₃)-CO-CH₂-SCH₃, -CH=C(C₂H₅)-CO-CH₃, -CH=C(C₂H₅)-CO-C₂H₅, -CH=C(C₂H₅)-CO-n-C₃H₇, -CH=C(C₂H₅)-CO-i-C₃H₇, -CH=C(C₂H₅)-CO-n-C₄H₉, -CH=C(C₂H₅)-CO-tert.-C₄H₉, -CH=C(C₂H₅)-CO-CH₂Cl, -CH=C(C₂H₅)-CO-CH₂Br, -CH=C(C₂H₅)-CO-CHCl₂, -CH=C(C₂H₅)-CO-CH₂-OCH₃, -CH=C(C₂H₅)-CO-CH(OCH₃)₂, -CH=C(C₂H₅)-CO-CH₂-SCH₃, -CH=C(Cl)-CO-CH₃, -CH=C(Cl)-CO-C₂H₅, -CH=C(Cl)-CO-n-C₃H₇, -CH=C(Cl)-CO-i-C₃H₇, -CH=C(Cl)-CO-n-C₄H₉, -CH=C(Cl)-CO-tert.-C₄H₉, -CH=C(Cl)-CO-CH₂Cl, -CH=C(Cl)-CO-CH₂Br, -CH=C(Cl)-CO-CHCl₂, -CH=C(Cl)-CO-CH₂-OCH₃, -CH=C(Cl)-CO-CH(OCH₃)₂, -CH=C(Cl)-CO-CH₂-SCH₃, -CH=C(Br)-CO-CH₃, -CH=C(Br)-CO-C₂H₅, -CH=C(Br)-CO-n-C₃H₇, -CH=C(Br)-CO-i-C₃H₇, -CH=C(Br)-CO-n-C₄H₉, -CH=C(Br)-CO-tert.-C₄H₉, -CH=C(Br)-CO-CH₂Cl, -CH=C(Br)-CO-CH₂Br, -CH=C(Br)-CO-CHCl₂, -CH=C(Br)-CO-CH₂-OCH₃, -CH=C(Br)-CO-CH(OCH₃)₂, -CH=C(Br)-CO-CH₂-SCH₃, -CH=C(CN)-CO-CH₃, -CH=C(CN)-CO-C₂H₅, -CH=C(CN)-CO-n-C₃H₇, -CH=C(CN)-CO-i-C₃H₇, -CH=C(CN)-CO-n-C₄H₉, -CH=C(CN)-CO-tert.-C₄H₉, -CH=C(CN)-CO-CH₂Cl, -CH=C(CN)-CO-CH₂Br, -CH=C(CN)-CO-CHCl₂, -CH=C(CN)-CO-CH₂-OCH₃, -CH=C(CN)-CO-CH(OCH₃)₂, -CH=C(CN)-CO-CH₂-SCH₃, -CH=CH-CO-C₆H₅, -CH=CH-CO-(4-Cl-C₆H₄), -CH=C(CH₃)-CO-C₆H₅, -CH=C(CH₃)-CO-(4-Cl-C₆H₄), -CH=C(C₂H₅)-CO-C₆H₅, -CH=C(C₂H₅)-CO-(4-Cl-C₆H₄), -CH=C(Cl)-CO-C₆H₅, -CH=C(Br)-CO-C₆H₅, -CH=C(CN)-CO-C₆H₅, -CH=CH-CO-NH₂, -CH=CH-CO-NHCH₃, -CH=CH-CO-N(CH₃)₂, -CH=CH-CO-NH-C₂H₅, -CH=CH-CO-N(C₂H₅)₂, -CH=CH-CO-NH-n-C₃H₇, -CH=CH-CO-NH-i-C₃H₇, -CH=CH-CO-NH-tert.-C₄H₉, -CH=CH-CO-NH-cyclopropyl, -CH=CH-CO-NH-cyclobutyl, -CH=CH-CO-NH-cyclopentyl, -CH=CH-CO-NH-cyclohexyl, -CH=CH-CO-NH-cycloheptyl, -CH=CH-CO-NH-cyclooctyl, -CH=CH-CO-pyrrolidin-1-yl, -CH=CH-CO-piperidin-1-yl, -CH=CH-CO-morpholin-4-yl, -CH=CH-CO-NH-CH₂CH=CH₂, -CH=CH-CO-NH-CH₂C≡CH, -CH=CH-CO-N(CH₃)-CH₂C≡CH, -CH=CH-CO-NH-(CH₂)₂Cl, -CH=CH-CO-NH-C₆H₅, -CH=C(CH₃)-CO-NH₂, -CH=C(CH₃)-CO-NHCH₃, -CH=C(CH₃)-CO-N(CH₃)₂, -CH=C(CH₃)-CO-NH-C₂H₅, -CH=C(CH₃)-CO-N(C₂H₅)₂, -CH=C(CH₃)-CO-NH-n-C₃H₇, -CH=C(CH₃)-CO-NH-i-C₃H₇, -CH=C(CH₃)-CO-NH-tert.-C₄H₉, -CH=C(CH₃)-CO-NH-cyclopropyl, -CH=C(CH₃)-CO-NH-cyclobutyl, -CH=C(CH₃)-CO-NH-cyclopentyl, -CH=C(CH₃)-CO-NH-cyclohexyl, -CH=C(CH₃)-CO-NH-cycloheptyl, -CH=C(CH₃)-CO-NH-cyclooctyl, -CH=C(CH₃)-CO-pyrrolidin-1-yl, -CH=C(CH₃)-CO-piperidin-1-yl, -CH=C(CH₃)-CO-morpholin-4-yl, -CH=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -CH=C(CH₃)-CO-NH-CH₂C≡CH, -CH=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CH₃)-CO-NH-(CH₂)₂Cl, -CH=C(CH₃)-CO-NH-C₆H₅, -CH=C(C₂H₅)-CO-NH₂, -CH=C(C₂H₅)-CO-NHCH₃, -CH=C(C₂H₅)-CO-N(CH₃)₂, -CH=C(C₂H₅)-CO-NH-C₂H₅, -CH=C(C₂H₅)-CO-N(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-n-C₃H₇, -CH=C(C₂H₅)-CO-NH-i-C₃H₇, -CH=C(C₂H₅)-CO-NH-tert.-C₄H₉, -CH=C(C₂H₅)-CO-NH-cyclopropyl, -CH=C(C₂H₅)-CO-NH-cyclobutyl, -CH=C(C₂H₅)-CO-NH-cyclopentyl, -CH=C(C₂H₅)-CO-NH-cyclohexyl, -CH=C(C₂H₅)-CO-NH-cycloheptyl, -CH=C(C₂H₅)-CO-NH-cyclooctyl, -CH=C(C₂H₅)-CO-pyrrolidin-1-yl, -CH=C(C₂H₅)-CO-piperidin-1-yl, -CH=C(C₂H₅)-CO-morpholin-4-yl, -CH=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-CH₂C≡CH, -CH=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -CH=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -CH=C(C₂H₅)-CO-NH-C₆H₅, -CH=C(Cl)-CO-NH₂, -CH=C(Cl)-CO-NHCH₃, -CH=C(Cl)-CO-N(CH₃)₂, -CH=C(Cl)-CO-NH-C₂H₅, -CH=C(Cl)-CO-N(C₂H₅)₂, -CH=C(Cl)-CO-NH-n-C₃H₇, -CH=C(Cl)-CO-NH-i-C₃H₇, -CH=C(Cl)-CO-NH-tert.-C₄H₉, -CH=C(Cl)-CO-NH-cyclopropyl, -CH=C(Cl)-CO-NH-cyclobutyl, -CH=C(Cl)-CO-NH-cyclopentyl, -CH=C(Cl)-CO-NH-cyclohexyl, -CH=C(Cl)-CO-NH-cycloheptyl, -CH=C(Cl)-CO-NH-cyclooctyl, -CH=C(Cl)-CO-pyrrolidin-1-yl, -CH=C(Cl)-CO-piperidin-1-yl, -CH=C(Cl)-CO-morpholin-4-yl, -CH=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -CH=C(Cl)-CO-NH-CH₂C≡CH, -CH=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Cl)-CO-NH-(CH₂)₂Cl, -CH=C(Cl)-CO-NH-C₆H₅, -CH=C(Br)-CO-NH₂, -CH=C(Br)-CO-NHCH₃, -CH=C(Br)-CO-N(CH₃)₂, -CH=C(Br)-CO-NH-C₂H₅, -CH=C(Br)-CO-N(C₂H₅)₂, -CH=C(Br)-CO-NH-n-C₃H₇, -CH=C(Br)-CO-NH-i-C₃H₇, -CH=C(Br)-CO-NH-tert.-C₄H₉, -CH=C(Br)-CO-NH-cyclopropyl, -CH=C(Br)-CO-NH-cyclobutyl, -CH=C(Br)-CO-NH-cyclopentyl, -CH=C(Br)-CO-NH-cyclohexyl, -CH=C(Br)-CO-NH-cycloheptyl, -CH=C(Br)-CO-NH-cyclooctyl, -CH=C(Br)-CO-pyrrolidin-1-yl, -CH=C(Br)-CO-piperidin-1-yl, -CH=C(Br)-CO-morpholin-4-yl, -CH=C(Br)-CO-NH-CH₂CH=C(Br)₂, -CH=C(Br)-CO-NH-CH₂C≡CH, -CH=C(Br)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Br)-CO-NH-(CH₂)₂Cl, -CH=C(Br)-CO-NH-C₆H₅, -CH=C(CN)-CO-NH₂, -CH=C(CN)-CO-NHCH₃, -CH=C(CN)-CO-N(CH₃)₂, -CH=C(CN)-CO-NH-C₂H₅, -CH=C(CN)-CO-N(C₂H₅)₂, -CH=C(CN)-CO-NH-n-C₃H₇, -CH=C(CN)-CO-NH-i-C₃H₇, -CH=C(CN)-CO-NH-tert.-C₄H₉, -CH=C(CN)-CO-NH-cyclopropyl, -CH=C(CN)-CO-NH-cyclobutyl, -CH=C(CN)-CO-NH-cyclopentyl, -CH=C(CN)-CO-NH-cyclohexyl, -CH=C(CN)-CO-NH-cycloheptyl, -CH=C(CN)-CO-NH-cyclooctyl, -CH=C(CN)-CO-pyrrolidin-1-yl, -CH=C(CN)-CO-piperidin-1-yl, -CH=C(CN)-CO-morpholin-4-yl, -CH=C(CN)-CO-NH-CH₂CH=C(CN)₂, -CH=C(CN)-CO-NH-CH₂C≡CH, -CH=C(CN)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CN)-CO-NH-(CH₂)₂Cl, -CH=C(CN)-CO-NH-C₆H₅, -CH=CH-CO-SCH₃, -CH=CH-CO-SC₂H₅, -CH=CH-CO-S-n-C₃H₇, -CH=CH-CO-S-i-C₃H₇, -CH=CH-CO-S-n-C₄H₉, -CH=CH-CO-S-tert.-C₄H₉, -CH=C(CH₃)-CO-SCH₃, -CH=C(CH₃)-CO-SC₂H₅, -CH=C(CH₃)-CO-S-n-C₃H₇, -CH=C(CH₃)-CO-S-i-C₃H₇, -CH=C(CH₃)-CO-S-n-C₄H₉, -CH=C(CH₃)-CO-S-tert.-C₄H₉, -CH=C(C₂H₅)-CO-SCH₃, -CH=C(C₂H₅)-CO-SC₂H₅, -CH=C(C₂H₅)-CO-S-n-C₃H₇, -CH=C(C₂H₅)-CO-S-i-C₃H₇, -CH=C(C₂H₅)-CO-S-n-C₄H₉, -CH=C(C₂H₅)-CO-S-tert.-C₄H₉, -CH=C(Cl)-CO-SCH₃, -CH=C(Cl)-CO-SC₂H₅, -CH=C(Cl)-CO-S-n-C₃H₇, -CH=C(Cl)-CO-S-i-C₃H₇, -CH=C(Cl)-CO-S-n-C₄H₉, -CH=C(Cl)-CO-S-tert.-C₄H₉, -CH=C(Br)-CO-SCH₃, -CH=C(Br)-CO-SC₂H₅, -CH=C(Br)-CO-S-n-C₃H₇, -CH=C(Br)-CO-S-i-C₃H₇, -CH=C(Br)-CO-S-n-C₄H₉, -CH=C(Br)-CO-S-tert.-C₄H₉, -CH=C(CN)-CO-SCH₃, -CH=C(CN)-CO-SC₂H₅, -CH=C(CN)-CO-S-n-C₃H₇, -CH=C(CN)-CO-S-i-C₃H₇, -CH=C(CN)-CO-S-n-C₄H₉, -CH=C(CN)-CO-S-tert.-C₄H₉, -CH=C(COCH₃)-CO-OCH₃, -CH=C(COC₂H₅)-CO-OCH₃, -CH=C(CO-n-C₃H₇)-CO-OCH₃, -CH=C(COCH₃)-CO-OC₂H₅, -CH=C(COC₂H₅)-CO-OC₂H₅, -CH=C(CO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COCH₃)-CO-O-n-C₃H₇, -CH=C(COC₂H₅)-CO-O-n-C₃H₇, -CH=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-OCH₃, -CH=C(CF₃)-CO-OC₂H₅, -CH=C(CF₃)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-O-i-C₃H₇, -CH=C(CF₃)-CO-O-n-C₄H₉, -CH=C(CF₃)-CO-O-tert.-C₄H₉, -CH=C(COOCH₃)₂, -CH=C(COOC₂H₅)₂, -CH=C(COOCH₃)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)-CO-OCH₃, -CH=C(COO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)₂, -CH=CH-CH=CH-COOH, -CH=CH-CH=CH-CO-OCH₃, -CH=CH-CH=CH-CO-OC₂H₅, -CH=CH-CH=C(COOCH₃)₂, -CH=CH-CH=C(CN)-CO-OCH₃, -CH=CH-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-OCH₃, -CH=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CH=C(Cl)-CO-OCH₃, -CH=C(CH₃)-CH=C(Br)-CO-OCH₃, -CH=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-NH₂, -CH=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -CH=CH-(CH₂)₂-COOH, -CH=CH-(CH₂)₂-CO-OCH₃, -CH=CH-(CH₂)₂-CO-OC₂H₅, -CH=CH-CH₂-CH(COOCH₃)₂, -CH=CH-CH₂-CH(COOC₂H₅)₂, -CH=CH-CH₂-CH(CN)-CO-OCH₃, -CH=CH-CH₂-CH(CN)-CO-OC₂H₅, -CH=CH-CH₂-CH(CH₃)-CO-OCH₃, -CH=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -CH=CH-(CH₂)₂-CO-NH₂, -CH=CH-(CH₂)₂-CO-NH-CH₃, -CH=CH-CH₂-COOH, -CH=CH-CH₂-CO-OCH₃, -CH=CH-CH₂-CO-OC₂H₅, -CH=C(COOCH₃)-CH₂-CO-OCH₃, -CH=C(COOCH₃)-CH₂-CO-OC₂H₅, -CH=CH-CH₂-CO-NH₂, -CH=CH-CH₂-CO-NH-CH₃, -CH=CH-CH₂-CO-N(CH₃)₂, -CH(OCH₃)₂, -CH(SCH₃)₂, -CH(OC₂H₅)₂, -CH(SC₂H₅)₂, -CH(O-n-C₃H₇)₂, -CH(O-i-C₃H₇)₂, -CH(S-n-C₃H₇)₂, -CH(S-i-C₃H₇)₂, -CH(O-n-C₄H₉)₂, -CH(O-i-C₄H₉)₂, -CH(O-s-C₄H₉)₂, -CH(O-tert.-C₄H₉)₂, -CH(S-n-C₄H₉)₂, -CH(S-i-C₄H₉)₂, -CH(S-s-C₄H₉)₂, -CH(S-tert.-C₄H₉)₂, -CH(OC₅H₁₁)₂, 1,3-Dioxolan-2-yl, 1,3-Dithio­ lan-2-yl, 1,3-Oxathiolan-2-yl, 4-Methyl-1,3-dioxolan-2-yl, 4-Methyl-1,3-dithiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 5-Methyl-1,3-oxathiolan-2-yl, 4-Ethyl-1,3-dioxolan-2-yl, 4-Ethyl- 1,4-dithiolan-2-yl, 4-Ethyl-1,3-oxathiolan-2-yl, 5-Ethyl-1,3-oxa­ thiolan-2-yl, 4,5-Dimethyl-1,3-dioxolan-2-yl, 4,4-Dimethyl-1,3- dioxolan-2-yl, 4,5-Dimethyl-1,3-dithiolan-2-yl, 5,5-Dimethyl-1,3- dithiolan-2-yl, 4,5-Dimethyl-1,3-oxathiolan-2-yl, 5,5-Dimethyl- 1,3-oxathiolan-2-yl, 4,4-Dimethyl-1,3-oxathiolan-2-yl, 4-Vinyl- 1,3-dioxolan-2-yl, 4-Vinyl-1,3-dithiolan-2-yl, 4-Vinyl-1,3-oxa­ thiolan-2-yl, 5-Vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3- dioxolan-2-yl, 4-Chlormethyl-1,3-dithiolan-2-yl, 4-Chlormethyl- 1,3-oxathiolan-2-yl, 5-Chlormethyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-1,3-dithio­ lan-2-yl, 4-Hydroxymethyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl- 1,3-oxathiolan-2-yl, 4-Methoxymethyl-1,3-dioxolan-2-yl, 4-Allyl­ oxymethyl-1,3-dioxolan-2-yl, 4-Propargyloxymethyl-1,3-dioxolan- 2-yl, 4-Acetoxymethyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-1,3-dithiolan-2-yl, 4-Propargyl­ oxymethyl-1,3-dithiolan-2-yl, 4-Acetoxymethyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-1,3-oxa­ thiolan-2-yl, 4-Allyloxymethyl-1,3-oxathiolan-2-yl, 5-Allyloxy­ methyl-1,3-oxathiolan-2-yl, 4-Propargyloxymethyl-1,3-oxathiolan- 2-yl, 5-Propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxymethyl- 1,3-oxathiolan-2-yl, 5-Acetoxymethyl-1,3-oxathiolan-2-yl, 4-Methylthiomethyl-1,3-dioxolan-2-yl, 4-Methylthiomethyl-1,3- dithiolan-2-yl, 4-Carboxy-1,3-dioxolan-2-yl, 4-Carboxy-1,3- dithiolan-2-yl, 4-Methoxycarbonyl-1,3-dioxolan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-1,3-di­ thiolan-2-yl, 4-n-Butoxycarbonyl-1,3-dithiolan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-4-methyl- 1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-di­ thiolan-2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-1,3- dithiolan-2-yl, 1,3-Dioxan-2-yl, 1,3-Dithian-2-yl, 1,3-Oxathian- 2-yl, 5-Methyl-1,3-dioxan-2-yl, 5-Methyl-1,3-dithian-2-yl, 5-Methyl-1,3-oxathian-2-yl, 5,5-Dimethyl-1,3-dioxan-2-yl, 4,6-Di­ methyl-1,3-dioxan-2-yl, 4,4-Dimethyl-1,3-dioxan-2-yl, 5,5-Di­ methyl-1,3-dithian-2-yl, 4,6-Dimethyl-1,3-dithian-2-yl, 4,4-Di­ methyl-1,3-dithian-2-yl, 5,5-Dimethyl-1,3-oxathian-2-yl, 4,4-Di­ methyl-1,3-oxathian-2-yl, 6,6-Dimethyl-1,3-oxathian-2-yl, 4-Hydroxymethyl-1,3-dioxan-2-yl, 4-Methoxymethyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-1,3-dioxan-2- yl, 4-Hydroxymethyl-1,3-dithian-2-yl, 4-Methoxymethyl-1,3-di­ thian-2-yl, 4-Allyloxymethyl-1,3-dithian-2-yl, 4-Acetoxymethyl- 1,3-dithian-2-yl, 4-Chlormethyl-1,3-dioxan-2-yl, 4-Chlormethyl- 1,3-dithian-2-yl, 1,3-Dioxepan-2-yl, 1,3-Dithiepan-2-yl, 1,3-Di­ oxep-5-en-2-yl, 4-Methoxycarbonyl-1,3-dioxan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-1,3-dithian- 4-yl, 4-n-Butoxycarbonyl-1,3-dithian-2-yl, 4-Methoxycarbonyl-4- methyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxan-2- yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-4-methyl- 1,3-dithian-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithian-2-yl, -C(CH₃)(OCH₃)₂, -C(CH₃)(SCH₃)₂, -C(CH₃)(OC₂H₅)₂, -C(CH₃)(SC₂H₅)₂, -C(CH₃)(O-n-C₃H₇)₂, -C(CH₃)(O-i-C₃H₇)₂, -C(CH₃)(S-n-C₃H₇)₂, -C(CH₃)(S-i-C₃H₇)₂, -C(CH₃)(O-n-C₄H₉)₂, -C(CH₃)(O-i-C₄H₉)₂, -C(CH₃)(O-s-C₄H₉)₂, -C(CH₃)(O-tert.-C₄H₉)₂, -C(CH₃)(S-n-C₄H₉)₂, -C(CH₃)(S-i-C₄H₉)₂, -C(CH₃)(S-s-C₄H₉)₂, -C(CH₃)(S-tert.-C₄H₉)₂, -C(CH₃)(O-n-C₅H₁₁)′′, 2-Methyl-1,3-dioxolan-2-yl, 2-Methyl-1,3-di­ thiolan-2-yl, 2-Methyl-1,3-oxathiolan-2-yl, 2,4-Dimethyl-1,3- dioxolan-2-yl, 2,4-Dimethyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-1,3- oxathiolan-2-yl, 2,5-Dimethyl-1,3-oxathiolan-2-yl, 4-Ethyl-2- methyl-1,3-dioxolan-2-yl, 4-Ethyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Ethyl-2-methyl-1,3- oxathiolan-2-yl, 2,4,5-Trimethyl-1,3-dioxolan-2-yl, 2,4,4-Tri­ methyl-1,3-dioxolan-2-yl, 2,4,5-Trimethyl-1,3-dithiolan-2-yl, 2,4,4-Trimethyl-1,3-dithiolan-2-yl, 2,4,5-Trimethyl-1,3-oxathio­ lan-2-yl, 2,4,4-Trimethyl-1,3-oxathiolan-2-yl, 2-Methyl-4-vinyl- 1,3-dioxolan-2-yl, 2-Methyl-4-vinyl-1,3-dithiolan-2-yl, 2-Methyl- 4-vinyl-1,3-oxathiolan-2-yl, 2-Methyl-5-vinyl-1,3-oxathiolan-2- yl, 4-Chlormethyl-2-methyl-1,3-dioxolan-2-yl, 4-Chlormethyl-2- methyl-1,3-dithiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-oxathio­ lan-2-yl, 5-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Hydroxy­ methyl-2-methyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-2- methyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dioxolan- 2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxy- 2-methyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dithiolan-2-yl, 4-Acetoxy-2- methyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-oxathio­ lan-2-yl, 5-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Allyl­ oxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Allyloxymethyl-2- methyl-1,3-oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3- oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3-oxathiolan-2- yl, 4-Acetoxy-2-methyl-1,3-oxathiolan-2-yl, 5-Acetoxy-2-methyl- 1,3-oxathiolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dioxolan-2- yl, 2-Methyl-4-methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-2- methyl-1,3-dioxolan-2-yl, 4-Carboxy-2-methyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-2- methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-2-methyl-1,3-dioxo­ lan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-Eth­ oxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-2- methyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-di­ oxolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-ethoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4- ethoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-n-butoxy­ carbony-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl-1,3- dithiolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-dioxan-2- yl, 2-Methyl-1,3-dithian-2-yl, 2-Methyl-1,3-oxathian-2-yl, 2,5- Dimethyl-1,3-dioxan-2-yl, 2,5-Dimethyl-1,3-dithian-2-yl, 2,5-Di­ methyl-1,3-oxathian-2-yl, 2,5,5-Trimethyl-1,3-dioxan-2-yl, 2,4,6- Trimethyl-1,3-dioxan-2-yl, 2,4,4-Trimethyl-1,3-dioxan-2-yl, 2,5,5-Trimethyl-1,3-dithian-2-yl, 2,4,6-Trimethyl-1,3-dithian-2- yl, 2,4,4-Trimethyl-1,3-dithian-2-yl, 2,5,5-Trimethyl-1,3-oxa­ thian-2-yl, 2,4,4-Trimethyl-1,3-oxathian-2-yl, 2,6,6-Trimethyl- 1,3-oxathian-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-2- methyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dithian-2-yl, 4-Methoxymethyl-2- methyl-1,3-dithian-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithian-2- yl, 4-Acetoxymethyl-2-methyl-1,3-dithian-2-yl, 4-Chlormethyl-2- methyl-1,3-dioxan-2-yl, 4-Chlormethyl-2-methyl-1,3-dithian-2-yl, -C(CH₃)=NH, -C(CH₃)=N-CH₃, -C(CH₃)=N-C₂H₅, -C(CH₃)=N-n-C₃H₇, -C(CH₃)=N-i-C₃H₇, -C(CH₃)=N-n-C₄H₉, -C(CH₃)=N-CH₂CH=CH₂, -C(CH₃)=N-CH₂CH=CH₂-CH₃, -C(CH₃)=N-CH₂C≡CH, -C(CH₃)=N-CH₂C≡C-CH₃, -C(CH₃)=N-cyclopropyl, -C(CH₃)=N-cyclobutyl, -C(CH₃)=N-cyclo­ pentyl, -C(CH₃)=N-cyclohexyl, -C(CH₃)=N-cycloheptyl, -C(CH₃)=N-CH₂-CH₂Cl, -C(CH₃)=N-CH₂Cl, -C(CH₃)=N-C₆H₅, -C(CH₃)=N-(2-F-C₆H₄), -C(CH₃)=N-(3-F-C₆H₄), -C(CH₃)=N-(4-F-C₆H₄), -C(CH₃)=N-(2-Cl-C₆H₄), -C(CH₃)=N-(3-Cl-C₆H₄), -C(CH₃)=N-(4-Cl-C₆H₄), -C(CH₃)=N-(2-CH₃-C₆H₄), -C(CH₃)=N-(3-CH₃-C₆H₄), -C(CH₃)=N-(4-CH₃-C₆H₄), -C(CH₃)=N-(2-CF₃-C₆H₄), -C(CH₃)=N-(3-CF₃-C₆H₄), -C(CH₃)=N-(4-CF₃-C₆H₄), -C(CH₃)=N-(2-OCH₃-C₆H₄), -C(CH₃)=N-(3-OCH₃-C₆H₄), -C(CH₃)=N-(4-OCH₃-C₆H₄), -C(CH₃)=N-(4-NO₂-C₆H₄), -C(CH₃)=N-(4-CN-C₆H₄), -C(CH₃)=N-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-(2,4-(CH₃)₂-C₆H₃), -C(CH₃)=N-CH₂-OCH₃, -C(CH₃)=N-CH₂-OC₂H₅, -C(CH₃)=N-CH₂CH₂-OCH₃, -C(CH₃)=N-CH₂CH-OC₂H₅, -C(CH₃)=N-OH, -C(CH₃)=N-OCH₃, -C(CH₃)=N-OC₂H₅, -C(CH₃)=N-O-n-C₃H₇, -C(CH₃)=N-O-i-C₃H₇, -C(CH₃)=N-O-n-C₄H₉, -C(CH₃)=N-O-i-C₄H₉, -C(CH₃)=N-O-s-C₄H₉, -C(CH₃)=N-O-tert.-C₄H₉, -C(CH₃)=N-OCH₂-CH=CH₂, -C(CH₃)=N-OCH(CH₃)-CH=CH₂, -C(CH₃)=N-OCH₂-C≡CH, -C(CH₃)=N-CH(CH₃)-C≡CH, -C(CH₃)=N-OCH₂-CH=C-CH₃, -C(CH₃)=N-OCH₂CH₂-Cl, -C(CH₃)=N-OCH₂CH₂-F, -C(CH₃)=N-OCH₂-CF₃, -C(CH₃)=N-OCH₂-CH=CHCl, -C(CH₃)=N-OCH₂-C(Cl)=CH₂, -C(CH₃)=N-OCH₂-C(Br)=CH₂, -C(CH₃)=N-OCH₂-CH=C(Cl)-CH₃, -C(CH₃)=N-O-CO-CH₃, -C(CH₃)=N-O-CO-C₂H₅, -C(CH₃)=N-OCH₂-CN, -C(CH₃)=N-OCH₂-CH=CH-CH₂-OCH₃, -C(CH₃)=N-OCH₂-CH=CH-CH₂-O-tert.-C₄H₉, -C(CH₃)=N-O-(CH₂)₃-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-(4-Cl-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-C₆H₅, -C(CH₃)=N-OCH₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(3-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-CH₂-(4-CH₃O-C₆H₄), -C(CH₃)=N-OCH₂-CH=C(CH₃)-C₆H₅, -C(CH₃)=N-O-(CH₂)₂-CH=CH-(3,4-Cl₂-C₆H₃), -C(CH₃)=N-O-(CH₂)₃-C≡C-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-OCH₃, -C(CH₃)=N-OCH₂CH₂-OCH₃, -C(CH₃)=N-OCH₂-OC₂H₅, -C(CH₃)=N-OCH(CH₃)-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=N-NH₂, -C(CH₃)=N-NH-CH₃, -C(CH₃)=N-NH-C₂H₅, -C(CH₃)=N-NH-n-C₃H₇, -C(CH₃)=N-NH-i-C₃H₇, -C(CH₃)=N-NH-n-C₄H₉, -C(CH₃)=N-NH-i-C₄H₉, -C(CH₃)=N-NH-s-C₄H₉, -C(CH₃)=N-NH-tert.-C₄H₉, -C(CH₃)=N-NH-cyclopropyl, -C(CH₃)=N-NH- cyclobutyl, -C(CH₃)=N-NH-cyclopentyl, -C(CH₃)=N-NH-cyclohexyl, -C(CH₃)=N-NH-cycloheptyl, -C(CH₃)=N-N(CH₃)₂, -C(CH₃)=N-N(C₂H₅)₂, -C(CH₃)=N-N(n-C₃H₇)₂, -C(CH₃)=N-N(i-C₃H₇)₂, -C(CH₃)=N-NH-CH₂-C=CH, -C(CH₃)=N-NH-CH₂-C≡CH, -C(CH₃)=N-N(CH₃)-CH₂-C≡CH, -C(CH₃)=N-NH-CH₂CF₃, -C(CH₃)=N-NH-CO-CH₃, -C(CH₃)=N-NH-CO-C₂H₅, -C(CH₃)=N-NH-CO-OCH₃, -C(CH₃)=N-NH-CO-OC₂H₅, -C(CH₃)=N-NH-CO-O-tert.-C₄H₉, -C(CH₃)=N- pyrrolidin-1-yl, -C(CH₃)=N-piperidin-1-yl, -C(CH₃)=N-morpholin- 4-yl, -C(CH₃)=N-NH-C₆H₅, -C(CH₃)=N-NH-(4-Cl-C₆H₄), -C(CH₃)=N-NH-(4-NO₂-C₆H₄), -C(CH₃)=N-NH-(4-F-C₆H₄), -C(CH₃)=N-NH-(4-CH₃O-C₆H₄), -C(CH₃)=N-NH-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-NH-(2,4-(NO₂)₂-C₆H₃), -C(CH₃)=N-NH-CO-NH₂, -C(CH₃)=N-NH-CO-NHCH₃, -C(CH₃)=N-NH-CO-NHC₂H₅, -C(CH₃)=N-NH-CO-N(CH₃)₂, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=CH-CO-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -(CH₃)=CH-CO-O-n-C₄H₉, -C(CH₃)=CH-CO-O-tert.-C₄H₉, -C(CH₃)=CH-CO-O-cyclopropyl, -C(CH₃)=CH-CO-O-cyclobutyl, -C(CH₃)=CH-CO-O-cyclopentyl, -C(CH₃)=CH-CO-O-cyclohexyl, -C(CH₃)=CH-CO-O-cycloheptyl, -C(CH₃)=C(CH₃)-COOH, -C(CH₃)=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-cyclopropyl, -C(CH₃)=C(CH₃)-CO-O-cyclobutyl, -C(CH₃)=C(CH₃)-CO-O-cyclopentyl, -C(CH₃)=C(CH₃)-CO-O-cyclohexyl, -C(CH₃)=C(CH₃)-CO-O-cycloheptyl, -C(CH₃)=C(C₂H₅)-COOH, -C(CH₃)=C(C₂H₅)-CO-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-cyclo­ propyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-O- cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-O-cycloheptyl, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=C(Cl)-CO-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-O-n-C₄H₉, -C(CH₃)=C(Cl)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-O-cyclopropyl, -C(CH₃)=C(Cl)-CO-O-cyclobutyl, -C(CH₃)=C(Cl)-CO-O-cyclopentyl, -C(CH₃)=C(Cl)-CO-O-cyclohexyl, -C(CH₃)=C(Cl)-CO-O-cycloheptyl, -C(CH₃)=C(Br)-COOH, -C(CH₃)=C(Br)-CO-OCH₃, -C(CH₃)=C(Br)-CO-OC₂H₅, -C(CH₃)=C(Br)-CO-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-O-n-C₄H₉, -C(CH₃)=C(Br)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-O-cyclopropyl, -C(CH₃)=C(Br)-CO-O-cyclobutyl, -C(CH₃)=C(Br)-CO-O-cyclopentyl, -C(CH₃)=C(Br)-CO-O-cyclohexyl, -C(CH₃)=C(Br)-CO-O-cycloheptyl, -C(CH₃)=C(CN)-COOH, -C(CH₃)=C(CN)-CO-OCH₃, -C(CH₃)=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CN)-CO-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-O-n-C₄H₉, -C(CH₃)=C(CN)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-O-cyclopropyl, -C(CH₃)=C(CN)-CO-O-cyclobutyl, -C(CH₃)=C(CN)-CO-O-cyclopentyl, -C(CH₃)=C(CN)-CO-O-cyclohexyl, -C(CH₃)=C(CN)-CO-O-cycloheptyl, -C(CH₃)=CH-CO-OCH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=CH-CO-O-i-C₃H₇, -C(CH₃)=CH-CO-OCH(CH₃)-OCH₃, -C(CH₃)=CH-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=CH-CO-OCH₂CH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=(C₂H₅)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-O-i-C₃H₇, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -(CH₃)=C(Cl)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-O-i-C₃H₇, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-O-i-C₃H₇, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-CF₃, -C(CH₃)=CH-CO-OCH₂-CCl₃, -C(CH₃)=CH-CO-OCH₂-oxiranyl, -C(CH₃)=CH-CO-O-(CH₂)₃-Br, -C(CH₃)=CH-CO-OCH₂-CH=CH₂, -C(CH₃)=CH-CO-OCH₂-C≡CH, -C(CH₃)=CH-CO-OCH₂-CN, -C(CH₃)=CH-CO-OCH₂CH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CF₃, -C(CH₃)=C(CH₃)-CO-OCH₂-CCl₃, -C(CH₃)=C(CH₃)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CH₃)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(CH₃)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CH₃)-CO-OCH₂-C≡CH, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CF₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CCl₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-oxiranyl, -C(CH₃)=C(C₂H₅)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(C₂H₅)-CO-OCH₂-C≡CH, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂-CF₃, -C(CH₃)=C(Cl)-CO-OCH₂-CCl₃, -C(CH₃)=C(Cl)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Cl)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Cl)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Cl)-CO-OCH₂-C≡CH, -C(CH₃)=C(Cl)-CO-OCH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂-CF₃, -C(CH₃)=C(Br)-CO-OCH₂-CCl₃, -C(CH₃)=C(Br)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Br)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Br)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Br)-CO-OCH₂-C≡CH, -C(CH₃)=C(Br)-CO-OCH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂CH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂-CF₃, -C(CH₃)=C(CN)-CO-OCH₂-CCl₃, -C(CH₃)=C(CN)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CN)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(CN)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CN)-CO-OCH₂-C≡CH, -C(CH₃)=C(CN)-CO-OCH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂CH₂-CN, -C(CH₃)=CH-CO-CH₃, -C(CH₃)=CH-CO-C₂H₅, -C(CH₃)=CH-CO-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-n-C₄H₉, -C(CH₃)=CH-CO-tert.-C₄H₉, -C(CH₃)=CH-CO-CH₂Cl, -C(CH₃)=CH-CO-CH₂Br, -C(CH₃)=CH-CO-CHCl₂, -C(CH₃)=CH-CO-CH₂-OCH₃, -C(CH₃)=CH-CO-CH(OCH₃)₂, -C(CH₃)=CH-CO-CH₂-SCH₃, -C(CH₃)=C(CH₃)-CO-CH₃, -C(CH₃)=C(CH₃)-CO-C₂H₅, -C(CH₃)=C(CH₃)-CO-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-CH₂Cl, -C(CH₃)=C(CH₃)-CO-CH₂Br, -C(CH₃)=C(CH₃)-CO-CHCl₂, -C(CH₃)=C(CH₃)-CO-CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-CH(OCH₃)₂, -C(CH₃)=C(CH₃)-CO-CH₂-SCH₃, -C(CH₃)=C(C₂H₅)-CO-CH₃, -C(CH₃)=C(C₂H₅)-CO-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-CH₂Cl, -C(CH₃)=C(C₂H₅)-CO-CH₂Br, -C(CH₃)=C(C₂H₅)-CO-CHCl₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-CH(OCH₃)₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-SCH₃, -C(CH₃)=C(Cl)-CO-CH₃, -C(CH₃)=C(Cl)-CO-C₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-n-C₄H₉, -C(CH₃)=C(Cl)-CO-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-CH₂Cl, -C(CH₃)=C(Cl)-CO-CHCl₂, -C(CH₃)=C(Cl)-CO-CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-CH(OCH₃)₂, -C(CH₃)=C(Cl)-CO-CH₂-SCH₃, -C(CH₃)=C(Br)-CO-CH₃, -C(CH₃)=C(Br)-CO-C₂H₅, -C(CH₃)=C(Br)-CO-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-n-C₄H₉, -C(CH₃)=C(Br)-CO-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-CH₂Cl, -C(CH₃)=C(Br)-CO-CH₂Br, -C(CH₃)=C(Br)-CO-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-CH(OCH₃)₂, -C(CH₃)=C(Br)-CO-CH₂-SCH₃, -C(CH₃)=C(CN)-CO-CH₃, -C(CH₃)=C(CN)-CO-C₂H₅, -C(CH₃)=C(CN)-CO-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-n-C₄H₉, -C(CH₃)=C(CN)-CO-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-CH₂Cl, -C(CH₃)=C(CN)-CO-CH₂Br, -C(CH₃)=C(CN)-CO-CHCl₂, -C(CH₃)=C(CN)-CO-CH₂-OCH₃, -C(CH₃)=C(CN)-CO-CH(OCH₃)₂, -C(CH₃)=C(CN)-CO-CH₂-SCH₃, -C(CH₃)=CH-CO-C₆H₅, -C(CH₃)=CH-CO-(4-Cl-C₆H₄), -C(CH₃)=C(CH₃)-CO-C₆H₅, -C(CH₃)=C(CH₃)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(C₂H₅)-CO-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(Cl)-CO-C₆H₅, -C(CH₃)=C(Br)-CO-C₆H₅, -C(CH₃)=C(CN)-CO-C₆H₅, -C(CH₃)=CH-CO-NH₂, -C(CH₃)=CH-CO-NHCH₃, -C(CH₃)=CH-CO-N(CH₃)₂, -C(CH₃)=CH-CO-NH-C₂H₅, -C(CH₃)=CH-CO-N(C₂H₅)₂, -C(CH₃)=CH-CO-NH-n-C₃H₇, -C(CH₃)=CH-CO-NH-i-C₃H₇, -C(CH₃)=CH-CO-NH-tert.-C₄H₉, -C(CH₃)=CH-CO-NH-cyclopropyl, -C(CH₃)=CH-CO-NH-cyclobutyl, -C(CH₃)=CH-CO-NH-cyclopentyl, -C(CH₃)=CH-CO-NH-cyclohexyl, -C(CH₃)=CH-CO-NH-cycloheptyl, -C(CH₃)=CH-CO-NH-cyclooctyl, -C(CH₃)=CH-CO-pyrrolidin-1-yl, -C(CH₃)=CH-CO-piperidin-1-yl, -C(CH₃)=CH-CO-morpholin-4-yl, -C(CH₃)=CH-CO-NH-CH₂CH=CH₂, -C(CH₃)=CH-CO-NH-CH₂C≡CH, -C(CH₃)=CH-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=CH-CO-NH-(CH₂)₂Cl, -C(CH₃)=CH-CO-NH-C₆H₅, -C(CH₃)=C(CH₃)-CO-NH₂, -C(CH₃)=C(CH₃)-CO-NHCH₃, -C(CH₃)=C(CH₃)-CO-N(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-C₂H₅, -C(CH₃)=C(CH₃)-CO-N(C₂H₅)₂, -C(CH₃)=C(CH₃)-CO-NH-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-NH- cyclopropyl, -C(CH₃)=C(CH₃)-CO-NH-cyclobutyl, -C(CH₃)=C(CH₃)-CO-NH-cyclopentyl, -C(CH₃)=C(CH₃)-CO-NH- cyclohexyl, -C(CH₃)=C(CH₃)-CO-NH-cycloheptyl, -C(CH₃)=C(CH₃)-CO-NH-cyclooctyl, -C(CH₃)=C(CH₃)-CO- pyrrolidin-1-yl, -C(CH₃)=C(CH₃)-CO-piperidin-1-yl, -C(CH₃)=C(CH₃)-CO-morpholin-4-yl, -C(CH₃)=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CH₃)-CO-NH-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-NH₂, -C(CH₃)=C(C₂H₅)-CO-NHCH₃, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)₂, -C(CH₃)=C(C₂H₅)-CO-NH-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-N(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-NH- cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclo­ hexyl, -C(CH₃)=C(C₂H₅)-CO-NH-cycloheptyl, -C(CH₃)=C(C₂H₅)-CO-NH- cyclooctyl, -C(CH₃)=C(C₂H₅)-CO-pyrrolidin-1-yl, -C(CH₃)=C(C₂H₅)-CO-piperidin-1-yl, -C(CH₃)=C(C₂H₅)-CO- morpholin-4-yl, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(C₂H₅)-CO-NH-C₆H₅, -C(CH₃)=C(Cl)-CO-NH₂, -C(CH₃)=C(Cl)-CO-NHCH₃, -C(CH₃)=C(Cl)-CO-N(CH₃)₂, -C(CH₃)=C(Cl)-CO-NH-C₂H₅, -C(CH₃)=C(Cl)-CO-N(C₂H₅)₂, -C(CH₃)=C(Cl)-CO-NH-n-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-i-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-NH-cyclopropyl, -C(CH₃)=C(Cl)-CO-NH-cyclobutyl, -C(CH₃)=C(Cl)-CO-NH-cyclopentyl, -C(CH₃)=C(Cl)-CO-NH-cyclohexyl, -C(CH₃)=C(Cl)-CO-NH-cycloheptyl, -C(CH₃)=C(Cl)-CO-NH-cyclooctyl, -C(CH₃)=C(Cl)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Cl)-CO-piperidin-1- yl, -C(CH₃)=C(Cl)-CO-morpholin-4-yl, -C(CH₃)=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -C(CH₃)=C(Cl)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-N(CH₃)-CH₂≡CH, -C(CH₃)=C(Cl)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Cl)-CO-NH-C₆H₅, -C(CH₃)=C(Br)-CO-NH₂, -C(CH₃)=C(Br)-CO-NHCH₃, -C(CH₃)=C(Br)-CO-N(CH₃)₂, -C(CH₃)=C(Br)-CO-NH-C₂H₅, -C(CH₃)=C(Br)-CO-N(C₂H₅)₂, -C(CH₃)=C(Br)-CO-NH-n-C₃H₇, -C(CH₃)=C(Br)-CO-NH-i-C₃H₇, -C(CH₃)=C(Br)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-NH-cyclopropyl, -C(CH₃)=C(Br)-CO-NH-cyclobutyl, -C(CH₃)=C(Br)-CO-NH-cyclopentyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cycloheptyl, -C(CH₃)=C(Br)-CO-NH-cyclooctyl, -C(CH₃)=C(Br)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Br)-CO-piperidin-1-yl, -C(CH₃)=C(Br)-CO-morpholin-4-yl, -C(CH₃)=C(Br)-CO-NH-CH₂CH=C(Br)₂, -C(CH₃)=C(Br)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Br)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Br)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Br)-CO-NH-C₆H₅, -C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CN)-CO-NHCH₃, -C(CH₃)=C(CN)-CO-N(CH₃)₂, -C(CH₃)=C(CN)-CO-NH-C₂H₅, -C(CH₃)=C(CN)-CO-N(C₂H₅)₂, -C(CH₃)=C(CN)-CO-NH-n-C₃H₇, -C(CH₃)=C(CN)-CO-NH-i-C₃H₇, -C(CH₃)=C(CN)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-NH-cyclopropyl, -C(CH₃)=C(CN)-CO-NH-cyclobutyl, -C(CH₃)=C(CN)-CO-NH-cyclopentyl, -C(CH₃)=C(CN)-CO-NH-cyclohexyl, -C(CH₃)=C(CN)-CO-NH-cycloheptyl, -C(CH₃)=C(CN)-CO-NH-cyclooctyl, -C(CH₃)=C(CN)-CO-pyrrolidin-1-yl, -C(CH₃)=C(CN)-CO-piperidin-1-yl, -C(CH₃)=C(CN)-CO-morpholin-4-yl, -C(CH₃)=C(CN)-CO-NH-CH₂CH=C(CN)₂, -C(CH₃)=C(CN)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CN)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CN)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CN)-CO-NH-C₆H₅, -C(CH₃)=CH-CO-SCH₃, -C(CH₃)=CH-CO-SC₂H₅, -C(CH₃)=CH-CO-S-n-C₃H₇, - C(CH₃)=CH-CO-S-i-C₃H₇, -C(CH₃)=CH-CO-S-n-C₄H₉, -C(CH₃)=CH-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-SCH₃, -C(CH₃)=C(CH₃)-CO-SC₂H₅, -C(CH₃)=C(CH₃)-CO-S-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-S-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-SCH₃, -C(CH₃)=C(C₂H₅)-CO-SC₂H₅, -C(CH₃)=C(C₂H₅)-CO-S-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-SCH₃, -C(CH₃)=C(Cl)-CO-SC₂H₅, -C(CH₃)=C(Cl)-CO-S-n-C₃H₇, -C(CH₃)=C(Cl)-CO-S-i-C₃H₇, -C(CH₃)=C(Cl)-CO-S-n-C₄H₉, -C(CH₃)=C(Cl)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-SCH₃, -C(CH₃)=C(Br)-CO-SC₂H₅, - ⁹⁹⁹⁹⁹ ⁰⁰⁰⁷⁰ ⁵⁵² ⁰⁰¹⁰⁰⁰²⁸⁰⁰⁰⁰⁰00200012000285919988800040 0002004131038 00004 99880 C(CH₃)=C(Br)-CO-S-n-C₃H₇, -C(CH₃)=C(Br)-CO-S-i-C₃H₇, -C(CH₃)=C(Br)-CO-S-n-C₄H₉, -C(CH₃)=C(Br)-CO-S-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-SCH₃, -C(CH₃)=C(CN)-CO-SC₂H₅, -C(CH₃)=C(CN)-CO-S-n-C₃H₇, -C(CH₃)=C(CN)-CO-S-i-C₃H₇, -C(CH₃)=C(CN)-CO-S-n-C₄H₉, -C(CH₃)=C(CN)-CO-S-tert.-C₄H₉, -C(CH₃)=C(COCH₃)-CO-OCH₃, -C(CH₃)=C(COC₂H₅)-CO-OCH₃, -C(CH₃)=C(CO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COCH₃)-CO-OC₂H₅, -C(CH₃)=C(COC₂H₅)-CO-OC₂H₅, -C(CH₃)=C(CO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COCH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(COC₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-OCH₃, -C(CH₃)=C(CF₃)-CO-OC₂H₅, -C(CH₃)=C(CF₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CF₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(COOCH₃)₂, -C(CH₃)=C(COOC₂H₅)₂, -C(CH₃)=C(COOCH₃)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)₂, -C(CH₃)=CH-CH=CH-COOH, -C(CH₃)=CH-CH=CH-CO-OCH₃, -C(CH₃)=CH-CH=CH-CO-OC₂H₅, -C(CH₃)=CH-CH=C(COOCH₃)₂, -C(CH₃)=CH-CH=C(CN)-CO-OCH₃, -C(CH₃)=CH-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH₂, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -C(CH₃)=CH-(CH₂)₂-COOH, -C(CH₃)=CH-(CH₂)₂-CO-OCH₃, -C(CH₃)=CH-(CH₂)₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(COOCH₃)₂, -C(CH₃)=CH-CH₂-CH(COOC₂H₅)₂, -C(CH₃)=CH-CH₂-CH(CN)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CN)-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -C(CH₃)=CH-(CH₂)₂-CO-NH₂, -C(CH₃)=CH-(CH₂)₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-COOH, -C(CH₃)=CH-CH₂-CO-OCH₃, -C(CH₃)=CH-CH₂-CO-OC₂H₅, -C(CH₃)=C(COOCH₃)-CH₂-CO-OCH₃, -C(CH₃)=C(COOCH₃)-CH₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CO-NH₂, -C(CH₃)=CH-CH₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-CO-N(CH₃)₂.
wobei W für eine der folgenden Bedeutungen steht:
-CHO, -COCH₃, -COC₂H₅, -CO-n-C₃H₇, -CO-i-C₃H₇, -CO-n-C₄H₉, -CO-i-C₄H₉, -CO-s-C₄H₉, -CO-tert.-C₄H₉, -CO-CH₂CH=CH₂, -CO-CF₃, -COCCl₃, -COCH₂C≡CH, -CO-cyclopropyl, -CO-cyclobutyl, -CO-cyclo­ pentyl, -CO-cyclohexyl, -CO-CN, -CO-COOCH₃, -CO-COOC₂H₅, -CH=NH, -CH=NCH₃, -CH=NC₂H₅, -CH=N-n-C₃H₅, -CH=N-i-C₃H₅, -CH=N-n-C₄H₉, -CH=NCH₂CH=CH₂, -CH=NCH₂CH=CH₂-CH₃, -CH=NCH₂C≡CH, -CH=NCH₂C≡C-CH₃, -CH=N-cyclopropyl, -CH=N-cyclobutyl, -CH=N-cyclopentyl, -CH=N-cyclohexyl, -CH=N-cycloheptyl, -CH=N-CH₂-CH₂Cl, -CH=N-CH₂Cl, -CH=N-₆H₅, -CH=N-4-Br-C₆H₄, -CH=N-3-F-C₆H₄, -CH=N-4-F-C₆H₄, -CH=N-2-Cl-C₆H₄, -CH=N-3-Cl-C₆H₄, -CH=N-4-Cl-C₆H₄, -CH=N-2-Br-C₆H₄, -CH=N-2-F-C₆H₄, -CH=N-2-CH₃-C₆H₄, -CH=N-3-CH₃-C₆H₄, -CH=N-4-CH₃-C₆H₄, -CH=N-2-CF₃-C₆H₄, -CH=N-3-CF₃-C₆H₄, -CH=N-4-CF₃-C₆H₄, -CH=N-2-OCH₃-C₆H₄, -CH=N-3-OCH₃-C₆H₄, -CH=N-4-OCH₃-C₆H₄, -CH=N-4-NO₂-C₆H₄, -CH=N-4-CN-C₆H₄, -CH=N-2,4-(Cl,Cl)-C₆H₄, -CH=N-2,4-(CH₃,CH₃)-C₆H₄, -CH=N-CH₂OCH₃ -CH=N-CH₂OC₂H₅, -CH=N-CH₂CH₂OCH₃, -CH=N-CH₂CH₂OC₂H₅, -CH=N-OH, -CH=N-OCH₃, -CH=N-OC₂H₅, -CH=N-O-n-C₃H₇, -CH=N-O-i-C₃H₇, -CH=N-O-n-C₄H₉, -CH=N-O-i-C₄H₉, -CH=N-O-s-C₄H₉, -CH=N-O-tert.-C₄H₉, -CH=N-O-CH₂CH=CH₂, -CH=N-O-CH(CH₃)CH=CH₂, -CH=N-O-CH₂C≡CH, -CH=N-O-CH(CH₃)-C≡CH, -CH=N-O-CH₂-CH=CH-CH₃, -CH=N-O-CH₂-CH₂-Cl, -CH=N-O-CH₂-CH₂-F, -CH=N-O-CH₂-CF₃, -CH=N-O-CH₂-CH=CHCl, -CH=N-O-CH₂-CCl=CH₂, -CH=N-O-CH₂-CBr=CH₂, -CH=N-O-CH₂-CH=CCl-CH₃, -CH=N-OC(O)CH₃, -CH=N-OC(O)C₂H₅, -CH=N-O-CH₂-CN, -CH=N-O-CH₂-CH=CH-CH₂-O-CH₃, -CH=N-O-CH₂-CH=CH-CH₂-O-tert.-C₄H₉, -CH=N-O-(CH₂)₃-C₆H₅, -CH=N-O-(CH₂)₄-C₆H₅, -CH=N-O-(CH₂)₄-4-Cl-C₆H₄, -CH=N-O-(CH₂)₄-4-OCH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-CH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-C₆H₅, -CH=N-O-CH₂CH=CH-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CH-3-OCH₃-C₆H₄, -CH=N-O-(CH₂)₂CH=CH-4-F-C₆H₄, -CH=N-O-(CH₂)CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH₂CH=CHCH₂-4-OCH₃-C₆H₄, -CH=N-O-CH₂-CH=C(CH₃)-C₆H₅, -CH=N-O-(CH₂)₂CH=CH-3,4(Cl,Cl)-C₆H₃, -CH=N-O-(CH₂)₃C≡C-4-F-C₆H₄, -CH₂=N-OCHOCH₃, -CH=N-OC₂H₄OCH₃, -CH=N-OCH₂OC₂H₅, -CH=N-OCH(CH₃)OCH₃, -CH=N-OCH(CH₃)COOCH₃, -CH=N-OCH(CH₃)COO-n-C₄H₉, -CH=N-NH₂, -CH=N-NHCH₃, -CH=N-NHC₂H₅, -CH=N-NH-n-C₃H₇, -CH=N-NH-i-C₃H₇, -CH=N-NH-n-C₄H₉, -CH=N-NH-i-C₄H₉, -CH=N-NH-s-C₄H₉, -CH=N-NH-tert.-C₄H₉, -CH=N-NH-cyclopropyl, -CH=N-NH-cyclobutyl, -CH=N-NH-cyclopentyl, -CH=N-NH-cyclohexyl, -CH=N-NH-cycloheptyl, -CH=N-N(CH₃)₂, -CH=N-N(C₂H₅)₂, -CH=N-N(C₃H₇)₂, -CH=N-N(i-C₃H₇)(CH₃), -CH=N-NHCH₂-C=CH, -CH=N-NHCH₂-C≡CH, -CH=N-N(CH₃)-CH₂-C≡CH, -CH=N-NHCH₂CF₃, -CH=N-NH-CO-CH₃, -CH=N-NH-CO-CH₂H₅, -CH=N-NH-COOCH₃, -CH=N-NH-COOC₂H₅, -CH=N-NH-COO-tert.-C₄H₉, -CH=N-pyrrolidin-1-yl, -CH=N-piperidin-1-yl, -CH=N-morpholin-4-yl, -CH=N-NH-C₆H₅, -CH=N-NH-(4-Cl-C₆H₄), -CH=N-NH-(4-NO₂-C₆H₄), -CH=N-NH-(4-F-C₆H₄), -CH=N-NH-(4-CH₃O-C₆H₄), -CH=N-NH-(2,4-Cl₂-C₆H₃), -CH=N-NH-(2,4-(NO₂)₂-C₆H₃), -CH=N-NH-CO-NH₂, -CH=N-NH-CO-NHCH₃, -CH=N-NH-CO-NHC₂H₅, -CH=N-NH-CO-N(CH₃)₂, -CH=CH-COOH, -CH=CH-CO-OCH₃, -CH=CH-CO-OC₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-O-i-C₃H₇, -CH=CH-CO-O-n-C₄H₉, -CH=CH-CO-O-tert.-C₄H₉, -CH=CH-CO-O-cyclopropyl, -CH=CH-CO-O-cyclobutyl, -CH=CH-CO-O-cyclopentyl, -CH=CH-CO-O-cyclohexyl, -CH=CH-CO-O-cycloheptyl, -CH=C(CH₃)-COOH, -CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CO-O-n-C₃H₇, -CH=C(CH₃)-CO-O-i-C₃H₇, -CH=C(CH₃)-CO-O-n-C₄H₉, -CH=C(CH₃)-CO-O-tert.-C₄H₉, -CH=C(CH₃)-CO-O-cyclopropyl, -CH=C(CH₃)-CO-O-cyclobutyl, -CH=C(CH₃)-CO-O-cyclopentyl, -CH=C(CH₃)-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cycloheptyl, -CH=C(C₂H₅)-COOH, -CH=C(C₂H₅)-CO-OCH₃, -CH=C(C₂H₅)-CO-OC₂H₅, -CH=C(C₂H₅)-CO-O-n-C₃H₇, -CH=C(C₂H₅)-CO-O-i-C₃H₇, -CH=C(C₂H₅)-CO-O-n-C₄H₉, -CH=C(C₂H₅)-CO-O-tert.-C₄H₉, -CH=C(C₂H₅)-CO-O-cyclopropyl, -CH=C(C₂H₅)-CO-O-cyclobutyl, -CH=C(C₂H₅)-CO-O-cyclopentyl, -CH=C(C₂H₅)-CO-O-cyclohexyl, -CH=C(C₂H₅)-CO-O-cycloheptyl, -CH=C(Cl)-COOH, -CH=C(Cl)-CO-OCH₃, -CH=C(Cl)-CO-OC₂H₅, -CH=C(Cl)-CO-O-n-C₃H₇, -CH=C(Cl)-CO-O-i-C₃H₇, -CH=C(Cl)-CO-O-n-C₄H₉, -CH=C(Cl)-CO-O-tert.-C₄H₉, -CH=C(Cl)-CO-O-cyclopropyl, -CH=C(Cl)-CO-O-cyclobutyl, -CH=C(Cl)-CO-O-cyclopentyl, -CH=C(Cl)-CO-O-cyclohexyl, -CH=C(Cl)-CO-O-cycloheptyl, -CH=C(Br)-COOH, -CH=C(Br)-CO-OCH₃, -CH=C(Br)-CO-OC₂H₅, -CH=C(Br)-CO-O-n-C₃H₇, -CH=C(Br)-CO-O-i-C₃H₇, -CH=C(Br)-CO-O-n-C₄H₉, -CH=C(Br)-CO-O-tert.-C₄H₉, -CH=C(Br)-CO-O-cyclopropyl, -CH=C(Br)-CO-O-cyclobutyl, -CH=C(Br)-CO-O-cyclopentyl, -CH=C(Br)-CO-O-cyclohexyl, -CH=C(Br)-CO-O-cycloheptyl, -CH=C(CN)-COOH, -CH=C(CN)-CO-OCH₃, -CH=C(CN)-CO-OC₂H₅, -CH=C(CN)-CO-O-n-C₃H₇, -CH=C(CN)-CO-O-i-C₃H₇, -CH=C(CN)-CO-O-n-C₄H₉, -CH=C(CN)-CO-O-tert.-C₄H₉, -CH=C(CN)-CO-O-cyclopropyl, -CH=C(CN)-CO-O-cyclobutyl, -CH=C(CN)-CO-O-cyclopentyl, -CH=C(CN)-CO-O-cyclohexyl, -CH=C(CN)-CO-O-cycloheptyl, -CH=CH-CO-OCH₂-OCH₃, -CH=CH-CO-OCH₂-OC₂H₅, -CH=CH-CO-OCH₂-O-n-C₃H₅, -CH=CH-CO-OCH₂-O-i-C₃H₅, -CH=CH-CO-OCH(CH₃)-OCH₃, -CH=CH-CO-OCH(CH₃)-OC₂H₅, -CH=CH-CO-O-CH₂CH₂-OCH₃, -CH=CH-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-OCH₃, -CH=C(CH₃)-CO-OCH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-O-n-C₃H₅, -CH=C(CH₃)-CO-OCH₂-O-i-C₃H₅, -CH=C(CH₃)-CO-OCH(CH₃)-OCH₃, -CH=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CH₃)-CO-O-CH₂CH₂-OCH₃, -CH=C(CH₃)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-OCH₃, -CH=C(C₂H₅)-CO-OCH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-O-n-C₃H₅, -CH=C(O₂H₅)-CO-OCH₂-O-i-C₃H₅, -CH=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -CH=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OCH₃, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-OCH₃, -CH=C(Cl)-CO-OCH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-O-n-C₃H₅, -CH=C(Cl)-CO-OCH₂-O-i-C₃H₅, -CH=C(Cl)-CO-OCH(CH₃)-OCH₃, -CH=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Cl)-CO-O-CH₂CH₂-OCH₃, -CH=C(Cl)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-OCH₃, -CH=C(Br)-CO-OCH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-O-n-C₃H₅, -CH=C(Br)-CO-OCH₂-O-i-C₃H₅, -CH=C(Br)-CO-OCH(CH₃)-OCH₃, -CH=C(Br)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Br)-CO-O-CH₂CH₂-OCH₃, -CH=C(Br)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-OCH₃, -CH=C(CN)-CO-OCH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-O-n-C₃H₅, -CH=C(CN)-CO-OCH₂-O-i-C₃H₅, -CH=C(CN)-CO-OCH(CH₃)-OCH₃, -CH=C(CN)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CN)-CO-O-CH₂CH₂-OCH₃, -CH=C(CN)-CO-O-CH₂CH₂-OC₂H₅, -CH=CH-CO-OCH₂-CF₃, -CH=CH-CO-OCH₂-CCl₃, -CH=CH-CO-OCH₂-oxiranyl, -CH=CH-CO-O(CH₂)₃-Br, -CH=CH-CO-OCH₂-CH=CH₂, -CH=CH-CO-OCH₂-C≡CH, -CH=CH-CO-OCH₂-CN, -CH=CH-CO-O(CH₂)₂-CN, -CH=C(CH₃)-CO-OCH₂-CF₃, -CH=C(CH₃)-CO-OCH₂-CCl₃, -CH=C(CH₃)-CO-OCH₂-oxiranyl, -CH=C(CH₃)-CO-O(CH₂)₃-Br, -CH=C(CH₃)-CO-OCH₂-CH=CH₂, -CH=C(CH₃)-CO-OCH₂-C≡CH, -CH=C(CH₃)-CO-OCH₂-CN, -CH=C(CH₃)-CO-O(CH₂)₂-CN, -CH=C(C₂H₅)-CO-OCH₂-CF₃, -CH=C(C₂H₅)-CO-OCH₂-CCl₃, -CH=C(C₂H₅)-CO-OCH₂-oxiranyl, -CH=C(C₂H₅)-CO-O(CH₂)₃-Br, -CH=C(C₂H₅)-CO-OCH₂-CH=CH₂, -CH=C(C₂H₅)-CO-OCH₂-C≡CH, -CH=C(C₂H₅)-CO-OCH₂-CN, -CH=C(C₂H₅)-CO-O(CH₂)₂-CN, -CH=C(Cl)-CO-OCH₂-CF₃, -CH=C(Cl)-CO-OCH₂-CCl₃, -CH=C(Cl)-CO-OCH₂-oxiranyl, -CH=C(Cl)-CO-O(CH₂)₃-Br, -CH=C(Cl)-CO-OCH₂-CH=CH₂, -CH=C(Cl)-CO-OCH₂-C≡CH, -CH=C(Cl)-CO-OCH₂-CN, -CH=C(Cl)-CO-O(CH₂)₂-CN, -CH=C(Br)-CO-OCH₂-CF₃, -CH=C(Br)-CO-OCH₂-CCl₃, -CH=C(Br)-CO-OCH₂-oxiranyl, -CH=C(Br)-CO-O(CH₂)₃-Br, -CH=C(Br)-CO-OCH₂-CH=CH₂, -CH=C(Br)-CO-OCH₂-C≡CH, -CH=C(Br)-CO-OCH₂-CN, -CH=C(Br)-CO-O(CH₂)₂-CN, -CH=C(CN)-CO-OCH₂-CF₃, -CH=C(CN)-CO-OCH₂-CCl₃, -CH=C(CN)-CO-OCH₂-oxiranyl, -CH=C(CN)-CO-O(CH₂)₃-Br, -CH=C(CN)-CO-OCH₂-CH=CH₂, -CH=C(CN)-CO-OCH₂-C≡CH, -CH=C(CN)-CO-OCH₂-CN, -CH=C(CN)-CO-O(CH₂)₂-CN, -CH=CH-CO-CH₃, -CH=CH-CO-C₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-i-C₃H₇, -CH=CH-CO-n-C₄H₉, -CH=CH-CO-tert.-C₄H₉, -CH=CH-CO-CH₂Cl, -CH=CH-CO-CH₂Br, -CH=CH-CO-CHCl₂, -CH=CH-CO-CH₂-OCH₃, -CH=CH-CO-CH(OCH₃)₂, -CH=CH-CO-CH₂-SCH₃, -CH=C(CH₃)-CO-CH₃, -CH=C(CH₃)-CO-C₂H₅, -CH=C(CH₃)-CO-n-C₃H₇, -CH=C(CH₃)-CO-i-C₃H₇, -CH=C(CH₃)-CO-n-C₄H₉, -CH=C(CH₃)-CO-tert.-C₄H₉, -CH=C(CH₃)-CO-CH₂Cl, -CH=C(CH₃)-CO-CH₂Br, -CH=C(CH₃)-CO-CHCl₂, -CH=C(CH₃)-CO-CH₂-OCH₃, -CH=C(CH₃)-CO-CH(OCH₃)₂, -CH=C(CH₃)-CO-CH₂-SCH₃, -CH=C(C₂H₅)-CO-CH₃, -CH=C(C₂H₅)-CO-C₂H₅, -CH=C(C₂H₅)-CO-n-C₃H₇, -CH=C(C₂H₅)-CO-i-C₃H₇, -CH=C(C₂H₅)-CO-n-C₄H₉, -CH=C(C₂H₅)-CO-tert.-C₄H₉, -CH=C(C₂H₅)-CO-CH₂Cl, -CH=C(C₂H₅)-CO-CH₂Br, -CH=C(C₂H₅)-CO-CHCl₂, -CH=C(C₂H₅)-CO-CH₂-OCH₃, -CH=C(C₂H₅)-CO-CH(OCH₃)₂, -CH=C(C₂H₅)-CO-CH₂-SCH₃, -CH=C(Cl)-CO-CH₃, -CH=C(Cl)-CO-C₂H₅, -CH=C(Cl)-CO-n-C₃H₇, -CH=C(Cl)-CO-i-C₃H₇, -CH=C(Cl)-CO-n-C₄H₉, -CH=C(Cl)-CO-tert.-C₄H₉, -CH=C(Cl)-CO-CH₂Cl, -CH=C(Cl)-CO-CH₂Br, -CH=C(Cl)-CO-CHCl₂, -CH=C(Cl)-CO- CH₂-OCH₃, -CH=C(Cl)-CO-CH(OCH₃)₂, -CH=C(Cl)-CO-CH₂-SCH₃, -CH=C(Br)-CO-CH₃, -CH=C(Br)-CO-C₂H₅, -CH=C(Br)-CO-n-C₃H₇, -CH=C(Br)-CO-i-C₃H₇, -CH=C(Br)-CO-n-C₄H₉, -CH=C(Br)-CO-tert.-C₄H₉, -CH=C(Br)-CO-CH₂Cl, -CH=C(Br)-CO-CH₂Br, -CH=C(Br)-CO-CHCl₂, -CH=C(Br)-CO-CH₂-OCH₃, -CH=C(Br)-CO-CH(OCH₃)₂, -CH=C(Br)-CO-CH₂-SCH₃, -CH=C(CN)-CO-CH₃, -CH=C(CN)-CO-C₂H₅, -CH=C(CN)-CO-n-C₃H₇, -CH=C(CN)-CO-i-C₃H₇, -CH=C(CN)-CO-n-C₄H₉, -CH=C(CN)-CO-tert.-C₄H₉, -CH=C(CN)-CO-CH₂Cl, -CH=C(CN)-CO-CH₂Br, -CH=C(CN)-CO-CHCl₂, -CH=C(CN)-CO-CH₂-OCH₃, -CH=C(CN)-CO-CH(OCH₃)₂, -CH=C(CN)-CO-CH₂-SCH₃, -CH=CH-CO-C₆H₅, -CH=CH-CO-(4-Cl-C₆H₄), -CH=C(CH₃)-CO-C₆H₅, -CH=C(CH₃)-CO-(4-Cl-C₆H₄), -CH=C(C₂H₅)-CO-C₆H₅, -CH=C(C₂H₅)-CO-(4-Cl-C₆H₄), -CH=C(Cl)-CO-C₆H₅, -CH=C(Br)-CO-C₆H₅, -CH=C(CN)-CO-C₆H₅, -CH=CH-CO-NH₂, -CH=CH-CO-NHCH₃, -CH=CH-CO-N(CH₃)₂, -CH=CH-CO-NH-C₂H₅, -CH=CH-CO-N(C₂H₅)₂, -CH=CH-CO-NH-n-C₃H₇, -CH=CH-CO-NH-i-C₃H₇, -CH=CH-CO-NH-tert.-C₄H₉, -CH=CH-CO-NH-cyclopropyl, -CH=CH-CO-NH-cyclobutyl, -CH=CH-CO-NH-cyclopentyl, -CH=CH-CO-NH-cyclohexyl, -CH=CH-CO-cycloheptyl, -CH=CH-CO-NH-cyclooctyl, -CH=CH-CO-pyrrolidin-1-yl, -CH=CH-CO-piperidin-1-yl, -CH=CH-CO-morpholin-4-yl, -CH=CH-CO-NH-CH₂CH=CH₂, -CH=CH-CO-NH-CH₂C≡CH, -CH=CH-CO-N(CH₃)-CH₂C≡CH, -CH=CH-CO-NH-(CH₂)₂Cl, -CH=CH-CO-NH-C₆H₅, -CH=C(CH₃)-CO-NH₂, -CH=C(CH₃)-CO-NHCH₃, -CH=C(CH₃)-CO-N(CH₃)₂, -CH=C(CH₃)-CO-NH-C₂H₅, -CH=C(CH₃)-CO-N(C₂H₅)₂, -CH=C(CH₃)-CO-NH-n-C₃H₇, -CH=C(CH₃)-CO-NH-i-C₃H₇, -CH=C(CH₃)-CO-NH-tert.-C₄H₉, -CH=C(CH₃)-CO-NH-cyclopropyl, -CH=C(CH₃)-CO-NH-cyclobutyl, -CH=C(CH₃)-CO-NH-cyclopentyl, -CH=C(CH₃)-CO-NH-cyclohexyl, -CH=C(CH₃)-CO-NH-cycloheptyl, -CH=C(CH₃)-CO-NH-cyclooctyl, -CH=C(CH₃)-CO-pyrolidin-1-yl, -CH=C(CH₃)-CO-piperidin-1-yl, -CH=C(CH₃)-CO-morpholin-4-yl, -CH=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -CH=C(CH₃)-CO-NH-CH₂C≡CH, -CH=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CH₃)-CO-NH-(CH₂)₂Cl, -CH=C(CH₃)-CO-NH-C₆H₅, -CH=C(C₂H₅)-CO-NH₂, -CH=C(C₂H₅)-CO-NHCH₃, -CH=C(C₂H₅)-CO-N(CH₃)₂, -CH=C(C₂H₅)-CO-NH-C₂H₅, -CH=C(C₂H₅)-CO-N(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-n-C₃H₇, -CH=C(C₂H₅)-CO-NH-i-C₃H₇, -CH=C(C₂H₅)-CO-NH-tert.-C₄H₉, -CH=C(C₂H₅)-CO-NH-cyclopropyl, -CH=C(C₂H₅)-CO-NH-cyclobutyl, -CH=C(C₂H₅)-CO-NH-cyclopentyl, -CH=C(C₂H₅)-CO-NH-cyclohexyl, -CH=C(C₂H₅)-CO-NH-cycloheptyl, -CH=C(C₂H₅)-CO-NH-cyclooctyl, -CH=C(C₂H₅)-CO-pyrrolidin-1-yl, -CH=C(C₂H₅)-CO-piperidin-1-yl, -CH=C(C₂H₅)-CO-morpholin-4-yl, -CH=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-CH₂C≡CH, -CH=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -CH=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -CH=C(C₂H₅)-CO-NH-C₆H₅, -CH=C(Cl)-CO-NH₂, -CH=C(Cl)-CO-NHCH₃, -CH=C(Cl)-CO-N(CH₃)₂, -CH=C(Cl)-CO-NH-C₂H₅, -CH=C(Cl)-CO-N(C₂H₅)₂, -CH=C(Cl)-CO-NH-n-C₃H₇, -CH=C(Cl)-CO-NH-i-C₃H₇, -CH=C(Cl)-CO-NH-tert.-C₄H₉, -CH=C(Cl)-CO-NH-cyclopropyl, -CH=C(Cl)-CO-NH-cyclobutyl, -CH=C(Cl)-CO-NH-cyclopentyl, -CH=C(Cl)-CO-NH-cyclohexyl, -CH=C(Cl)-CO-NH-cycloheptyl, -CH=C(Cl)-CO-NH-cyclooctyl, -CH=C(Cl)-CO-pyrrolidin-1-yl, -CH=C(Cl)-CO-piperidin-1-yl, -CH=C(Cl)-CO-morpholin-4-yl, -CH=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -CH=C(Cl)-CO-NH-CH₂C≡CH, -CH=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Cl)-CO-NH-(CH₂)₂Cl, -CH=C(Cl)-CO-NH-C₆H₅, -CH=C(Br)-CO-NH₂, -CH=C(Br)-CO-NHCH₃, -CH=C(Br)-CO-N(CH₃)₂, -CH=C(Br)-CO-NH-C₂H₅, -CH=C(Br)-CO-N(C₂H₅)₂, -CH=C(Br)-CO-NH-n-C₃H₇, -CH=C(Br)-CO-NH-i-C₃H₇, -CH=C(Br)-CO-NH-tert.-C₄H₉, -CH=C(Br)-CO-NH-cyclopropyl, -CH=C(Br)-CO-NH-cyclobutyl, -CH=C(Br)-CO-NH-cyclopentyl, -CH=C(Br)-CO-NH-cyclohexyl, -CH=C(Br)-CO-NH-cycloheptyl, -CH=C(Br)-CO-NH-cyclooctyl, -CH=C(Br)-CO-pyrrolidin-1-yl, -CH=C(Br)-CO-piperidin-1-yl, -CH=C(Br)-CO-morpholin-4-yl, -CH=C(Br)-CO-NH-CH₂CH=C(Br)₂, -CH=C(Br)-CO-NH-CH₂C≡CH, -CH=C(Br)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Br)-CO-NH-(CH₂)₂Cl, -CH=C(Br)-CO-NH-C₆H₅, -CH=C(CN)-CO-NH₂, -CH=C(CN)-CO-NHCH₃, -CH=C(CN)-CO-N(CH₃)₂, -CH=C(CN)-CO-NH-C₂H₅, -CH=C(CN)-CO-N(C₂H₅)₂, -CH=C(CN)-CO-NH-n-C₃H₇, -CH=C(CN)-CO-NH-i-C₃H₇, -CH=C(CN)-CO-NH-tert.-C₄H₉, -CH=C(CN)-CO-NH-cyclopropyl, -CH=C(CN)-CO-NH-cyclobutyl, -CH=C(CN)-CO-NH-cyclopentyl, -CH=C(CN)-CO-NH-cyclohexyl, -CH=C(CN)-CO-NH-cycloheptyl, -CH=C(CN)-CO-NH-cyclooctyl, -CH=C(CN)-CO-pyrrolidin-1-yl, -CH=C(CN)-CO-piperidin-1-yl, -CH=C(CN)-CO-morpholin-4-yl, -CH=C(CN)-CO-NH-CH₂CH=C(CN)₂, -CH=C(CN)-CO-NH-CH₂C≡CH, -CH=C(CN)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CN)-CO-NH-(CH₂)₂Cl, -CH=C(CN)-CO-NH-C₆H₅, -CH=CH-CO-SCH₃, -CH=CH-CO-SC₂H₅, -CH=CH-CO-S-n-C₃H₇, -CH=CH-CO-S-i-C₃H₇, -CH=CH-CO-S-n-C₄H₉, -CH=CH-CO-S-tert.-C₄H₉, -CH=C(CH₃)-CO-SCH₃, -CH=C(CH₃)-CO-SC₂H₅, -CH=C(CH₃)-CO-S-n-C₃H₇, -CH=C(CH₃)-CO-S-i-C₃H₇, -CH=C(CH₃)-CO-S-n-C₄H₉, -CH=C(CH₃)-CO-S-tert.-C₄H₉, -CH=C(C₂H₅)-CO-SCH₃, -CH=C(C₂H₅)-CO-SC₂H₅, -CH=C(C₂H₅)-CO-S-n-C₃H₇, -CH=C(C₂H₅)-CO-S-i-C₃H₇, -CH=C(C₂H₅)-CO-S-n-C₄H₉, -CH=C(C₂H₅)-CO-S-tert.-C₄H₉, -CH=C(Cl)-CO-SCH₃, -CH=C(Cl)-CO-SC₂H₅, -CH=C(Cl)-CO-S-n-C₃H₇, -CH=C(Cl)-CO-S-i-C₃H₇, -CH=C(Cl)-CO-S-n-C₄H₉, -CH=C(Cl)-CO-S-tert.-C₄H₉, -CH=C(Br)-CO-SCH₃, -CH=C(Br)-CO-SC₂H₅, -CH=C(Br)-CO-S-n-C₃H₇, -CH=C(Br)-CO-S-i-C₃H₇, -CH=C(Br)-CO-S-n-C₄H₉, -CH=C(Br)-CO-S-tert.-C₄H₉, -CH=C(CN)-CO-SCH₃, -CH=C(CN)-CO-SC₂H₅, -CH=C(CN)-CO-S-n-C₃H₇, -CH=C(CN)-CO-S-i-C₃H₇, -CH=C(CN)-CO-S-n-C₄H₉, -CH=C(CN)-CO-S-tert.-C₄H₉, -CH=C(COCH₃)-CO-OCH₃, -CH=C(COC₂H₅)-CO-OCH₃, -CH=C(CO-n-C₃H₇)-CO-OCH₃, -CH=C(COCH₃)-CO-OC₂H₅, -CH=C(COC₂H₅)-CO-OC₂H₅, -CH=C(CO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COCH₃)-CO-O-n-C₃H₇, -CH=C(COC₂H₅)-CO-O-n-C₃H₇, -CH=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-OCH₃, -CH=C(CF₃)-CO-OC₂H₅, -CH=C(CF₃)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-O-i-C₃H₇, -CH=C(CF₃)-CO-O-n-C₄H₉, -CH=C(CF₃)-CO-O-tert.-C₄H₉, -CH=C(COOCH₃)₂, -CH=C(COOC₂H₅)₂, -CH=C(COOCH₃)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)-CO-OCH₃, -CH=C(COO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)₂, -CH=CH-CH=CH-COOH, -CH=CH-CH=CH-CO-OCH₃, -CH=CH-CH=CH-CO-OC₂H₅, -CH=CH-CH=C(COOCH₃)₂, -CH=CH-CH=C(CN)-CO-OCH₃, -CH=CH-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-OCH₃, -CH=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CH=C(Cl)-CO-OCH₃, -CH=C(CH₃)-CH=C(Br)-CO-OCH₃, -CH=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-NH₂, -CH=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -CH=CH-(CH₂)₂-COOH, -CH=CH-(CH₂)₂-CO-OCH₃, -CH=CH-(CH₂)₂-CO-OC₂H₅, -CH=CH-CH₂-CH(COOCH₃)₂, -CH=CH-CH₂-CH(COOC₂H₅)₂, -CH=CH-CH₂-CH(CN)-CO-OCH₃, -CH=CH-CH₂-CH(CN)-CO-OC₂H₅, -CH=CH-CH₂-CH(CH₃)-CO-OCH₃, -CH=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -CH=CH-(CH₂)₂-CO-NH₂, -CH=CH-(CH₂)₂-CO-NH-CH₃, -CH=CH-CH₂-COOH, -CH=CH-CH₂-CO-OCH₃, -CH=CH-CH₂-CO-OC₂H₅, -CH=C(COOCH₃)-CH₂-CO-OCH₃, -CH=C(COOCH₃)-CH₂-CO-OC₂H₅, -CH=CH-CH₂-CO-NH₂, -CH=CH-CH₂-CO-NH-CH₃, -CH=CH-CH₂-CO-N(CH₃)₂, -CH(OCH₃)₂, -CH(SCH₃)₂, -CH(OC₂H₅)₂, -CH(SC₂H₅)₂, -CH(O-n-C₃H₇)₂, -CH(O-i-C₃H₇)₂, -CH(S-n-C₃H₇)₂, -CH(S-i-C₃H₇)₂, -CH(O-n-C₄H₉)₂, -CH(O-i-C₄H₉)₂, -CH(O-s-C₄H₉)₂, -CH(O-tert.-C₄H₉)₂, -CH(S-n-C₄H₉)₂, -CH(S-i-C₄H₉)₂, -CH(S-s-C₄H₉)₂, -CH(S-tert.-C₄H₉)₂, -CH(OC₅H₁₁)₂, 1,3-Dioxolan-2-yl, 1,3-Dithio­ lan-2-yl, 1,3-Oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 4-Methyl-1,3-dithiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 5-Methyl-1,3-oxathiolan-2-yl, 4-Ethyl-1,3-dioxolan-2-yl, 4-Ethyl- 1,4-dithiolan-2-yl, 4-Ethyl-1,3-oxathiolan-2-yl, 5-Ethyl-1,3-oxa­ thiolan-2-yl, 4,5-Dimethyl-1,3-dioxolan-2-yl, 4,4-Dimethyl-1,3- dioxolan-2-yl, 4,5-Dimethyl-1,3-dithiolan-2-yl, 5,5-Dimethyl-1,3- dithiolan-2-yl, 4,5-Dimethyl-1,3-oxathiolan-2-yl, 5,5-Dimethyl- 1,3-oxathiolan-2-yl, 4,4-Dimethyl-1,3-oxathiolan-2-yl, 4-Vinyl- 1,3-dioxolan-2-yl, 4-Vinyl-1,3-dithiolan-2-yl, 4-Vinyl-1,3-oxa­ thiolan-2-yl, 5-Vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3- dioxolan-2-yl, 4-Chlormethyl-1,3-dithiolan-2-yl, 4-Chlormethyl- 1,3-oxathiolan-2-yl, 5-Chlormethyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-1,3-dithio­ lan-2-yl, 4-Hydroxymethyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl- 1,3-oxathiolan-2-yl, 4-Methoxymethyl-1,3-dioxolan-2-yl, 4-Allyl­ oxymethyl-1,3-dioxolan-2-yl, 4-Propargyloxymethyl-1,3-dioxolan- 2-yl, 4-Acetoxymethyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-1,3-dithiolan-2-yl, 4-Propargyl­ oxymethyl-1,3-dithiolan-2-yl, 4-Acetoxymethyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl-1,3-oxathiolan-2-yl, 5-Allyloxy­ methyl-1,3-oxathiolan-2-yl, 4-Propargyloxymethyl-1,3-oxathiolan-2-yl, 5-Propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxymethyl- 1,3-oxathiolan-2-yl, 5-Acetoxymethyl-1,3-oxathiolan-2-yl, 4-Methylthiomethyl-1,3-dioxolan-2-yl, 4-Methylthiomethyl-1,3- dithiolan-2-yl, 4-Carboxy-1,3-dioxolan-2-yl, 4-Carboxy-1,3- dithiolan-2-yl, 4-Methoxycarbonyl-1,3-dioxolan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-1,3-dithiolan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-4-methyl- 1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-di­ thiolan-2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-1,3- dithiolan-2-yl, 1,3-Dioxan-2-yl, 1,3-Dithian-2-yl, 1,3-Oxathian- 2-yl, 5-Methyl-1,3-dioxan-2-yl, 5-Methyl-1,3-dithian-2-yl, 5-Methyl-1,3-oxathian-2-yl, 5,5-Dimethyl-1,3-dioxan-2-yl, 4,6-Dimethyl- 1,3-dioxan-2-yl, 4,4-Dimethyl-1,3-dioxan-2-yl, 5,5-Dimethyl- 1,3-dithian-2-yl, 4,6-Dimethyl-1,3-dithian-2-yl, 4,4-Dimethyl- 1,3-dithian-2-yl, 5,5-Dimethyl-1,3-oxathian-2-yl, 4,4-Dimethyl- 1,3-oxathian-2-yl, 6,6-Dimethyl-1,3-oxathian-2-yl, 4-Hydroxymethyl-1,3-dioxan-2-yl, 4-Methoxymethyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-1,3-dithian-2-yl, 4-Methoxymethyl-1,3-dithian-2-yl, 4-Allyloxymethyl-1,3-dithian-2-yl, 4-Acetoxymethyl- 1,3-dithian-2-yl, 4-Chlormethyl-1,3-dioxan-2-yl, 4-Chlormethyl- 1,3-dithian-2-yl, 1,3-Dioxepan-2-yl, 1,3-Dithiepan-2-yl, 1,3-Dioxep-5-en-2-yl, 4-Methoxycarbonyl-1,3-dioxan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-1,3-dithian-2-yl, 4-n-Butoxycarbonyl-1,3-dithian-2-yl, 4-Methoxycarbonyl-4- methyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-4-methyl- 1,3-dithian-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithian-2-yl, -C(CH₃)(OCH₃)₂, -C(CH₃)(SCH₃)₂, -C(CH₃)(OC₂H₅)₂, -C(CH₃)(SC₂H₅)₂, -C(CH₃)(O-n-C₃H₇)₂, -C(CH₃)(O-i-C₃H₇)₂, -C(CH₃)(S-n-C₃H₇)₂, -C(CH₃)(S-i-C₃H₇)₂, -C(CH₃)(O-n-C₄H₉)₂, -C(CH₃)(O-i-C₄H₉)₂, -C(CH₃)(O-s-C₄H₉)₂, -C(CH₃)(O-tert.-C₄H₉)₂, -C(CH₃)(S-n-C₄H₉)₂, -C(CH₃)(S-i-C₄H₉)₂, -C(CH₃)(S-s-C₄H₉)₂, -C(CH₃)(S-tert.-C₄H₉)₂, -C(CH₃)(O-n-C₅H₁₁)′′, 2-Methyl-1,3-dioxolan-2-yl, 2-Methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-oxathiolan-2-yl, 2,4-Dimethyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-1,3- oxathiolan-2-yl, 2,5-Dimethyl-1,3-oxathiolan-2-yl, 4-Ethyl-2- methyl-1,3-dioxolan-2-yl, 4-Ethyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Ethyl-2-methyl-1,3- oxathiolan-2-yl, 2,4,5-Trimethyl-1,3-dioxolan-2-yl, 2,4,4-Trimethyl- 1,3-dioxolan-2-yl, 2,4,5-Trimethyl-1,3-dithiolan-2-yl, 2,4,4-Trimethyl-1,3-dithiolan-2-yl, 2,4,5-Trimethyl-1,3-oxathiolan-2-yl, 2,4,4-Trimethyl-1,3-oxathiolan-2-yl, 2-Methyl-4-vinyl- 1,3-dioxolan-2-yl, 2-Methyl-4-vinyl-1,3-dithiolan-2-yl, 2-Methyl- 4-vinyl-1,3-oxathiolan-2-yl, 2-Methyl-5-vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-dioxolan-2-yl, 4-Chlormethyl-2- methyl-1,3-dithiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl- 2-methyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-2- methyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dioxolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxy- 2-methyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dithiolan-2-yl, 4-Acetoxy-2- methyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl- 2-methyl-1,3-oxathiolan-2-yl, 5-Allyloxymethyl-2- methyl-1,3-oxathiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3- oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxy-2-methyl-1,3-oxathiolan-2-yl, 5-Acetoxy-2-methyl- 1,3-oxathiolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dioxolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-2- methyl-1,3-dioxolan-2-yl, 4-Carboxy-2-methyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-2- methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl- 2-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-2- methyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-ethoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4- ethoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-n-butoxy­ carbony-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl-1,3- dithiolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-dioxan-2-yl, 2-Methyl-1,3-dithian-2-yl, 2-Methyl-1,3-oxathian-2-yl, 2,5- Dimethyl-1,3-dioxan-2-yl, 2,5-Dimethyl-1,3-dithian-2-yl, 2,5-Dimethyl- 1,3-oxathian-2-yl, 2,5,5-Trimethyl-1,3-dioxan-2-yl, 2,4,6- Trimethyl-1,3-dioxan-2-yl, 2,2,4-Trimethyl-1,3-dioxan-2-yl, 2,5,5-Trimethyl-1,3-dithian-2-yl, 2,4,6-Trimethyl-1,3-dithian-2-yl, 2,4,4-Trimethyl-1,3-dithian-2-yl, 2,5,5-Trimethyl-1,3-oxathian-2-yl, 2,4,4-Trimethyl-1,3-oxathian-2-yl, 2,6,6-Trimethyl- 1,3-oxathian-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-2- methyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dithian-2-yl, 4-Methoxymethyl-2- methyl-1,3-dithian-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithian-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dithian-2-yl, 4-Chlormethyl-2- methyl-1,3-dioxan-2-yl, 4-Chlormethyl-2-methyl-1,3-dithian-2-yl, -C(CH₃)=NH, -C(CH₃)=N-CH₃, -C(CH₃)=N-C₂H₅, -C(CH₃)=N-n-C₃H₇, -(CH₃)=N-i-C₃H₇, -C(CH₃)=N-n-C₄H₉, -C(CH₃)=N-CH₂CH=CH₂, -C(CH₃)=N-CH₂CH=CH₂-CH₃, -C(CH₃)=N-CH₂C≡CH, -C(CH₃)=N-CH₂C≡C-CH₃, -C(CH₃)=N-cyclopropyl, -C(CH₃)=N-cyclobutyl, -C(CH₃)=N-cyclopentyl, -C(CH₃)=N-cyclohexyl, -C(CH₃)=N-cycloheptyl, -C(CH₃)=N-CH₂-CH₂Cl, -C(CH₃)=N-CH₂Cl, -C(CH₃)=N-C₆H₅, -C(CH₃)=N-(2-F-C₆H₄), -C(CH₃)=N-(3-F-C₆H₄), -C(CH₃)=N-(4-F-C₆H₄), -C(CH₃)=N-(2-Cl-C₆H₄), -C(CH₃)=N-(3-Cl-C₆H₄), -C(CH₃)=N-(4-Cl-C₆H₄), -C(CH₃)=N-(2-CH₃-C₆H₄), -C(CH₃)=N-(3-CH₃-C₆H₄), -C(CH₃)=N-(4-CH₃-C₆H₄), -C(CH₃)=N-(2-CF₃-C₆H₄), -C(CH₃)=N-(3-CF₃-C₆H₄), -C(CH₃)=N-(4-CF₃-C₆H₄), -C(CH₃)=N-(2-OCH₃-C₆H₄), -C(CH₃)=N-(3-OCH₃-C₆H₄), -C(CH₃)=N-(4-OCH₃-C₆H₄), -C(CH₃)=N-(4-NO₂-C₆H₄), -C(CH₃)=N-(4-CN-C₆H₄), -C(CH₃)=N-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-(2,4-(CH₃)₂-C₆H₃), -C(CH₃)=N-CH₂-OCH₃, -C(CH₃)=N-CH₂-OC₂H₅, -C(CH₃)=N-CH₂CH₂-OCH₃, -C(CH₃)=N-CH₂CH₂-OC₂H₅, -C(CH₃)=N-OH, -C(CH₃)=N-OCH₃, -C(CH₃)=N-OC₂H₅, -C(CH₃)=N-O-n-C₃H₇, -C(CH₃)=N-O-i-C₃H₇, -C(CH₃)=N-O-n-C₄H₉, -C(CH₃)=N-O-i-C₄H₉, -C(CH₃)=N-O-s-C₄H₉, -C(CH₃)=N-O-tert.-C₄H₉, -C(CH₃)=N-OCH₂-CH=CH₂, -C(CH₃)=N-OCH(CH₃)-CH=CH₂, -C(CH₃)=N-OCH₂-C≡CH, -C(CH₃)=N-CH(CH₃)-C≡CH, -C(CH₃)=N-OCH₂-CH=C-CH₃, -C(CH₃)=N-OCH₂CH₂-Cl, -C(CH₃)=N-OCH₂CH₂-F, -C(CH₃)=N-OCH₂-CF₃, -C(CH₃)=N-OCH₂-CH=CHCl, -C(CH₃)=N-OCH₂-C(Cl)=CH₂, -C(CH₃)=N-OCH₂-C(Br)=CH₂, -C(CH₃)=N-OCH₂-CH=C(Cl)-CH₃, -C(CH₃)=N-O-CO-CH₃, -C(CH₃)=N-O-CO-C₂H₅, -C(CH₃)=N-OCH₂-CN, -C(CH₃)=N-OCH₂-CH=CH-CH₂-OCH₃, -C(CH₃)=N-OCH₂-CH=CH-CH₂-O-tert.-C₄H₉, -C(CH₃)=N-O-(CH₂)₃-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-(4-Cl-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-C₆H₅, -C(CH₃)=N-OCH₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(3-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-CH₂-(4-CH₃O-C₆H₄), -C(CH₃)=N-OCH₂-CH=C(CH₃)-C₆H₅, -C(CH₃)=N-O-(CH₂)₂-CH=CH-(3,4-Cl₂-C₆H₃), -C(CH₃)=N-O-(CH₂)₃-C≡C-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-OCH₃, -C(CH₃)=N-OCH₂CH₂-OCH₃, -C(CH₃)=N-OCH₂-OC₂H₅, -C(CH₃)=N-OCH(CH₃)-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=N-NH₂, -C(CH₃)=N-NH-CH₃, -C(CH₃)=N-NH-C₂H₅, -C(CH₃)=N-NH-n-C₃H₇, -C(CH₃)=N-NH-i-C₃H₇, -C(CH₃)=N-NH-n-C₄H₉, -C(CH₃)=N-NH-i-C₄H₉, -C(CH₃)=N-NH-s-C₄H₉, -C(CH₃)=N-NH-tert.-C₄H₉, -C(CH₃)=N-NH-cyclopropyl, -C(CH₃)=N-NH-cyclobutyl, -C(CH₃)=N-NH-cyclopentyl, -C(CH₃)=N-NH-cyclohexyl, -C(CH₃)=N-NH-cycloheptyl, -C(CH₃)=N-N(CH₃)₂, -C(CH₃)=N-N(C₂H₅)₂, -C(CH₃)=N-N(n-C₃H₇)₂, -C(CH₃)=N-N(i-C₃H₇)₂, -C(CH₃)=N-NH-CH₂-C=CH, -C(CH₃)=N-NH-CH₂-C≡CH, -C(CH₃)=N-N(CH₃)-CH₂-C≡CH, -C(CH₃)=N-NH-CH₂CF₃, -C(CH₃)=N-NH-CO-CH₃, -C(CH₃)=N-NH-CO-C₂H₅, -C(CH₃)=N-NH-CO-OCH₃, -C(CH₃)=N-NH-CO-OC₂H₅, -C(CH₃)=N-NH-CO-O-tert.-C₄H₉, -C(CH₃)=N-pyrrolidin-1-yl, -C(CH₃)=N-piperidin-1-yl, -C(CH₃)=N-morpholin-4-yl, -C(CH₃)=N-NH-C₆H₅, -C(CH₃)=N-NH-(4-Cl-C₆H₄), -C(CH₃)=N-NH-(4-NO₂-C₆H₄), -C(CH₃)=N-NH-(4-F-C₆H₄), -C(CH₃)=N-NH-(4-CH₃O-C₆H₄), -C(CH₃)=N-NH-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-NH-(2,4-(NO₂)₂-C₆H₃), -C(CH₃)=N-NH-CO-NH₂, -C(CH₃)=N-NH-CO-NHCH₃, -C(CH₃)=N-NH-CO-NHC₂H₅, -C(CH₃)=N-NH-CO-N(CH₃)₂, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=CH-CO-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -(CH₃)=CH-CO-O-n-C₄H₉, -C(CH₃)=CH-CO-O-tert.-C₄H₉, -C(CH₃)=CH-CO-O-cyclopropyl, -C(CH₃)=CH-CO-O-cyclobutyl, -C(CH₃)=CH-CO-O-cyclopentyl, -C(CH₃)=CH-CO-O-cyclohexyl, -C(CH₃)=CH-CO-O-cycloheptyl, -C(CH₃)=C(CH₃)-COOH, -C(CH₃)=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-cyclopropyl, -C(CH₃)=C(CH₃)-CO-O-cyclobutyl, -C(CH₃)=C(CH₃)-CO-O-cyclopentyl, -C(CH₃)=C(CH₃)-CO-O-cyclohexyl, -C(CH₃)=C(CH₃)-CO-O-cycloheptyl, -C(CH₃)=C(C₂H₅)-COOH, -C(CH₃)=C(C₂H₅)-CO-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-cyclo­ propyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-O- cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-O-cycloheptyl, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-O-n-C₄H₉, -C(CH₃)=C(Cl)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-O-cyclopropyl, -C(CH₃)=C(Cl)-CO-O-cyclobutyl, -C(CH₃)=C(Cl)-CO-O-cyclopentyl, -C(CH₃)=C(Cl)-CO-O-cyclohexyl, -C(CH₃)=C(Cl)-CO-O-cycloheptyl, -C(CH₃)=C(Br)-COOH, -C(CH₃)=C(Br)-CO-OCH₃, -C(CH₃)=C(Br)-CO-OC₂H₅, -C(CH₃)=C(Br)-CO-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-O-n-C₄H₉, -C(CH₃)=C(Br)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-O-cyclopropyl, -C(CH₃)=C(Br)-CO-O-cyclobutyl, -C(CH₃)=C(Br)-CO-O-cyclopentyl, -C(CH₃)=C(Br)-CO-O-cyclohexyl, -C(CH₃)=C(Br)-CO-O-cycloheptyl, -C(CH₃)=C(CN)-COOH, -C(CH₃)=C(CN)-CO-OCH₃, -C(CH₃)=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CN)-CO-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-O-n-C₄H₉, -C(CH₃)=C(CN)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-O-cyclopropyl, -C(CH₃)=C(CN)-CO-O-cyclobutyl, -C(CH₃)=C(CN)-CO-O-cyclopentyl, -C(CH₃)=C(CN)-CO-O-cyclohexyl, -C(CH₃)=C(CN)-CO-O-cycloheptyl, -C(CH₃)=CH-CO-OCH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-OCH(CH₃)-OCH₃, -C(CH₃)=CH-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=CH-CO-OCH₂CH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-O-i-C₃H₇, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-O-i-C₃H₇, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-O-i-C₃H₇, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-CF₃, -C(CH₃)=CH-CO-OCH₂-CCl₃, -C(CH₃)=CH-CO-OCH₂-oxiranyl, -C(CH₃)=CH-CO-O-(CH₂)₃-Br, -C(CH₃)=CH-CO-OCH₂-CH=CH₂, -C(CH₃)=CH-CO-OCH₂-C≡CH, -C(CH₃)=CH-CO-OCH₂-CN, -C(CH₃)=CH-CO-OCH₂CH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CF₃, -C(CH₃)=C(CH₃)-CO-OCH₂-CCl₃, -C(CH₃)=C(CH₃)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CH₃)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(CH₃)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CH₃)-CO-OCH₂-C≡CH, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CF₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CCl₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-oxiranyl, -C(CH₃)=C(C₂H₅)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(C₂H₅)-CO-OCH₂-C≡CH, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂-CF₃, -C(CH₃)=C(Cl)-CO-OCH₂-CCl₃, -C(CH₃)=C(Cl)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Cl)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Cl)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Cl)-CO-OCH₂-C≡CH, -C(CH₃)=C(Cl)-CO-OCH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂-CF₃, -C(CH₃)=C(Br)-CO-OCH₂-CCl₃, -C(CH₃)=C(Br)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Br)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Br)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Br)-CO-OCH₂-C≡CH, -C(CH₃)=C(Br)-CO-OCH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂CH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂-CF₃, -C(CH₃)=C(CN)-CO-OCH₂-CCl₃, -C(CH₃)=C(CN)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CN)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CN)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CN)-CO-OCH₂-C≡CH, -C(CH₃)=C(CN)-CO-OCH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂CH₂-CN, -C(CH₃)=CH-CO-CH₃, -C(CH₃)=CH-CO-C₂H₅, -C(CH₃)=CH-CO-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-n-C₄H₉, -C(CH₃)=CH-CO-tert.-C₄H₉, -C(CH₃)=CH-CO-CH₂Cl, -C(CH₃)=CH-CO-CH₂Br, -C(CH₃)=CH-CO-CHCl₂, -C(CH₃)=CH-CO-CH₂-OCH₃, -C(CH₃)=CH-CO-CH(OCH₃)₂, -C(CH₃)=CH-CO-CH₂-SCH₃, -C(CH₃)=C(CH₃)-CO-CH₃, -C(CH₃)=C(CH₃)-CO-C₂H₅, -C(CH₃)=C(CH₃)-CO-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-CH₂Cl, -C(CH₃)=C(CH₃)-CO-CH₂Br, -C(CH₃)=C(CH₃)-CO-CHCl₂, -C(CH₃)=C(CH₃)-CO-CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-CH(OCH₃)₂, -C(CH₃)=C(CH₃)-CO-CH₂-SCH₃, -C(CH₃)=C(C₂H₅)-CO-CH₃, -C(CH₃)=C(C₂H₅)-CO-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-CH₂Cl, -C(CH₃)=C(C₂H₅)-CO-CH₂Br, -C(CH₃)=C(C₂H₅)-CO-CHCl₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-CH(OCH₃)₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-SCH₃, -C(CH₃)=C(Cl)-CO-CH₃, -C(CH₃)=C(Cl)-CO-C₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-n-C₄H₉, -C(CH₃)=C(Cl)-CO-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-CH₂Cl, -C(CH₃)=C(Cl)-CO-CHCl₂, -C(CH₃)=C(Cl)-CO-CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-CH(OCH₃)₂, -C(CH₃)=C(Cl)-CO-CH₂-SCH₃, -C(CH₃)=C(Br)-CO-CH₃, -C(CH₃)=C(Br)-CO-C₂H₅, -C(CH₃)=C(Br)-CO-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-n-C₄H₉, -C(CH₃)=C(Br)-CO-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-CH₂Cl, -C(CH₃)=C(Br)-CO-CH₂Br, -C(CH₃)=C(Br)-CO-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-CH(OCH₃)₂, -C(CH₃)=C(Br)-CO-CH₂-SCH₃, -C(CH₃)=C(CN)-CO-CH₃, -C(CH₃)=C(CN)-CO-C₂H₅, -C(CH₃)=C(CN)-CO-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-n-C₄H₉, -C(CH₃)=C(CN)-CO-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-CH₂Cl, -C(CH₃)=C(CN)-CO-CH₂Br, -C(CH₃)=C(CN)-CO-CHCl₂, -C(CH₃)=C(CN)-CO-CH₂-OCH₃, -C(CH₃)=C(CN)-CO-CH(OCH₃)₂, -C(CH₃)=C(CN)-CO-CH₂-SCH₃, -C(CH₃)=CH-CO-C₆H₅, -C(CH₃)=CH-CO-(4-Cl-C₆H₄), -C(CH₃)=C(CH₃)-CO-C₆H₅, -C(CH₃)=C(CH₃)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(C₂H₅)-CO-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(Cl)-CO-C₆H₅, -C(CH₃)=C(Br)-CO-C₆H₅, -C(CH₃)=C(CN)-CO-C₆H₅, -C(CH₃)=CH-CO-NH₂, -C(CH₃)=CH-CO-NHCH₃, -C(CH₃)=CH-CO-N(CH₃)₂, -C(CH₃)=CH-CO-NH-C₂H₅, -C(CH₃)=CH-CO-N(C₂H₅)₂, -C(CH₃)=CH-CO-NH-n-C₃H₇, -C(CH₃)=CH-CO-NH-i-C₃H₇, -C(CH₃)=CH-CO-NH-tert.-C₄H₉, -C(CH₃)=CH-CO-NH-cyclopropyl, -C(CH₃)=CH-CO-NH-cyclobutyl, -C(CH₃)=CH-CO-NH-cyclopentyl, -C(CH₃)=CH-CO-NH-cyclohexyl, -C(CH₃)=CH-CO-NH-cycloheptyl, -C(CH₃)=CH-CO-NH-cyclooctyl, -C(CH₃)=CH-CO-pyrrolidin-1-yl, -C(CH₃)=CH-CO-piperidin-1-yl, -C(CH₃)=CH-CO-morpholin-4-yl, -C(CH₃)=CH-CO-NH-CH₂CH=CH₂, -C(CH₃)=CH-CO-NH-CH₂C≡CH, -C(CH₃)=CH-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=CH-CO-NH-(CH₂)₂Cl, -C(CH₃)=CH-CO-NH-C₆H₅, -C(CH₃)=C(CH₃)-CO-NH₂, -C(CH₃)=C(CH₃)-CO-NHCH₃, -C(CH₃)=C(CH₃)-CO-N(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-C₂H₅, -C(CH₃)=C(CH₃)-CO-N(C₂H₅)₂, -C(CH₃)=C(CH₃)-CO-NH-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-NH- cyclopropyl, -C(CH₃)=C(CH₃)-CO-NH-cyclobutyl, -C(CH₃)=C(CH₃)-CO-NH-cyclopentyl, -C(CH₃)=C(CH₃)-CO-NH- cyclohexyl, -C(CH₃)=C(CH₃)-CO-NH-cycloheptyl, -C(CH₃)=C(CH₃)-CO-NH-cyclooctyl, -C(CH₃)=C(CH₃)-CO- pyrrolidin-1-yl, -C(CH₃)=C(CH₃)-CO-piperidin-1-yl, -C(CH₃)=C(CH₃)-CO-morpholin-4-yl, -C(CH₃)=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-NH(CH₂)₂Cl, -C(CH₃)=C(CH₃)-CO-NH-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-NH₂, -C(CH₃)=C(C₂H₅)-CO-NHCH₃, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)₂, -C(CH₃)=C(C₂H₅)-CO-NH-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-N(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-NH- cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclo­ hexyl, -C(CH₃)=C(C₂H₅)-CO-NH-cycloheptyl, -C(CH₃)=C(C₂H₅)-CO-NH- cyclooctyl, -C(CH₃)=C(C₂H₅)-CO-pyrrolidin-1-yl, -C(CH₃)=C(C₂H₅)-CO-piperidin-1-yl, -C(CH₃)=C(C₂H₅)-CO- morpholin-4-yl, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(C₂H₅)-CO-NH-C₆H₅, -C(CH₃)=C(Cl)-CO-NH₂, -C(CH₃)=C(CH₃)=C(Cl)-CO-NHCH₃, -C(CH₃)=C(Cl)-CO-N(CH₃)₂, -C(CH₃)=C(Cl)-CO-NH-C₂H₅, -C(CH₃)=C(Cl)-CO-N(C₂H₅)₂, -C(CH₃)=C(Cl)-CO-NH-n-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-i-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-NH-cyclopropyl, -C(CH₃)=C(Cl)-CO-NH-cyclobutyl, -C(CH₃)=C(Cl)-CO-NH-cyclopentyl, -C(CH₃)=C(Cl)-CO-NH-cyclohexyl, -C(CH₃)=C(Cl)-CO-NH-cycloheptyl, -C(CH₃)=C(Cl)-CO-NH-cyclooctyl, -C(CH₃)=C(Cl)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Cl)-CO-piperidin-1- yl,-C(CH₃)=C(Cl)-CO-morpholin-4-yl, -C(CH₃)=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -C(CH₃)=C(Cl)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-N(CH₃)-CH₂≡CH, -C(CH₃)=C(Cl)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Cl)-CO-NH-C₆H₅, -C(CH₃)=C(Br)-CO-NH₂, -C(CH₃)=C(Br)-CO-NHCH₃, -C(CH₃)=C(Br)-CO-N(CH₃)₂, -C(CH₃)=C(Br)-CO-NH-C₂H₅, -C(CH₃)=C(Br)-CO-N(C₂H₅)₂, -C(CH₃)=C(Br)-CO-NH-n-C₃H₇, -C(CH₃)=C(Br)-CO-NH-i-C₃H₇, -C(CH₃)=C(Br)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-NH-cyclopropyl, -C(CH₃)=C(Br)-CO-NH-cyclobutyl, -C(CH₃)=C(Br)-CO-NH-cyclopentyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cycloheptyl, -C(CH₃)=C(Br)-CO-NH-cyclooctyl, -C(CH₃)=C(Br)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Br)-CO-piperidin-1-yl, -C(CH₃)=C(Br)-CO-morpholin-4-yl, -C(CH₃)=C(Br)-CO-NH-CH₂CH=C(Br)₂, -C(CH₃)=C(Br)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Br)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Br)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Br)-CO-NH-C₆H₅, -C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CN)-CO-NHCH₃, -C(CH₃)=C(CN)-CO-N(CH₃)₂, -C(CH₃)=C(CN)-CO-NH-C₂H₅, -C(CH₃)=C(CN)-CO-N(C₂H₅)₂, -C(CH₃)=C(CN)-CO-NH-n-C₃H₇, -C(CH₃)=C(CN)-CO-NH-i-C₃H₇, -C(CH₃)=C(CN)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-NH-cyclopropyl, -C(CH₃)=C(CN)-CO-NH-cyclobutyl, -C(CH₃)=C(CN)-CO-NH-cyclopentyl, -C(CH₃)=C(CN)-CO-NH-cyclohexyl, -C(CH₃)=C(CN)-CO-NH-cycloheptyl, -C(CH₃)=C(CN)-CO-NH-cyclooctyl, -C(CH₃)=C(CN)-CO-pyrrolidin-1-yl, -C(CH₃)=C(CN)-CO-piperidin-1-yl, -C(CH₃)=C(CN)-CO-morpholin-4-yl, -C(CH₃)=C(CN)-CO-NH-CH₂CH=C(CN)₂, -C(CH₃)=C(CN)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CN)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)=(CN)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CN)-CO-NH-C₆H₅, -C(CH₃)=CH-SO-SCH₃, -C(CH₃)=CH-CO-SC₂H₅, -C(CH₃)=CH-CO-S-n-C₃H₇, -C(CH₃)=CH-CO-S-i-C₃H₇, -C(CH₃)=CH-CO-S-n-C₄H₉, -C(CH₃)=CH-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-SCH₃, -C(CH₃)=C(CH₃)-CO-SC₂H₅, -C(CH₃)=C(CH₃)CO-S-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-S-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-SCH₃, -C(CH₃)=C(C₂H₅)-CO-SC₂H₅, -C(CH₃)=C(C₂H₅)-CO-S-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-SCH₃, -C(CH₃)=C(Cl)-CO-SC₂H₅, -C(CH₃)=C(Cl)-CO-S-n-C₃H₇, -C(CH₃)=C(Cl)-CO-S-i-C₃H₇, -C(CH₃)=C(Cl)-CO-S-n-C₄H₉, -C(CH₃)=C(Cl)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-SCH₃, -C(CH₃)=C(Br)-CO-SC₂H₅, -C(CH₃)=C(Br)-CO-S-n-C₃H₇, -C(CH₃)=C(Br)-CO-S-i-C₃H₇, -C(CH₃)=C(Br)-CO-S-n-C₄H₉, -C(CH₃)=C(Br)-CO-S-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-SCH₃, -C(CH₃)=C(CN)-CO-SC₂H₅, -C(CH₃)=C(CN)-CO-S-n-C₃H₇, -C(CH₃)=C(CN)-CO-S-i-C₃H₇, -C(CH₃)=C(CN)-CO-S-N-C₄H₉, -C(CH₃)=C(CN)-CO-S-tert.-C₄H₉, -C(CH₃)=C(COCH₃)-CO-OCH₃, -C(CH₃)=C(COC₂H₅)-CO-OCH₃, -C(CH₃)=C(CO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COCH₃)-CO-OC₂H₅, -C(CH₃)=C(COC₂H₅)-CO-OC₂H₅, -C(CH₃)=C(CO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COCH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(COC₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-OCH₃, -C(CH₃)=C(CF₃)-CO-OC₂H₅, -C(CH₃)=C(CF₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CF₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(COOCH₃)₂, -C(CH₃)=C(COOC₂H₅)₂, -C(CH₃)=C(COOCH₃)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)₂, -C(CH₃)=CH-CH=CH-COOH, -C(CH₃)=CH-CH=CH-CO-OCH₃, -C(CH₃)=CH-CH=CH-CO-OC₂H₅, -C(CH₃)=CH-CH=C(COOCH₃)₂, -C(CH₃)=CH-CH=C(CN)-CO-OCH₃, -C(CH₃)=CH-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CN)CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH₂, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -C(CH₃)=CH-(CH₂)₂-COOH, -C(CH₃)=CH-(CH₂)₂-CO-OCH₃, -C(CH₃)=CH-(CH₂)₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(COOCH₃)₂, -C(CH₃)=CH-CH₂-CH(COOC₂H₅)₂, -C(CH₃)=CH-CH₂-CH(CN)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CN)-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -C(CH₃)=CH-(CH₂)₂-CO-NH₂, -C(CH₃)=CH-(CH₂)₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-COOH, -C(CH₃)=CH-CH₂-CO-OCH₃, -C(CH₃)=CH-CH₂-CO-OC₂H₅, -C(CH₃)=C(COOCH₃)-CH₂-CO-OCH₃, -C(CH₃)=C(COOCH₃)-CH₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CO-NH₂, -C(CH₃)=CH-CH₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-CO-N(CH₃)₂.
wobei W für eine der folgenden Bedeutungen steht:
-CHO, -COCH₃, -COC₂H₅, -CO-n-C₃H₇, -CO-i-C₃H₇, -CO-n-C₄H₉, -CO-i-C₄H₉, -CO-s-C₄H₉, -CO-tert.-C₄H₉, -CO-CH₂CH=CH₂, -CO-CF₃, -COCCl₃, -COCH₂C≡CH, -CO-cyclopropyl, -CO-cyclobutyl, -CO-cyclopentyl, -CO-cyclohexyl, -CO-CN, -CO-COOCH₃, -CO-COOC₂H₅, -CH=NH, -CH=NCH₃, -CH=NC₂H₅, -CH=N-n-C₃H₅, -CH=N-i-C₃H₅, -CH=N-n-C₄H₉, -CH=NCH₂CH=CH₂, -CH=NCH₂CH=CH₂-CH₃, -CH=NCH₂≡CH, -CH=NCH₂C≡C-CH₃, -CH=N-cyclopropyl, -CH=N-cyclobutyl, -CH=N-cyclopentyl, -CH=N-cyclohexyl, -CH=N-cycloheptyl, -CH=N-CH₂-CH₂Cl, -CH=N-CH₂Cl, -CH=N-₆H₅, -CH=N-(4-Br-C₆H₄), -CH=N-3-F-C₆H₄, -CH=N-4-F-C₆H₄, -CH=N-2-Cl-C₆H₄, -CH=N-3-Cl-C₆H₄, -CH=N-4-Cl-C₆H₄, -CH=N-2-Br-C₆H₄, -CH=N-2-F-C₆H₄, -CH=N-2-CH₃-C₆H₄, -CH=N-3-CH₃-C₆H₄, -CH=N-4-CH₃-C₆H₄, -CH=N-2-CF₃-C₆H₄, -CH=N-3-CF₃-C₆H₄, -CH=N-4-CF₃-C₆H₄, -CH=N-2-OCH₃-C₆H₄, -CH=N-3-OCH₃-C₆H₄, -CH=N-4-OCH₃-C₆H₄, -CH=N-4-NO₂-C₆H₄, -CH=N-4-CN-C₆H₄, -CH=N-2,4-(Cl,Cl)-C₆H₄, -CH=N-2,4-(CH₃,CH₃)-C₆H₄, -CH=N-CH₂OCH₃ -CH=N-CH₂OC₂H₅, -CH=N-CH₂CH₂OCH₃, -CH=N-CH₂CH₂OC₂H₅, -CH=N-OH, -CH=N-OCH₃, -CH=N-OC₂H₅, -CH=N-O-n-C₃H₇, -CH=N-O-i-C₃H₇, -CH=N-O-n-C₄H₉, -CH=N-O-i-C₄H₉, -CH=N-O-s-C₄H₉, -CH=N-O-tert.-C₄H₉, -CH=N-O-CH₂CH=CH₂, -CH=N-O-CH(CH₃)CH=CH₂, -CH=N-O-CH₂C≡CH, -CH=N-O-CH(CH₃)-C≡CH, -CH=N-O-CH₂-CH=CH-CH₃, -CH=N-O-CH₂-CH₂-Cl, -CH=N-O-CH₂-CH₂-F, -CH=N-O-CH₂-CF₃, -CH=N-O-CH₂-CH=CHCl, -CH=N-O-CH₂-CCl=CH₂, -CH=N-O-CH₂-CBr=CH₂, -CH=N-O-CH₂-CH=CCl-CH₃, -CH=N-OC(O)CH₃, -CH=N-OC(O)C₂H₅, -CH=N-O-CH₂-CN, -CH=N-O-CH₂-CH=CH-CH₂-O-CH₃, -CH=N-O-CH₂-CH=CH-CH₂-O-tert.-C₄H₉, -CH=N-O-(CH₂)₃-C₆H₅, -CH=N-O-(CH₂)₄-C₆H₅, -CH=N-O-(CH₂)₄-4-Cl-C₆H₄, -CH=N-O-(CH₂)₄-4-OCH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-CH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-C₆H₅, -CH=N-O-CH₂CH=CH-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CH-3-OCH₃-C₆H₄, -CH=N-O-(CH₂)₂CH=CH-4-F-C₆H₄, -CH=N-O-(CH₂)CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CHCH₂-4-OCH₃-C₆H₄, -CH=N-O-CH₂-CH=C(CH₃)-C₆H₅, -CH=N-O-(CH₂)₂CH=CH-3,4(Cl,Cl)-C₆H₃, -CH=N-O-(CH₂)₃C≡C-4-F-C₆H₄, -CH₂=N-OCHOCH₃, -CH=N-OC₂H₄OCH₃, -CH=N-OCH₂OC₂H₅, -CH=N-OCH(CH₃)OCH₃, -CH=N-OCH(CH₃)COOCH₃, -CH=N-OCH(CH₃)COO-n-C₄H₉, -CH=N-NH₂, -CH=N-NHCH₃, -CH=N-NHC₂H₅, -CH=N-NH-n-C₃H₇, -CH=N-NH-i-C₃H₇, -CH=N-NH-n-C₄H₉, -CH=N-NH-i-C₄H₉, -CH=N-NH-s-C₄H₉, -CH=N-NH-tert.-C₄H₉, -CH=N-NH-cyclopropyl, -CH=N-NH-cyclobutyl, -CH=N-NH-cyclopentyl, -CH=N-NH-cyclohexyl, -CH=N-NH-cycloheptyl, -CH=N-N(CH₃)₂, -CH=N-N(C₂H₅)₂, -CH=N-N(C₃H₇)₂, -CH=N-N(i-C₃H₇)(CH₃), -CH=N-NHCH₂-C=CH, -CH=N-NHCH₂-C≡CH, -CH=N-N(CH₃)-CH₂-C≡CH, -CH=N-NHCH₂CF₃, -CH=N-NH-CO-CH₃, -CH=N-NH-CO-CH₂H₅, -CH=N-NH-COOCH₃, -CH=N-NH-COOC₂H₅, -CH=N-NH-COO-tert.-C₄H₉, -CH=N-pyrrolidin-1-yl, -CH=N-piperidin-1-yl, -CH=N-morpholin-4-yl, -CH=N-NH-C₆H₅, -CH=N-NH-(4-Cl-C₆H₄), -CH=N-NH-(4-NO₂-C₆H₄), -CH=N-NH-(4-F-C₆H₄), -CH=N-NH-(4-CH₃O-C₆H₄), -CH=N-NH-(2,4-Cl₂-C₆H₃), -CH=N-NH-(2,4-(NO₂)₂-C₆H₃), -CH=N-NH-CO-NH₂, -CH=N-NH-CO-NHCH₃, -CH=N-NH-CO-NHC₂H₅, -CH=N-NH-CO-N(CH₃)₂, -CH=CH-COOH, -CH=CH-CO-OCH₃, -CH=CH-CO-OC₂H₅, -CH=CH-CO-O-n-C₃H₇, -CH=CH-CO-O-i-C₃H₇, -CH=CH-CO-O-n-C₄H₉, -CH=CH-CO-O-tert.-C₄H₉, -CH=CH-CO-O-cyclopropyl, -CH=CH-CO-O-cyclobutyl, -CH=CH-CO-O-cyclopentyl, -CH=CH-CO-O-cyclohexyl, -CH=CH-CO-O-cycloheptyl, -CH=C(CH₃)-COOH, -CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CO-O-n-C₃H₇, -CH=C(CH₃)-CO-O-i-C₃H₇, -CH=C(CH₃)-CO-O-n-C₄H₉, -CH=C(CH₃)-CO-O-tert.-C₄H₉, -CH=C(CH₃)-CO-O-cyclopropyl, -CH=C(CH₃)-CO-O-cyclobutyl, -CH=C(CH₃)-CO-O-cyclopentyl, -CH=C(CH₃)-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cycloheptyl, -CH=C(C₂H₅)-COOH, -CH=C(C₂H₅)-CO-OCH₃, -CH=C(C₂H₅)-CO-OC₂H₅, -CH=C(C₂H₅)-CO-O-n-C₃H₇, -CH=C(C₂H₅)-CO-O-i-C₃H₇, -CH=C(C₂H₅)-CO-O-n-C₄H₉, -CH=C(C₂H₅)-CO-O-tert.-C₄H₉, -CH=C(C₂H₅)-CO-O-cyclopropyl, -CH=C(C₂H₅)-CO-O-cyclobutyl, -CH=C(C₂H₅)-CO-O-cyclopentyl, -CH=C(C₂H₅)-CO-O-cyclohexyl, -CH=C(C₂H₅)-CO-O-cycloheptyl, -CH=C(Cl)-COOH, -CH=C(Cl)-CO-OCH₃, -CH=C(Cl)-CO-OC₂H₅, -CH=C(Cl)-CO-O-n-C₃H₇, -CH=C(Cl)-CO-O-i-C₃H₇, -CH=C(Cl)-CO-O-n-C₄H₉, -CH=C(Cl)-CO-O-tert.-C₄H₉, -CH=C(Cl)-CO-O-cyclopropyl, -CH=C(Cl)-CO-O-cyclobutyl, -CH=C(Cl)-CO-O-cyclopentyl, -CH=C(Cl)-CO-O-cyclohexyl, -CH=C(Cl)-CO-O-cycloheptyl, -CH=C(Br)-COOH, -CH=C(Br)-CO-OCH₃, -CH=C(Br)-CO-OC₂H₅, -CH=C(Br)-CO-O-n-C₃H₇, -CH=C(Br)-CO-O-i-C₃H₇, -CH=C(Br)-CO-O-n-C₄H₉, -CH=C(Br)-CO-O-tert.-C₄H₉, -CH=C(Br)-CO-O-cyclopropyl, -CH=C(Br)-CO-O-cyclobutyl, -CH=C(Br)-CO-O-cyclopentyl, -CH=C(Br)-CO-O-cyclohexyl, -CH=C(Br)-CO-O-cycloheptyl, -CH=C(CN)-COOH, -CH=C(CN)-CO-OCH₃, -CH=C(CN)-CO-OC₂H₅, -CH=C(CN)-CO-O-n-C₃H₇, -CH=C(CN)-CO-O-i-C₃H₇, -CH=C(CN)-CO-O-n-C₄H₉, -CH=C(CN)-CO-O-tert.-C₄H₉, -CH=C(CN)-CO-O-cyclopropyl, -CH=C(CN)-CO-O-cyclobutyl, -CH=C(CN)-CO-O-cyclopentyl, -CH=C(CN)-CO-O-cyclohexyl, -CH=C(CN)-CO-O-cycloheptyl, -CH=CH-CO-OCH₂-OCH₃, -CH=CH-CO-OCH₂-OC₂H₅, -CH=CH-CO-OCH₂-O-n-C₃H₅, -CH=CH-CO-OCH₂-O-i-C₃H₅, -CH=CH-CO-OCH(CH₃)-OCH₃, -CH=CH-CO-OCH(CH₃)-OC₂H₅, -CH=CH-CO-O-CH₂CH₂-OCH₃, -CH=CH-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-OCH₃, -CH=C(CH₃)-CO-OCH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-O-n-C₃H₅, -CH=C(CH₃)-CO-OCH₂-O-i-C₃H₅, -CH=C(CH₃)-CO-OCH(CH₃)-OCH₃, -CH=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CH₃)-CO-O-CH₂CH₂-OCH₃, -CH=C(CH₃)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-OCH₃, -CH=C(C₂H₅)-CO-OCH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-O-n-C₃H₅, -CH=C(C₂H₅)-CO-OCH₂-O-i-C₃H₅, -CH=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -CH=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OCH₃, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-OCH₃, -CH=C(Cl)-CO-OCH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-O-n-C₃H₅, -CH=C(Cl)-CO-OCH₂-O-i-C₃H₅, -CH=C(Cl)-CO-OCH(CH₃)-OCH₃, -CH=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Cl)-CO-O-CH₂CH₂-OCH₃, -CH=C(Cl)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-OCH₃, -CH=C(Br)-CO-OCH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-O-n-C₃H₅, -CH=C(Br)-CO-OCH₂-O-i-C₃H₅, -CH=C(Br)-CO-OCH(CH₃)-OCH₃, -CH=C(Br)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Br)-CO-O-CH₂CH₂-OCH₃, -CH=C(Br)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-OCH₃, -CH=C(CN)-CO-OCH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-O-n-C₃H₅, -CH=C(CN)-CO-OCH₂-O-i-C₃H₅, -CH=C(CN)-CO-OCH(CH₃)-OCH₃, -CH=C(CN)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CN)-CO-O-CH₂CH₂-OCH₃, -CH=C(CN)-CO-O-CH₂CH₂-OC₂H₅, -CH=CH-CO-OCH₂-CF₃, -CH=CH-CO-OCH₂-CCl₃, -CH=CH-CO-OCH₂-oxiranyl, -CH=CH-CO-O(CH₂)₃-Br, -CH=CH-CO-OCH₂-CH=CH₂, -CH=CH-CO-OCH₂-C≡CH, -CH=CH-CO-OCH₂-CN, -CH=CH-CO-O(CH₂)₂-CN, -CH=C(CH₃)-CO-OCH₂-CF₃, -CH=C(CH₃)-CO-OCH₂-CCl₃, -CH=C(CH₃)-CO-OCH₂-oxiranyl, -CH=C(CH₃)-CO-O(CH₂)₃-Br, -CH=C(CH₃)-CO-OCH₂-CH=CH₂, -CH=C(CH₃)-CO-OCH₂-C≡CH, -CH=C(CH₃)-CO-OCH₂-CN, -CH=C(CH₃)-CO-O(CH₂)₂-CN, -CH=C(C₂H₅)-CO-OCH₂-CF₃, -CH=C(C₂H₅)-CO-OCH₂-CCl₃, -CH=C(C₂H₅)-CO-OCH₂-oxiranyl, -CH=C(C₂H₅)-CO-O(CH₂)₃-Br, -CH=C(C₂H₅)-CO-OCH₂-CH=CH₂, -CH=C(C₂H₅)-CO-OCH₂-C≡CH, -CH=C(C₂H₅)-CO-OCH₂-CN, -CH=C(C₂H₅)-CO-O(CH₂)₂-CN, -CH=C(Cl)-CO-OCH₂-CF₃, -CH=C(Cl)-CO-OCH₂-CCl₃, -CH=C(Cl)-CO-OCH₂-oxiranyl, -CH=C(Cl)-CO-O(CH₂)₃-Br, -CH=C(Cl)-CO-OCH₂-CH=CH₂, -CH=C(Cl)-CO-OCH₂-C≡CH, -CH=C(Cl)-CO-OCH₂-CN, -CH=C(Cl)-CO-O(CH₂)₂-CN, -CH=C(Br)-CO-OCH₂-CF₃, -CH=C(Br)-CO-OCH₂-CCl₃, -CH=C(Br)-CO-OCH₂-oxiranyl, -CH=C(Br)-CO-O(CH₂)₃-Br, -CH=C(Br)-CO-OCH₂-CH=CH₂, -CH=C(Br)-CO-OCH₂-C≡CH, -CH=C(Br)-CO-OCH₂-CN, -CH=C(Br)-CO-O(CH₂)₂-CN, -CH=C(CN)-CO-OCH₂-CF₃, -CH=C(CN)-CO-OCH₂-CCl₃, -CH=C(CN)-CO-OCH₂-oxiranyl -CH=C(CN)-CO-O(CH₂)₃-Br, -CH=C(CN)-CO-OCH₂-CH=CH₂, -CH=C(CN)-CO-OCH₂-C≡CH, -CH=C(CN)-CO-OCH₂-CN, -CH=C(CN)-CO-O(CH₂)₂-CN, -CH=CH-CO-CH₃, -CH=CH-CO-C₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-i-C₃H₇, -CH=CH-CO-n-C₄H₉, -CH=CH-CO-tert.-C₄H₉, -CH=CH-CO-CH₂Cl, -CH=CH-CO-CH₂Br, -CH=CH-CO-CHCl₂, -CH=CH-CO-CH₂-OCH₃, -CH=CH-CO-CH(OCH₃)₂, -CH=CH-CO-CH₂-SCH₃, -CH=C(CH₃)-CO-CH₃, -CH=C(CH₃)-CO-C₂H₅, -CH=C(CH₃)-CO-n-C₃H₇, -CH=C(CH₃)-CO-i-C₃H₇, -CH=C(CH₃)-CO-n-C₄H₉, -CH=C(CH₃)-CO-tert.-C₄H₉, -CH=C(CH₃)-CO-CH₂Cl, -CH=C(CH₃)-CO-CH₂Br, -CH=C(CH₃)-CO-CHCl₂, -CH=C(CH₃)-CO-CH₂-OCH₃, -CH=C(CH₃)-CO-CH(OCH₃)₂, -CH=C(CH₃)-CO-CH₂-SCH₃, -CH=C(C₂H₅)-CO-CH₃, -CH=C(C₂H₅)-CO-C₂H₅, -CH=C(C₂H₅)-CO-n-C₃H₇, -CH=C(C₂H₅)-CO-i-C₃H₇, -CH=C(C₂H₅)-CO-n-C₄H₉, -CH=C(C₂H₅)-CO-tert.-C₄H₉, -CH=C(C₂H₅)-CO-CH₂Cl, -CH=C(C₂H₅)-CO-CH₂Br, -CH=C(C₂H₅)-CO-CHCl₂, -CH=C(C₂H₅)-CO-CH₂-OCH₃, -CH=C(C₂H₅)-CO-CH(OCH₃)₂, -CH=C(C₂H₅)-CO-CH₂-SCH₃, -CH=C(Cl)-CO-CH₃, -CH=C(Cl)-CO-C₂H₅, -CH=C(Cl)-CO-n-C₃H₇, -CH=C(Cl)-CO-i-C₃H₇, -CH=C(Cl)-CO-n-C₄H₉, -CH=C(Cl)-CO-tert.-C₄H₉, -CH=C(Cl)-CO-CH₂Cl, -CH=C(Cl)-CO-CH₂Br, -CH=C(Cl)-CO-CHCl₂, -CH=C(Cl)-CO-CH₂-OCH₃, -CH=C(Cl)-CO-CH(OCH₃)₂, -CH=C(Cl)-CO-CH₂-SCH₃, -CH=C(Br)-CO-CH₃, -CH=C(Br)-CO-C₂H₅, -CH=C(Br)-CO-n-C₃H₇, -CH=C(Br)-CO-i-C₃H₇, -CH=C(Br)-CO-n-C₄H₉, -CH=C(Br)-CO-tert.-C₄H₉, -CH=C(Br)-CO-CH₂Cl, -CH=C(Br)-CO-CH₂Br, -CH=C(Br)-CO-CHCl₂, -CH=C(Br)-CO-CH₂-OCH₃, -CH=C(Br)-CO-CH(OCH₃)₂, -CH=C(Br)-CO-CH₂-SCH₃, -CH=C(CN)-CO-CH₃, -CH=C(CN)-CO-C₂H₅, -CH=C(CN)-CO-n-C₃H₇, -CH=C(CN)-CO-i-C₃H₇, -CH=C(CN)-CO-n-C₄H₉, -CH=C(CN)-CO-tert.-C₄H₉, -CH=C(CN)-CO-CH₂Cl, -CH=C(CN)-CO-CH₂Br, -CH=C(CN)-CO-CHCl₂, -CH=C(CN)-CO-CH₂-OCH₃, -CH=C(CN)-CO-CH(OCH₃)₂, -CH=C(CN)-CO-CH₂-SCH₃, -CH=CH-CO-C₆H₅, -CH=CH-CO-(4-Cl-C₆H₄), -CH=C(CH₃)-CO-C₆H₅, -CH=C(CH₃)-CO-(4-Cl-C₆H₄), -CH=C(C₂H₅)-CO-C₆H₅, -CH=C(C₂H₅)-CO-(4-Cl-C₆H₄), -CH=C(Cl)-CO-C₆H₅, -CH=C(Br)-CO-C₆H₅, -CH=C(CN)-CO-C₆H₅ -CH=CH-CO-NH₂, -CH=CH-CO-NHCH₃, -CH=CH-CO-N(CH₃)₂, -CH=CH-CO-NH-C₂H₅, -CH=CH-CO-N(C₂H₅)₂, -CH=CH-CO-NH-n-C₃H₇, -CH=CH-CO-NH-i-C₃H₇, -CH=CH-CO-NH-tert.-C₄H₉, -CH=CH-CO-NH-cyclopropyl, -CH=CH-CO-NH-cyclobutyl, -CH=CH-CO-NH-cyclopentyl, -CH=CH-CO-NH-cyclohexyl, -CH=CH-CO-NH-cycloheptyl, -CH=CH-CO-NH-cyclooctyl, -CH=CH-CO-pyrrolidin-1-yl, -CH=CH-CO-piperidin-1-yl, -CH=CH-CO-morpholin-4-yl, -CH=CH-CO-NH-CH₂CH=CH₂, -CH=CH-CO-NH-CH₂C≡CH, -CH=CH-CO-N(CH₃)-CH₂C≡CH, -CH=CH-CO-NH-(CH₂)₂Cl, -CH=CH-CO-NH-C₆H₅, -CH=C(CH₃)-CO-NH₂, -CH=C(CH₃)-CO-NHCH₃, -CH=C(CH₃)-CO-N(CH₃)₂, -CH=C(CH₃)-CO-NH-C₂H₅, -CH=C(CH₃)-CO-N(C₂H₅)₂, -CH=C(CH₃)-CO-NH-n-C₃H₇, -CH=C(CH₃)-CO-NH-i-C₃H₇, -CH=C(CH₃)-CO-NH-tert.-C₄H₉, -CH=C(CH₃)-CO-NH-cyclopropyl, -CH=C(CH₃)-CO-NH-cyclobutyl, -CH=C(CH₃)-CO-NH-cyclopentyl, -CH=C(CH₃)-CO-NH-cyclohexyl, -CH=C(CH₃)-CO-NH-cycloheptyl, -CH=C(CH₃)-CO-NH-cyclooctyl, -CH=C(CH₃)-CO-pyrrolidin-1-yl, -CH=C(CH₃)-CO-piperidin-1-yl, -CH=C(CH₃)-CO-morpholin-4-yl, -CH=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -CH=C(CH₃)-CO-NH-CH₂C≡CH, -CH=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CH₃)-CO-NH-(CH₂)₂Cl, -CH=C(CH₃)-CO-NH-C₆H₅, -CH=C(C₂H₅)-CO-NH₂, -CH=C(C₂H₅)-CO-NHCH₃, -CH=C(C₂H₅)-CO-N(CH₃)₂, -CH=C(C₂H₅)-CO-NH-C₂H₅, -CH=C(C₂H₅)-CO-N(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-n-C₃H₇, -CH=C(C₂H₅)-CO-NH-i-C₃H₇, -CH=C(C₂H₅)-CO-NH-tert.-C₄H₉, -CH=C(C₂H₅)-CO-NH-cyclopropyl, -CH=C(C₂H₅)-CO-NH-cyclobutyl, -CH=C(C₂H₅)-CO-NH-cyclopentyl, -CH=C(C₂H₅)-CO-NH-cyclohexyl, -CH=C(C₂H₅)-CO-NH-cycloheptyl, -CH=C(C₂H₅)-CO-NH-cyclooctyl, -CH=C(C₂H₅)-CO-pyrrolidin-1-yl, -CH=C(C₂H₅)-CO-piperidin-1-yl, -CH=C(C₂H₅)-CO-morpholin-4-yl, -CH=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-CH₂C≡CH, -CH=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -CH=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -CH=C(C₂H₅)-CO-NH-C₆H₅, -CH=C(Cl)-CO-NH₂, -CH=C(Cl)-CO-NHCH₃, -CH=C(Cl)-CO-N(CH₃)₂, -CH=C(Cl)-CO-NH-C₂H₅, -CH=C(Cl)-CO-N(C₂H₅)₂, -CH=C(Cl)-CO-NH-n-C₃H₇, -CH=C(Cl)-CO-NH-i-C₃H₇, -CH=C(Cl)-CO-NH-tert.-C₄H₉, -CH=C(Cl)-CO-NH-cyclopropyl, -CH=C(Cl)-CO-NH-cyclobutyl, -CH=C(Cl)-CO-NH-cyclopentyl, -CH=C(Cl)-CO-NH-cyclohexyl, -CH=C(Cl)-CO-NH-cycloheptyl, -CH=C(Cl)-CO-NH-cyclooctyl, -CH=C(Cl)-CO-pyrrolidin-1-yl, -CH=C(Cl)-CO-piperidin-1-yl, -CH=C(Cl)-CO-morpholin-4-yl, -CH=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -CH=C(Cl)-CO-NH-CH₂C≡CH, -CH=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Cl)-CO-NH-(CH₂)₂Cl, -CH=C(Cl)-CO-NH-C₆H₅, -CH=C(Br)-CO-NH₂, -CH=C(Br)-CO-NHCH₃, -CH=C(Br)-CO-N(CH₃)₂, -CH=C(Br)-CO-NH-C₂H₅, -CH=C(Br)-CO-N(C₂H₅)₂, -CH=C(Br)-CO-NH-n-C₃H₇, -CH=C(Br)-CO-NH-i-C₃H₇, -CH=C(Br)-CO-NH-tert.-C₄H₉, -CH=C(Br)-CO-NH-cyclopropyl, -CH=C(Br)-CO-NH-cyclobutyl, -CH=C(Br)-CO-NH-cyclopentyl, -CH=C(Br)-CO-NH-cyclohexyl, -CH=C(Br)-CO-NH-cycloheptyl, -CH=C(Br)-CO-NH-cyclooctyl, -CH=C(Br)-CO-pyrrolidin-1-yl, -CH=C(Br)-CO-piperidin-1-yl, -CH=C(Br)-CO-morpholin-4-yl, -CH=C(Br)-CO-NH-CH₂CH=C(Br)₂, -CH=C(Br)-CO-NH-CH₂C≡CH, -CH=C(Br)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Br)-CO-NH-(CH₂)₂Cl, -CH=C(Br)-CO-NH-C₆H₅, -CH=C(CN)-CO-NH₂, -CH=C(CN)-CO-NHCH₃, -CH=C(CN)-CO-N(CH₃)₂, -CH=C(CN)-CO-NH-C₂H₅, -CH=C(CN)-CO-N(C₂H₅)₂, -CH=C(CN)-CO-NH-n-C₃H₇, -CH=C(CN)-CO-NH-i-C₃H₇, -CH=C(CN)-CO-NH-tert.-C₄H₉, -CH=C(CN)-CO-NH-cyclopropyl, -CH=C(CN)-CO-NH-cyclobutyl, -CH=C(CN)-CO-NH-cyclopentyl, -CH=C(CN)-CO-NH-cyclohexyl, -CH=C(CN)-CO-NH-cycloheptyl, -CH=C(CN)-CO-NH-cyclooctyl, -CH=C(CN)-CO-pyrrolidin-1-yl, -CH=C(CN)-CO-piperidin-1-yl, -CH=C(CN)-CO-morpholin-4-yl, -CH=C(CN)-CO-NH-CH₂CH=C(CN)₂, -CH=C(CN)-CO-NH-CH₂C≡CH, -CH=C(CN)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CN)-CO-NH-(CH₂)₂Cl, -CH=C(CN)-CO-NH-C₆H₅, -CH=CH-CO-SCH₃, -CH=CH-CO-SC₂H₅, -CH=CH-CO-S-n-C₃H₇, -CH=CH-CO-S-i-C₃H₇, -CH=CH-CO-S-n-C₄H₉, -CH=CH-CO-S-tert.-C₄H₉, -CH=C(CH₃)-CO-SCH₃, -CH=C(CH₃)-CO-SC₂H₅, -CH=C(CH₃)-CO-S-n-C₃H₇, -CH=C(CH₃)-CO-S-i-C₃H₇, -CH=C(CH₃)-CO-S-n-C₄H₉, -CH=C(CH₃)-CO-S-tert.-C₄H₉, -CH=C(C₂H₅)-CO-SCH₃, -CH=C(C₂H₅)-CO-SC₂H₅, -CH=C(C₂H₅)-CO-S-n-C₃H₇, -CH=C(C₂H₅)-CO-S-i-C₃H₇, -CH=C(C₂H₅)-CO-S-n-C₄H₉, -CH=C(C₂H₅)-CO-S-tert.-C₄H₉, -CH=C(Cl)-CO-SCH₃, -CH=C(Cl)-CO-SC₂H₅, -CH=C(Cl)-CO-S-n-C₃H₇, -CH=C(Cl)-CO-S-i-C₃H₇, -CH=C(Cl)-CO-S-n-C₄H₉, -CH=C(Cl)-CO-S-tert.-C₄H₉, -CH=C(Br)-CO-SCH₃, -CH=C(Br)-CO-SC₂H₅, -CH=C(Br)-CO-S-n-C₃H₇, -CH=C(Br)-CO-S-i-C₃H₇, -CH=C(Br)-CO-S-n-C₄H₉, -CH=C(Br)-CO-S-tert.-C₄H₉, -CH=C(CN)-CO-SCH₃, -CH=C(CN)-CO-SC₂H₅, -CH=C(CN)-CO-S-n-C₃H₇, -CH=C(CN)-CO-S-i-C₃H₇, -CH=C(CN)-CO-S-n-C₄H₉, -CH=C(CN)-CO-S-tert.-C₄H₉, -CH=C(COCH₃)-CO-OCH₃, -CH=C(COC₂H₅)-CO-OCH₃, -CH=C(CO-n-C₃H₇)-CO-OCH₃, -CH=C(COCH₃)-CO-OC₂H₅, -CH=C(COC₂H₅)-CO-OC₂H₅, -CH=C(CO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COCH₃)-CO-O-n-C₃H₇, -CH=C(COC₂H₅)-CO-O-n-C₃H₇, -CH=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-OCH₃, -CH=C(CF₃)-CO-OC₂H₅, -CH=C(CF₃)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-O-i-C₃H₇, -CH=C(CF₃)-CO-O-n-C₄H₉, -CH=C(CF₃)-CO-O-tert.-C₄H₉, -CH=C(COOCH₃)₂, -CH=C(COOC₂H₅)₂, -CH=C(COOCH₃)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)-CO-OCH₃, -CH=C(COO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)₂, -CH=CH-CH=CH-COOH, -CH=CH-CH=CH-CO-OCH₃, -CH=CH-CH=CH-CO-OC₂H₅, -CH=CH-CH=C(COOCH₃)₂, -CH=CH-CH=C(CN)-CO-OCH₃, -CH=CH-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-OCH₃, -CH=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CH=C(Cl)-CO-OCH₃, -CH=C(CH₃)-CH=C(Br)-CO-OCH₃, -CH=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-NH₂, -CH=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -CH=CH-(CH₂)₂-COOH, -CH=CH-(CH₂)₂-CO-OCH₃, -CH=CH-(CH₂)₂-CO-OC₂H₅, -CH=CH-CH₂-CH(COOCH₃)₂, -CH=CH-CH₂-CH(COOC₂H₅)₂, -CH=CH-CH₂-CH(CN)-CO-OCH₃, -CH=CH-CH₂-CH(CN)-CO-OC₂H₅, -CH=CH-CH₂-CH(CH₃)-CO-OCH₃, -CH=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -CH=CH-(CH₂)₂-CO-NH₂, -CH=CH-(CH₂) 99999 00070 552 001000280000000200012000285919988800040 0002004131038 00004 99880 ¥äCO-NH-CH₃, -CH=CH-CH₂-COOH, -CH=CH-CH₂-CO-OCH₃, -CH=CH-CH₂-CO-OC₂H₅, -CH=C(COOCH₃)-CH₂-CO-OCH₃, -CH=C(COOCH₃)-CH₂-CO-OC₂H₅, -CH=CH-CH₂-CO-NH₂, -CH=CH-CH₂-CO-NH-CH₃, -CH=CH-CH₂-CO-N(CH₃)₂, -CH(OCH₃)₂, -CH(SCH₃)₂, -CH(OC₂H₅)₂, -CH(SC₂H₅)₂, -CH(O-n-C₃H₇)₂, -CH(O-i-C₃H₇)₂, -CH(S-n-C₃H₇)₂, -CH(S-i-C₃H₇)₂, -CH(O-n-C₄H₉)₂, -CH(O-i-C₄H₉)₂, -CH(O-s-C₄H₉)₂, -CH(O-tert.-C₄H₉)₂, -CH(S-n-C₄H₉)₂, -CH(S-i-C₄H₉)₂, -CH(S-s-C₄H₉)₂, -CH(S-tert.-C₄H₉)₂, -CH(OC₅H₁₁)₂, 1,3-Dioxolan-2-yl, 1,3-Dithiolan-2-yl, 1,3-Oxathiolan-2-yl, 4-Methyl-1,3-dioxolan-2-yl, 4-Methyl-1,3-dithiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 5-Methyl-1,3-oxathiolan-2-yl, 4-Ethyl-1,3-dioxolan-2-yl, 4-Ethyl-1,4-dithiolan-2-yl, 4-Ethyl-1,3-oxathiolan-2-yl, 5-Ethyl-1,3-oxathiolan-2-yl, 4,5-Dimethyl-1,3-dioxolan-2-yl, 4,4-Dimethyl-1,3-dioxolan-2-yl, 4,5-Dimethyl-1,3-dithiolan-2-yl, 5,5-Dimethyl-1,3-dithiolan-2-yl, 4,5-Dimethyl-1,3-oxathiolan-2-yl, 5,5-Dimethyl-1,3-oxathiolan-2-yl, 4,4-Dimethyl-1,3-oxathiolan-2-yl, 4-Vinyl-1,3-dioxolan-2-yl, 4-Vinyl-1,3-dithiolan-2-yl, 4-Vinyl-1,3-oxathiolan-2-yl, 5-Vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3-dioxolan-2-yl, 5-Chlormethyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3-dithiolan-2-yl, 4-Chlormethyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-1,3-dithiolan-2-yl, 4-Hydroxymethyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl- 1,3-dioxolan-2-yl, 4-Propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxymethyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-1,3-dithiolan-2-yl, 4-Allyloxymethyl-1,3-dithiolan-2-yl, 4-Propargyloxymethyl- 1,3-dithiolan-2-yl, 4-Acetoxymethyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl-1,3-oxathiolan-2-yl, 5-Allyloxymethyl- 1,3-oxathiolan-2-yl, 4-Propargyloxymethyl-1,3-oxathiolan-2-yl, 5-Propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxymethyl- 1,3-oxathiolan-2-yl, 5-Acetoxymethyl-1,3-oxathiolan-2-yl, 4-Methylthiomethyl-1,3-dioxolan-2-yl, 4-Methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-1,3-dioxolan-2-yl, 4-Carboxy-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-4-methyl- 1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-1,3-dithiolan-2-yl, 1,3-Dioxan-2-yl, 1,3-Dithian-2-yl, 1,3-Oxathian-2-yl, 5-Methyl-1,3-dioxan-2-yl, 5-Methyl-1,3-dithian-2-yl, 5-Methyl-1,3-oxathian-2-yl, 5,5-Dimethyl-1,3-dioxan-2-yl, 4,6-Dimethyl- 1,3-dioxan-2-yl, 4,4-Dimethyl-1,3-dioxan-2-yl, 5,5-Dimethyl- 1,3-dithian-2-yl, 4,6-Dimethyl-1,3-dithian-2-yl, 4,4-Dimethyl- 1,3-dithian-2-yl, 5,5-Dimethyl-1,3-oxathian-2-yl, 4,4-Dimethyl- 1,3-oxathian-2-yl, 6,6-Dimethyl-1,3-oxathian-2-yl, 4-Hydroxymethyl-1,3-dioxan-2-yl, 4-Methoxymethyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-1,3-dithian-2-yl, 4-Methoxymethyl-1,3-dithian-2-yl, 4-Allyloxymethyl-1,3-dithian-2-yl, 4-Acetoxymethyl- 1,3-dithian-2-yl, 4-Chlormethyl-1,3-dioxan-2-yl, 4-Chlormethyl- 1,3-dithian-2-yl, 1,3-Dioxepan-2-yl, 1,3-Dithiepan-2-yl, 1,3-Dioxep-5-en-2-yl, 4-Methoxycarbonyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl- 1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-1,3-dithian-4-yl, 4-n-Butoxycarbonyl-1,3-dithian-2-yl, 4-Methoxycarbonyl-4- methyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl- 4-methyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-4-methyl- 1,3-dithian-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithian-2-yl, -C(CH₃)(OCH₃)₂, -C(CH₃)(SCH₃)₂, -C(CH₃)(OC₂H₅)₂, -C(CH₃)(SC₂H₅)₂, -C(CH₃)(O-n-C₃H₇)₂, -C(CH₃)(O-i-C₃H₇)₂, -C(CH₃)(S-n-C₃H₇)₂, -C(CH₃)(S-i-C₃H₇)₂, -C(CH₃)(O-n-C₄H₉)₂, -C(CH₃)(O-i-C₄H₉)₂, -C(CH₃)(O-s-C₄H₉)₂, -C(CH₃)(O-tert.-C₄H₉)₂, -C(CH₃)(S-n-C₄H₉)₂, -C(CH₃)(S-i-C₄H₉)₂, -C(CH₃)(S-s-C₄H₉)₂, -C(CH₃)(S-tert.-C₄H₉)₂, -C(CH₃)(O-n-C₅H₁₁)′′, 2-Methyl-1,3-dioxolan-2-yl, 2-Methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-oxathiolan-2-yl, 2,4-Dimethyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-1,3- oxathiolan-2-yl, 2,5-Dimethyl-1,3-oxathiolan-2-yl, 4-Ethyl-2- methyl-1,3-dioxolan-2-yl, 4-Ethyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Ethyl-2-methyl-1,3- oxathiolan-2-yl, 2,4,5-Trimethyl-1,3-dioxolan-2-yl, 2,4,4-Trimethyl- 1,3-dioxolan-2-yl, 2,4,5-Trimethyl-1,3-dithiolan-2-yl, 2,4,4-Trimethyl-1,3-dithiolan-2-yl, 2,4,5-Trimethyl-1,3-oxathiolan-2-yl, 2,4,4-Trimethyl-1,3-oxathiolan-2-yl, 2-Methyl-4-vinyl- 1,3-dioxolan-2-yl, 2-Methyl-4-vinyl-1,3-dithiolan-2-yl, 2-Methyl- 4-vinyl-1,3-oxathiolan-2-yl, 2-Methyl-5-vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-dioxolan-2-yl, 4-Chlormethyl-2- methyl-1,3-dithiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl- 2-methyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-2- methyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dioxolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxy- 2-methyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dithiolan-2-yl, 4-Acetoxy-2- methyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl- 2-methyl-1,3-oxathiolan-2-yl, 5-Allyloxymethyl-2- methyl-1,3-oxathiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3- oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxy-2-methyl-1,3-oxathiolan-2-yl, 5-Acetoxy-2-methyl- 1,3-oxathiolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dioxolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-2- methyl-1,3-dioxolan-2-yl, 4-Carboxy-2-methyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-2- methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl- 2-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-2- methyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-ethoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4- ethoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl- 1,3-dioxolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl-1,3- dithiolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-dioxan-2-yl, 2-Methyl-1,3-dithian-2-yl, 2-Methyl-1,3-oxathian-2-yl, 2,5- Dimethyl-1,3-dioxan-2-yl, 2,5-Dimethyl-1,3-dithian-2-yl, 2,5-Dimethyl- 1,3-oxathian-2-yl, 2,5,5-Trimethyl-1,3-dioxan-2-yl, 2,4,6- Trimethyl-1,3-dioxan-2-yl, 2,2,4-Trimethyl-1,3-dioxan-2-yl, 2,5,5-Trimethyl-1,3-dithian-2-yl, 2,4,6-Trimethyl-1,3-dithian-2-yl, 2,4,4-Trimethyl-1,3-dithian-2-yl, 2,5,5-Trimethyl-1,3-oxathian-2-yl, 2,4,4-Trimethyl-1,3-oxathian-2-yl, 2,6,6-Trimethyl- 1,3-oxathian-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-2- methyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dithian-2-yl, 4-Methoxymethyl-2- methyl-1,3-dithian-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithian-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dithian-2-yl, 4-Chlormethyl-2- methyl-1,3-dioxan-2-yl, 4-Chlormethyl-2-methyl-1,3-dithian-2-yl, -C(CH₃)=NH, -C(CH₃)=N-CH₃, -C(CH₃)=N-C₂H₅, -C(CH₃)=N-n-C₃H₇, -(CH₃)=N-i-C₃H₇, -C(CH₃)=N-n-C₄H₉, -C(CH₃)=N-CH₂CH=CH₂, -C(CH₃)=N-CH₂CH=CH₂-CH₃, -C(CH₃)=N-CH₂C≡CH, -C(CH₃)=N-CH₂C≡C-CH₃, -C(CH₃)=N-cyclopropyl, -C(CH₃)=N-cyclobutyl, -C(CH₃)=N-cyclopentyl, -C(CH₃)=N-cyclohexyl, -C(CH₃)=N-cycloheptyl, -C(CH₃)=N-CH₂-CH₂Cl, -C(CH₃)=N-CH₂Cl, -C(CH₃)=N-C₆H₅, -C(CH₃)=N-(2-F-C₆H₄), -C(CH₃)=N-(3-F-C₆H₄), -C(CH₃)=N-(4-F-C₆H₄), -C(CH₃)=N-(2-Cl-C₆H₄), -C(CH₃)=N-(3-Cl-C₆H₄), -C(CH₃)=N-(4-Cl-C₆H₄), -C(CH₃)=N-(2-CH₃-C₆H₄), -C(CH₃)=N-(3-CH₃-C₆H₄), -C(CH₃)=N-(4-CH₃-C₆H₄), -C(CH₃)=N-(2-CF₃-C₆H₄), -C(CH₃)=N-(3-CF₃-C₆H₄), -C(CH₃)=N-(4-CF₃-C₆H₄), -C(CH₃)=N-(2-OCH₃-C₆H₄), -C(CH₃)=N-(3-OCH₃-C₆H₄), -C(CH₃)=N-(4-OCH₃-C₆H₄), -C(CH₃)=N-(4-NO₂-C₆H₄), -C(CH₃)=N-(4-CN-C₆H₄), -C(CH₃)=N-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-(2,4-(CH₃)₂-C₆H₃), -C(CH₃)=N-CH₂-OCH₃, -C(CH₃)=N-CH₂-OC₂H₅, -C(CH₃)=N-CH₂CH₂-OCH₃, -C(CH₃)=N-CH₂CH₂-OC₂H₅, -C(CH₃)=N-OH, -C(CH₃)=N-OCH₃, -C(CH₃)=N-OC₂H₅, -C(CH₃)=N-O-n-C₃H₇, -C(CH₃)=N-O-i-C₃H₇, -C(CH₃)=N-O-n-C₄H₉, -C(CH₃)=N-O-i-C₄H₉, -C(CH₃)=N-O-s-C₄H₉, -C(CH₃)=N-O-tert.-C₄H₉, -C(CH₃)=N-OCH₂-CH=CH₂, -C(CH₃)=N-OCH(CH₃)-CH=CH₂, -C(CH₃)=N-OCH₂-C≡CH, -C(CH₃)=N-CH(CH₃)-C≡CH, -C(CH₃)=N-OCH₂-CH=C-CH₃, -C(CH₃)=N-OCH₂CH₂-Cl, -C(CH₃)=N-OCH₂CH₂-F, -C(CH₃)=N-OCH₂-CF₃, -C(CH₃)=N-OCH₂-CH=CHCl, -C(CH₃)=N-OCH₂-C(Cl)=CH₂, -C(CH₃)=N-OCH₂-C(Br)=CH₂, -C(CH₃)=N-OCH₂-CH=C(Cl)-CH₃, -C(CH₃)=N-O-CO-CH₃, -C(CH₃)=N-O-CO-C₂H₅, -C(CH₃)=N-OCH₂-CN, -C(CH₃)=N-OCH₂-CH=CH-CH₂-OCH₃, -C(CH₃)=N-OCH₂-CH=CH-CH₂-O-tert.-C₄H₉, -C(CH₃)=N-O-(CH₂)₃-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-(4-Cl-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-C₆H₅, -C(CH₃)=N-OCH₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(3-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-CH₂-(4-CH₃O-C₆H₄), -C(CH₃)=N-OCH₂-CH=C(CH₃)-C₆H₅, -C(CH₃)=N-O-(CH₂)₂-CH=CH-(3,4-Cl₂-C₆H₃), -C(CH₃)=N-O-(CH₂)₃-C≡C-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-OCH₃, -C(CH₃)=N-OCH₂CH₂-OCH₃, -C(CH₃)=N-OCH₂-OC₂H₅, -C(CH₃)=N-OCH(CH₃)-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=N-NH₂, -C(CH₃)=N-NH-CH₃, -C(CH₃)=N-NH-C₂H₅, -C(CH₃)=N-NH-n-C₃H₇, -C(CH₃)=N-NH-i-C₃H₇, -C(CH₃)=N-NH-n-C₄H₉, -C(CH₃)=N-NH-i-C₄H₉, -C(CH₃)=N-NH-s-C₄H₉, -C(CH₃)=N-NH-tert.-C₄H₉, -C(CH₃)=N-NH-cyclopropyl, -C(CH₃)=N-NH-cyclobutyl, -C(CH₃)=N-NH-cyclopentyl, -C(CH₃)=N-NH-cyclohexyl, -C(CH₃)=N-NH-cycloheptyl, -C(CH₃)=N-N(CH₃)₂, -C(CH₃)=N-N(C₂H₅)₂, -C(CH₃)=N-N(n-C₃H₇)₂, -C(CH₃)=N-N(i-C₃H₇)₂, -C(CH₃)=N-NH-CH₂-C=CH, -C(CH₃)=N-NH-CH₂-C≡CH, -C(CH₃)=N-N(CH₃)-CH₂-C≡CH, -C(CH₃)=N-NH-CH₂CF₃, -C(CH₃)=N-NH-CO-CH₃, -C(CH₃)=N-NH-CO-C₂H₅, -C(CH₃)=N-NH-CO-OCH₃, -C(CH₃)=N-NH-CO-OC₂H₅, -C(CH₃)=N-NH-CO-O-tert.-C₄H₉, -C(CH₃)=N-pyrrolidin-1-yl, -C(CH₃)=N-piperidin-1-yl, -C(CH₃)=N-morpholin-4-yl, -C(CH₃)=N-NH-C₆H₅, -C(CH₃)=N-NH-(4-Cl-C₆H₄), -C(CH₃)=N-NH-(4-NO₂-C₆H₄), -C(CH₃)=N-NH-(4-F-C₆H₄), -C(CH₃)=N-NH-(4-CH₃O-C₆H₄), -C(CH₃)=N-NH-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-NH-(2,4-(NO₂)₂-C₆H₃), -C(CH₃)=N-NH-CO-NH₂, -C(CH₃)=N-NH-CO-NHCH₃, -C(CH₃)=N-NH-CO-NHC₂H₅, -C(CH₃)=N-NH-CO-N(CH₃)₂, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=CH-CO-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-O-n-C₄H₉, -C(CH₃)=CH-CO-O-tert.-C₄H₉, -C(CH₃)=CH-CO-O-cyclopropyl, -C(CH₃)=CH-CO-O-cyclobutyl, -C(CH₃)=CH-CO-O-cyclopentyl, -C(CH₃)=CH-CO-O-cyclohexyl, -C(CH₃)=CH-CO-O-cycloheptyl, -C(CH₃)=C(CH₃)-COOH, -C(CH₃)=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-cyclopropyl, -C(CH₃)=C(CH₃)-CO-O-cyclobutyl, -C(CH₃)=C(CH₃)-CO-O-cyclopentyl, -C(CH₃)=C(CH₃)-CO-O-cyclohexyl, -C(CH₃)=C(CH₃)-CO-O-cycloheptyl, -C(CH₃)=C(C₂H₅)-COOH, -C(CH₃)=C(C₂H₅)-CO-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-cyclo­ propyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-O- cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-O-cycloheptyl, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=C(Cl)-CO-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-O-n-C₄H₉, -C(CH₃)=C(Cl)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-O-cyclopropyl, -C(CH₃)=C(Cl)-CO-O-cyclobutyl, -C(CH₃)=C(Cl)-CO-O-cyclopentyl, -C(CH₃)=C(Cl)-CO-O-cyclohexyl, -C(CH₃)=C(Cl)-CO-O-cycloheptyl, -C(CH₃)=C(Br)-COOH, -C(CH₃)=C(Br)-CO-OCH₃, -C(CH₃)=C(Br)-CO-OC₂H₅, -C(CH₃)=C(Br)-CO-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-O-n-C₄H₉, -C(CH₃)=C(Br)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-O-cyclopropyl, -C(CH₃)=C(Br)-CO-O-cyclobutyl, -C(CH₃)=C(Br)-CO-O-cyclopentyl, -C(CH₃)=C(Br)-CO-O-cyclohexyl, -C(CH₃)=C(Br)-CO-O-cycloheptyl, -C(CH₃)=C(CN)-COOH, -C(CH₃)=C(CN)-CO-OCH₃, -C(CH₃)=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CN)-CO-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-O-n-C₄H₉, -C(CH₃)=C(CN)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-O-cyclopropyl, -C(CH₃)=C(CN)-CO-O-cyclobutyl, -C(CH₃)=C(CN)-CO-O-cyclopentyl, -C(CH₃)=C(CN)-CO-O-cyclohexyl, -C(CH₃)=C(CN)-CO-O-cycloheptyl, -C(CH₃)=CH-CO-OCH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=CH-CO-O-i-C₃H₇, -C(CH₃)=CH-CO-OCH(CH₃)-OCH₃, -C(CH₃)=CH-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=CH-CO-OCH₂CH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=(C₂H₅)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-O-i-C₃H₇, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-O-i-C₃H₇, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-O-i-C₃H₇, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-CF₃, -C(CH₃)=CH-CO-OCH₂-CCl₃, -C(CH₃)=CH-CO-OCH₂-oxiranyl, -C(CH₃)=CH-CO-O-(CH₂)₃-Br, -C(CH₃)=CH-CO-OCH₂-CH=CH₂, -C(CH₃)=CH-CO-OCH₂-C≡CH, -C(CH₃)=CH-CO-OCH₂-CN, -C(CH₃)=CH-CO-OCH₂CH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CF₃, -C(CH₃)=C(CH₃)-CO-OCH₂-CCl₃, -C(CH₃)=C(CH₃)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CH₃)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CH₃)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CH₃)-CO-OCH₂-C≡CH, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CF₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CCl₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-oxiranyl, -C(CH₃)=C(C₂H₅)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(C₂H₅)-CO-OCH₂-C≡CH, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂-CF₃, -C(CH₃)=C(Cl)-CO-OCH₂-CCl₃, -C(CH₃)=C(Cl)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Cl)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Cl)-CO-OCH₂-CH≡CH₂, -C(CH₃)=C(Cl)-CO-OCH₂-C≡CH, -C(CH₃)=C(Cl)-CO-OCH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂-CF₃, -C(CH₃)=C(Br)-CO-OCH₂-CCl₃, -C(CH₃)=C(Br)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Br)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Br)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Br)-CO-OCH₂-C≡CH, -C(CH₃)=C(Br)-CO-OCH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂CH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂-CF₃, -C(CH₃)=C(CN)-CO-OCH₂-CCl₃, -C(CH₃)=C(CN)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CN)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(CN)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CN)-CO-OCH₂-C≡CH, -C(CH₃)=C(CN)-CO-OCH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂CH₂-CN, -C(CH₃)=CH-CO-CH₃, -C(CH₃)=CH-CO-C₂H₅, -C(CH₃)=CH-CO-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-n-C₄H₉, -C(CH₃)=CH-CO-tert.-C₄H₉, -C(CH₃)=CH-CO-CH₂Cl, -C(CH₃)=CH-CO-CH₂Br, -C(CH₃)=CH-CO-CHCl₂, -C(CH₃)=CH-CO-CH₂-OCH₃, -C(CH₃)=CH-CO-CH(OCH₃)₂, -C(CH₃)=CH-CO-CH₂-SCH₃, -C(CH₃)=C(CH₃)-CO-CH₃, -C(CH₃)=C(CH₃)-CO-C₂H₅, -C(CH₃)=C(CH₃)-CO-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-CH₂Cl, -C(CH₃)=C(CH₃)-CO-CH₂Br, -C(CH₃)=C(CH₃)-CO-CHCl₂, -C(CH₃)=C(CH₃)-CO-CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-CH(OCH₃)₂, -C(CH₃)=C(CH₃)-CO-CH₂-SCH₃, -C(CH₃)=C(C₂H₅)-CO-CH₃, -C(CH₃)=C(C₂H₅)-CO-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-CH₂Cl, -C(CH₃)=C(C₂H₅)-CO-CH₂Br, -C(CH₃)=C(C₂H₅)-CO-CHCl₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-CH(OCH₃)₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-SCH₃, -C(CH₃)=C(Cl)-CO-CH₃, -C(CH₃)=C(Cl)-CO-C₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-n-C₄H₉, -C(CH₃)=C(Cl)-CO-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-CH₂Cl, -C(CH₃)=C(Cl)-CO-CHCl₂, -C(CH₃)=C(Cl)-CO-CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-CH(OCH₃)₂, -C(CH₃)=C(Cl)-CO-CH₂-SCH₃, -C(CH₃)=C(Br)-CO-CH₃, -C(CH₃)=C(Br)-CO-C₂H₅, -C(CH₃)=C(Br)-CO-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-n-C₄H₉, -C(CH₃)=C(Br)-CO-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-CH₂Cl, -C(CH₃)=C(Br)-CO-CH₂Br, -C(CH₃)=C(Br)-CO-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-CH(OCH₃)₂, -C(CH₃)=C(Br)-CO-CH₂-SCH₃, -C(CH₃)=C(CN)-CO-CH₃, -C(CH₃)=C(CN)-CO-C₂H₅, -C(CH₃)=C(CN)-CO-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-n-C₄H₉, -C(CH₃)=C(CN)-CO-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-CH₂Cl, -C(CH₃)=C(CN)-CO-CH₂Br, -C(CH₃)=C(CN)-CO-CHCl₂, -C(CH₃)=C(CN)-CO-CH₂-OCH₃, -C(CH₃)=C(CN)-CO-CH(OCH₃)₂, -C(CH₃)=C(CN)-CO-CH₂-SCH₃, -C(CH₃)=CH-CO-C₆H₅, -C(CH₃)=CH-CO-(4-Cl-C₆H₄), -C(CH₃)=C(CH₃)-CO-C₆H₅, -C(CH₃)=C(CH₃)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(C₂H₅)-CO-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(Cl)-CO-C₆H₅, -C(CH₃)=C(Br)-CO-C₆H₅, -C(CH₃)=C(CN)-CO-C₆H₅, -C(CH₃)=CH-CO-NH₂, -C(CH₃)=CH-CO-NHCH₃, -C(CH₃)=CH-CO-N(CH₃)₂, -C(CH₃)=CH-CO-NH-C₂H₅, -C(CH₃)=CH-CO-N(C₂H₅)₂, -C(CH₃)=CH-CO-NH-n-C₃H₇, -C(CH₃)=CH-CO-NH-i-C₃H₇, -C(CH₃)=CH-CO-NH-tert.-C₄H₉, -C(CH₃)=CH-CO-NH-cyclopropyl, -C(CH₃)=CH-CO-NH-cyclobutyl, -C(CH₃)=CH-CO-NH-cyclopentyl, -C(CH₃)=CH-CO-NH-cyclohexyl, -C(CH₃)=CH-CO-NH-cycloheptyl, -C(CH₃)=CH-CO-NH-cyclooctyl, -C(CH₃)=CH-CO-pyrrolidin-1-yl, -C(CH₃)=CH-CO-piperidin-1-yl, -C(CH₃)=CH-CO-morpholin-4-yl, -C(CH₃)=CH-CO-NH-CH₂CH=CH₂, -C(CH₃)=CH-CO-NH-CH₂C≡CH, -C(CH₃)=CH-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=CH-CO-NH-(CH₂)₂Cl, -C(CH₃)=CH-CO-NH-C₆H₅, -C(CH₃)=C(CH₃)-CO-NH₂, -C(CH₃)=C(CH₃)-CO-NHCH₃, -C(CH₃)=C(CH₃)-CO-N(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-C₂H₅, -C(CH₃)=C(CH₃)-CO-N(C₂H₅)₂, -C(CH₃)=C(CH₃)-CO-NH-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-NH- cyclopropyl, -C(CH₃)=C(CH₃)-CO-NH-cyclobutyl, -C(CH₃)=C(CH₃)-CO-NH-cyclopentyl, -C(CH₃)=C(CH₃)-CO-NH- cyclohexyl, -C(CH₃)=C(CH₃)-CO-NH-cycloheptyl, -C(CH₃)=C(CH₃)-CO-NH-cyclooctyl, -C(CH₃)=C(CH₃)-CO- pyrrolidin-1-yl, -C(CH₃)=C(CH₃)-CO-piperidin-1-yl, -C(CH₃)=C(CH₃)-CO-morpholin-4-yl, -C(CH₃)=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CH₃)-CO-NH-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-NH₂, -C(CH₃)=C(C₂H₅)-CO-NHCH₃, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)₂, -C(CH₃)=C(C₂H₅)-CO-NH-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-N(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-NH- cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclo­ hexyl, -C(CH₃)=C(C₂H₅)-CO-NH-cycloheptyl, -C(CH₃)=C(C₂H₅)-CO-NH- cyclooctyl, -C(CH₃)=C(C₂H₅)-CO-pyrrolidin-1-yl, -C(CH₃)=C(C₂H₅)-CO-piperidin-1-yl, -C(CH₃)=C(C₂H₅)-CO- morpholin-4-yl, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(C₂H₅)-CO-NH-C₆H₅, -C(CH₃)=C(Cl)-CO-NH₂, -C(CH₃)=C(Cl)-CO-NHCH₃, -C(CH₃)=C(Cl)-CO-N(CH₃)₂, -C(CH₃)=C(Cl)-CO-NH-C₂H₅, -C(CH₃)=C(Cl)-CO-N(C₂H₅)₂, -C(CH₃)=C(Cl)-CO-NH-n-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-i-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-NH-cyclopropyl, -C(CH₃)=C(Cl)-CO-NH-cyclobutyl, -C(CH₃)=C(Cl)-CO-NH-cyclopentyl, -C(CH₃)=C(Cl)-CO-NH-cyclohexyl, -C(CH₃)=C(Cl)-CO-NH-cycloheptyl, -C(CH₃)=C(Cl)-CO-NH-cyclooctyl, -C(CH₃)=C(Cl)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Cl)-CO-piperidin-1- yl, -C(CH₃)=C(Cl)-CO-morpholin-4-yl, -C(CH₃)=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -C(CH₃)=C(Cl)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Cl)-CO-NH-C₆H₅, -C(CH₃)=C(Br)-CO-NH₂, -C(CH₃)=C(Br)-CO-NHCH₃, -C(CH₃)=C(Br)-CO-N(CH₃)₂, -C(CH₃)=C(Br)-CO-NH-C₂H₅, -C(CH₃)=C(Br)-CO-N(C₂H₅)₂, -C(CH₃)=C(Br)-CO-NH-n-C₃H₇, -C(CH₃)=C(Br)-CO-NH-i-C₃H₇, -C(CH₃)=C(Br)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-NH-cyclopropyl, -C(CH₃)=C(Br)-CO-NH-cyclobutyl, -C(CH₃)=C(Br)-CO-NH-cyclopentyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cycloheptyl, -C(CH₃)=C(Br)-CO-NH-cyclooctyl, -C(CH₃)=C(Br)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Br)-CO-piperidin-1-yl, -C(CH₃)=C(Br)-CO-morpholin-4-yl, -C(CH₃)=C(Br)-CO-NH-CH₂CH=C(Br)₂, -C(CH₃)=C(Br)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Br)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Br)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Br)-CO-NH-C₆H₅, -C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CN)-CO-NHCH₃, -C(CH₃)=C(CN)-CO-N(CH₃)₂, -C(CH₃)=C(CN)-CO-NH-C₂H₅, -C(CH₃)=C(CN)-CO-N(C₂H₅)₂, -C(CH₃)=C(CN)-CO-NH-n-C₃H₇, -C(CH₃)=C(CN)-CO-NH-i-C₃H₇, -C(CH₃)=C(CN)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-NH-cyclopropyl, -C(CH₃)=C(CN)-CO-NH-cyclobutyl, -C(CH₃)=C(CN)-CO-NH-cyclopentyl, -C(CH₃)=C(CN)-CO-NH-cyclohexyl, -C(CH₃)=C(CN)-CO-NH-cycloheptyl, -C(CH₃)=C(CN)-CO-NH-cyclooctyl, -C(CH₃)=C(CN)-CO-pyrrolidin-1-yl, -C(CH₃)=C(CN)-CO-piperidin-1-yl, -C(CH₃)=C(CN)-CO-morpholin-4-yl, -C(CH₃)=C(CN)-CO-NH-CH₂CH=C(CN)₂, -C(CH₃)=C(CN)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CN)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CN)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CN)-CO-NH-C₆H₅, -C(CH₃)=CH-CO-SCH₃, -C(CH₃)=CH-CO-SC₂H₅, -C(CH₃)=CH-CO-S-n-C₃H₇, -C(CH₃)=CH-CO-S-i-C₃H₇, -C(CH₃)=CH-CO-S-n-C₄H₉, -C(CH₃)=CH-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-SCH₃, -C(CH₃)=C(CH₃)-CO-SC₂H₅, -C(CH₃)=C(CH₃)-CO-S-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-S-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-SCH₃, -C(CH₃)=C(C₂H₅)-CO-SC₂H₅, -C(CH₃)=C(C₂H₅)-CO-S-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-SCH₃, -C(CH₃)=C(Cl)-CO-SC₂H₅, -C(CH₃)=C(Cl)-CO-S-n-C₃H₇, -C(CH₃)=C(Cl)-CO-S-i-C₃H₇, -C(CH₃)=C(Cl)-CO-S-n-C₄H₉, -C(CH₃)=C(Cl)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-SCH₃, -C(CH₃)=C(Br)-CO-SC₂H₅, -C(CH₃)=C(Br)-CO-S-n-C₃H₇, -C(CH₃)=C(Br)-CO-S-i-C₃H₇, -C(CH₃)=C(Br)-CO-S-n-C₄H₉, -C(CH₃)=C(Br)-CO-S-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-SCH₃, -C(CH₃)=C(CN)-CO-SC₂H₅, -C(CH₃)=C(CN)-CO-S-n-C₃H₇, -C(CH₃)=C(CN)-CO-S-i-C₃H₇, -C(CH₃)=C(CN)-CO-S-n-C₄H₉, -C(CH₃)=C(CN)-CO-S-tert.-C₄H₉, -C(CH₃)=C(COCH₃)-CO-OCH₃, -C(CH₃)=C(COC₂H₅)-CO-OCH₃, -C(CH₃)=C(CO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COCH₃)-CO-OC₂H₅, -C(CH₃)=C(COC₂H₅)-CO-OC₂H₅, -C(CH₃)=C(CO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COCH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(COC₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-OCH₃, -C(CH₃)=C(CF₃)-CO-OC₂H₅, -C(CH₃)=C(CF₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CF₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(COOCH₃)₂, -C(CH₃)=C(COOC₂H₅)₂, -C(CH₃)=C(COOCH₃)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)₂, -C(CH₃)=CH-CH=CH-COOH, -C(CH₃)=CH-CH=CH-CO-OCH₃, -C(CH₃)=CH-CH=CH-CO-OC₂H₅, -C(CH₃)=CH-CH=C(COOCH₃)₂, -C(CH₃)=CH-CH=C(CN)-CO-OCH₃, -C(CH₃)=CH-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH₂, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -C(CH₃)=CH-(CH₂)₂-COOH, -C(CH₃)=CH-(CH₂)₂-CO-OCH₃, -C(CH₃)=CH-(CH₂)₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(COOCH₃)₂, -C(CH₃)=CH-CH₂-CH(COOC₂H₅)₂, -C(CH₃)=CH-CH₂-CH(CN)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CN)-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -C(CH₃)=CH-(CH₂)₂-CO-NH₂, -C(CH₃)=CH-(CH₂)₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-COOH, -C(CH₃)=CH-CH₂-CO-OCH₃, -C(CH₃)=CH-CH₂-CO-OC₂H₅, -C(CH₃)=C(COOCH₃)-CH₂-CO-OCH₃, -C(CH₃)=C(COOCH₃)-CH₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CO-NH₂, -C(CH₃)=CH-CH₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-CO-N(CH₃)₂.
wobei W für eine der folgenden Bedeutungen steht:
-CHO, -COCH₃, -COC₂H₅, -CO-n-C₃H₇, -CO-i-C₃H₇, -CO-n-C₄H₉, -CO-i-C₄H₉, -CO-s-C₄H₉, -CO-tert.-C₄H₉, -CO-CH₂CH=CH₂, -CO-CF₃, -COCCl₃, -COCH₂C≡CH, -CO-cyclopropyl, -CO-cyclobutyl, -CO-cyclopentyl, -CO-cyclohexyl, -CO-CN, -CO-COOCH₃, -CO-COOC₂H₅, -CH=NH, -CH=NCH₃, -CH=NC₂H₅, -CH=N-n-C₃H₅, -CH=N-i-C₃H₅, -CH=N-n-C₄H₉, -CH=NCH₂CH=CH₂, -CH=NCH₂CH=CH₂-CH₃, -CH=NCH₂C≡CH, -CH=NCH₂C≡C-CH₃, -CH=N-cyclopropyl, -CH=N-cyclobutyl, -CH=N-cyclopentyl, -CH=N-cyclohexyl, -CH=N-cycloheptyl, -CH=N-CH₂-CH₂Cl, -CH=N-CH₂Cl, -CH=N-C₆H₅, -CH=N-4-Br-C₆H₄, -CH=N-3-F-C₆H₄, -CH=N-4-F-C₆H₄, -CH=N-2-Cl-C₆H₄, -CH=N-3-Cl-C₆H₄, -CH=N-4-Cl-C₆H₄, -CH=N-2-Br-C₆H₄, -CH=N-2-F-C₆H₄, -CH=N-2-CH₃-C₆H₄, -CH=N-3-CH₃-C₆H₄, -CH=N-4-CH₃-C₆H₄, -CH=N-2-CF₃-C₆H₄, -CH=N-3-CF₃-C₆H₄, -CH=N-4-CF₃-C₆H₄, -CH=N-2-OCH₃-C₆H₄, -CH=N-3-OCH₃-C₆H₄, -CH=N-4-OCH₃-C₆H₄, -CH=N-4-NO₂-C₆H₄, -CH=N-4-CN-C₆H₄, -CH=N-2,4-(Cl,Cl)-C₆H₄, -CH=N-2,4-(CH₃,CH₃)-C₆H₄, -CH=N-CH₂OCH₃, -CH=N-CH₂OC₂H₅, -CH=N-CH₂CH₂OCH₃, -CH=N-CH₂CH₂OC₂H₅, -CH=N-OH, -CH=N-OCH₃, -CH=N-OC₂H₅, -CH=N-O-n-C₃H₇, -CH=N-O-i-C₃H₇, -CH=N-O-n-C₄H₉, -CH=N-O-i-C₄H₉, -CH=N-O-s-C₄H₉, -CH=N-O-tert.-C₄H₉, -CH=N-O-CH₂CH=CH₂, -CH=N-O-CH(CH₃)CH=CH₂, -CH=N-O-CH₂C≡CH, -CH=N-O-CH(CH₃)-C≡CH, -CH=N-O-CH₂-CH=CH-CH₃, -CH=N-O-CH₂-CH₂-Cl, -CH=N-O-CH₂-CH₂-F, -CH=N-O-CH₂-CF₃, -CH=N-O-CH₂-CH=CHCl, -CH=N-O-CH₂-CCl=CH₂, -CH=N-O-CH₂-CBr=CH₂, -CH=N-O-CH₂-CH=CCl-CH₃, -CH=N-OC(O)CH₃, -CH=N-OC(O)C₂H₅, -CH=N-O-CH₂-CN, -CH=N-O-CH₂-CH=CH-CH₂-O-CH₃, -CH=N-O-CH₂-CH=CH-CH₂-O-tert.-C₄H₉, -CH=N-O-(CH₂)₃-C₆H₅, -CH=N-O-(CH₂)₄-C₆H₅, -CH=N-O-(CH₂)₄-4-Cl-C₆H₄, -CH=N-O-(CH₂)₄-4-OCH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-CH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-C₆H₅, -CH=N-O-CH₂CH=CH-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CH-3-OCH₃-C₆H₄, -CH=N-O-(CH₂)₂CH=CH-4-F-C₆H₄, -CH=N-O-(CH₂)CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CHCH₂-4-OCH₃-C₆H₄, -CH=N-O-CH₂-CH=C(CH₃)-C₆H₄ -CH=N-O-(CH₂)₂CH=CH-3,4(Cl,Cl)-C₆H₃, -CH=N-O-(CH₂)₃C≡C-4-F-C₆H₄, -CH₂=N-OCHOCH₃, -CH=N-OC₂H₄OCH₃, -CH=N-OCH₂OC₂H₅, -CH=N-OCH(CH₃)OCH₃, -CH=N-OCH(CH₃)COOCH₃, -CH=N-OCH(CH₃)COO-n-C₄H₉, -CH=N-NH₂, -CH=N-NHCH₃, -CH=N-NHC₂H₅, -CH=N-NH-n-C₃H₇, -CH=N-NH-i-C₃H₇, -CH=N-NH-n-C₄H₉, -CH=N-NH-i-C₄H₉, -CH=N-NH-s-C₄H₉, -CH=N-NH-tert.-C₄H₉, -CH=N-NH-cyclopropyl, -CH=N-NH-cyclobutyl, -CH=N-NH-cyclopentyl, -CH=N-NH-cyclohexyl, -CH=N-NH-cycloheptyl, -CH=N-N(CH₃)₂, -CH=N-N(C₂H₅)₂, -CH=N-N(C₃H₇)₂, -CH=N-N(i-C₃H₇)(CH₃), -CH=N-NHCH₂-C=CH, -CH=N-NHCH₂-C≡CH, -CH=N-N(CH₃)-CH₂-C≡CH, -CH=N-NHCH₂CF₃, -CH=N-NH-CO-CH₃, -CH=N-NH-CO-CH₂H₅, -CH=N-NH-COOCH₃, -CH=N-NH-COOC₂H₅, -CH=N-NH-COO-tert.-C₄H₉, -CH=N-pyrrolidin-1-yl, -CH=N-piperidin-1-yl, -CH=N-morpholin-4-yl, -CH=N-NH-C₆H₅, -CH=N-NH-(4-Cl-C₆H₄), -CH=N-NH-(4-NO₂-C₆H₄), -CH=N-NH-(4-F-C₆H₄), -CH=N-NH-(4-CH₃O-C₆H₄), -CH=N-NH-(2,4-Cl₂-C₆H₃), -CH=N-NH-(2,4-(NO₂)₂-C₆H₃), -CH=N-NH-CO-NH₂, -CH=N-NH-CO-NHCH₃, -CH=N-NH-CO-NHC₂H₅, -CH=N-NH-CO-N(CH₃)₂, -CH=CH-COOH, -CH=CH-CO-OCH₃, -CH=C-CO-OC₂H₅, -CH=CH-CO-O-n-C₃H₇, -CH=CH-CO-O-i-C₃H₇, -CH=CH-CO-O-n-C₄H₉, -CH=CH-CO-O-tert.-C₄H₉, -CH=CH-CO-O-cyclopropyl, -CH=CH-CO-O-cyclobutyl, -CH=CH-CO-O-cyclopentyl, -CH=CH-CO-O-cyclohexyl, -CH=CH-CO-O-cycloheptyl, -CH=C(CH₃)-COOH, -CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CO-O-n-C₃H₇, -CH=C(CH₃)-CO-O-i-C₃H₇, -CH=C(CH₃)-CO-O-n-C₄H₉, -CH=C(CH₃)-CO-O-tert.-C₄H₉, -CH=C(CH₃)-CO-O-cyclopropyl, -CH=C(CH₃)-CO-O-cyclobutyl, -CH=C(CH₃)-CO-O-cyclopentyl, -CH=C(CH₃)-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cycloheptyl, -CH=C(C₂H₅)-COOH, -CH=C(C₂H₅)-CO-OCH₃, -CH=C(C₂H₅)-CO-OC₂H₅, -CH=C(C₂H₅)-CO-O-n-C₃H₇, -CH=C(C₂H₅)-CO-O-i-C₃H₇, -CH=C(C₂H₅)-CO-O-n-C₄H₉, -CH=C(C₂H₅)-CO-O-tert.-C₄H₉, -CH=C(C₂H₅)-CO-O-cyclopropyl, -CH=C(C₂H₅)-CO-O-cyclobutyl, -CH=C(C₂H₅)-CO-O-cyclopentyl, -CH=C(C₂H₅)-CO-O-cyclohexyl, -CH=C(C₂H₅)-CO-O-cycloheptyl, -CH=C(Cl)-COOH, -CH=C(Cl)-CO-OCH₃, -CH=C(Cl)-CO-OC₂H₅, -CH=C(Cl)-CO-O-n-C₃H₇, -CH=C(Cl)-CO-O-i-C₃H₇, -CH=C(Cl)-CO-O-n-C₄H₉, -CH=C(Cl)-CO-O-tert.-C₄H₉, -CH=C(Cl)-CO-O-cyclopropyl, -CH=C(Cl)-CO-O-cyclobutyl, -CH=C(Cl)-CO-O-cyclopentyl, -CH=C(Cl)-CO-O-cyclohexyl, -CH=C(Cl)-CO-O-cycloheptyl, -CH=C(Br)-COOH, -CH=C(Br)-CO-OCH₃, -CH=C(Br)-CO-OC₂H₅, -CH=C(Br)-CO-O-n-C₃H₇, -CH=C(Br)-CO-O-i-C₃H₇, -CH=C(Br)-CO-O-n-C₄H₉, -CH=C(Br)-CO-O-tert.-C₄H₉, -CH=C(Br)-CO-O-cyclopropyl, -CH=C(Br)-CO-O-cyclobutyl, -CH=C(Br)-CO-O-cyclopentyl, -CH=C(Br)-CO-O-cyclohexyl, -CH=C(Br)-CO-O-cycloheptyl, -CH=C(CN)-COOH, -CH=C(CN)-CO-OCH₃, -CH=C(CN)-CO-OC₂H₅, -CH=C(CN)-CO-O-n-C₃H₇, -CH=C(CN)-CO-O-i-C₃H₇, -CH=C(CN)-CO-O-n-C₄H₉, -CH=C(CN)-CO-O-tert.-C₄H₉, -CH=C(CN)-CO-O-cyclopropyl, -CH=C(CN)-CO-O-cyclobutyl, -CH=C(CN)-CO-O-cyclopentyl, -CH=C(CN)-CO-O-cyclohexyl, -CH=C(CN)-CO-O-cycloheptyl, -CH=CH-CO-OCH₂-OCH₃, -CH=CH-CO-OCH₂-OC₂H₅, -CH=CH-CO-OCH₂-O-n-C₃H₅, -CH=CH-CO-OCH₂-O-i-C₃H₅, -CH=CH-CO-OCH(CH₃)-OCH₃, -CH=CH-CO-OCH(CH₃)-OC₂H₅, -CH=CH-CO-O-CH₂CH₂-OCH₃, -CH=CH-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-OCH₃, -CH=C(CH₃)-CO-OCH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-O-n-C₃H₅, -CH=C(CH₃)-CO-OCH₂-O-i-C₃H₅, -CH=C(CH₃)-CO-OCH(CH₃)-OCH₃, -CH=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CH₃)-CO-O-CH₂CH₂-OCH₃, -CH=C(CH₃)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-OCH₃, -CH=C(C₂H₅)-CO-OCH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-O-n-C₃H₅, -CH=C(C₂H₅)-CO-OCH₂-O-i-C₃H₅, -CH=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -CH=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OCH₃, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-OCH₃, -CH=C(Cl)-CO-OCH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-O-n-C₃H₅, -CH=C(Cl)-CO-OCH₂-O-i-C₃H₅, -CH=C(Cl)-CO-OCH(CH₃)-OCH₃, -CH=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Cl)-CO-O-CH₂CH₂-OCH₃, -CH=C(Cl)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-OCH₃, -CH=C(Br)-CO-OCH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-O-n-C₃H₅, -CH=C(Br)-CO-OCH₂-O-i-C₃H₅, -CH=C(Br)-CO-OCH(CH₃)-OCH₃, -CH=C(Br)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Br)-CO-O-CH₂CH₂-OCH₃, -CH=C(Br)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-OCH₃, -CH=C(CN)-CO-OCH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-O-n-C₃H₅, -CH=C(CN)-CO-OCH₂-O-i-C₃H₅, -CH=C(CN)-CO-OCH(CH₃)-OCH₃, -CH=C(CN)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CN)-CO-O-CH₂CH₂-OCH₃, -CH=C(CN)-CO-O-CH₂CH₂-OC₂H₅, -CH=CH-CO-OCH₂-CF₃, -CH=CH-CO-OCH₂-CCl₃, -CH=CH-CO-OCH₂-oxiranyl, -CH=CH-CO-O(CH₂)₃-Br, -CH=CH-CO-OCH₂-CH=CH₂, -CH=CH-CO-OCH₂-C≡CH, -CH=CH-CO-OCH₂-CN, -CH=CH-CO-O(CH₂)₂-CN, -CH=C(CH₃)-CO-OCH₂-CF₃, -CH=C(CH₃)-CO-OCH₂-CCl₃, -CH=C(CH₃)-CO-OCH₂-oxiranyl, -CH=C(CH₃)-CO-O(CH₂)₃-Br, -CH=C(CH₃)-CO-OCH₂-CH=CH₂, -CH=C(CH₃)-CO-OCH₂-C≡CH, -CH=C(CH₃)-CO-OCH₂-CN, -CH=C(CH₃)-CO-O(CH₂)₂-CN, -CH=C(C₂H₅)-CO-OCH₂-CF₃, -CH=C(C₂H₅)-CO-OCH₂-CCl₃, -CH=C(C₂H₅)-CO-OCH₂-oxiranyl, -CH=C(C₂H₅)-CO-O(CH₂)₃-Br, -CH=C(C₂H₅)-CO-OCH₂-CH=CH₂, -CH=C(C₂H₅)-CO-OCH₂-C≡CH, -CH=C(C₂H₅)-CO-OCH₂-CN, -CH=C(C₂H₅)-CO-O(CH₂)₂-CN, -CH=C(Cl)-CO-OCH₂-CF₃, -CH=C(Cl)-CO-OCH₂-CCl₃, -CH=C(Cl)-CO-OCH₂-oxiranyl, -CH=C(Cl)-CO-O(CH₂)₃-Br, -CH=C(Cl)-CO-OCH₂-CH=CH₂, -CH=C(Cl)-CO-OCH₂-C≡CH, -CH=C(Cl)-CO-OCH₂-CN, -CH=C(Cl)-CO-O(CH₂)₂-CN, -CH=C(Br)-CO-OCH₂-CF₃, -CH=C(Br)-CO-OCH₂-CCl₃, -CH=C(Br)-CO-OCH₂-oxiranyl, -CH=C(Br)-CO-O(CH₂)₃-Br, -CH=C(Br)-CO-OCH₂-CH=CH₂, -CH=C(Br)-CO-OCH₂-C≡CH, -CH=C(Br)-CO-OCH₂-CN, -CH=C(Br)-CO-O(CH₂)₂-CN, -CH=C(CN)-CO-OCH₂-CF₃, -CH=C(CN)-CO-OCH₂-CCl₃, -CH=C(CN)-CO-OCH₂-oxiranyl -CH=C(CN)-CO-O(CH₂)₃-Br, -CH=C(CN)-CO-OCH₂-CH=CH₂, -CH=C(CN)-CO-OCH₂-C≡CH, -CH=C(CN)-CO-OCH₂-CN, -CH=C(CN)-CO-O(CH₂)₂-CN, -CH=CH-CO-CH₃, -CH=CH-CO-C₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-i-C₃H₇, -CH=CH-CO-n-C₄H₉, -CH=CH-CO-tert.-C₄H₉, -CH=CH-CO-CH₂Cl, -CH=CH-CO-CH₂Br, -CH=CH-CO-CHCl₂, -CH=CH-CO-CH₂-OCH₃, -CH=CH-CO-CH(OCH₃)₂, -CH=CH-CO-CH₂-SCH₃, -CH=C(CH₃)-CO-CH₃, -CH=C(CH₃)-CO-C₂H₅, -CH=C(CH₃)-CO-n-C₃H₇, -CH=C(CH₃)-CO-i-C₃H₇, -CH=C(CH₃)-CO-n-C₄H₉, -CH=C(CH₃)-CO-tert.-C₄H₉, -CH=C(CH₃)-CO-CH₂Cl, -CH=C(CH₃)-CO-CH₂Br, -CH=C(CH₃)-CO-CHCl₂, -CH=C(CH₃)-CO-CH₂-OCH₃, -CH=C(CH₃)-CO-CH(OCH₃)₂, -CH=C(CH₃)-CO-CH₂-SCH₃, -CH=C(C₂H₅)-CO-CH₃, -CH=C(C₂H₅)-CO-C₂H₅, -CH=C(C₂H₅)-CO-n-C₃H₇, -CH=C(C₂H₅)-CO-i-C₃H₇, -CH=C(C₂H₅)-CO-n-C₄H₉, -CH=C(C₂H₅)-CO-tert.-C₄H₉, -CH=C(C₂H₅)-CO-CH₂Cl, -CH=C(C₂H₅)-CO-CH₂Br, -CH=C(C₂H₅)-CO-CHCl₂, -CH=C(C₂H₅)-CO-CH₂-OCH₃, -CH=C(C₂H₅)-CO-CH(OCH₃)₂, -CH=C(C₂H₅)-CO-CH₂-SCH₃, -CH=C(Cl)-CO-CH₃, -CH=C(Cl)-CO-C₂H₅, -CH=C(Cl)-CO-n-C₃H₇, -CH=C(Cl)-CO-i-C₃H₇, -CH=C(Cl)-CO-n-C₄H₉, -CH=C(Cl)-CO-tert.-C₄H₉, -CH=C(Cl)-CO-CH₂Cl, -CH=C(Cl)-CO-CH₂Br, -CH=C(Cl)-CO-CHCl₂, -CH=C(Cl)-CO-CH₂-OCH₃, -CH=C(Cl)-CO-CH(OCH₃)₂, -CH=C(Cl)-CO-CH₂-SCH₃, -CH=C(Br)-CO-CH₃, -CH=C(Br)-CO-C₂H₅, -CH=C(Br)-CO-n-C₃H₇, -CH=C(Br)-CO-i-C₃H₇, -CH=C(Br)-CO-n-C₄H₉, -CH=C(Br)-CO-tert.-C₄H₉, -CH=C(Br)-CO-CH₂Cl, -CH=C(Br)-CO-CH₂Br, -CH=C(Br)-CO-CHCl₂, -CH=C(Br)-CO-CH₂-OCH₃, -CH=C(Br)-CO-CH(OCH₃)₂, -CH=C(Br)-CO-CH₂-SCH₃, -CH=C(CN)-CO-CH₃, -CH=C(CN)-CO-C₂H₅, -CH=C(CN)-CO-n-C₃H₇, -CH=C(CN)-CO-i-C₃H₇, -CH=C(CN)-CO-n-C₄H₉, -CH=C(CN)-CO-tert.-C₄H₉, -CH=C(CN)-CO-CH₂Cl, -CH=C(CN)-CO-CH₂Br, -CH=C(CN)-CO-CHCl₂, -CH=C(CN)-CO-CH₂-OCH₃, -CH=C(CN)-CO-CH(OCH₃)₂, -CH=C(CN)-CO-CH₂-SCH₃, -CH=CH-CO-C₆H₅, -CH=CH-CO-(4-Cl-C₆H₄), -CH=C(CH₃)-CO-C₆H₅, -CH=C(CH₃)-CO-(4-Cl-C₆H₄), -CH=C(C₂H₅)-CO-C₆H₅, -CH=C(C₂H₅)-CO-(4-Cl-C₆H₄), -CH=C(Cl)-CO-C₆H₅, -CH=C(Br)-CO-C₆H₅, -CH=C(CN)-CO-C₆H₅, -CH=CH-CO-NH₂, -CH=CH-CO-NHCH₃, -CH=CH-CO-N(CH₃)₂, -CH=CH-CO-NH-C₂H₅, -CH=CH-CO-N(C₂H₅)₂, -CH=CH-CO-NH-n-C₃H₇, -CH=CH-CO-NH-i-C₃H₇, -CH=CH-CO-NH-tert.-C₄H₉, -CH=CH-CO-NH-cyclopropyl, -CH=CH-CO-NH-cyclobutyl, -CH=CH-CO-NH-cyclopentyl, -CH=CH-CO-NH-cyclohexyl, -CH=CH-CO-NH-cycloheptyl, -CH=CH-CO-NH-cyclooctyl, -CH=CH-CO-pyrrolidin-1-yl, -CH=CH-CO-piperidin-1-yl, -CH=CH-CO-morpholin-4-yl, -CH=CH-CO-NH-CH₂CH=CH₂, -CH=CH-CO-NH-CH₂C≡CH, -CH=CH-CO-N(CH₃)-CH₂C≡CH, -CH=CH-CO-NH-(CH₂)₂Cl, -CH=CH-CO-NH-C₆H₅, -CH=C(CH₃)-CO-NH₂, -CH=C(CH₃)-CO-NHCH₃, -CH=C(CH₃)-CO-N(CH₃)₂, -CH=C(CH₃)-CO-NH-C₂H₅, -CH=C(CH₃)-CO-N(C₂H₅)₂, -CH=C(CH₃)-CO-NH-n-C₃H₇, -CH=C(CH₃)-CO-NH-i-C₃H₇, -CH=C(CH₃)-CO-NH-tert.-C₄H₉, -CH=C(CH₃)-CO-NH-cyclopropyl, -CH=C(CH₃)-CO-NH-cyclobutyl, -CH=C(CH₃)-CO-NH-cyclopentyl, -CH=C(CH₃)-CO-NH-cyclohexyl, -CH=C(CH₃)-CO-NH-cycloheptyl, -CH=C(CH₃)-CO-NH-cyclooctyl, -CH=C(CH₃)-CO-pyrrolidin-1-yl, -CH=C(CH₃)-CO-piperidin-1-yl, -CH=C(CH₃)-CO-morpholin-4-yl, -CH=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -CH=C(CH₃)-CO-NH-CH₂C≡CH, -CH=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CH₃)-CO-NH-(CH₂)₂Cl, -CH=C(CH₃)-CO-NH-C₆H₅, -CH=C(C₂H₅)-CO-NH₂, -CH=C(C₂H₅)-CO-NHCH₃, -CH=C(C₂H₅)-CO-N(CH₃)₂, -CH=C(C₂H₅)-CO-NH-C₂H₅, -CH=C(C₂H₅)-CO-N(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-n-C₃H₇, -CH=C(C₂H₅)-CO-NH-i-C₃H₇, -CH=C(C₂H₅)-CO-NH-tert.-C₄H₉, -CH=C(C₂H₅)-CO-NH-cyclopropyl, -CH=C(C₂H₅)-CO-NH-cyclobutyl, -CH=C(C₂H₅)-CO-NH-cyclopentyl, -CH=C(C₂H₅)-CO-NH-cyclohexyl, -CH=C(C₂H₅)-CO-NH-cycloheptyl, -CH=C(C₂H₅)-CO-NH-cyclooctyl, -CH=C(C₂H₅)-CO-pyrrolidin-1-yl, -CH=C(C₂H₅)-CO-piperidin-1-yl, -CH=C(C₂H₅)-CO-morpholin-4-yl, -CH=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-CH₂C≡CH -CH=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -CH=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -CH=C(C₂H₅)-CO-NH-C₆H₅, -CH=C(Cl)-CO-NH₂, -CH=C(Cl)-CO-NHCH₃, -CH=C(Cl)-CO-N(CH₃)₂, -CH=C(Cl)-CO-NH-C₂H₅, -CH=C(Cl)-CO-N(C₂H₅)₂, -CH=C(Cl)-CO-NH-n-C₃H₇, -CH=C(Cl)-CO-NH-i-C₃H₇, -CH=C(Cl)-CO-NH-tert.-C₄H₉, -CH=C(Cl)-CO-NH-cyclopropyl, -CH=C(Cl)-CO-NH-cyclobutyl, -CH=C(Cl)-CO-NH-cyclopentyl, -CH=C(Cl)-CO-NH-cyclohexyl, -CH=C(Cl)-CO-NH-cycloheptyl, -CH=C(Cl)-CO-NH-cyclooctyl, -CH=C(Cl)-CO-pyrrolidin-1-yl, -CH=C(Cl)-CO-piperidin-1-yl, -CH=C(Cl)-CO-morpholin-4-yl, -CH=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -CH=C(Cl)-CO-NH-CH₂C≡CH, -CH=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Cl)-CO-NH-(CH₂)₂Cl, -CH=C(Cl)-CO-NH-C₆H₅, -CH=C(Br)-CO-NH₂, -CH=C(Br)-CO-NHCH₃, -CH=C(Br)-CO-N(CH₃)₂, -CH=C(Br)-CO-NH-C₂H₅, -CH=C(Br)-CO-N(C₂H₅)₂, -CH=C(Br)-CO-NH-n-C₃H₇, -CH=C(Br)-CO-NH-i-C₃H₇, -CH=C(Br)-CO-NH-tert.-C₄H₉, -CH=C(Br)-CO-NH-cyclopropyl, -CH=C(Br)-CO-NH-cyclobutyl, -CH=C(Br)-CO-NH-cyclopentyl, -CH=C(Br)-CO-NH-cyclohexyl, -CH=C(Br)-CO-NH-cycloheptyl, -CH=C(Br)-CO-NH-cyclooctyl, -CH=C(Br)-CO-pyrrolidin-1-yl, -CH=C(Br)-CO-piperidin-1-yl, -CH=C(Br)-CO-morpholin-4-yl, -CH=C(Br)-CO-NH-CH₂CH=C(Br)₂, -CH=C(Br)-CO-NH-CH₂C≡CH, -CH=C(Br)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Br)-CO-NH-(CH₂)₂Cl, -CH=C(Br)-CO-NH-C₆H₅, -CH=C(CN)-CO-NH₂, -CH=C(CN)-CO-NHCH₃, -CH=C(CN)-CO-N(CH₃)₂, -CH=C(CN)-CO-NH-C₂H₅, -CH=C(CN)-CO-N(C₂H₅)₂, -CH=C(CN)-CO-NH-n-C₃H₇, -CH=C(CN)-CO-NH-i-C₃H₇, -CH=C(CN)-CO-NH-tert.-C₄H₉, -CH=C(CN)-CO-NH-cyclopropyl, -CH=C(CN)-CO-NH-cyclobutyl, -CH=C(CN)-CO-NH-cyclopentyl, -CH=C(CN)-CO-NH-cyclohexyl, -CH=C(CN)-CO-NH-cycloheptyl, -CH=C(CN)-CO-NH-cyclooctyl, -CH=C(CN)-CO-pyrrolidin-1-yl, -CH=C(CN)-CO-piperidin-1-yl, -CH=C(CN)-CO-morpholin-4-yl, -CH=C(CN)-CO-NH-CH₂CH=C(CN)₂, -CH=C(CN)-CO-NH-CH₂C≡CH, -CH=C(CN)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CN)-CO-NH-(CH₂)₂Cl, -CH=C(CN)-CO-NH-C₆H₅, -CH=CH-CO-SCH₃, -CH=CH-CO-SC₂H₅, -CH=CH-CO-S-n-C₃H₇, -CH=CH-CO-S-i-C₃H₇, -CH=CH-CO-S-n-C₄H₉, -CH=CH-CO-S-tert.-C₄H₉, -CH=C(CH₃)-CO-SCH₃, -CH=C(CH₃)-CO-SC₂H₅, -CH=C(CH₃)-CO-S-n-C₃H₇, -CH=C(CH₃)-CO-S-i-C₃H₇, -CH=C(CH₃)-CO-S-n-C₄H₉, -CH=C(CH₃)-CO-S-tert.-C₄H₉, -CH=C(C₂H₅)-CO-SCH₃, -CH=C(C₂H₅)-CO-SC₂H₅, -CH=C(C₂H₅)-CO-S-n-C₃H₇, -CH=C(C₂H₅)-CO-S-i-C₃H₇, -CH=C(C₂H₅)-CO-S-n-C₄H₉, -CH=C(C₂H₅)-CO-S-tert.-C₄H₉, -CH=C(Cl)-CO-SCH₃, -CH=C(Cl)-CO-SC₂H₅, -CH=C(Cl)-CO-S-n-C₃H₇, -CH=C(Cl)-CO-S-i-C₃H₇, -CH=C(Cl)-CO-S-n-C₄H₉, -CH=C(Cl)-CO-S-tert.-C₄H₉, -CH=C(Br)-CO-SCH₃, -CH=C(Br)-CO-SC₂H₅, -CH=C(Br)-CO-S-n-C₃H₇, -CH=C(Br)-CO-S-i-C₃H₇, -CH=C(Br)-CO-S-n-C₄H₉, -CH=C(Br)-CO-S-tert.-C₄H₉, -CH=C(CN)-CO-SCH₃, -CH=C(CN)-CO-SC₂H₅, -CH=C(CN)-CO-S-n-C₃H₇, -CH=C(CN)-CO-S-i-C₃H₇, -CH=C(CN)-CO-S-n-C₄H₉, -CH=C(CN)-CO-S-tert.-C₄H₉, -CH=C(COCH₃)-CO-OCH₃, -CH=C(COC₂H₅)-CO-OCH₃, -CH=C(CO-n-C₃H₇)-CO-OCH₃, -CH=C(COCH₃)-CO-OC₂H₅, -CH=C(COC₂H₅)-CO-OC₂H₅, -CH=C(CO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COCH₃)-CO-O-n-C₃H₇, -CH=C(COC₂H₅)-CO-O-n-C₃H₇, -CH=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-OCH₃, -CH=C(CF₃)-CO-OC₂H₅, -CH=C(CF₃)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-O-i-C₃H₇, -CH=C(CF₃)-CO-O-n-C₄H₉, -CH=C(CF₃)-CO-O-tert.-C₄H₉, -CH=C(COOCH₃)₂, -CH=C(COOC₂H₅)₂, -CH=C(COOCH₃)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)-CO-OCH₃, -CH=C(COO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)₂, -CH=CH-CH=CH-COOH, -CH=CH-CH=CH-CO-OCH₃, -CH=CH-CH=CH-CO-OC₂H₅, -CH=CH-CH=C(COOCH₃)₂, -CH=CH-CH=C(CN)-CO-OCH₃, -CH=CH-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-OCH₃, -CH=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CH=C(Cl)-CO-OCH₃, -CH=C(CH₃)-CH=C(Br)-CO-OCH₃, -CH=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-NH₂, -CH=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -CH=CH-(CH₂)₂-COOH, -CH=CH-(CH₂)₂-CO-OCH₃, -CH=CH-(CH₂)₂-CO-OC₂H₅, -CH=CH-CH₂-CH(COOCH₃)₂, -CH=CH-CH₂-CH(COOC₂H₅)₂, -CH=CH-CH₂-CH(CN)-CO-OCH₃, -CH=CH-CH₂-CH(CN)-CO-OC₂H₅, -CH=CH-CH₂-CH(CH₃)-CO-OCH₃, -CH=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -CH=CH-(CH₂)₂-CO-NH₂, -CH=CH-(CH₂)₂-CO-NH-CH₃, -CH=CH-CH₂-COOH, -CH=CH-CH₂-CO-OCH₃, -CH=CH-CH₂-CO-OC₂H₅, -CH=C(COOCH₃)-CH₂-CO-OCH₃, -CH=C(COOCH₃)-CH₂-CO-OC₂H₅, -CH=CH-CH₂-CO-NH₂, -CH=CH-CH₂-CO-NH-CH₃, -CH=CH-CH₂-CO-N(CH₃)₂, -CH(OCH₃)₂, -CH(SCH₃)₂, -CH(OC₂H₅)₂, -CH(SC₂H₅)₂, -CH(O-n-C₃H₇)₂, -CH(O-i-C₃H₇)₂, -CH(S-n-C₃H₇)₂, -CH(S-i-C₃H₇)₂, -CH(O-n-C₄H₉)₂, -CH(O-i-C₄H₉)₂, -CH(O-s-C₄H₉)₂, -CH(O-tert.-C₄H₉)₂, -CH(S-n-C₄H₉)₂, -CH(S-i-C₄H₉)₂, -CH(S-s-C₄H₉)₂, -CH(S-tert.-C₄H₉)₂, -CH(OC₅H₁₁)₂, 1,3-Dioxolan-2-yl, 1,3-Dithio­ lan-2-yl, 1,3-Oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 5-Methyl-1,3-oxathiolan-2-yl, 4-Ethyl-1,3-dioxolan-2-yl, 4-Ethyl- 1,4-dithiolan-2-yl, 4-Ethyl-1,3-oxathiolan-2-yl, 5-Ethyl-1,3-oxa­ thiolan-2-yl, 4,5-Dimethyl-1,3-dioxolan-2-yl, 4,4-Dimethyl-1,3- dioxolan-2-yl, 4,5-Dimethyl-1,3-dithiolan-2-yl, 5,5-Dimethyl-1,3- dithiolan-2-yl, 4,5-Dimethyl-1,3-oxathiolan-2-yl, 5,5-Dimethyl- 1,3-oxathiolan-2-yl, 4,4-Dimethyl-1,3-oxathiolan-2-yl, 4-Vinyl- 1,3-dioxolan-2-yl, 4-Vinyl-1,3-dithiolan-2-yl, 4-Vinyl-1,3-oxa­ thiolan-2-yl, 5-Vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3- dioxolan-2-yl, 4-Chlormethyl-1,3-dithiolan-2-yl, 4-Chlormethyl- 1,3-oxathiolan-2-yl, 5-Chlormethyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-1,3-dithio­ lan-2-yl, 4-Hydroxymethyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl- 1,3-oxathiolan-2-yl, 4-Methoxymethyl-1,3-dioxolan-2-yl, 4-Allyl­ oxymethyl-1,3-dioxolan-2-yl, 4-Propargyloxymethyl-1,3-dioxolan- 2-yl, 4-Acetoxymethyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-1,3-dithiolan-2-yl, 4-Propargyl­ oxymethyl-1,3-dithiolan-2-yl, 4-Acetoxymethyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl-1,3-oxathiolan-2-yl, 5-Allyloxy­ methyl-1,3-oxathiolan-2-yl, 4-Propargyloxymethyl-1,3-oxathiolan-2-yl, 5-Propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxymethyl- 1,3-oxathiolan-2-yl, 5-Acetoxymethyl-1,3-oxathiolan-2-yl, 4-Methylthiomethyl-1,3-dioxolan-2-yl, 4-Methylthiomethyl-1,3- dithiolan-2-yl, 4-Carboxy-1,3-dioxolan-2-yl, 4-Carboxy-1,3- dithiolan-2-yl, 4-Methoxycarbonyl-1,3-dioxolan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-4-methyl- 1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithiolan- 2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-1,3- dithiolan-2-yl, 1,3-Dioxan-2-yl, 1,3-Dithian-2-yl, 1,3-Oxathian- 2-yl, 5-Methyl-1,3-dioxan-2-yl, 5-Methyl-1,3-dithian-2-yl, 5-Methyl-1,3-oxathian-2-yl, 5,5-Dimethyl-1,3-dioxan-2-yl, 4,6-Dimethyl- 1,3-dioxan-2-yl, 4,4-Dimethyl-1,3-dioxan-2-yl, 5,5-Dimethyl- 1,3-dithian-2-yl, 4,6-Dimethyl-1,3-dithian-2-yl, 4,4-Dimethyl- 1,3-dithian-2-yl, 5,5-Dimethyl-1,3-oxathian-2-yl, 4,4-Dimethyl- 1,3-oxathian-2-yl, 6,6-Dimethyl-1,3-oxathian-2-yl, 4-Hydroxymethyl-1,3-dioxan-2-yl, 4-Methoxymethyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-1,3-dithian-2-yl, 4-Methoxymethyl-1,3-dithian-2-yl, 4-Allyloxymethyl-1,3-dithian-2-yl, 4-Acetoxymethyl- 1,3-dithian-2-yl, 4-Chlormethyl-1,3-dioxan-2-yl, 4-Chlormethyl- 1,3-dithian-2-yl, 1,3-Dioxepan-2-yl, 1,3-Dithiepan-2-yl, 1,3-Dioxep-5-en-2-yl, 4-Methoxycarbonyl-1,3-dioxan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-1,3-dithian-2-yl, 4-n-Butoxycarbonyl-1,3-dithian-2-yl, 4-Methoxycarbonyl-4- methyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-Methoxy- carbonyl-4-methyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-4-methyl- 1,3-dithian-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithian-2-yl, -C(CH₃)(OCH₃)₂, -C(CH₃)(SCH₃)₂, -C(CH₃)(OC₂H₅)₂, -C(CH₃)(SC₂H₅)₂, -C(CH₃)(O-n-C₃H₇)₂, -C(CH₃)(O-i-C₃H₇)₂, -C(CH₃)(S-n-C₃H₇)₂, -C(CH₃)(S-i-C₃H₇)₂, -C(CH₃)(O-n-C₄H₉)₂, -C(CH₃)(O-i-C₄H₉)₂, -C(CH₃)(O-s-C₄H₉)₂, -C(CH₃)(O-tert.-C₄H₉)₂, -C(CH₃)(S-n-C₄H₉)₂, -C(CH₃)(S-i-C₄H₉)₂, -C(CH₃)(S-s-C₄H₉)₂, -C(CH₃)(S-tert.-C₄H₉)₂, -C(CH₃)(O-n-C₅H₁₁)′′, 2-Methyl-1,3-dioxolan-2-yl, 2-Methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-oxathiolan-2-yl, 2,4-Dimethyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-1,3- oxathiolan-2-yl, 2,5-Dimethyl-1,3-oxathiolan-2-yl, 4-Ethyl-2- methyl-1,3-dioxolan-2-yl, 4-Ethyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Ethyl-2-methyl-1,3- oxathiolan-2-yl, 2,4,5-Trimethyl-1,3-dioxolan-2-yl, 2,4,4-Trimethyl- 1,3-dioxolan-2-yl, 2,4,5-Trimethyl-1,3-dithiolan-2-yl, 2,4,4-Trimethyl-1,3-dithiolan-2-yl, 2,4,5-Trimethyl-1,3-oxathiolan-2-yl, 2,4,4-Trimethyl-1,3-oxathiolan-2-yl, 2-Methyl-4-vinyl- 1,3-dioxolan-2-yl, 2-Methyl-4-vinyl-1,3-dithiolan-2-yl, 2-Methyl- 4-vinyl-1,3-oxathiolan-2-yl, 2-Methyl-5-vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-dioxolan-2-yl, 4-Chlormethyl-2- methyl-1,3-dithiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl- 2-methyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-2- methyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dioxolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxy- 2-methyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dithiolan-2-yl, 4-Acetoxy-2- methyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl- 2-methyl-1,3-oxathiolan-2-yl, 5-Allyloxymethyl-2- methyl-1,3-oxathiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3- oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxy-2-methyl-1,3-oxathiolan-2-yl, 5-Acetoxy-2-methyl- 1,3-oxathiolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dioxolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-2- methyl-1,3-dioxolan-2-yl, 4-Carboxy-2-methyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-2- methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl- 2-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-2- methyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-ethoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4- ethoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl- 1,3-dioxolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl-1,3- dithiolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-dioxan-2-yl, 2-Methyl-1,3-dithian-2-yl, 2-Methyl-1,3-oxathian-2-yl, 2,5- Dimethyl-1,3-dioxan-2-yl, 2,5-Dimethyl-1,3-dithian-2-yl, 2,5-Dimethyl- 1,3-oxathian-2-yl, 2,5,5-Trimethyl-1,3-dioxan-2-yl, 2,4,6- Trimethyl-1,3-dioxan-2-yl, 2,2,4-Trimethyl-1,3-dioxan-2-yl, 2,5,5-Trimethyl-1,3-dithian-2-yl, 2,4,6-Trimethyl-1,3-dithian-2-yl, 2,4,4-Trimethyl-1,3-dithian-2-yl, 2,5,5-Trimethyl-1,3-oxathian-2-yl, 2,4,4-Trimethyl-1,3-oxathian-2-yl, 2,6,6-Trimethyl- 1,3-oxathian-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-2- methyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dithian-2-yl, 4-Methoxymethyl-2- methyl-1,3-dithian-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithian-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dithian-2-yl, 4-Chlormethyl-2- methyl-1,3-dioxan-2-yl, 4-Chlormethyl-2-methyl-1,3-dithian-2-yl, -C(CH₃)=NH, -C(CH₃)=N-CH₃, -C(CH₃)=N-C₂H₅, -C(CH₃)=N-n-C₃H₇, -(CH₃)=N-i-C₃H₇, -C(CH₃)=N-n-C₄H₉, -C(CH₃)=N-CH₂CH=CH₂, -C(CH₃)=N-CH₂CH=CH₂-CH₃, -C(CH₃)=N-CH₂C≡CH, -C(CH₃)=N-CH₂C≡C-CH₃, -C(CH₃)=N-cyclopropyl, -C(CH₃)=N-cyclobutyl, -C(CH₃)=N-cyclopentyl, -C(CH₃)=N-cyclohexyl, -C(CH₃)=N-cycloheptyl, -C(CH₃)=N-CH₂-CH₂Cl, -C(CH₃)=N-CH₂Cl, -C(CH₃)=N-C₆H₅, -C(CH₃)=N-(2-F-C₆H₄), -C(CH₃)=N-(3-F-C₆H₄), -C(CH₃)=N-(4-F-C₆H₄), -C(CH₃)=N-(2-Cl-C₆H₄), -C(CH₃)=N-(3-Cl-C₆H₄), -C(CH₃)=N-(4-Cl-C₆H₄), -C(CH₃)=N-(2-CH₃-C₆H₄), -C(CH₃)=N-(3-CH₃-C₆H₄), -C(CH₃)=N-(4-CH₃-C₆H₄), -C(CH₃)=N-(2-CF₃-C₆H₄), -C(CH₃)=N-(3-CF₃-C₆H₄), -C(CH₃)=N-(4-CF₃-C₆H₄), -C(CH₃)=N-(2-OCH₃-C₆H₄), -C(CH₃)=N-(3-OCH₃-C₆H₄), -C(CH₃)=N-(4-OCH₃-C₆H₄), -C(CH₃)=N-(4-NO₂-C₆H₄), -C(CH₃)=N-(4-CN-C₆H₄), -C(CH₃)=N-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-(2,4-(CH₃)₂-C₆H₃), -C(CH₃)=N-CH₂-OCH₃, -C(CH₃)=N-CH₂-OC₂H₅, -C(CH₃)=N-CH₂CH₂-OCH₃, -C(CH₃)=N-CH₂CH₂-OC₂H₅, -C(CH₃)=N-OH, -C(CH₃)=N-OCH₃, -C(CH₃)=N-OC₂H₅, -C(CH₃)=N-O-n-C₃H₇, -C(CH₃)=N-O-i-C₃H₇, -C(CH₃)=N-O-n-C₄H₉, -C(CH₃)=N-O-i-C₄H₉, -C(CH₃)=N-O-s-C₄H₉, -C(CH₃)=N-O-tert.-C₄H₉, -C(CH₃)=N-OCH₂-CH=CH₂, -C(CH₃)=N-OCH(CH₃)-CH=CH₂, -C(CH₃)=N-OCH₂-C≡CH, -C(CH₃)=N-CH(CH₃)-C≡CH, -C(CH₃)=N-OCH₂-CH=C-CH₃, -C(CH₃)=N-OCH₂CH₂-Cl, -C(CH₃)=N-OCH₂CH₂-F, -C(CH₃)=N-OCH₂-CF₃, -C(CH₃)=N-OCH₂-CH=CHCl, -C(CH₃)=N-OCH₂-C(Cl)=CH₂, -C(CH₃)=N-OCH₂-C(Br)=CH₂, -C(CH₃)=N-OCH₂-CH=C(Cl)-CH₃, -C(CH₃)=N-O-CO-CH₃, -C(CH₃)=N-O-CO-C₂H₅, -C(CH₃)=N-OCH₂-CN, -C(CH₃)=N-OCH₂-CH=CH-CH₂-OCH₃, -C(CH₃)=N-OCH₂-CH=CH-CH₂-O-tert.-C₄H₉, -C(CH₃)=N-O-(CH₂)₃-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-(4-Cl-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-C₆H₅, -C(CH₃)=N-OCH₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(3-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-CH₂-(4-CH₃O-C₆H₄), -C(CH₃)=N-OCH₂-CH=C(CH₃)-C₆H₅, -C(CH₃)=N-O-(CH₂)₂-CH=CH-(3,4-Cl₂-C₆H₃), -C(CH₃)=N-O-(CH₂)₃-C≡C-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-OCH₃, -C(CH₃)=N-OCH₂CH₂-OCH₃, -C(CH₃)=N-OCH₂-OC₂H₅, -C(CH₃)=N-OCH(CH₃)-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=N-NH₂, -C(CH₃)=N-NH-CH₃, -C(CH₃)=N-NH-C₂H₅, -C(CH₃)=N-NH-n-C₃H₇, -C(CH₃)=N-NH-i-C₃H₇, -C(CH₃)=N-NH-n-C₄H₉, -C(CH₃)=N-NH-i-C₄H₉, -C(CH₃)=N-NH-s-C₄H₉, -C(CH₃)=N-NH-tert.-C₄H₉, -C(CH₃)=N-NH-cyclopropyl, -C(CH₃)=N-NH-cyclobutyl, -C(CH₃)=N-NH-cyclopentyl, -C(CH₃)=N-NH-cyclohexyl, -C(CH₃)=N-NH-cycloheptyl, -C(CH₃)=N-N(CH₃)₂, -C(CH₃)=N-N(C₂H₅)₂, -C(CH₃)=N-N(n-C₃H₇)₂, -C(CH₃)=N-N(i-C₃H₇)₂, -C(CH₃)=N-NH-CH₂-C=CH, -C(CH₃)=N-NH-CH₂-C≡CH, -C(CH₃)=N-N(CH₃)-CH₂-C≡CH, -C(CH₃)=N-NH-CH₂CF₃, -C(CH₃)=N-NH-CO-CH₃, -C(CH₃)=N-NH-CO-C₂H₅, -C(CH₃)=N-NH-CO-OCH₃, -C(CH₃)=N-NH-CO-OC₂H₅, -C(CH₃)=N-NH-CO-O-tert.-C₄H₉, -C(CH₃)=N-pyrrolidin-1-yl, -C(CH₃)=N-piperidin-1-yl, -C(CH₃)=N-morpholin-4-yl, -C(CH₃)=N-NH-C₆H₅, -C(CH₃)=N-NH-(4-Cl-C₆H₄), -C(CH₃)=N-NH-(4-NO₂-C₆H₄), -C(CH₃)=N-NH-(4-F-C₆H₄), -C(CH₃)=N-NH-(4-CH₃O-C₆H₄), -C(CH₃)=N-NH-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-NH-(2,4-(NO₂)₂-C₆H₃), -C(CH₃)=N-NH-CO-NH₂, -C(CH₃)=N-NH-CO-NHCH₃, -C(CH₃)=N-NH-CO-NHC₂H₅, -C(CH₃)=N-NH-CO-N(CH₃)₂, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=CH-CO-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-O-n-C₄H₉, -C(CH₃)=CH-CO-O-tert.-C₄H₉, -C(CH₃)=CH-CO-O-cyclopropyl, -C(CH₃)=CH-CO-O-cyclobutyl, -C(CH₃)=CH-CO-O-cyclopentyl, -C(CH₃)=CH-CO-O-cyclohexyl, -C(CH₃)=CH-CO-O-cycloheptyl, -C(CH₃)=C(CH₃)-COOH, -C(CH₃)=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-cyclopropyl, -C(CH₃)=C(CH₃)-CO-O-cyclobutyl, -C(CH₃)=C(CH₃)-CO-O-cyclopentyl, -C(CH₃)=C(CH₃)-CO-O-cyclohexyl, -C(CH₃)=C(CH₃)-CO-O-cycloheptyl, -C(CH₃)=C(C₂H₅)-COOH, -C(CH₃)=C(C₂H₅)-CO-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-O- cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-O-cycloheptyl, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=C(Cl)-CO-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-O-n-C₄H₉, -C(CH₃)=C(Cl)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-O-cyclopropyl, -C(CH₃)=C(Cl)-CO-O-cyclobutyl, -C(CH₃)=C(Cl)-CO-O-cyclopentyl, -C(CH₃)=C(Cl)-CO-O-cyclohexyl, -C(CH₃)=C(Cl)-CO-O-cycloheptyl, -C(CH₃)=C(Br)-COOH, -C(CH₃)=C(Br)-CO-OCH₃, -C(CH₃)=C(Br)-CO-OC₂H₅, -C(CH₃)=C(Br)-CO-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-O-n-C₄H₉, -C(CH₃)=C(Br)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-O-cyclopropyl, -C(CH₃)=C(Br)-CO-O-cyclobutyl, -C(CH₃)=C(Br)-CO-O-cyclopentyl, -C(CH₃)=C(Br)-CO-O-cyclohexyl, -C(CH₃)=C(Br)-CO-O-cycloheptyl, -C(CH₃)=C(CN)-COOH, -C(CH₃)=C(CN)-CO-OCH₃, -C(CH₃)=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CN)-CO-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-O-n-C₄H₉, -C(CH₃)=C(CN)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-O-cyclopropyl, -C(CH₃)=C(CN)-CO-O-cyclobutyl, -C(CH₃)=C(CN)-CO-O-cyclopentyl, -C(CH₃)=C(CN)-CO-O-cyclohexyl, -C(CH₃)=C(CN)-CO-O-cycloheptyl, -C(CH₃)=CH-CO-OCH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=CH-CO-O-i-C₃H₇, -C(CH₃)=CH-CO-OCH(CH₃)-OCH₃, -C(CH₃)=CH-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=CH-CO-OCH₂CH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-O-i-C₃H₇, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -(CH₃)=C(Cl)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-O-i-C₃H₇, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-O-i-C₃H₇, -C(CH₃)=C(CN)-CO-OCH(CH₃)OCH₃, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-CF₃, -C(CH₃)=CH-CO-OCH₂-CCl₃, -C(CH₃)=CH-CO-OCH₂-oxiranyl, -C(CH₃)=CH-CO-(CH₂)₃-Br,-C(CH₃)=CH-CO-OCH₂-CH=CH₂, -C(CH₃)=CH-CO-OCH₂-C≡CH, -C(CH₃)=CH-CO-OCH₂-CN, -C(CH₃)=CH-CO-OCH₂CH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CF₃, -C(CH₃)=C(CH₃)-CO-OCH₂-CCl₃, -C(CH₃)=C(CH₃)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CH₃)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(CH₃)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CH₃)-CO-OCH₂-C≡CH, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CF₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CCl₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-oxiranyl, -C(CH₃)=C(C₂H₅)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(C₂H₅)-CO-OCH₂-C≡CH, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂-CF₃, -C(CH₃)=C(Cl)-CO-OCH₂-CCl₃, -C(CH₃)=C(Cl)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Cl)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Cl)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Cl)-CO-OCH₂-C≡CH, -C(CH₃)=C(Cl)-CO-OCH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂-CF₃, -C(CH₃)=C(Br)-CO-OCH₂-CCl₃, -C(CH₃)=C(Br)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Br)-CO-O(CH₂)₃-Br, -C(CH₃)=C(Br)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Br)-CO-OCH₂-C≡CH, -C(CH₃)=C(Br)-CO-OCH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂CH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂-CF₃, -C(CH₃)=C(CN)-CO-OCH₂-CCl₃, -C(CH₃)=C(CN)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CN)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(CN)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CN)-CO-OCH₂-C≡CH, -C(CH₃)=C(CN)-CO-OCH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂CH₂-CN, -C(CH₃)=CH-CO-CH₃, -C(CH₃)=CH-CO-C₂H₅, -C(CH₃)=CH-CO-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-n-C₄H₉, -C(CH₃)=CH-CO-tert.-C₄H₉, -C(CH₃)=CH-CO-CH₂Cl, -C(CH₃)=CH-CO-CH₂Br, -C(CH₃)=CH-CO-CHCl₂, -C(CH₃)=CH-CO-CH₂-OCH₃, -C(CH₃)=CH-CO-CH(OCH₃)₂, -C(CH₃)=CH-CO-CH₂-SCH₃, -C(CH₃)=C(CH₃)-CO-CH₃, -C(CH₃)=C(CH₃)-CO-C₂H₅, -C(CH₃)=C(CH₃)-CO-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-CH₂Cl, -C(CH₃)=C(CH₃)-CO-CH₂Br, -C(CH₃)=C(CH₃)-CO-CHCl₂, -C(CH₃)=C(CH₃)-CO-CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-CH(OCH₃)₂, -C(CH₃)=C(CH₃)-CO-CH₂-SCH₃, -C(CH₃)=C(C₂H₅)-CO-CH₃, -C(CH₃)=C(C₂H₅)-CO-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-CH₂Cl, -C(CH₃)=C(C₂H₅)-CO-CH₂Br, -C(CH₃)=C(C₂H₅)-CO-CHCl₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-CH(OCH₃)₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-SCH₃, -C(CH₃)=C(Cl)-CO-CH₃, -C(CH₃)=C(Cl)-CO-C₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-n-C₄H₉, -C(CH₃)=C(Cl)-CO-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-CH₂Cl, -C(CH₃)=C(Cl)-CO-CHCl₂, -C(CH₃)=C(Cl)-CO-CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-CH(OCH₃)₂, -C(CH₃)=C(Cl)-CO-CH₂-SCH₃, -C(CH₃)=C(Br)-CO-CH₃, -C(CH₃)=C(Br)-CO-C₂H₅, -C(CH₃)=C(Br)-CO-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-n-C₄H₉, -C(CH₃)=C(Br)-CO-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-CH₂Cl, -C(CH₃)=C(Br)-CO-CH₂Br, -C(CH₃)=C(Br)-CO-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-CH(OCH₃)₂, -C(CH₃)=C(Br)-CO-CH₂-SCH₃, -C(CH₃)=C(CN)-CO-CH₃, -C(CH₃)=C(CN)-CO-C₂H₅, -C(CH₃)=C(CN)-CO-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-n-C₄H₉, -C(CH₃)=C(CN)-CO-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-CH₂Cl, -C(CH₃)=C(CN)-CO-CH₂Br, -C(CH₃)=C(CN)-CO-CHCl₂, -C(CH₃)=C(CN)-CO-CH₂-OCH₃, -C(CH₃)=C(CN)-CO-CH(OCH₃)₂, -C(CH₃)=C(CN)-CO-CH₂-SCH₃, -C(CH₃)=CH-CO-C₆H₅, -C(CH₃)=CH-CO-(4-Cl-C₆H₄), -C(CH₃)=C(CH₃)-CO-C₆H₅, -C(CH₃)=C(CH₃)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(C₂H₅)-CO-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(Cl)-CO-C₆H₅, -C(CH₃)=C(Br)-CO-C₆H₅, -C(CH₃)=C(CN)-CO-C₆H₅, -C(CH₃)=CH-CO-NH₂, -C(CH₃)=CH-CO-NHCH₃, -C(CH₃)=CH-CO-N(CH₃)₂, -C(CH₃)=CH-CO-NH-C₂H₅, -C(CH₃)=CH-CO-N(C₂H₅)₂, -C(CH₃)=CH-CO-NH-n-C₃H₇, -C(CH₃)=CH-CO-NH-i-C₃H₇, -C(CH₃)=CH-CO-NH-tert.-C₄H₉, -C(CH₃)=CH-CO-NH-cyclopropyl, -C(CH₃)=CH-CO-NH-cyclobutyl, -C(CH₃)=CH-CO-NH-cyclopentyl, -C(CH₃)=CH-CO-NH-cyclohexyl, -C(CH₃)=CH-CO-NH-cycloheptyl, -C(CH₃)=CH-CO-NH-cyclooctyl, -C(CH₃)=CH-CO-pyrrolidin-1-yl, -C(CH₃)=CH-CO-piperidin-1-yl, -C(CH₃)=CH-CO-morpholin-4-yl, -C(CH₃)=CH-CO-NH-CH₂CH=CH₂, -C(CH₃)=CH-CO-NH-CH₂C≡CH, -C(CH₃)=CH-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=CH-CO-NH-(CH₂)₂Cl, -C(CH₃)=CH-CO-NH-C₆H₅, -C(CH₃)=C(CH₃)-CO-NH₂, -C(CH₃)=C(CH₃)-CO-NHCH₃, -C(CH₃)=C(CH₃)-CO-N(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-C₂H₅, -C(CH₃)=C(CH₃)-CO-N(C₂H₅)₂, -C(CH₃)=C(CH₃)-CO-NH-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-tert.-C₄H₉, -C(CH )=C(CH₃)-CO-NH- cyclopropyl, -C(CH₃)=C(CH₃)-CO-NH-cyclobutyl, -C(CH₃)=C(CH₃)-CO-NH-cyclopentyl, -C(CH₃)=C(CH₃)-CO-NH- cyclohexyl, -C(CH₃)=C(CH₃)-CO-NH-cycloheptyl, -C(CH₃)=C(CH₃)-CO-NH-cyclooctyl, -C(CH₃)=C(CH₃)-CO- pyrrolidin-1-yl, -C(CH₃)=C(CH₃)-CO-piperidin-1-yl, -C(CH₃)=C(CH₃)-CO-morpholin-4-yl, -C(CH₃)=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CH₃)-CO-NH-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-NH₂, -C(CH₃)=C(C₂H₅)-CO-NHCH₃, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)₂, -C(CH₃)=C(C₂H₅)-CO-NH-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-N(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-tert.-C₄H₉, 99999 00070 552 001000280000000200012000285919988800040 0002004131038 00004 99880 -C(CH₃)=C(C₂H₅)-CO-NH- cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-NH-cycloheptyl, -C(CH₃)=C(C₂H₅)-CO-NH- cyclooctyl, -C(CH₃)=C(C₂H₅)-CO-pyrrolidin-1-yl, -C(CH₃)=C(C₂H₅)-CO-piperidin-1-yl, -C(CH₃)=C(C₂H₅)-CO- morpholin-4-yl, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(C₂H₅)-CO-NH-C₆H₅, -C(CH₃)=C(Cl)-CO-NH₂, -C(CH₃)=C(Cl)-CO-NHCH₃, -C(CH₃)=C(Cl)-CO-N(CH₃)₂, -C(CH₃)=C(Cl)-CO-NH-C₂H₅, -C(CH₃)=C(Cl)-CO-N(C₂H₅)₂, -C(CH₃)=C(Cl)-CO-NH-n-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-i-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-NH-cyclopropyl, -C(CH₃)=C(Cl)-CO-NH-cyclobutyl, -C(CH₃)=C(Cl)-CO-NH-cyclopentyl, -C(CH₃)=C(Cl)-CO-NH-cyclohexyl, -C(CH₃)=C(Cl)-CO-NH-cycloheptyl, -C(CH₃)=C(Cl)-CO-NH-cyclooctyl, -C(CH₃)=C(Cl)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Cl)-CO-piperidin-1- yl, -C(CH₃)=C(Cl)-CO-morpholin-4-yl, -C(CH₃)=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -C(CH₃)=C(Cl)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Cl)-CO-NH-C₆H₅, -C(CH₃)=C(Br)-CO-NH₂, -C(CH₃)=C(Br)-CO-NHCH₃, -C(CH₃)=C(Br)-CO-N(CH₃)₂, -C(CH₃)=C(Br)-CO-NH-C₂H₅, -C(CH₃)=C(Br)-CO-N(C₂H₅)₂, -C(CH₃)=C(Br)-CO-NH-n-C₃H₇, -C(CH₃)=C(Br)-CO-NH-i-C₃H₇, -C(CH₃)=C(Br)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-NH-cyclopropyl, -C(CH₃)=C(Br)-CO-NH-cyclobutyl, -C(CH₃)=C(Br)-CO-NH-cyclopentyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cycloheptyl, -C(CH₃)=C(Br)-CO-NH-cyclooctyl, -C(CH₃)=C(Br)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Br)-CO-piperidin-1-yl, -C(CH₃)=C(Br)-CO-morpholin-4-yl, -C(CH₃)=C(Br)-CO-NH-CH₂CH=C(Br)₂, -C(CH₃)=C(Br)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Br)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Br)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Br)-CO-NH-C₆H₅, -C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CN)-CO-NHCH₃, -C(CH₃)=C(CN)-CO-N(CH₃)₂, -C(CH₃)=C(CN)-CO-NH-C₂H₅, -C(CH₃)=C(CN)-CO-N(C₂H₅)₂, -C(CH₃)=C(CN)-CO-NH-n-C₃H₇, -C(CH₃)=C(CN)-CO-NH-i-C₃H₇, -C(CH₃)=C(CN)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-NH-cyclopropyl, -C(CH₃)=C(CN)-CO-NH-cyclobutyl, -C(CH₃)=C(CN)-CO-NH-cyclopentyl, -C(CH₃)=C(CN)-CO-NH-cyclohexyl, -C(CH₃)=C(CN)-CO-NH-cycloheptyl, -C(CH₃)=C(CN)-CO-NH-cyclooctyl, -C(CH₃)=C(CN)-CO-pyrrolidin-1-yl, -C(CH₃)=C(CN)-CO-piperidin-1-yl, -C(CH₃)=C(CN)-CO-morpholin-4-yl, -C(CH₃)=C(CN)-CO-NH-CH₂CH=C(CN)₂, -C(CH₃)=C(CN)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CN)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CN)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CN)-CO-NH-C₆H₅, -C(CH₃)=CH-SO-SCH₃, -C(CH₃)=CH-CO-SC₂H₅, -C(CH₃)=CH-CO-S-n-C₃H₇, -C(CH₃)=CH-CO-S-i-C₃H₇, -C(CH₃)=CH-CO-S-n-C₄H₉, -C(CH₃)=CH-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-SCH₃, -C(CH₃)=C(CH₃)-CO-SC₂H₅, -C(CH₃)=C(CH₃)-CO-S-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-S-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-SCH₃, -C(CH₃)=C(C₂H₅)-CO-SC₂H₅, -C(CH₃)=C(C₂H₅)-CO-S-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-SCH₃, -C(CH₃)=C(Cl)-CO-SC₂H₅, -C(CH₃)=C(Cl)-CO-S-n-C₃H₇, -C(CH₃)=C(Cl)-CO-S-i-C₃H₇, -C(CH₃)=C(Cl)-CO-S-n-C₄H₉, -C(CH₃)=C(Cl)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-SCH₃, -C(CH₃)=C(Br)-CO-SC₂H₅, -C(CH₃)=C(Br)-CO-S-n-C₃H₇, -C(CH₃)=C(Br)-CO-S-i-C₃H₇, -C(CH₃)=C(Br)-CO-S-n-C₄H₉, -C(CH₃)=C(Br)-CO-S-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-SCH₃, -C(CH₃)=C(CN)-CO-SC₂H₅, -C(CH₃)=C(CN)-CO-S-n-C₃H₇, -C(CH₃)=C(CN)-CO-S-i-C₃H₇, -C(CH₃)=C(CN)-CO-S-n-C₄H₉, -C(CH₃)=C(CN)-CO-S-tert.-C₄H₉, -C(CH₃)=C(COCH₃)-CO-OCH₃, -C(CH₃)=C(COC₂H₅)-CO-OCH₃, -C(CH₃)=C(CO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COCH₃)-CO-OC₂H₅, -C(CH₃)=C(COC₂H₅)-CO-OC₂H₅, -C(CH₃)=C(CO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COCH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(COC₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-OCH₃, -C(CH₃)=C(CF₃)-CO-OC₂H₅, -C(CH₃)=C(CF₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CF₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(COOCH₃)₂, -C(CH₃)=C(COOC₂H₅)₂, -C(CH₃)=C(COOCH₃)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)₂, -C(CH₃)=CH-CH=CH-COOH, -C(CH₃)=CH-CH=CH-CO-OCH₃, -C(CH₃)=CH-CH=CH-CO-OC₂H₅, -C(CH₃)=CH-CH=C(COOCH₃)₂, -C(CH₃)=CH-CH=C(CN)-CO-OCH₃, -C(CH₃)=CH-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH₂, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -C(CH₃)=CH-(CH₂)₂-COOH, -C(CH₃)=CH-(CH₂)₂-CO-OCH₃, -C(CH₃)=CH-(CH₂)₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(COOCH₃)₂, -C(CH₃)=CH-CH₂-CH(COOC₂H₅)₂, -C(CH₃)=CH-CH₂-CH(CN)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CN)-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -C(CH₃)=CH-(CH₂)₂-CO-NH₂, -C(CH₃)=CH-(CH₂)₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-COOH, -C(CH₃)=CH-CH₂-CO-OCH₃, -C(CH₃)=CH-CH₂-CO-OC₂H₅, -C(CH₃)=C(COOCH₃)-CH₂-CO-OCH₃, -C(CH₃)=C(COOCH₃)-CH₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CO-NH₂, -C(CH₃)=CH-CH₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-CO-N(CH₃)₂.
wobei W für eine der folgenden Bedeutungen steht:
-CHO, -COCH₃, -COC₂H₅, -CO-n-C₃H₇, -CO-i-C₃H₇, -CO-n-C₄H₉, -CO-i-C₄H₉, -CO-s-C₄H₉, -CO-tert.-C₄H₉, -CO-CH₂CH=CH₂, -CO-CF₃, -COCCl₃, -COCH₂C≡CH, -CO-cyclopropyl, -CO-cyclobutyl, -CO-cyclopentyl, -CO-cyclohexyl, -CO-CN, -CO-COOCH₃, -CO-COOC₂H₅, -CH=NH, -CH=NCH₃, -CH=NC₂H₅, -CH=N-n-C₃H₅, -CH=N-i-C₃H₅, -CH=N-n-C₄H₉, -CH=NCH₂CH=CH₂, -CH=NCH₂CH=CH₂-CH₃, -CH=NCH₂C≡CH, -CH=NCH₂C≡C-CH₃, -CH=N-cyclopropyl, -CH=N-cyclobutyl, -CH=N-cyclopentyl, -CH=N-cyclohexyl, -CH=N-cycloheptyl, -CH=N-CH₂-CH₂Cl, -CH=N-CH₂Cl, -CH=N-C₆H₅, -CH=N-4-Br-C₆H₄, -CH=N-3-F-C₆H₄, -CH=N-4-F-C₆H₄, -CH=N-2-Cl-C₆H₄, -CH=N-3-Cl-C₆H₄, -CH=N-4-Cl-C₆H₄, -CH=N-2-Br-C₆H₄, -CH=N-2-F-C₆H₄, -CH=N-2-CH₃-C₆H₄, -CH=N-3-CH₃-C₆H₄, -CH=N-4-CH₃-C₆H₄, -CH=N-2-CF₃-C₆H₄, -CH=N-3-CF₃-C₆H₄, -CH=N-4-CF₃-C₆H₄, -CH=N-2-OCH₃-C₆H₄, -CH=N-3-OCH₃-C₆H₄, -CH=N-4-OCH₃-C₆H₄, -CH=N-4-NO₂-C₆H₄, -CH=N-4-CN-C₆H₄, -CH=N-2,4-(Cl,Cl)-C₆H₄, -CH=N-2,4-(CH₃,CH₃)-C₆H₄, -CH=N-CH₂OCH₃ -CH=N-CH₂OC₂H₅, -CH=N-CH₂CH₂OCH₃, -CH=N-CH₂CH₂OC₂H₅, -CH=N-OH, -CH=N-OCH₃, -CH=N-OC₂H₅, -CH=N-O-n-C₃H₇, -CH=N-O-i-C₃H₇, -CH=N-O-n-C₄H₉, -CH=N-O-i-C₄H₉, -CH=N-O-s-C₄H₉, -CH=N-O-tert.-C₄H₉, -CH=N-O-CH₂CH=CH₂, -CH=N-O-CH(CH₃)CH=CH₂, -CH=N-O-CH₂C≡CH, -CH=N-O-CH(CH₃)-C≡CH, -CH=N-O-CH₂-CH=CH-CH₃, -CH=N-O-CH₂-CH₂-Cl, -CH=N-O-CH₂-CH₂-F, -CH=N-O-CH₂-CF₃, -CH=N-O-CH₂-CH=CHCl, -CH=N-O-CH₂-CCl=CH₂, -CH=N-O-CH₂-CBr=CH₂, -CH=N-O-CH₂-CH=CCl-CH₃, -CH=N-OC(O)CH₃, -CH=N-OC(O)C₂H₅, -CH=N-O-CH₂-CN, -CH=N-O-CH₂-CH=CH-CH₂-O-CH₃, -CH=N-O-CH₂-CH=CH-CH₂-O-tert.-C₄H₉, -CH=N-O-(CH₂)₃-C₆H₅, -CH=N-O-(CH₂)₄-C₆H₅, -CH=N-O-(CH₂)₄-4-Cl-C₆H₄, -CH=N-O-(CH₂)₄-4-OCH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-CH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-C₆H₅, -CH=N-O-CH₂CH=CH-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CH-3-OCH₃-C₆H₄, -CH=N-O-(CH₂)₂CH=CH-4-F-C₆H₄, -CH=N-O-(CH₂)CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CHCH₂-4-OCH₃-C₆H₄, -CH=N-O-CH₂-CH=C(CH₃)-C₆H₅ -CH=N-O-(CH₂)₂CH=CH-3,4(Cl,Cl)-C₆H₃, -CH=N-O-(CH₂)₃C≡C-4-F-C₆H₄, -CH₂=N-OCHOCH₃, -CH=N-OC₂H₄OCH₃, -CH=N-OCH₂OC₂H₅, -CH=N-OCH(CH₃)OCH₃, -CH=N-OCH(CH₃)COOCH₃, -CH=N-OCH(CH₃)COO-n-C₄H₉, -CH=N-NH₂, -CH=N-NHCH₃, -CH=N-NHC₂H₅, -CH=N-NH-n-C₃H₇, -CH=N-NH-i-C₃H₇, -CH=N-NH-n-C₄H₉, -CH=N-NH-i-C₄H₉, -CH=N-NH-s-C₄H₉, -CH=N-NH-tert.-C₄H₉, -CH=N-NH-cyclopropyl, -CH=N-NH-cyclobutyl, -CH=N-NH-cyclopentyl, -CH=N-NH-cyclohexyl, -CH=N-NH-cycloheptyl, -CH=N-N(CH₃)₂, -CH=N-N(C₂H₅)₂, -CH=N-N(C₃H₇)₂, -CH=N-N(i-C₃H₇)(CH₃), -CH=N-NHCH₂-C=CH, -CH=N-NHCH₂-C≡CH, -CH=N-N(CH₃)-CH₂-C≡CH, -CH=N-NHCH₂CF₃, -CH=N-NH-CO-CH₃, -CH=N-NH-CO-CH₂H₅, -CH=N-NH-COOCH₃, -CH=N-NH-COOC₂H₅, -CH=N-NH-COO-tert.-C₄H₉, -CH=N-pyrrolidin-1-yl, -CH=N-piperidin-1-yl, -CH=N-morpholin-4-yl, -CH=N-NH-C₆H₅, -CH=N-NH-(4-Cl-C₆H₄), -CH=N-NH-(4-NO₂-C₆H₄), -CH=N-NH-(4-F-C₆H₄), -CH=N-NH-(4-CH₃O-C₆H₄), -CH=N-NH-(2,4-Cl₂-C₆H₃), -CH=N-NH-(2,4-(NO₂)₂-C₆H₃), -CH=N-NH-CO-NH₂, -CH=N-NH-CO-NHCH₃, -CH=N-NH-CO-NHC₂H₅, -CH=N-NH-CO-N(CH₃)₂, -CH=CH-COOH, -CH=CH-CO-OCH₃, -CH=CH-CO-OC₂H₅, -CH=CH-CO-O-n-C₃H₇, -CH=CH-CO-O-i-C₃H₇, -CH=CH-CO-O-n-C₄H₉, -CH=CH-CO-O-tert.-C₄H₉, -CH=CH-CO-O-cyclopropyl, -CH=CH-CO-O-cyclobutyl, -CH=CH-CO-O-cyclopentyl, -CH=CH-CO-O-cyclohexyl, -CH=CH-CO-O-cycloheptyl, -CH=C(CH₃)-COOH, -CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CO-O-n-C₃H₇, -CH=C(CH₃)-CO-O-i-C₃H₇, -CH=C(CH₃)-CO-O-n-C₄H₉, -CH=C(CH₃)-CO-O-tert.-C₄H₉, -CH=C(CH₃)-CO-O-cyclopropyl, -CH=C(CH₃)-CO-O-cyclobutyl, -CH=C(CH₃)-CO-O-cyclopentyl, -CH=C(CH₃)-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cycloheptyl, -CH=C(C₂H₅)-COOH, -CH=C(C₂H₅)-CO-OCH₃, -CH=C(C₂H₅)-CO-OC₂H₅, -CH=C(C₂H₅)-CO-O-n-C₃H₇, -CH=C(C₂H₅)-CO-O-i-C₃H₇, -CH=C(C₂H₅)-CO-O-n-C₄H₉, -CH=C(C₂H₅)-CO-O-tert.-C₄H₉, -CH=C(C₂H₅)-CO-O-cyclopropyl, -CH=C(C₂H₅)-CO-O-cyclobutyl, -CH=C(C₂H₅)-CO-O-cyclopentyl, -CH=C(C₂H₅)-CO-O-cyclohexyl, -CH=C(C₂H₅)-CO-O-cycloheptyl, -CH=C(Cl)-COOH, -CH=C(Cl)-CO-OCH₃, -CH=C(Cl)-CO-OC₂H₅, -CH=C(Cl)-CO-O-n-C₃H₇, -CH=C(Cl)-CO-O-i-C₃H₇, -CH=C(Cl)-CO-O-n-C₄H₉, -CH=C(Cl)-CO-O-tert.-C₄H₉, -CH=C(Cl)-CO-O-cyclopropyl, -CH=C(Cl)-CO-O-cyclobutyl, -CH=C(Cl)-CO-O-cyclopentyl, -CH=C(Cl)-CO-O-cyclohexyl, -CH=C(Cl)-CO-O-cycloheptyl, -CH=C(Br)-COOH, -CH=C(Br)-CO-OCH₃, -CH=C(Br)-CO-OC₂H₅, -CH=C(Br)-CO-O-n-C₃H₇, -CH=C(Br)-CO-O-i-C₃H₇, -CH=C(Br)-CO-O-n-C₄H₉, -CH=C(Br)-CO-O-tert.-C₄H₉, -CH=C(Br)-CO-O-cyclopropyl, -CH=C(Br)-CO-O-cyclobutyl, -CH=C(Br)-CO-O-cyclopentyl, -CH=C(Br)-CO-O-cyclohexyl, -CH=C(Br)-CO-O-cycloheptyl, -CH=C(CN)-COOH, -CH=C(CN)-CO-OCH₃, -CH=C(CN)-CO-OC₂H₅, -CH=C(CN)-CO-O-n-C₃H₇, -CH=C(CN)-CO-O-i-C₃H₇, -CH=C(CN)-CO-O-n-C₄H₉, -CH=C(CN)-CO-O-tert.-C₄H₉, -CH=C(CN)-CO-O-cyclopropyl, -CH=C(CN)-CO-O-cyclobutyl, -CH=C(CN)-CO-O-cyclopentyl, -CH=C(CN)-CO-O-cyclohexyl, -CH=C(CN)-CO-O-cycloheptyl, -CH=CH-CO-OCH₂-OCH₃, -CH=CH-CO-OCH₂-OC₂H₅, -CH=CH-CO-OCH₂-O-n-C₃H₅, -CH=CH-CO-OCH₂-O-i-C₃H₅, -CH=CH-CO-OCH(CH₃)-OCH₃, -CH=CH-CO-OCH(CH₃)-OC₂H₅, -CH=CH-CO-O-CH₂CH₂-OCH₃, -CH=CH-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-OCH₃, -CH=C(CH₃)-CO-OCH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-O-n-C₃H₅, -CH=C(CH₃)-CO-OCH₂-O-i-C₃H₅, -CH=C(CH₃)-CO-OCH(CH₃)-OCH₃, -CH=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OCH₃, -CH=C(CH₃)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-OCH₃, -CH=C(C₂H₅)-CO-OCH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-O-n-C₃H₅, -CH=C(C₂H₅)-CO-OCH₂-O-i-C₃H₅, -CH=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -CH=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OCH₃, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-OCH₃, -CH=C(Cl)-CO-OCH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-O-n-C₃H₅, -CH=C(Cl)-CO-OCH₂-O-i-C₃H₅, -CH=C(Cl)-CO-OCH(CH₃)-OCH₃, -CH=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Cl)-CO-O-CH₂CH₂-OCH₃, -CH=C(Cl)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-OCH₃, -CH=C(Br)-CO-OCH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-O-n-C₃H₅, -CH=C(Br)-CO-OCH₂-O-i-C₃H₅, -CH=C(Br)-CO-OCH(CH₃)-OCH₃, -CH=C(Br)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Br)-CO-O-CH₂CH₂-OCH₃, -CH=C(Br)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-OCH₃, -CH=C(CN)-CO-OCH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-O-n-C₃H₅, -CH=C(CN)-CO-OCH₂-O-i-C₃H₅, -CH=C(CN)-CO-OCH(CH₃)-OCH₃, -CH=C(CN)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CN)-CO-O-CH₂CH₂-OCH₃, -CH=C(CN)-CO-O-CH₂CH₂-OC₂H₅, -CH=CH-CO-OCH₂-CF₃, -CH=CH-CO-OCH₂-CCl₃, -CH=CH-CO-OCH₂-oxiranyl, -CH=CH-CO-O(CH₂)₃-Br, -CH=CH-CO-OCH₂-CH=CH₂, -CH=CH-CO-OCH₂-C≡CH, -CH=CH-CO-OCH₂-CN, -CH=CH-CO-O(CH₂)₂-CN, -CH=C(CH₃)-CO-OCH₂-CF₃, -CH=C(CH₃)-CO-OCH₂-CCl₃, -CH=C(CH₃)-CO-OCH₂-oxiranyl, -CH=C(CH₃)-CO-O(CH₂)₃-Br, -CH=C(CH₃)-CO-OCH₂-CH=CH₂, -CH=C(CH₃)-CO-OCH₂-C≡CH, -CH=C(CH₃)-CO-OCH₂-CN, -CH=C(CH₃)-CO-O(CH₂)₂-CN, -CH=C(C₂H₅)-CO-OCH₂-CF₃, -CH=C(C₂H₅)-CO-OCH₂-CCl₃, -CH=C(C₂H₅)-CO-OCH₂-oxiranyl, -CH=C(C₂H₅)-CO-O(CH₂)₃-Br, -CH=C(C₂H₅)-CO-OCH₂-CH=CH₂, -CH=C(C₂H₅)-CO-OCH₂-C≡CH, -CH=C(C₂H₅)-CO-OCH₂-CN, -CH=C(C₂H₅)-CO-O(CH₂)₂-CN, -CH=C(Cl)-CO-OCH₂-CF₃, -CH=C(Cl)-CO-OCH₂-CCl₃, -CH=C(Cl)-CO-OCH₂-oxiranyl, -CH=C(Cl)-CO-O(CH₂)₃-Br, -CH=C(Cl)-CO-OCH₂-CH=CH₂, -CH=C(Cl)-CO-OCH₂-C≡CH, -CH=C(Cl)-CO-OCH₂-CN, -CH=C(Cl)-CO-O(CH₂)₂-CN, -CH=C(Br)-CO-OCH₂-CF₃, -CH=C(Br)-CO-OCH₂-CCl₃, -CH=C(Br)-CO-OCH₂-oxiranyl, -CH=C(Br)-CO-O(CH₂)₃-Br, -CH=C(Br)-CO-OCH₂-CH=CH₂, -CH=C(Br)-CO-OCH₂-C≡CH, -CH=C(Br)-CO-OCH₂-CN, -CH=C(Br)-CO-O(CH₂)₂-CN, -CH=C(CN)-CO-OCH₂-CF₃, -CH=C(CN)-CO-OCH₂-CCl₃, -CH=C(CN)-CO-OCH₂-oxiranyl -CH=C(CN)-CO-O(CH₂)₃-Br, -CH=C(CN)-CO-OCH₂-CH=CH₂, -CH=C(CN)-CO-OCH₂-C≡CH, -CH=C(CN)-CO-OCH₂-CN, -CH=C(CN)-CO-O(CH₂)₂-CN, -CH=CH-CO-CH₃, -CH=CH-CO-C₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-i-C₃H₇, -CH=CH-CO-n-C₄H₉, -CH=CH-CO-tert.-C₄H₉, -CH=CH-CO-CH₂Cl, -CH=CH-CO-CH₂Br, -CH=CH-CO-CHCl₂, -CH=CH-CO-CH₂-OCH₃, -CH=CH-CO-CH(OCH₃)₂, -CH=CH-CO-CH₂-SCH₃, -CH=C(CH₃)-CO-CH₃, -CH=C(CH₃)-CO-C₂H₅, -CH=C(CH₃)-CO-n-C₃H₇, -CH=C(CH₃)-CO-i-C₃H₇, -CH=C(CH₃)-CO-n-C₄H₉, -CH=C(CH₃)-CO-tert.-C₄H₉, -CH=C(CH₃)-CO-CH₂Cl, -CH=C(CH₃)-CO-CH₂Br, -CH=C(CH₃)-CO-CHCl₂, -CH=C(CH₃)-CO-CH₂-OCH₃, -CH=C(CH₃)-CO-CH(OCH₃)₂, -CH=C(CH₃)-CO-CH₂-SCH₃, -CH=C(C₂H₅)-CO-CH₃, -CH=C(C₂H₅)-CO-C₂H₅, -CH=C(C₂H₅)-CO-n-C₃H₇, -CH=C(C₂H₅)-CO-i-C₃H₇, -CH=C(C₂H₅)-CO-n-C₄H₉, -CH=C(C₂H₅)-CO-tert.-C₄H₉, -CH=C(C₂H₅)-CO-CH₂Cl, -CH=C(C₂H₅)-CO-CH₂Br, -CH=C(C₂H₅)-CO-CHCl₂, -CH=C(C₂H₅)-CO-CH₂-OCH₃, -CH=C(C₂H₅)-CO-CH(OCH₃)₂, -CH=C(C₂H₅)-CO-CH₂-SCH₃, -CH=C(Cl)-CO-CH₃, -CH=C(Cl)-CO-C₂H₅, -CH=C(Cl)-CO-n-C₃H₇, -CH=C(Cl)-CO-i-C₃H₇, -CH=C(Cl)-CO-n-C₄H₉, -CH=C(Cl)-CO-tert.-C₄H₉, -CH=C(Cl)-CO-CH₂Cl, -CH=C(Cl)-CO-CH₂Br, -CH=C(Cl)-CO-CHCl₂, -CH=C(Cl)-CO-CH₂-OCH₃, -CH=C(Cl)-CO-CH(OCH₃)₂, -CH=C(Cl)-CO-CH₂-SCH₃, -CH=C(Br)-CO-CH₃, -CH=C(Br)-CO-C₂H₅, -CH=C(Br)-CO-n-C₃H₇, -CH=C(Br)-CO-i-C₃H₇, -CH=C(Br)-CO-n-C₄H₉, -CH=C(Br)-CO-tert.-C₄H₉, -CH=C(Br)-CO-CH₂Cl, -CH=C(Br)-CO-CH₂Br, -CH=C(Br)-CO-CHCl₂, -CH=C(Br)-CO-CH₂-OCH₃, -CH=C(Br)-CO-CH(OCH₃)₂, -CH=C(Br)-CO-CH₂-SCH₃, -CH=C(CN)-CO-CH₃, -CH=C(CN)-CO-C₂H₅, -CH=C(CN)-CO-n-C₃H₇, -CH=C(CN)-CO-i-C₃H₇, -CH=C(CN)-CO-n-C₄H₉, -CH=C(CN)-CO-tert.-C₄H₉, -CH=C(CN)-CO-CH₂Cl, -CH=C(CN)-CO-CH₂Br, -CH=C(CN)-CO-CHCl₂, -CH=C(CN)-CO-CH₂-OCH₃, -CH=C(CN)-CO-CH(OCH₃)₂, -CH=C(CN)-CO-CH₂-SCH₃, -CH=CH-CO-C₆H₅, -CH=CH-CO-(4-Cl-C₆H₄), -CH=C(CH₃)-CO-C₆H₅, -CH=C(CH₃)-CO-(4-Cl-C₆H₄), -CH=C(C₂H₅)-CO-C₆H₅, -CH=C(C₂H₅)-CO-(4-Cl-C₆H₄), -CH=C(Cl)-CO-C₆H₅, -CH=C(Br)-CO-C₆H₅, -CH=C(CN)-CO-C₆H₅, -CH=CH-CO-NH₂, -CH=CH-CO-NHCH₃, -CH=CH-CO-N(CH₃)₂, -CH=CH-CO-NH-C₂H₅, -CH=CH-CO-N(C₂H₅)₂, -CH=CH-CO-NH-n-C₃H₇, -CH=CH-CO-NH-i-C₃H₇, -CH=CH-CO-NH-tert.-C₄H₉, -CH=CH-CO-NH-cyclopropyl, -CH=CH-CO-NH-cyclobutyl, -CH=CH-CO-NH-cyclopentyl, -CH=CH-CO-NH-cyclohexyl, -CH=CH-CO-NH-cycloheptyl, -CH=CH-CO-NH-cyclooctyl, -CH=CH-CO-pyrrolidin-1-yl, -CH=CH-CO-piperidin-1-yl, -CH=CH-CO-morpholin-4-yl, -CH=CH-CO-NH-CH₂CH=CH₂, -CH=CH-CO-NH-CH₂C≡CH, -CH=CH-CO-N(CH₃)-CH₂C≡CH, -CH=CH-CO-NH-(CH₂)₂Cl, -CH=CH-CO-NH-C₆H₅, -CH=C(CH₃)-CO-NH₂, -CH=C(CH₃)-CO-NHCH₃, -CH=C(CH₃)-CO-N(CH₃)₂, -CH=C(CH₃)-CO-NH-C₂H₅, -CH=C(CH₃)-CO-N(C₂H₅)₂, -CH=C(CH₃)-CO-NH-n-C₃H₇, -CH=C(CH₃)-CO-NH-i-C₃H₇, -CH=C(CH₃)-CO-NH-tert.-C₄H₉, -CH=C(CH₃)-CO-NH-cyclopropyl, -CH=C(CH₃)-CO-NH-cyclobutyl, -CH=C(CH₃)-CO-NH-cyclopentyl, -CH=C(CH₃)-CO-NH-cyclohexyl, -CH=C(CH₃)-CO-NH-cycloheptyl, -CH=C(CH₃)-CO-NH-cyclooctyl, -CH=C(CH₃)-CO-pyrrolidin-1-yl, -CH=C(CH₃)-CO-piperidin-1-yl, -CH=C(CH₃)-CO-morpholin-4-yl, -CH=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -CH=C(CH₃)-CO-NH-CH₂C≡CH, -CH=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CH₃)-CO-NH-(CH₂)₂Cl, -CH=C(CH₃)-CO-NH-C₆H₅, -CH=C(C₂H₅)-CO-NH₂, -CH=C(C₂H₅)-CO-NHCH₃, -CH=C(C₂H₅)-CO-N(CH₃)₂, -CH=C(C₂H₅)-CO-NH-C₂H₅, -CH=C(C₂H₅)-CO-N(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-n-C₃H₇, -CH=C(C₂H₅)-CO-NH-i-C₃H₇, -CH=C(C₂H₅)-CO-NH-tert.-C₄H₉, -CH=C(C₂H₅)-CO-NH-cyclopropyl, -CH=C(C₂H₅)-CO-NH-cyclobutyl, -CH=C(C₂H₅)-CO-NH-cyclopentyl, -CH=C(C₂H₅)-CO-NH-cyclohexyl, -CH=C(C₂H₅)-CO-NH-cycloheptyl, -CH=C(C₂H₅)-CO-NH-cyclooctyl, -CH=C(C₂H₅)-CO-pyrrolidin-1-yl, -CH=C(C₂H₅)-CO-piperidin-1-yl, -CH=C(C₂H₅)-CO-morpholin-4-yl, -CH=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-CH₂C≡CH, -CH=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -CH=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -CH=C(C₂H₅)-CO-NH-C₆H₅, -CH=C(Cl)-CO-NH₂, -CH=C(Cl)-CO-NHCH₃, -CH=C(Cl)-CO-N(CH₃)₂, -CH=C(Cl)-CO-NH-C₂H₅, -CH=C(Cl)-CO-N(C₂H₅)₂, -CH=C(Cl)-CO-NH-n-C₃H₇, -CH=C(Cl)-CO-NH-i-C₃H₇, -CH=C(Cl)-CO-NH-tert.-C₄H₉, -CH=C(Cl)-CO-NH-cyclopropyl, -CH=C(Cl)-CO-NH-cyclobutyl, -CH=C(Cl)-CO-NH-cyclopentyl, -CH=C(Cl)-CO-NH-cyclohexyl, -CH=C(Cl)-CO-NH-cycloheptyl, -CH=C(Cl)-CO-NH-cyclooctyl, -CH=C(Cl)-CO-pyrrolidin-1-yl, -CH=C(Cl)-CO-piperidin-1-yl, -CH=C(Cl)-CO-morpholin-4-yl, -CH=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -CH=C(Cl)-CO-NH-CH₂C≡CH, -CH=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Cl)-CO-NH-(CH₂)₂Cl, -CH=C(Cl)-CO-NH-C₆H₅, -CH=C(Br)-CO-NH₂, -CH=C(Br)-CO-NHCH₃, -CH=C(Br)-CO-N(CH₃)₂, -CH=C(Br)-CO-NH-C₂H₅, -CH=C(Br)-CO-N(C₂H₅)₂, -CH=C(Br)-CO-NH-n-C₃H₇, -CH=C(Br)-CO-NH-i-C₃H₇, -CH=C(Br)-CO-NH-tert.-C₄H₉, -CH=C(Br)-CO-NH-cyclopropyl, -CH=C(Br)-CO-NH-cyclobutyl, -CH=C(Br)-CO-NH-cyclopentyl, -CH=C(Br)-CO-NH-cyclohexyl, -CH=C(Br)-CO-NH-cycloheptyl, -CH=C(Br)-CO-NH-cyclooctyl, -CH=C(Br)-CO-pyrrolidin-1-yl, -CH=C(Br)-CO-piperidin-1-yl, -CH=C(Br)-CO-morpholin-4-yl, -CH=C(Br)-CO-NH-CH₂CH=C(Br)₂, -CH=C(Br)-CO-NH-CH₂C≡CH, -CH=C(Br)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Br)-CO-NH-(CH₂)₂Cl, -CH=C(Br)-CO-NH-C₆H₅, -CH=C(CN)-CO-NH₂, -CH=C(CN)-CO-NHCH₃, -CH=C(CN)-CO-N(CH₃)₂, -CH=C(CN)-CO-NH-C₂H₅, -CH=C(CN)-CO-N(C₂H₅)₂, -CH=C(CN)-CO-NH-n-C₃H₇, -CH=C(CN)-CO-NH-i-C₃H₇, -CH=C(CN)-CO-NH-tert.-C₄H₉, -CH=C(CN)-CO-NH-cyclopropyl, -CH=C(CN)-CO-NH-cyclobutyl, -CH=C(CN)-CO-NH-cyclopentyl, -CH=C(CN)-CO-NH-cyclohexyl, -CH=C(CN)-CO-NH-cycloheptyl, -CH=C(CN)-CO-NH-cyclooctyl, -CH=C(CN)-CO-pyrrolidin-1-yl, -CH=C(CN)-CO-piperidin-1-yl, -CH=C(CN)-CO-morpholin-4-yl, -CH=C(CN)-CO-NH-CH₂CH=C(CN)₂, -CH=C(CN)-CO-NH-CH₂C≡CH, -CH=C(CN)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CN)-CO-NH-(CH₂)₂Cl, -CH=C(CN)-CO-NH-C₆H₅, -CH=CH-CO-SCH₃, -CH=CH-CO-SC₂H₅, -CH=CH-CO-S-n-C₃H₇, -CH=CH-CO-S-i-C₃H₇, -CH=CH-CO-S-n-C₄H₉, -CH=CH-CO-S-tert.-C₄H₉, -CH=C(CH₃)-CO-SCH₃, -CH=C(CH₃)-CO-SC₂H₅, -CH=C(CH₃)-CO-S-n-C₃H₇, -CH=C(CH₃)-CO-S-i-C₃H₇, -CH=C(CH₃)-CO-S-n-C₄H₉, -CH=C(CH₃)-CO-S-tert.-C₄H₉, -CH=C(C₂H₅)-CO-SCH₃, -CH=C(C₂H₅)-CO-SC₂H₅, -CH=C(C₂H₅)-CO-S-n-C₃H₇, -CH=C(C₂H₅)-CO-S-i-C₃H₇, -CH=C(C₂H₅)-CO-S-n-C₄H₉, -CH=C(C₂H₅)-CO-S-tert.-C₄H₉, -CH=C(Cl)-CO-SCH₃, -CH=C(Cl)-CO-SC₂H₅, -CH=C(Cl)-CO-S-n-C₃H₇, -CH=C(Cl)-CO-S-i-C₃H₇, -CH=C(Cl)-CO-S-n-C₄H₉, -CH=C(Cl)-CO-S-tert.-C₄H₉, -CH=C(Br)-CO-SCH₃, -CH=C(Br)-CO-SC₂H₅, -CH=C(Br)-CO-S-n-C₃H₇, -CH=C(Br)-CO-S-i-C₃H₇, -CH=C(Br)-CO-S-n-C₄H₉, -CH=C(Br)-CO-S-tert.-C₄H₉, -CH=C(CN)-CO-SCH₃, -CH=C(CN)-CO-SC₂H₅, -CH=C(CN)-CO-S-n-C₃H₇, -CH=C(CN)-CO-S-i-C₃H₇, -CH=C(CN)-CO-S-n-C₄H₉, -CH=C(CN)-CO-S-tert.-C₄H₉, -CH=C(COCH₃)-CO-OCH₃, -CH=C(COC₂H₅)-CO-OCH₃, -CH=C(CO-n-C₃H₇)-CO-OCH₃, -CH=C(COCH₃)-CO-OC₂H₅, -CH=C(COC₂H₅)-CO-OC₂H₅, -CH=C(CO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COCH₃)-CO-O-n-C₃H₇, -CH=C(COC₂H₅)-CO-O-n-C₃H₇, -CH=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-OCH₃, -CH=C(CF₃)-CO-OC₂H₅, -CH=C(CF₃)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-O-i-C₃H₇, -CH=C(CF₃)-CO-O-n-C₄H₉, -CH=C(CF₃)-CO-O-tert.-C₄H₉, -CH=C(COOCH₃)₂, -CH=C(COOC₂H₅)₂, -CH=C(COOCH₃)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)-CO-OCH₃, -CH=C(COO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)₂, -CH=CH-CH=CH-COOH, -CH=CH-CH=CH-CO-OCH₃, -CH=CH-CH=CH-CO-OC₂H₅, -CH=CH-CH=C(COOCH₃)₂, -CH=CH-CH=C(CN)-CO-OCH₃, -CH=CH-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-OCH₃, -CH=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CH=C(Cl)-CO-OCH₃, -CH=C(CH₃)-CH=C(Br)-CO-OCH₃, -CH=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-NH₂, -CH=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -CH=CH-(CH₂)₂-COOH, -CH=CH-(CH₂)₂-CO-OCH₃, -CH=CH-(CH₂)₂-CO-OC₂H₅, -CH=CH-CH₂-CH(COOCH₃)₂, -CH=CH-CH₂-CH(COOC₂H₅)₂, -CH=CH-CH₂-CH(CN)-CO-OCH₃, -CH=CH-CH₂-CH(CN)-CO-OC₂H₅, -CH=CH-CH₂-CH(CH₃)-CO-OCH₃, -CH=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -CH=CH-(CH₂)₂-CO-NH₂, -CH=CH-(CH₂)₂-CO-NH-CH₃, -CH=CH-CH₂-COOH, -CH=CH-CH₂-CO-OCH₃, -CH=CH-CH₂-CO-OC₂H₅, -CH=C(COOCH₃)-CH₂-CO-OCH₃, -CH=C(COOCH₃)-CH₂-CO-OC₂H₅, -CH=CH-CH₂-CO-NH₂, -CH=CH-CH₂-CO-NH-CH₃, -CH=CH-CH₂-CO-N(CH₃)₂, -CH(OCH₃)₂, -CH(SCH₃)₂, -CH(OC₂H₅)₂, -CH(SC₂H₅)₂, -CH(O-n-C₃H₇)₂, -CH(O-i-C₃H₇)₂, -CH(S-n-C₃H₇)₂, -CH(S-i-C₃H₇)₂, -CH(O-n-C₄H₉)₂, -CH(O-i-C₄H₉)₂, -CH(O-s-C₄H₉)₂, -CH(O-tert.-C₄H₉)₂, -CH(S-n-C₄H₉)₂, -CH(S-i-C₄H₉)₂, -CH(S-s-C₄H₉)₂, -CH(S-tert.-C₄H₉)₂, -CH(OC₅H₁₁)₂, 1,3-Dioxolan-2-yl, 1,3-Dithiolan- 2-yl, 1,3-Oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 5-Methyl-1,3-oxathiolan-2-yl, 4-Ethyl-1,3-dioxolan-2-yl, 4-Ethyl- 1,4-dithiolan-2-yl, 4-Ethyl-1,3-oxathiolan-2-yl, 5-Ethyl-1,3-oxathiolan- 2-yl, 4,5-Dimethyl-1,3-dioxolan-2-yl, 4,4-Dimethyl-1,3- dioxolan-2-yl, 4,5-Dimethyl-1,3-dithiolan-2-yl, 5,5-Dimethyl-1,3- dithiolan-2-yl, 4,5-Dimethyl-1,3-oxathiolan-2-yl, 5,5-Dimethyl- 1,3-oxathiolan-2-yl, 4,4-Dimethyl-1,3-oxathiolan-2-yl, 4-Vinyl- 1,3-dioxolan-2-yl, 4-Vinyl-1,3-dithiolan-2-yl, 4-Vinyl-1,3-oxathiolan- 2-yl, 5-Vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3- dioxolan-2-yl, 4-Chlormethyl-1,3-dithiolan-2-yl, 4-Chlormethyl- 1,3-oxathiolan-2-yl, 5-Chlormethyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-1,3-dithiolan- 2-yl, 4-Hydroxymethyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl- 1,3-oxathiolan-2-yl, 4-Methoxymethyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl- 1,3-dioxolan-2-yl, 4-Propargyloxymethyl-1,3-dioxolan- 2-yl, 4-Acetoxymethyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-1,3-dithiolan-2-yl, 4-Propargyl­ oxymethyl-1,3-dithiolan-2-yl, 4-Acetoxymethyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl-1,3-oxathiolan-2-yl, 5-Allyloxy­ methyl-1,3-oxathiolan-2-yl, 4-Propargyloxymethyl-1,3-oxathiolan-2-yl, 5-Propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxymethyl- 1,3-oxathiolan-2-yl, 5-Acetoxymethyl-1,3-oxathiolan-2-yl, 4-Methylthiomethyl-1,3-dioxolan-2-yl, 4-Methylthiomethyl-1,3- dithiolan-2-yl, 4-Carboxy-1,3-dioxolan-2-yl, 4-Carboxy-1,3- dithiolan-2-yl, 4-Methoxycarbonyl-1,3-dioxolan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-4-methyl- 1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithiolan- 2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-1,3- dithiolan-2-yl, 1,3-Dioxan-2-yl, 1,3-Dithian-2-yl, 1,3-Oxathian- 2-yl, 5-Methyl-1,3-dioxan-2-yl, 5-Methyl-1,3-dithian-2-yl, 5-Methyl-1,3-oxathian-2-yl, 5,5-Dimethyl-1,3-dioxan-2-yl, 4,6-Dimethyl- 1,3-dioxan-2-yl, 4,4-Dimethyl-1,3-dioxan-2-yl, 5,5-Dimethyl- 1,3-dithian-2-yl, 4,6-Dimethyl-1,3-dithian-2-yl, 4,4-Dimethyl- 1,3-dithian-2-yl, 5,5-Dimethyl-1,3-oxathian-2-yl, 4,4-Dimethyl- 1,3-oxathian-2-yl, 6,6-Dimethyl-1,3-oxathian-2-yl, 4-Hydroxymethyl-1,3-dioxan-2-yl, 4-Methoxymethyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-1,3-dithian-2-yl, 4-Methoxymethyl-1,3-dithian-2-yl, 4-Allyloxymethyl-1,3-dithian-2-yl, 4-Acetoxymethyl- 1,3-dithian-2-yl, 4-Chlormethyl-1,3-dioxan-2-yl, 4-Chlormethyl- 1,3-dithian-2-yl, 1,3-Dioxepan-2-yl, 1,3-Dithiepan-2-yl, 1,3-Dioxep-5-en-2-yl, 4-Methoxycarbonyl-1,3-dioxan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-1,3-dithian-2-yl, 4-n-Butoxycarbonyl-1,3-dithian-2-yl, 4-Methoxycarbonyl-4- methyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-4-methyl- 1,3-dithian-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithian-2-yl, -C(CH₃)(OCH₃)₂, -C(CH₃)(SCH₃)₂, -C(CH₃)(OC₂H₅)₂, -C(CH₃)(SC₂H₅)₂, -C(CH₃)(O-n-C₃H₇)₂, -C(CH₃)(O-i-C₃H₇)₂, -C(CH₃)(S-n-C₃H₇)₂, -C(CH₃)(S-i-C₃H₇)₂, -C(CH₃)(O-n-C₄H₉)₂, -C(CH₃)(O-i-C₄H₉)₂, -C(CH₃)(O-s-C₄H₉)₂, -C(CH₃)(O-tert.-C₄H₉)₂, -C(CH₃)(S-n-C₄H₉)₂, -C(CH₃)(S-i-C₄H₉)₂, -C(CH₃)(S-s-C₄H₉)₂, -C(CH₃)(S-tert.-C₄H₉)₂, -C(CH₃)(O-n-C₅H₁₁)′′, 2-Methyl-1,3-dioxolan-2-yl, 2-Methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-oxathiolan-2-yl, 2,4-Dimethyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-1,3- oxathiolan-2-yl, 2,5-Dimethyl-1,3-oxathiolan-2-yl, 4-Ethyl-2- methyl-1,3-dioxolan-2-yl, 4-Ethyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Ethyl-2-methyl-1,3- oxathiolan-2-yl, 2,4,5-Trimethyl-1,3-dioxolan-2-yl, 2,4,4-Trimethyl- 1,3-dioxolan-2-yl, 2,4,5-Trimethyl-1,3-dithiolan-2-yl, 2,4,4-Trimethyl-1,3-dithiolan-2-yl, 2,4,5-Trimethyl-1,3-oxathiolan-2-yl, 2,4,4-Trimethyl-1,3-oxathiolan-2-yl, 2-Methyl-4-vinyl- 1,3-dioxolan-2-yl, 2-Methyl-4-vinyl-1,3-dithiolan-2-yl, 2-Methyl- 4-vinyl-1,3-oxathiolan-2-yl, 2-Methyl-5-vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-dioxolan-2-yl, 4-Chlormethyl-2- methyl-1,3-dithiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl- 2-methyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-2- methyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dioxolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxy- 2-methyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dithiolan-2-yl, 4-Acetoxy-2- methyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl- 2-methyl-1,3-oxathiolan-2-yl, 5-Allyloxymethyl-2- methyl-1,3-oxathiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3- oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxy-2-methyl-1,3-oxathiolan-2-yl, 5-Acetoxy-2-methyl- 1,3-oxathiolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dioxolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-2- methyl-1,3-dioxolan-2-yl, 4-Carboxy-2-methyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-2- methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl- 2-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-2- methyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-ethoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4- ethoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-n-butoxy- carbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl-1,3- dithiolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-dioxan-2-yl, 2-Methyl-1,3-dithian-2-yl, 2-Methyl-1,3-oxathian-2-yl, 2,5- Dimethyl-1,3-dioxan-2-yl, 2,5-Dimethyl-1,3-dithian-2-yl, 2,5-Dimethyl- 1,3-oxathian-2-yl, 2,5,5-Trimethyl-1,3-dioxan-2-yl, 2,4,6- Trimethyl-1,3-dioxan-2-yl, 2,2,4-Trimethyl-1,3-dioxan-2-yl, 2,5,5-Trimethyl-1,3-dithian-2-yl, 2,4,6-Trimethyl-1,3-dithian-2-yl, 2,4,4-Trimethyl-1,3-dithian-2-yl, 2,5,5-Trimethyl-1,3-oxathian-2-yl, 2,4,4-Trimethyl-1,3-oxathian-2-yl, 2,6,6-Trimethyl- 1,3-oxathian-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-2- methyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dithian-2-yl, 4-Methoxymethyl-2- methyl-1,3-dithian-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithian-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dithian-2-yl, 4-Chlormethyl-2- methyl-1,3-dioxan-2-yl, 4-Chlormethyl-2-methyl-1,3-dithian-2-yl, -C(CH₃)=NH, -C(CH₃)=N-CH₃, -C(CH₃)=N-C₂H₅, -C(CH₃)=N-n-C₃H₇, -(CH₃)=N-i-C₃H₇, -C(CH₃)=N-n-C₄H₉, -C(CH₃)=N-CH₂CH=CH₂, -C(CH₃)=N-CH₂CH=CH₂-CH₃, -C(CH₃)=N-CH₂C≡CH, -C(CH₃)=N-CH₂C≡C-CH₃, -C(CH₃)=N-cyclopropyl, -C(CH₃)=N-cyclobutyl, -C(CH₃)=N-cyclopentyl, -C(CH₃)=N-cyclohexyl, -C(CH₃)=N-cycloheptyl, -C(CH₃)=N-CH₂-CH₂Cl, -C(CH₃)=N-CH₂Cl, -C(CH₃)=N-C₆H₅, -C(CH₃)=N-(2-F-C₆H₄), -C(CH₃)=N-(3-F-C₆H₄), -C(CH₃)=N-(4-F-C₆H₄), -C(CH₃)=N-(2-Cl-C₆H₄), -C(CH₃)=N-(3-Cl-C₆H₄), -C(CH₃)=N-(4-Cl-C₆H₄), -C(CH₃)=N-(2-CH₃-C₆H₄), -C(CH₃)=N-(3-CH₃-C₆H₄), -C(CH₃)=N-(4-CH₃-C₆H₄), -C(CH₃)=N-(2-CF₃-C₆H₄), -C(CH₃)=N-(3-CF₃-C₆H₄), -C(CH₃)=N-(4-CF₃-C₆H₄), -C(CH₃)=N-(2-OCH₃-C₆H₄), -C(CH₃)=N-(3-OCH₃-C₆H₄), -C(CH₃)=N-(4-OCH₃-C₆H₄), -C(CH₃)=N-(4-NO₂-C₆H₄), -C(CH₃)=N-(4-CN-C₆H₄), -C(CH₃)=N-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-(2,4-(CH₃)₂-C₆H₃), -C(CH₃)=N-CH₂-OCH₃, -C(CH₃)=N-CH₂-OC₂H₅, -C(CH₃)=N-CH₂CH₂-OCH₃, -C(CH₃)=N-CH₂CH₂-OC₂H₅, -C(CH₃)=N-OH, -C(CH₃)=N-OCH₃, -C(CH₃)=N-OC₂H₅, -C(CH₃)=N-O-n-C₃H₇, -C(CH₃)=N-O-i-C₃H₇, -C(CH₃)=N-O-n-C₄H₉, -C(CH₃)=N-O-i-C₄H₉, -C(CH₃)=N-O-s-C₄H₉, -C(CH₃)=N-O-tert.-C₄H₉, -C(CH₃)=N-OCH₂-CH=CH₂, -C(CH₃)=N-OCH(CH₃)-CH=CH₂, -C(CH₃)=N-OCH₂-C≡CH, -C(CH₃)=N-CH(CH₃)-C≡CH, -C(CH₃)=N-OCH₂-CH=C-CH₃, -C(CH₃)=N-OCH₂CH₂-Cl, -C(CH₃)=N-OCH₂CH₂-F, -C(CH₃)=N-OCH₂-CF₃, -C(CH₃)=N-OCH₂-CH=CHCl, -C(CH₃)=N-OCH₂-C(Cl)=CH₂, -C(CH₃)=N-OCH₂-C(Br)=CH₂, -C(CH₃)=N-OCH₂-CH=C(Cl)-CH₃, -C(CH₃)=N-O-CO-CH₃, -C(CH₃)=N-O-CO-C₂H₅, -C(CH₃)=N-OCH₂-CN, -C(CH₃)=N-OCH₂-CH=CH-CH₂-OCH₃, -C(CH₃)=N-OCH₂-CH=CH-CH₂-O-tert.-C₄H₉, -C(CH₃)=N-O-(CH₂)₃-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-(4-Cl-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-C₆H₅, -C(CH₃)=N-OCH₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(3-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-CH₂-(4-CH₃O-C₆H₄), -C(CH₃)=N-OCH₂-CH=C(CH₃)-C₆H₅, -C(CH₃)=N-O-(CH₂)₂-CH=CH-(3,4-Cl₂-C₆H₃), -C(CH₃)=N-O-(CH₂)₃-C≡C-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-OCH₃, -C(CH₃)=N-OCH₂CH₂-OCH₃, -C(CH₃)=N-OCH₂-OC₂H₅, -C(CH₃)=N-OCH(CH₃)-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=N-NH₂, -C(CH₃)=N-NH-CH₃, -C(CH₃)=N-NH-C₂H₅, -C(CH₃)=N-NH-n-C₃H₇, -C(CH₃)=N-NH-i-C₃H₇, -C(CH₃)=N-NH-n-C₄H₉, -C(CH₃)=N-NH-i-C₄H₉, -C(CH₃)=N-NH-s-C₄H₉, -C(CH₃)=N-NH-tert.-C₄H₉, -C(CH₃)=N-NH-cyclopropyl, -C(CH₃)=N-NH- cyclobutyl, -C(CH₃)=N-NH-cyclopentyl, -C(CH₃)=N-NH-cyclohexyl, -C(CH₃)=N-NH-cycloheptyl, -C(CH₃)=N-N(CH₃)₂, -C(CH₃)=N-N(C₂H₅)₂, -C(CH₃)=N-N(n-C₃H₇)₂, -C(CH₃)=N-N(i-C₃H₇)₂, -C(CH₃)=N-NH-CH₂-C=CH, -C(CH₃)=N-NH-CH₂-C≡CH, -C(CH₃)=N-N(CH₃)-CH₂-C≡CH, -C(CH₃)=N-NH-CH₂CF₃, -C(CH₃)=N-NH-CO-CH₃, -C(CH₃)=N-NH-CO-C₂H₅, -C(CH₃)=N-NH-CO-OCH₃, -C(CH₃)=N-NH-CO-OC₂H₅, -C(CH₃)=N-NH-CO-O-tert.-C₄H₉, -C(CH₃)=N- pyrrolidin-1-yl, -C(CH₃)=N-piperidin-1-yl, -C(CH₃)=N-morpholin- 4-yl, -C(CH₃)=N-NH-C₆H₅, -C(CH₃)=N-NH-(4-Cl-C₆H₄), -C(CH₃)=N-NH-(4-NO₂-C₆H₄), -C(CH₃)=N-NH-(4-F-C₆H₄), -C(CH₃)=N-NH-(4-CH₃O-C₆H₄), -C(CH₃)=N-NH-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-NH-(2,4-(NO₂)₂-C₆H₃), -C(CH₃)=N-NH-CO-NH₂, -C(CH₃)=N-NH-CO-NHCH₃, -C(CH₃)=N-NH-CO-NHC₂H₅, -C(CH₃)=N-NH-CO-N(CH₃)₂, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=CH-CO-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-O-n-C₄H₉, -C(CH₃)=CH-CO-O-tert.-C₄H₉, -C(CH₃)=CH-CO-O-cyclopropyl, -C(CH₃)=CH-CO-O-cyclobutyl, -C(CH₃)=CH-CO-O-cyclopentyl, -C(CH₃)=CH-CO-O-cyclohexyl, -C(CH₃)=CH-CO-O-cycloheptyl, -C(CH₃)=C(CH₃)-COOH, -C(CH₃)=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-cyclopropyl, -C(CH₃)=C(CH₃)-CO-O-cyclobutyl, -C(CH₃)=C(CH₃)-CO-O-cyclopentyl, -C(CH₃)=C(CH₃)-CO-O-cyclohexyl, -C(CH₃)=C(CH₃)-CO-O-cycloheptyl, -C(CH₃)=C(C₂H₅)-COOH, -C(CH₃)=C(C₂H₅)-CO-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-cyclo­ propyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-O- cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-O-cycloheptyl, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=C(Cl)-CO-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-O-n-C₄H₉, -C(CH₃)=C(Cl)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-O-cyclopropyl, -C(CH₃)=C(Cl)-CO-O-cyclobutyl, -C(CH₃)=C(Cl)-CO-O-cyclopentyl, -C(CH₃)=C(Cl)-CO-O-cyclohexyl, -C(CH₃)=C(Cl)-CO-O-cycloheptyl, -C(CH₃)=C(Br)-COOH, -C(CH₃)=C(Br)-CO-OCH₃, -C(CH₃)=C(Br)-CO-OC₂H₅, -C(CH₃)=C(Br)-CO-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-O-n-C₄H₉, -C(CH₃)=C(Br)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-O-cyclopropyl, -C(CH₃)=C(Br)-CO-O-cyclobutyl, -C(CH₃)=C(Br)-CO-O-cyclopentyl, -C(CH₃)=C(Br)-CO-O-cyclohexyl, -C(CH₃)=C(Br)-CO-O-cycloheptyl, -C(CH₃)=C(CN)-COOH, -C(CH₃)=C(CN)-CO-OCH₃, -C(CH₃)=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CN)-CO-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-O-n-C₄H₉, -C(CH₃)=C(CN)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-O-cyclopropyl, -C(CH₃)=C(CN)-CO-O-cyclobutyl, -C(CH₃)=C(CN)-CO-O-cyclopentyl, -C(CH₃)=C(CN)-CO-O-cyclohexyl, -C(CH₃)=C(CN)-CO-O-cycloheptyl, -C(CH₃)=CH-CO-OCH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=CH-CO-O-i-C₃H₇, -C(CH₃)=CH-CO-OCH(CH₃)-OCH₃, -C(CH₃)=CH-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=CH-CO-OCH₂CH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=(C₂H₅)-CO-OCH₂CH₂-OCH₃, -(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-O-i-C₃H₇, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -(CH₃)=C(Cl)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-O-i-C₃H₇, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-O-i-C₃H₇, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-CF₃, -C(CH₃)=CH-CO-OCH₂-CCl₃, -C(CH₃)=CH-CO-OCH₂-oxiranyl, -C(CH₃)=CH-CO-O-(CH₂)₃-Br,-C(CH₃)=CH-CO-OCH₂-CH=CH₂, -C(CH₃)=CH-CO-OCH₂-C≡CH, -C(CH₃)=CH-CO-OCH₂-CN, -C(CH₃)=CH-CO-OCH₂CH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CF₃, -C(CH₃)=C(CH₃)-CO-OCH₂-CCl₃, -C(CH₃)=C(CH₃)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CH₃)-CO-O -(CH₂)₃-Br, -C(CH₃)=C(CH₃)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CH₃)-CO-OCH₂-C≡CH, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CF₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CCl₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-oxiranyl, -C(CH₃)=C(C₂H₅)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(C₂H₅)-CO-OCH₂-C≡CH, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂-CF₃, -C(CH₃)=C(Cl)-CO-OCH₂-CCl₃, -C(CH₃)=C(Cl)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Cl)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Cl)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Cl)-CO-OCH₂-C≡CH, -C(CH₃)=C(Cl)-CO-OCH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂-CF₃, -C(CH₃)=C(Br)-CO-OCH₂-CCl₃, -C(CH₃)=C(Br)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Br)-CO-O(CH₂)₃-Br, -C(CH₃)=C(Br)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Br)-CO-OCH₂-C≡CH, -C(CH₃)=C(Br)-CO-OCH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂CH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂-CF₃, -C(CH₃)=C(CN)-CO-OCH₂-CCl₃, -C(CH₃)=C(CN)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CN)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CN)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CN)-CO-OCH₂-C≡CH, -C(CH₃)=C(CN)-CO-OCH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂CH₂-CN, -C(CH₃)=CH-CO-CH₃, -C(CH₃)=CH-CO-C₂H₅, -C(CH₃)=CH-CO-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-n-C₄H₉, -C(CH₃)=CH-CO-tert.-C₄H₉, -C(CH₃)=CH-CO-CH₂Cl, -C(CH₃)=CH-CO-CH₂Br, -C(CH₃)=CH-CO-CHCl₂, -C(CH₃)=CH-CO-CH₂-OCH₃, -C(CH₃)=CH-CO-CH(OCH₃)₂, -C(CH₃)=CH-CO-CH₂-SCH₃, -C(CH₃)=C(CH₃)-CO-CH₃, -C(CH₃)=C(CH₃)-CO-C₂H₅, -C(CH₃)=C(CH₃)-CO-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-CH₂Cl, -C(CH₃)=C(CH₃)-CO-CH₂Br, -C(CH₃)=C(CH₃)-CO-CHCl₂, -C(CH₃)=C(CH₃)-CO-CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-CH(OCH₃)₂, -C(CH₃)=C(CH₃)-CO-CH₂-SCH₃, -C(CH₃)=C(C₂H₅)-CO-CH₃, -C(CH₃)=C(C₂H₅)-CO-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-CH₂Cl, -C(CH₃)=C(C₂H₅)-CO-CH₂Br, -C(CH₃)=C(C₂H₅)-CO-CHCl₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-CH(OCH₃)₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-SCH₃, -C(CH₃)=C(Cl)-CO-CH₃, -C(CH₃)=C(Cl)-CO-C₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-n-C₄H₉, -C(CH₃)=C(Cl)-CO-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-CH₂Cl, -C(CH₃)=C(Cl)-CO-CHCl₂, -C(CH₃)=C(Cl)-CO-CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-CH(OCH₃)₂, -C(CH₃)=C(Cl)-CO-CH₂-SCH₃, -C(CH₃)=C(Br)-CO-CH₃, -C(CH₃)=C(Br)-CO-C₂H₅, -C(CH₃)=C(Br)-CO-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-n-C₄H₉, -C(CH₃)=C(Br)-CO-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-CH₂Cl, -C(CH₃)=C(Br)-CO-CH₂Br, -C(CH₃)=C(Br)-CO-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-CH(OCH₃)₂, -C(CH₃)=C(Br)-CO-CH₂-SCH₃, -C(CH₃)=C(CN)-CO-CH₃, -C(CH₃)=C(CN)-CO-C₂H₅, -C(CH₃)=C(CN)-CO-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-n-C₄H₉, -C(CH₃)=C(CN)-CO-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-CH₂Cl, -C(CH₃)=C(CN)-CO-CH₂Br, -C(CH₃)=C(CN)-CO-CHCl₂, -C(CH₃)=C(CN)-CO-CH₂-OCH₃, -C(CH₃)=C(CN)-CO-CH(OCH₃)₂, -C(CH₃)=C(CN)-CO-CH₂-SCH₃, -C(CH₃)=CH-CO-C₆H₅, -C(CH₃)=CH-CO-(4-Cl-C₆H₄), -C(CH₃)=C(CH₃)-CO-C₆H₅, -C(CH₃)=C(CH₃)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(C₂H₅)-CO-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(Cl)-CO-C₆H₅, -C(CH₃)=C(Br)-CO-C₆H₅, -C(CH₃)=C(CN)-CO-C₆H₅, -C(CH₃)=CH-CO-NH₂, -C(CH₃)=CH-CO-NHCH₃, -C(CH₃)=CH-CO-N(CH₃)₂, -C(CH₃)=CH-CO-NH-C₂H₅, -C(CH₃)=CH-CO-N(C₂H₅)₂, -C(CH₃)=CH-CO-NH-n-C₃H₇, -C(CH₃)=CH-CO-NH-i-C₃H₇, -C(CH₃)=CH-CO-NH-tert.-C₄H₉, -C(CH₃)=CH-CO-NH-cyclopropyl, -C(CH₃)=CH-CO-NH-cyclobutyl, -C(CH₃)=CH-CO-NH-cyclopentyl, -C(CH₃)=CH-CO-NH-cyclohexyl, -C(CH₃)=CH-CO-NH-cycloheptyl, -C(CH₃)=CH-CO-NH-cyclooctyl, -C(CH₃)=CH-CO-pyrrolidin-1-yl, -C(CH₃)=CH-CO-piperidin-1-yl, -C(CH₃)=CH-CO-morpholin-4-yl, -C(CH₃)=CH-CO-NH-CH₂CH=CH₂, -C(CH₃)=CH-CO-NH-CH₂C≡CH, -C(CH₃)=CH-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=CH-CO-NH-(CH₂)₂Cl, -C(CH₃)=CH-CO-NH-C₆H₅, -C(CH₃)=C(CH₃)-CO-NH₂, -C(CH₃)=C(CH₃)-CO-NHCH₃, -C(CH₃)=C(CH₃)-CO-N(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-C₂H₅, -C(CH₃)=C(CH₃)-CO-N(C₂H₅)₂, -C(CH₃)=C(CH₃)-CO-NH-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-NH- cyclopropyl, -C(CH₃)=C(CH₃)-CO-NH-cyclobutyl, -C(CH₃)=C(CH₃)-CO-NH-cyclopentyl, -C(CH₃)=C(CH₃)-CO-NH- cyclohexyl, -C(CH₃)=C(CH₃)-CO-NH-cycloheptyl, -C(CH₃)=C(CH₃)-CO-NH-cyclooctyl, -C(CH₃)=C(CH₃)-CO- pyrrolidin-1-yl, -C(CH₃)=C(CH₃)-CO-piperidin-1-yl, -C(CH₃)=C(CH₃)-CO-morpholin-4-yl, -C(CH₃)=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-NH(CH₂)₂Cl, -C(CH₃)=C(CH₃)-CO-NH-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-NH₂, -C(CH₃)=C(C₂H₅)-CO-NHCH₃, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)₂, -C(CH₃)=C(C₂H₅)-CO-NH-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-N(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-NH- cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclo­ hexyl, -C(CH₃)=C(C₂H₅)-CO-NH-cycloheptyl, -C(CH₃)=C(C₂H₅)-CO-NH- cyclooctyl, -C(CH₃)=C(C₂H₅)-CO-pyrrolidin-1-yl, -C(CH₃)=C(C₂H₅)-CO-piperidin-1-yl, -C(CH₃)=C(C₂H₅)-CO- morpholin-4-yl, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(C₂H₅)-CO-NH-C₆H₅, -C(CH₃)=C(Cl)-CO-NH₂, -C(CH₃)=C(Cl)-CO-NHCH₃, -C(CH₃)=C(Cl)-CO-N(CH₃)₂, -C(CH₃)=C(Cl)-CO-NH-C₂H₅, -C(CH₃)=C(Cl)-CO-N(C₂H₅)₂, -C(CH₃)=C(Cl)-CO-NH-n-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-i-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-NH-cyclopropyl, -C(CH₃)=C(Cl)-CO-NH-cyclobutyl, -C(CH₃)=C(Cl)-CO-NH-cyclopentyl, -C(CH₃)=C(Cl)-CO-NH-cyclohexyl, -C(CH₃)=C(Cl)-CO-NH-cycloheptyl, -C(CH₃)=C(Cl)-CO-NH-cyclooctyl, -C(CH₃)=C(Cl)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Cl)-CO-piperidin-1- yl, -C(CH₃)=C(Cl)-CO-morpholin-4-yl, -C(CH₃)=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -C(CH₃)=C(Cl)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Cl)-CO-NH-C₆H₅, -C(CH₃)=C(Br)-CO-NH₂, -C(CH₃)=C(Br)-CO-NHCH₃, -C(CH₃)=C(Br)-CO-N(CH₃)₂, -C(CH₃)=C(Br)-CO-NH-C₂H₅, -C(CH₃)=C(Br)-CO-N(C₂H₅)₂, -C(CH₃)=C(Br)-CO-NH-n-C₃H₇, -C(CH₃)=C(Br)-CO-NH-i-C₃H₇, -C(CH₃)=C(Br)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-NH-cyclopropyl, -C(CH₃)=C(Br)-CO-NH-cyclobutyl, -C(CH₃)=C(Br)-CO-NH-cyclopentyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cycloheptyl, -C(CH₃)=C(Br)-CO-NH-cyclooctyl, -C(CH₃)=C(Br)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Br)-CO-piperidin-1-yl, -C(CH₃)=C(Br)-CO-morpholin-4-yl, -C(CH₃)=C(Br)-CO-NH-CH₂CH=C(Br)₂, -C(CH₃)=C(Br)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Br)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Br)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Br)-CO-NH-C₆H₅, -C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CN)-CO-NHCH₃, -C(CH₃)=C(CN)-CO-N(CH₃)₂, -C(CH₃)=C(CN)-CO-NH-C₂H₅, -C(CH₃)=C(CN)-CO-N(C₂H₅)₂, -C(CH₃)=C(CN)-CO-NH-n-C₃H₇, -C(CH₃)=C(CN)-CO-NH-i-C₃H₇, -C(CH₃)=C(CN)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-NH-cyclopropyl, -C(CH₃)=C(CN)-CO-NH-cyclobutyl, -C(CH₃)=C(CN)-CO-NH-cyclopentyl, -C(CH₃)=C(CN)-CO-NH-cyclohexyl, -C(CH₃)=C(CN)-CO-NH-cycloheptyl, -C(CH₃)=C(CN)-CO-NH-cyclooctyl, -C(CH₃)=C(CN)-CO-pyrrolidin-1-yl, -C(CH₃)=C(CN)-CO-piperidin-1-yl, -C(CH₃)=C(CN)-CO-morpholin-4-yl, -C(CH₃)=C(CN)-CO-NH-CH₂CH=C(CN)₂, -C(CH₃)=C(CN)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CN)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=(CN)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CN)-CO-NH-C₆H₅, -C(CH₃)=CH-SO-SCH₃, -C(CH₃)=CH-CO-SC₂H₅, -C(CH₃)=CH-CO-S-n-C₃H₇, -C(CH₃)=CH-CO-S-i-C₃H₇, -C(CH₃)=CH-CO-S-n-C₄H₉, -C(CH₃)=CH-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-SCH₃, -C(CH₃)=C(CH₃)-CO-SC₂H₅, -C(CH₃)=C(CH₃)-CO-S-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-S-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-SCH₃, -C(CH₃)=C(C₂H₅)-CO-SC₂H₅, -C(CH₃)=C(C₂H₅)-CO-S-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-SCH₃, -C(CH₃)=C(Cl)-CO-SC₂H₅, -C(CH₃)=C(Cl)-CO-S-n-C₃H₇, -C(CH₃)=C(Cl)-CO-S-i-C₃H₇, -C(CH₃)=C(Cl)-CO-S-n-C₄H₉, -C(CH₃)=C(Cl)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-SCH₃, -C(CH₃)=C(Br)-CO-SC₂H₅, -C(CH₃)=C(Br)-CO-S-n-C₃H₇, -C(CH₃)=C(Br)-CO-S-i-C₃H₇, -C(CH₃)=C(Br)-CO-S-n-C₄H₉, -C(CH₃)=C(Br)-CO-S-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-SCH₃, -C(CH₃)=C(CN)-CO-SC₂H₅, -C(CH₃)=C(CN)-CO-S-n-C₃H₇, -C(CH₃)=C(CN)-CO-S-i-C₃H₇, -C(CH₃)=C(CN)-CO-S-n-C₄H₉, -C(CH₃)=C(CN)-CO-S-tert.-C₄H₉, -C(CH₃)=C(COCH₃)-CO-OCH₃, -C(CH₃)=C(COC₂H₅)-CO-OCH₃, -C(CH₃)=C(CO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COCH₃)-CO-OC₂H₅, -C(CH₃)=C(COC₂H₅)-CO-OC₂H₅, -C(CH₃)=C(CO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COCH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(COC₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-OCH₃, -C(CH₃)=C(CF₃)-CO-OC₂H₅, -C(CH₃)=C(CF₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CF₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(COOCH₃)₂, -C(CH₃)=C(COOC₂H₅)₂, -C(CH₃)=C(COOCH₃)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇))-CO-OCH₃, -C(CH₃)=C(COO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)₂, -C(CH₃)=CH-CH=CH-COOH, -C(CH₃)=CH-CH=CH-CO-OCH₃, -C(CH₃)=CH-CH=CH-CO-OC₂H₅, -C(CH₃)=CH-CH=C(COOCH₃)₂, -C(CH₃)=CH-CH=C(CN)-CO-OCH₃, -C(CH₃)=CH-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CN)CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH₂, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -C(CH₃)=CH-(CH₂)₂-COOH, -C(CH₃)=CH-(CH₂)₂-CO-OCH₃, -C(CH₃)=CH-(CH₂)₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(COOCH₃)₂, -C(CH₃)=CH-CH₂-CH(COOC₂H₅)₂, -C(CH₃)=CH-CH₂-CH(CN)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CN)-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -C(CH₃)=CH-(CH₂)₂-CO-NH₂, -C(CH₃)=CH-(CH₂)₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-COOH, -C(CH₃)=CH-CH₂-CO-OCH₃, -C(CH₃)=CH-CH₂-CO-OC₂H₅, -C(CH₃)=C(COOCH₃)-CH₂-CO-OCH₃, -C(CH₃)=C(COOCH₃)-CH₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CO-NH₂, -C(CH₃)=CH-CH₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-CO-N(CH₃)₂.
wobei W für eine der folgenden Bedeutungen steht:
-CHO, -COCH₃, -COC₂H₅, -CO-n-C₃H₇, -CO-i-C₃H₇, -CO-n-C₄H₉, -CO-i-C₄H₉, -CO-s-C₄H₉, -CO-tert.-C₄H₉, -CO-CH₂CH=CH₂, -CO-CF₃, -COCCl₃, -COCH₂C≡CH, -CO-cyclopropyl, -CO-cyclobutyl, -CO-cyclopentyl, -CO-cyclohexyl, -CO-CN, -CO-COOCH₃, -CO-COOC₂H₅, -CH=NH, -CH=NCH₃, -CH=NC₂H₅, -CH=N-n-C₃H₅, -CH=N-i-C₃H₅, -CH=N-n-C₄H₉, -CH=NCH₂CH=CH₂, -CH=NCH₂CH=CH₂-CH₃, -CH=NCH₂C≡CH, -CH=NCH₂C≡C-CH₃, -CH=N-cyclopropyl, -CH=N-cyclobutyl, -CH=N-cyclopentyl, -CH=N-cyclohexyl, -CH=N-cycloheptyl, -CH=N-CH₂-CH₂Cl, -CH=N-CH₂Cl, -CH=N-C₆H₅, -CH=N-4-Br-C₆H₄, -CH=N-3-F-C₆H₄, -CH=N-4-F-C₆H₄, -CH=N-2-Cl-C₆H₄, -CH=N-3-Cl-C₆H₄, -CH=N-4-Cl-C₆H₄, -CH=N-2-Br-C₆H₄, -CH=N-2-F-C₆H₄, -CH=N-2-CH₃-C₆H₄, -CH=N-3-CH₃-C₆H₄, -CH=N-4-CH₃-C₆H₄, -CH=N-2-CF₃-C₆H₄, -CH=N-3-CF₃-C₆H₄, -CH=N-4-CF₃-C₆H₄, -CH=N-2-OCH₃-C₆H₄, -CH=N-3-OCH₃-C₆H₄, -CH=N-4-OCH₃-C₆H₄, -CH=N-4-NO₂-C₆H₄, -CH=N-4-CN-C₆H₄, -CH=N-2,4-(Cl,Cl)-C₆H₄, -CH=N-2,4-(CH₃,CH₃)-C₆H₄, -CH=N-CH₂OCH₃ -CH=N-CH₂OC₂H₅, -CH=N-CH₂CH₂OCH₃, -CH=N-CH₂CH₂OC₂H₅, -CH=N-OH, -CH=N-OCH₃, -CH=N-OC₂H₅, -CH=N-O-n-C₃H₇, -CH=N-O-i-C₃H₇, -CH=N-O-n-C₄H₉, -CH=N-O-i-C₄H₉, -CH=N-O-s-C₄H₉, -CH=N-O-tert.-C₄H₉, -CH=N-O-CH₂CH=CH₂, -CH=N-O-CH(CH₃)CH=CH₂, -CH=N-O-CH₂C≡CH, -CH=N-O-CH(CH₃)-C≡CH, -CH=N-O-CH₂-CH=CH-CH₃, -CH=N-O-CH₂-CH₂-Cl, -CH=N-O-CH₂-CH₂-F, -CH=N-O-CH₂-CF₃, -CH=N-O-CH₂-CH=CHCl, -CH=N-O-CH₂-CCl=CH₂, -CH=N-O-CH₂-CBr=CH₂, -CH=N-O-CH₂-CH=CCl-CH₃, -CH=N-OC(O)CH₃, -CH=N-OC(O)C₂H₅, -CH=N-O-CH₂-CN, -CH=N-O-CH₂-CH=CH-CH₂-O-CH₃, -CH=N-O-CH₂-CH=CH-CH₂-O-tert.-C₄H₉, -CH=N-O-(CH₂)₃-C₆H₅, -CH=N-O-(CH₂)₄-C₆H₅, -CH=N-O-(CH₂)₄-4-Cl-C₆H₄, -CH=N-O-(CH₂)₄-4-OCH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-CH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-C₆H₅, -CH=N-O-CH₂CH=CH-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CH-3-OCH₃-C₆H₄, -CH=N-O-(CH₂)₂CH=CH-4-F-C₆H₄, -CH=N-O-(CH₂)CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CHCH₂-4-OCH₃-C₆H₄, -CH=N-O-CH₂-CH=C(CH₃)-C₆H₅ -CH=N-O-(CH₂)₂CH=CH-3,4(Cl,Cl)-C₆H₃, -CH=N-O-(CH₂)₃C≡C-4-F-C₆H₄, -CH₂=N-OCHOCH₃, -CH=N-OC₂H₄OCH₃, -CH=N-OCH₂OC₂H₅, -CH=N-OCH(CH₃)OCH₃, -CH=N-OCH(CH₃)COOCH₃, -CH=N-OCH(CH₃)COO-n-C₄H₉, -CH=N-NH₂, -CH=N-NHCH₃, -CH=N-NHC₂H₅, -CH=N-NH-n-C₃H₇, -CH=N-NH-i-C₃H₇, -CH=N-NH-n-C₄H₉, -CH=N-NH-i-C₄H₉, -CH=N-NH-s-C₄H₉, -CH=N-NH-tert.-C₄H₉, -CH=N-NH-cyclopropyl, -CH=N-NH-cyclobutyl, -CH=N-NH-cyclopentyl, -CH=N-NH-cyclohexyl, -CH=N-NH-cycloheptyl, -CH=N-N(CH₃)₂, -CH=N-N(C₂H₅)₂, -CH=N-N(C₃H₇)₂, -CH=N-N(i-C₃H₇)(CH₃), -CH=N-NHCH₂-C=CH, -CH=N-NHCH₂-C≡CH, -CH=N-N(CH₃)-CH₂-C≡CH, -CH=N-NHCH₂CF₃, -CH=N-NH-CO-CH₃, -CH=N-NH-CO-CH₂H₅, -CH=N-NH-COOCH₃, -CH=N-NH-COOC₂H₅, -CH=N-NH-COO-tert.-C₄H₉, -CH=N-pyrrolidin-1-yl, -CH=N-piperidin-1-yl, -CH=N-morpholin-4-yl, -CH=N-NH-C₆H₅, -CH=N-NH-(4-Cl-C₆H₄), -CH=N-NH-(4-NO₂-C₆H₄), -CH=N-NH-(4-F-C₆H₄), -CH=N-NH-(4-CH₃O-C₆H₄), -CH=N-NH-(2,4-Cl₂-C₆H₃), -CH=N-NH-(2,4-(NO₂)₂-C₆H₃), -CH=N-NH-CO-NH₂, -CH=N-NH-CO-NHCH₃, -CH=N-NH-CO-NHC₂H₅, -CH=N-NH-CO-N(CH₃)₂, -CH=CH-COOH, -CH=CH-CO-OCH₃, -CH=CH-CO-OC₂H₅, -CH=CH-CO-O-n-C₃H₇, -CH=CH-CO-O-i-C₃H₇, -CH=CH-CO-O-n-C₄H₉, -CH=CH-CO-O-tert.-C₄H₉, -CH=CH-CO-O-cyclopropyl, -CH=CH-CO-O-cyclobutyl, -CH=CH-CO-O-cyclopentyl, -CH=CH-CO-O-cyclohexyl, -CH=CH-CO-O-cycloheptyl, -CH=C(CH₃)-COOH, -CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CO-O-n-C₃H₇, -CH=C(CH₃)-CO-O-i-C₃H₇, -CH=C(CH₃)-CO-O-n-C₄H₉, -CH=C(CH₃)-CO-O-tert.-C₄H₉, -CH=C(CH₃)-CO-O-cyclopropyl, -CH=C(CH₃)-CO-O-cyclobutyl, -CH=C(CH₃)-CO-O-cyclopentyl, -CH=C(CH₃)-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cycloheptyl, -CH=C(C₂H₅)-COOH, -CH=C(C₂H₅)-CO-OCH₃, -CH=C(C₂H₅)-CO-OC₂H₅, -CH=C(C₂H₅)-CO-O-n-C₃H₇, -CH=C(C₂H₅)-CO-O-i-C₃H₇, -CH=C(C₂H₅)-CO-O-n-C₄H₉, -CH=C(C₂H₅)-CO-O-tert.-C₄H₉, -CH=C(C₂H₅)-CO-O-cyclopropyl, -CH=C(C₂H₅)-CO-O-cyclobutyl, -CH=C(C₂H₅)-CO-O-cyclopentyl, -CH=C(C₂H₅)-CO-O-cyclohexyl, -CH=C(C₂H₅)-CO-O-cycloheptyl, -CH=C(Cl)-COOH, -CH=C(Cl)-CO-OCH₃, -CH=C(Cl)-CO-OC₂H₅, -CH=C(Cl)-CO-O-n-C₃H₇, -CH=C(Cl)-CO-O-i-C₃H₇, -CH=C(Cl)-CO-O-n-C₄H₉, -CH=C(Cl)-CO-O-tert.-C₄H₉, -CH=C(Cl)-CO-O-cyclopropyl, -CH=C(Cl)-CO-O-cyclobutyl, -CH=C(Cl)-CO-O-cyclopentyl, -CH=C(Cl)-CO-O-cyclohexyl, -CH=C(Cl)-CO-O-cycloheptyl, -CH=C(Br)-COOH, -CH=C(Br)-CO-OCH₃, -CH=C(Br)-CO-OC₂H₅, -CH=C(Br)-CO-O-n-C₃H₇, -CH=C(Br)-CO-O-i-C₃H₇, -CH=C(Br)-CO-O-n-C₄H₉, -CH=C(Br)-CO-O-tert.-C₄H₉, -CH=C(Br)-CO-O-cyclopropyl, -CH=C(Br)-CO-O-cyclobutyl, -CH=C(Br)-CO-O-cyclopentyl, -CH=C(Br)-CO-O-cyclohexyl, -CH=C(Br)-CO-O-cycloheptyl, -CH=C(CN)-COOH, -CH=C(CN)-CO-OCH₃, -CH=C(CN)-CO-OC₂H₅, -CH=C(CN)-CO-O-n-C₃H₇, -CH=C(CN)-CO-O-i-C₃H₇, -CH=C(CN)-CO-O-n-C₄H₉, -CH=C(CN)-CO-O-tert.-C₄H₉, -CH=C(CN)-CO-O-cyclopropyl, -CH=C(CN)-CO-O-cyclobutyl, -CH=C(CN)-CO-O-cyclopentyl, -CH=C(CN)-CO-O-cyclohexyl, -CH=C(CN)-CO-O-cycloheptyl, -CH=CH-CO-OCH₂-OCH₃, -CH=CH-CO-OCH₂-OC₂H₅, -CH=CH-CO-OCH₂-O-n-C₃H₅, -CH=CH-CO-OCH₂-O-i-C₃H₅, -CH=CH-CO-OCH(CH₃)-OCH₃, -CH=CH-CO-OCH(CH₃)-OC₂H₅, -CH=CH-CO-O-CH₂CH₂-OCH₃, -CH=CH-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-OCH₃, -CH=C(CH₃)-CO-OCH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-O-n-C₃H₅, -CH=C(CH₃)-CO-OCH₂-O-i-C₃H₅, -CH=C(CH₃)-CO-OCH(CH₃)-OCH₃, -CH=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CH₃)-CO-O-CH₂CH₂-OCH₃, -CH=C(CH₃)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-OCH₃, -CH=C(C₂H₅)-CO-OCH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-O-n-C₃H₅, -CH=C(C₂H₅)-CO-OCH₂-O-i-C₃H₅, -CH=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -CH=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OCH₃, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-OCH₃, -CH=C(Cl)-CO-OCH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-O-n-C₃H₅, -CH=C(Cl)-CO-OCH₂-O-i-C₃H₅, -CH=C(Cl)-CO-OCH(CH₃)-OCH₃, -CH=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Cl)-CO-O-CH₂CH₂-OCH₃, -CH=C(Cl)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-OCH₃, -CH=C(Br)-CO-OCH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-O-n-C₃H₅, -CH=C(Br)-CO-OCH₂-O-i-C₃H₅, -CH=C(Br)-CO-OCH(CH₃)-OCH₃, -CH=C(Br)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Br)-CO-O-CH₂CH₂-OCH₃, -CH=C(Br)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-OCH₃, -CH=C(CN)-CO-OCH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-O-n-C₃H₅, -CH=C(CN)-CO-OCH₂-O-i-C₃H₅, -CH=C(CN)-CO-OCH(CH₃)-OCH₃, -CH=C(CN)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CN)-CO-O-CH₂CH₂-OCH₃, -CH=C(CN)-CO-O-CH₂CH₂-OC₂H₅, -CH=CH-CO-OCH₂-CF₃, -CH=CH-CO-OCH₂-CCl₃, -CH=CH-CO-OCH₂-oxiranyl, -CH=CH-CO-O(CH₂)₃-Br, -CH=CH-CO-OCH₂-CH=CH₂, -CH=CH-CO-OCH₂-C≡CH, -CH=CH-CO-OCH₂-CN, -CH=CH-CO-O(CH₂)₂-CN, -CH=C(CH₃)-CO-OCH₂-CF₃, -CH=C(CH₃)-CO-OCH₂-CCl₃, -CH=C(CH₃)-CO-OCH₂-oxiranyl, -CH=C(CH₃)-CO-O(CH₂)₃-Br, -CH=C(CH₃)-CO-OCH₂-CH=CH₂, -CH=C(CH₃)-CO-OCH₂-C≡CH, -CH=C(CH₃)-CO-OCH₂-CN, -CH=C(CH₃)-CO-O(CH₂)₂-CN, -CH=C(C₂H₅)-CO-OCH₂-CF₃, -CH=C(C₂H₅)-CO-OCH₂-CCl₃, -CH=C(C₂H₅)-CO-OCH₂-oxiranyl, -CH=C(C₂H₅)-CO-O(CH₂)₃-Br, -CH=C(C₂H₅)-CO-OCH₂-CH=CH₂, -CH=C(C₂H₅)-CO-OCH₂-C≡CH, -CH=C(C₂H₅)-CO-OCH₂-CN, -CH=C(C₂H₅)-CO-O(CH₂)₂-CN, -CH=C(Cl)-CO-OCH₂-CF₃, -CH=C(Cl)-CO-OCH₂-CCl₃, -CH=C(Cl)-CO-OCH₂-oxiranyl, -CH=C(Cl)-CO-O(CH₂)₃-Br, -CH=C(Cl)-CO-OCH₂-CH=CH₂, -CH=C(Cl)-CO-OCH₂-C≡CH, -CH=C(Cl)-CO-OCH₂-CN, -CH=C(Cl)-CO-O(CH₂)₂-CN, -CH=C(Br)-CO-OCH₂-CF₃, -CH=C(Br)-CO-OCH₂-CCl₃, -CH=C(Br)-CO-OCH₂-oxiranyl, -CH=C(Br)-CO-O(CH₂)₃-Br, -CH=C(Br)-CO-OCH₂-CH=CH₂, -CH=C(Br)-CO-OCH₂-C≡CH, -CH=C(Br)-CO-OCH₂-CN, -CH=C(Br)-CO-O(CH₂)₂-CN, -CH=C(CN)-CO-OCH₂-CF₃, -CH=C(CN)-CO-OCH₂-CCl₃, -CH=C(CN)-CO-OCH₂-oxiranyl -CH=C(CN)-CO-O(CH₂)₃-Br, -CH=C(CN)-CO-OCH₂-CH=CH₂, -CH=C(CN)-CO-OCH₂-C≡CH, -CH=C(CN)-CO-OCH₂-CN, -CH=C(CN)-CO-O(CH₂)₂-CN, -CH=CH-CO-CH₃, -CH=CH-CO-C₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-i-C₃H₇, -CH=CH-CO-n-C₄H₉, -CH=CH-CO-tert.-C₄H₉, -CH=CH-CO-CH₂Cl, -CH=CH-CO-CH₂Br, -CH=CH-CO-CHCl₂, -CH=CH-CO-CH₂-OCH₃, -CH=CH-CO-CH(OCH₃)₂, -CH=CH-CO-CH₂-SCH₃, -CH=C(CH₃)-CO-CH₃, -CH=C(CH₃)-CO-C₂H₅, -CH=C(CH₃)-CO-n-C₃H₇, -CH=C(CH₃)-CO-i-C₃H₇, -CH=C(CH₃)-CO-n-C₄H₉, -CH=C(CH₃)-CO-tert.-C₄H₉, -CH=C(CH₃)-CO-CH₂Cl, -CH=C(CH₃)-CO-CH₂Br, -CH=C(CH₃)-CO-CHCl₂, -CH=C(CH₃)-CO-CH₂-OCH₃, -CH=C(CH₃)-CO-CH(OCH₃)₂, -CH=C(CH₃)-CO-CH₂-SCH₃, -CH=C(C₂H₅)-CO-CH₃, -CH=C(C₂H₅)-CO-C₂H₅, -CH=C(C₂H₅)-CO-n-C₃H₇, -CH=C(C₂H₅)-CO-i-C₃H₇, -CH=C(C₂H₅)-CO-n-C₄H₉, -CH=C(C₂H₅)-CO-tert.-C₄H₉, -CH=C(C₂H₅)-CO-CH₂Cl, -CH=C(C₂H₅)-CO-CH₂Br, -CH=C(C₂H₅)-CO-CHCl₂, -CH=C(C₂H₅)-CO-CH₂-OCH₃, -CH=C(C₂H₅)-CO-CH(OCH₃)₂, -CH=C(C₂H₅)-CO-CH₂-SCH₃, -CH=C(Cl)-CO-CH₃, -CH=C(Cl)-CO-C₂H₅, -CH=C(Cl)-CO-n-C₃H₇, -CH=C(Cl)-CO-i-C₃H₇, -CH=C(Cl)-CO-n-C₄H₉, -CH=C(Cl)-CO-tert.-C₄H₉, -CH=C(Cl)-CO-CH₂Cl, -CH=C(Cl)-CO-CH₂Br, -CH=C(Cl)-CO-CHCl₂, -CH=C(Cl)-CO-CH₂-OCH₃, -CH=C(Cl)-CO-CH(OCH₃)₂, -CH=C(Cl)-CO-CH₂-SCH₃, -CH=C(Br)-CO-CH₃, -CH=C(Br)-CO-C₂H₅, -CH=C(Br)-CO-n-C₃H₇, -CH=C(Br)-CO-i-C₃H₇, -CH=C(Br)-CO-n-C₄H₉, -CH=C(Br)-CO-tert.-C₄H₉, -CH=C(Br)-CO-CH₂Cl, -CH=C(Br)-CO-CH₂Br, -CH=C(Br)-CO-CHCl₂, -CH=C(Br)-CO-CH₂-OCH₃, -CH=C(Br)-CO-CH(OCH₃)₂, -CH=C(Br)-CO-CH₂-SCH₃, -CH=C(CN)-CO-CH₃, -CH=C(CN)-CO-C₂H₅, -CH=C(CN)-CO-n-C₃H₇, -CH=C(CN)-CO-i-C₃H₇, -CH=C(CN)-CO-n-C₄H₉, -CH=C(CN)-CO-tert.-C₄H₉, -CH=C(CN)-CO-CH₂Cl, -CH=C(CN)-CO-CH₂Br, -CH=C(CN)-CO-CHCl₂, -CH=C(CN)-CO-CH₂-OCH₃, -CH=C(CN)-CO-CH(OCH₃)₂, -CH=C(CN)-CO-CH₂-SCH₃, -CH=CH-CO-C₆H₅, -CH=CH-CO-(4-Cl-C₆H₄), -CH=C(CH₃)-CO-C₆H₅, -CH=C(CH₃)-CO-(4-Cl-C₆H₄), -CH=C(C₂H₅)-CO-C₆H₅, -CH=C(C₂H₅)-CO-(4-Cl-C₆H₄), -CH=C(Cl)-CO-C₆H₅, -CH=C(Br)-CO-C₆H₅, -CH=C(CN)-CO-C₆H₅, -CH=CH-CO-NH₂, -CH=CH-CO-NHCH₃, -CH=CH-CO-N(CH₃)₂, -CH=CH-CO-NH-C₂H₅, -CH=CH-CO-N(C₂H₅)₂, -CH=CH-CO-NH-n-C₃H₇, -CH=CH-CO-NH-i-C₃H₇, -CH=CH-CO-NH-tert.-C₄H₉, -CH=CH-CO-NH-cyclopropyl, -CH=CH-CO-NH-cyclobutyl, -CH=CH-CO-NH-cyclopentyl, -CH=CH-CO-NH-cyclohexyl, -CH=CH-CO-NH-cycloheptyl, -CH=CH-CO-NH-cyclooctyl, -CH=CH-CO-pyrrolidin-1-yl, -CH=CH-CO-piperidin-1-yl, -CH=CH-CO-morpholin-4-yl, -CH=CH-CO-NH-CH₂CH=CH₂, -CH=CH-CO-NH-CH₂C≡CH, -CH=CH-CO-N(CH₃)-CH₂C≡CH, -CH=CH-CO-NH-(CH₂)₂Cl, -CH=CH-CO-NH-C₆H₅, -CH=C(CH₃)-CO-NH₂, -CH=C(CH₃)-CO-NHCH₃, -CH=C(CH₃)-CO-N(CH₃)₂, -CH=C(CH₃)-CO-NH-C₂H₅, -CH=C(CH₃)-CO-N(C₂H₅)₂, -CH=C(CH₃)-CO-NH-n-C₃H₇, -CH=C(CH₃)-CO-NH-i-C₃H₇, -CH=C(CH₃)-CO-NH-tert.-C₄H₉, -CH=C(CH₃)-CO-NH-cyclopropyl, -CH=C(CH₃)-CO-NH-cyclobutyl, -CH=C(CH₃)-CO-NH-cyclopentyl, -CH=C(CH₃)-CO-NH-cyclohexyl, -CH=C(CH₃)-CO-NH-cycloheptyl, -CH=C(CH₃)-CO-NH-cyclooctyl, -CH=C(CH₃)-CO-pyrrolidin-1-yl, -CH=C(CH₃)-CO-piperidin-1-yl, -CH=C(CH₃)-CO-morpholin-4-yl, -CH=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -CH=C(CH₃)-CO-NH-CH₂C≡CH, -CH=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CH₃)-CO-NH-(CH₂)₂Cl, -CH=C(CH₃)-CO-NH-C₆H₅, -CH=C(C₂H₅)-CO-NH₂, -CH=C(C₂H₅)-CO-NHCH₃, -CH=C(C₂H₅)-CO-N(CH₃)₂, -CH=C(C₂H₅)-CO-NH-C₂H₅, -CH=C(C₂H₅)-CO-N(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-n-C₃H₇, -CH=C(C₂H₅)-CO-NH-i-C₃H₇, -CH=C(C₂H₅)-CO-NH-tert.-C₄H₉, -CH=C(C₂H₅)-CO-NH-cyclopropyl, -CH=C(C₂H₅)-CO-NH-cyclobutyl, -CH=C(C₂H₅)-CO-NH-cyclopentyl, -CH=C(C₂H₅)-CO-NH-cyclohexyl, -CH=C(C₂H₅)-CO-NH-cycloheptyl, -CH=C(C₂H₅)-CO-NH-cyclooctyl, -CH=C(C₂H₅)-CO-pyrrolidin-1-yl, -CH=C(C₂H₅)-CO-piperidin-1-yl, -CH=C(C₂H₅)-CO-morpholin-4-yl, -CH=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-CH₂C≡CH, -CH=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -CH=C(C₂H₅)-CO-NH-(CH₂)₂Cl, äCH=C(C₂H₅)-CO-NH-C₆H₅, -CH=C(Cl)-CO-NH₂, -CH=C(Cl)-CO-NHCH₃, -CH=C(Cl)-CO-N(CH₃)₂, -CH=C(Cl)-CO-NH-C₂H₅, -CH=C(Cl)-CO-N(C₂H₅)₂, -CH=C(Cl)-CO-NH-n-C₃H₇, -CH=C(Cl)-CO-NH-i-C₃H₇, -CH=C(Cl)-CO-NH-tert.-C₄H₉, -CH=C(Cl)-CO-NH-cyclopropyl, -CH=C(Cl)-CO-NH-cyclobutyl, -CH=C(Cl)-CO-NH-cyclopentyl, -CH=C(Cl)-CO-NH-cyclohexyl, -CH=C(Cl)-CO-NH-cycloheptyl, -CH=C(Cl)-CO-NH-cyclooctyl, -CH=C(Cl)-CO-pyrrolidin-1-yl, -CH=C(Cl)-CO-piperidin-1-yl, -CH=C(Cl)-CO-morpholin-4-yl, -CH=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -CH=C(Cl)-CO-NH-CH₂C≡CH, -CH=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Cl)-CO-NH-(CH₂)₂Cl, -CH=C(Cl)-CO-NH-C₆H₅, -CH=C(Br)-CO-NH₂, -CH=C(Br)-CO-NHCH₃, -CH=C(Br)-CO-N(CH₃)₂, -CH=C(Br)-CO-NH-C₂H₅, -CH=C(Br)-CO-N(C₂H₅)₂, -CH=C(Br)-CO-NH-n-C₃H₇, 99999 00070 552 001000280000000200012000285919988800040 0002004131038 00004 99880 -CH=C(Br)-CO-NH-i-C₃H₇, -CH=C(Br)-CO-NH-tert.-C₄H₉, -CH=C(Br)-CO-NH-cyclopropyl, -CH=C(Br)-CO-NH-cyclobutyl, -CH=C(Br)-CO-NH-cyclopentyl, -CH=C(Br)-CO-NH-cyclohexyl, -CH=C(Br)-CO-NH-cycloheptyl, -CH=C(Br)-CO-NH-cyclooctyl, -CH=C(Br)-CO-pyrrolidin-1-yl, -CH=C(Br)-CO-piperidin-1-yl, -CH=C(Br)-CO-morpholin-4-yl, -CH=C(Br)-CO-NH-CH₂CH=C(Br)₂, -CH=C(Br)-CO-NH-CH₂C≡CH, -CH=C(Br)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Br)-CO-NH-(CH₂)₂Cl, -CH=C(Br)-CO-NH-C₆H₅, -CH=C(CN)-CO-NH₂, -CH=C(CN)-CO-NHCH₃, -CH=C(CN)-CO-N(CH₃)₂, -CH=C(CN)-CO-NH-C₂H₅, -CH=C(CN)-CO-N(C₂H₅)₂, -CH=C(CN)-CO-NH-n-C₃H₇, -CH=C(CN)-CO-NH-i-C₃H₇, -CH=C(CN)-CO-NH-tert.-C₄H₉, -CH=C(CN)-CO-NH-cyclopropyl, -CH=C(CN)-CO-NH-cyclobutyl, -CH=C(CN)-CO-NH-cyclopentyl, -CH=C(CN)-CO-NH-cyclohexyl, -CH=C(CN)-CO-NH-cycloheptyl, -CH=C(CN)-CO-NH-cyclooctyl, -CH=C(CN)-CO-pyrrolidin-1-yl, -CH=C(CN)-CO-piperidin-1-yl, -CH=C(CN)-CO-morpholin-4-yl, -CH=C(CN)-CO-NH-CH₂CH=C(CN)₂, -CH=C(CN)-CO-NH-CH₂C≡CH, -CH=C(CN)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CN)-CO-NH-(CH₂)₂Cl, -CH=C(CN)-CO-NH-C₆H₅, -CH=CH-CO-SCH₃, -CH=CH-CO-SC₂H₅, -CH=CH-CO-S-n-C₃H₇, -CH=CH-CO-S-i-C₃H₇, -CH=CH-CO-S-n-C₄H₉, -CH=CH-CO-S-tert.-C₄H₉, -CH=C(CH₃)-CO-SCH₃, -CH=C(CH₃)-CO-SC₂H₅, -CH=C(CH₃)-CO-S-n-C₃H₇, -CH=C(CH₃)-CO-S-i-C₃H₇, -CH=C(CH₃)-CO-S-n-C₄H₉, -CH=C(CH₃)-CO-S-tert.-C₄H₉, -CH=C(C₂H₅)-CO-SCH₃, -CH=C(C₂H₅)-CO-SC₂H₅, -CH=C(C₂H₅)-CO-S-n-C₃H₇, -CH=C(C₂H₅)-CO-S-i-C₃H₇, -CH=C(C₂H₅)-CO-S-n-C₄H₉, -CH=C(C₂H₅)-CO-S-tert.-C₄H₉, -CH=C(Cl)-CO-SCH₃, -CH=C(Cl)-CO-SC₂H₅, -CH=C(Cl)-CO-S-n-C₃H₇, -CH=C(Cl)-CO-S-i-C₃H₇, -CH=C(Cl)-CO-S-n-C₄H₉, -CH=C(Cl)-CO-S-tert.-C₄H₉, -CH=C(Br)-CO-SCH₃, -CH=C(Br)-CO-SC₂H₅, -CH=C(Br)-CO-S-n-C₃H₇, -CH=C(Br)-CO-S-i-C₃H₇, -CH=C(Br)-CO-S-n-C₄H₉, -CH=C(Br)-CO-S-tert.-C₄H₉, -CH=C(CN)-CO-SCH₃, -CH=C(CN)-CO-SC₂H₅, -CH=C(CN)-CO-S-n-C₃H₇, -CH=C(CN)-CO-S-i-C₃H₇, -CH=C(CN)-CO-S-n-C₄H₉, -CH=C(CN)-CO-S-tert.-C₄H₉, -CH=C(COCH₃)-CO-OCH₃, -CH=C(COC₂H₅)-CO-OCH₃, -CH=C(CO-n-C₃H₇)-CO-OCH₃, -CH=C(COCH₃)-CO-OC₂H₅, -CH=C(COC₂H₅)-CO-OC₂H₅, -CH=C(CO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COCH₃)-CO-O-n-C₃H₇, -CH=C(COC₂H₅)-CO-O-n-C₃H₇, -CH=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-OCH₃, -CH=C(CF₃)-CO-OC₂H₅, -CH=C(CF₃)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-O-i-C₃H₇, -CH=C(CF₃)-CO-O-n-C₄H₉, -CH=C(CF₃)-CO-O-tert.-C₄H₉, -CH=C(COOCH₃)₂, -CH=C(COOC₂H₅)₂, -CH=C(COOCH₃)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)-CO-OCH₃, -CH=C(COO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)₂, -CH=CH-CH=CH-COOH, -CH=CH-CH=CH-CO-OCH₃, -CH=CH-CH=CH-CO-OC₂H₅, -CH=CH-CH=C(COOCH₃)₂, -CH=CH-CH=C(CN)-CO-OCH₃, -CH=CH-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-OCH₃, -CH=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CH=C(Cl)-CO-OCH₃, -CH=C(CH₃)-CH=C(Br)-CO-OCH₃, -CH=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-NH₂, -CH=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -CH=CH-(CH₂)₂-COOH, -CH=CH-(CH₂)₂-CO-OCH₃, -CH=CH-(CH₂)₂-CO-OC₂H₅, -CH=CH-CH₂-CH(COOCH₃)₂, -CH=CH-CH₂-CH(COOC₂H₅)₂, -CH=CH-CH₂-CH(CN)-CO-OCH₃, -CH=CH-CH₂-CH(CN)-CO-OC₂H₅, -CH=CH-CH₂-CH(CH₃)-CO-OCH₃, -CH=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -CH=CH-(CH₂)₂-CO-NH₂, -CH=CH-(CH₂)₂-CO-NH-CH₃, -CH=CH-CH₂-COOH, -CH=CH-CH₂-CO-OCH₃, -CH=CH-CH₂-CO-OC₂H₅, -CH=C(COOCH₃)-CH₂-CO-OCH₃, -CH=C(COOCH₃)-CH₂-CO-OC₂H₅, -CH=CH-CH₂-CO-NH₂, -CH=CH-CH₂-CO-NH-CH₃, -CH=CH-CH₂-CO-N(CH₃)₂, -CH(OCH₃)₂, -CH(SCH₃)₂, -CH(OC₂H₅)₂, -CH(SC₂H₅)₂, -CH(O-n-C₃H₇)₂, -CH(O-i-C₃H₇)₂, -CH(S-n-C₃H₇)₂, -CH(S-i-C₃H₇)₂, -CH(O-n-C₄H₉)₂, -CH(O-i-C₄H₉)₂, -CH(O-s-C₄H₉)₂, -CH(O-tert.-C₄H₉)₂, -CH(S-n-C₄H₉)₂, -CH(S-i-C₄H₉)₂, -CH(S-s-C₄H₉)₂, -CH(S-tert.-C₄H₉)₂, -CH(OC₅H₁₁)₂, 1,3-Dioxolan-2-yl, 1,3-Dithio­ lan-2-yl, 1,3-Oxathiolan-2-yl, 4-Methyl-1,3-dioxolan-2-yl, 4-Methyl-1,3-dithiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 5-Methyl-1,3-oxathiolan-2-yl, 4-Ethyl-1,3-dioxolan-2-yl, 4-Ethyl- 1,4-dithiolan-2-yl, 4-Ethyl-1,3-oxathiolan-2-yl, 5-Ethyl-1,3-oxa­ thiolan-2-yl, 4,5-Dimethyl-1,3-dioxolan-2-yl, 4,4-Dimethyl-1,3- dioxolan-2-yl, 4,5-Dimethyl-1,3-dithiolan-2-yl, 5,5-Dimethyl-1,3- dithiolan-2-yl, 4,5-Dimethyl-1,3-oxathiolan-2-yl, 5,5-Dimethyl- 1,3-oxathiolan-2-yl, 4,4-Dimethyl-1,3-oxathiolan-2-yl, 4-Vinyl- 1,3-dioxolan-2-yl, 4-Vinyl-1,3-dithiolan-2-yl, 4-Vinyl-1,3-oxa­ thiolan-2-yl, 5-Vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3- dioxolan-2-yl, 4-Chlormethyl-1,3-dithiolan-2-yl, 4-Chlormethyl- 1,3-oxathiolan-2-yl, 5-Chlormethyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-1,3-dithio­ lan-2-yl, 4-Hydroxymethyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl- 1,3-oxathiolan-2-yl, 4-Methoxymethyl-1,3-dioxolan-2-yl, 4-Allyl­ oxymethyl-1,3-dioxolan-2-yl, 4-Propargyloxymethyl-1,3-dioxolan- 2-yl, 4-Acetoxymethyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-1,3-dithiolan-2-yl, 4-Propargyl­ oxymethyl-1,3-dithiolan-2-yl, 4-Acetoxymethyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl-1,3-oxathiolan-2-yl, 5-Allyloxy­ methyl-1,3-oxathiolan-2-yl, 4-Propargyloxymethyl-1,3-oxathiolan-2-yl, 5-Propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxymethyl- 1,3-oxathiolan-2-yl, 5-Acetoxymethyl-1,3-oxathiolan-2-yl, 4-Methylthiomethyl-1,3-dioxolan-2-yl, 4-Methylthiomethyl-1,3- dithiolan-2-yl, 4-Carboxy-1,3-dioxolan-2-yl, 4-Carboxy-1,3- dithiolan-2-yl, 4-Methoxycarbonyl-1,3-dioxolan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-1,3-dithiolan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-4-methyl- 1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-di­ thiolan-2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-1,3- dithiolan-2-yl, 1,3-Dioxan-2-yl, 1,3-Dithian-2-yl, 1,3-Oxathian- 2-yl, 5-Methyl-1,3-dioxan-2-yl, 5-Methyl-1,3-dithian-2-yl, 5-Methyl-1,3-oxathian-2-yl, 5,5-Dimethyl-1,3-dioxan-2-yl, 4,6-Dimethyl- 1,3-dioxan-2-yl, 4,4-Dimethyl-1,3-dioxan-2-yl, 5,5-Dimethyl- 1,3-dithian-2-yl, 4,6-Dimethyl-1,3-dithian-2-yl, 4,4-Dimethyl- 1,3-dithian-2-yl, 5,5-Dimethyl-1,3-oxathian-2-yl, 4,4-Dimethyl- 1,3-oxathian-2-yl, 6,6-Dimethyl-1,3-oxathian-2-yl, 4-Hydroxymethyl-1,3-dioxan-2-yl, 4-Methoxymethyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-1,3-dithian-2-yl, 4-Methoxymethyl-1,3-dithian-2-yl, 4-Allyloxymethyl-1,3-dithian-2-yl, 4-Acetoxymethyl- 1,3-dithian-2-yl, 4-Chlormethyl-1,3-dioxan-2-yl, 4-Chlormethyl- 1,3-dithian-2-yl, 1,3-Dioxepan-2-yl, 1,3-Dithiepan-2-yl, 1,3-Dioxep-5-en-2-yl, 4-Methoxycarbonyl-1,3-dioxan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-1,3-dithian-2-yl, 4-n-Butoxycarbonyl-1,3-dithian-2-yl, 4-Methoxycarbonyl-4- methyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-Methoxy- carbonyl-4-methyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-4-methyl- 1,3-dithian-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithian-2-yl, -C(CH₃)(OCH₃)₂, -C(CH₃)(SCH₃)₂, -C(CH₃)(OC₂H₅)₂, -C(CH₃)(SC₂H₅)₂, -C(CH₃)(O-n-C₃H₇)₂, -C(CH₃)(O-i-C₃H₇)₂, -C(CH₃)(S-n-C₃H₇)₂, -C(CH₃)(S-i-C₃H₇)₂, -C(CH₃)(O-n-C₄H₉)₂, -C(CH₃)(O-i-C₄H₉)₂, -C(CH₃)(O-s-C₄H₉)₂, -C(CH₃)(O-tert.-C₄H₉)₂, -C(CH₃)(S-n-C₄H₉)₂, -C(CH₃)(S-i-C₄H₉)₂, -C(CH₃)(S-s-C₄H₉)₂, -C(CH₃)(S-tert.-C₄H₉)₂, -C(CH₃)(O-n-C₅H₁₁)′′, 2-Methyl-1,3-dioxolan-2-yl, 2-Methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-oxathiolan-2-yl, 2,4-Dimethyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-1,3- oxathiolan-2-yl, 2,5-Dimethyl-1,3-oxathiolan-2-yl, 4-Ethyl-2- methyl-1,3-dioxolan-2-yl, 4-Ethyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Ethyl-2-methyl-1,3- oxathiolan-2-yl, 2,4,5-Trimethyl-1,3-dioxolan-2-yl, 2,4,4-Trimethyl- 1,3-dioxolan-2-yl, 2,4,5-Trimethyl-1,3-dithiolan-2-yl, 2,4,4-Trimethyl-1,3-dithiolan-2-yl, 2,4,5-Trimethyl-1,3-oxathiolan-2-yl, 2,4,4-Trimethyl-1,3-oxathiolan-2-yl, 2-Methyl-4-vinyl- 1,3-dioxolan-2-yl, 2-Methyl-4-vinyl-1,3-dithiolan-2-yl, 2-Methyl- 4-vinyl-1,3-oxathiolan-2-yl, 2-Methyl-5-vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-dioxolan-2-yl, 4-Chlormethyl-2- methyl-1,3-dithiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl- 2-methyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-2- methyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dioxolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxy- 2-methyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dithiolan-2-yl, 4-Acetoxy-2- methyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl- 2-methyl-1,3-oxathiolan-2-yl, 5-Allyloxymethyl-2-methyl-1,3- oxathiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3- oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxy-2-methyl-1,3-oxathiolan-2-yl, 5-Acetoxy-2-methyl- 1,3-oxathiolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dioxolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-2- methyl-1,3-dioxolan-2-yl, 4-Carboxy-2-methyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-2- methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl- 2-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-2- methyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-ethoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4- ethoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-n-butoxy­ carbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl-1,3- dithiolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-dioxan-2-yl, 2-Methyl-1,3-dithian-2-yl, 2-Methyl-1,3-oxathian-2-yl, 2,5- Dimethyl-1,3-dioxan-2-yl, 2,5-Dimethyl-1,3-dithian-2-yl, 2,5-Dimethyl- 1,3-oxathian-2-yl, 2,5,5-Trimethyl-1,3-dioxan-2-yl, 2,4,6- Trimethyl-1,3-dioxan-2-yl, 2,2,4-Trimethyl-1,3-dioxan-2-yl, 2,5,5-Trimethyl-1,3-dithian-2-yl, 2,4,6-Trimethyl-1,3-dithian-2-yl, 2,4,4-Trimethyl-1,3-dithian-2-yl, 2,5,5-Trimethyl-1,3-oxathian-2-yl, 2,4,4-Trimethyl-1,3-oxathian-2-yl, 2,6,6-Trimethyl- 1,3-oxathian-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-2- methyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dithian-2-yl, 4-Methoxymethyl-2- methyl-1,3-dithian-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithian-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dithian-2-yl, 4-Chlormethyl-2- methyl-1,3-dioxan-2-yl, 4-Chlormethyl-2-methyl-1,3-dithian-2-yl, -C(CH₃)=NH, -C(CH₃)=N-CH₃, -C(CH₃)=N-C₂H₅, -C(CH₃)=N-n-C₃H₇, -C(CH₃)=N-i-C₃H₇, -C(CH₃)=N-n-C₄H₉, -C(CH₃)=N-CH₂CH=CH₂, -C(CH₃)=N-CH₂CH=CH₂-CH₃, -C(CH₃)=N-CH₂C≡CH, -C(CH₃)=N-CH₂C≡C-CH₃, -C(CH₃)=N-cyclopropyl, -C(CH₃)=N-cyclobutyl, -C(CH₃)=N-cyclopentyl, -C(CH₃)=N-cyclohexyl, -C(CH₃)=N-cycloheptyl, -C(CH₃)=N-CH₂-CH₂Cl, -C(CH₃)=N-CH₂Cl, -C(CH₃)=N-C₆H₅, -C(CH₃)=N-(2-F-C₆H₄), -C(CH₃)=N-(3-F-C₆H₄), -C(CH₃)=N-(4-F-C₆H₄), -C(CH₃)=N-(2-Cl-C₆H₄), -C(CH₃)=N-(3-Cl-C₆H₄), -C(CH₃)=N-(4-Cl-C₆H₄), -C(CH₃)=N-(2-CH₃-C₆H₄), -C(CH₃)=N-(3-CH₃-C₆H₄), -C(CH₃)=N-(4-CH₃-C₆H₄), -C(CH₃)=N-(2-CF₃-C₆H₄), -C(CH₃)=N-(3-CF₃-C₆H₄), -C(CH₃)=N-(4-CF₃-C₆H₄), -C(CH₃)=N-(2-OCH₃-C₆H₄), -C(CH₃)=N-(3-OCH₃-C₆H₄), -C(CH₃)=N-(4-OCH₃-C₆H₄), -C(CH₃)=N-(4-NO₂-C₆H₄), -C(CH₃)=N-(4-CN-C₆H₄), -C(CH₃)=N-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-(2,4-(CH₃)₂-C₆H₃), -C(CH₃)=N-CH₂-OCH₃, -C(CH₃)=N-CH₂-OC₂H₅, -C(CH₃)=N-CH₂CH₂-OCH₃, -C(CH₃)=N-CH₂CH₂-OC₂H₅, -C(CH₃)=N-OH, -C(CH₃)=N-OCH₃, -C(CH₃)=N-OC₂H₅, -C(CH₃)=N-O-n-C₃H₇, -C(CH₃)=N-O-i-C₃H₇, -C(CH₃)=N-O-n-C₄H₉, -C(CH₃)=N-O-i-C₄H₉, -C(CH₃)=N-O-s-C₄H₉, -C(CH₃)=N-O-tert.-C₄H₉, -C(CH₃)=N-OCH₂-CH=CH₂, -C(CH₃)=N-OCH(CH₃)-CH=CH₂, -C(CH₃)=N-OCH₂-C≡CH, -C(CH₃)=N-CH(CH₃)-C≡CH, -C(CH₃)=N-OCH₂-CH=C-CH₃, -C(CH₃)=N-OCH₂CH₂-Cl, -C(CH₃)=N-OCH₂CH₂-F, -C(CH₃)=N-OCH₂-CF₃, -C(CH₃)=N-OCH₂-CH=CHCl, -C(CH₃)=N-OCH₂-C(Cl)=CH₂, -C(CH₃)=N-OCH₂-C(Br)=CH₂, -C(CH₃)=N-OCH₂-CH=C(Cl)-CH₃, -C(CH₃)=N-O-CO-CH₃, -C(CH₃)=N-O-CO-C₂H₅, -C(CH₃)=N-OCH₂-CN, -C(CH₃)=N-OCH₂-CH=CH-CH₂-OCH₃, -C(CH₃)=N-OCH₂-CH=CH-CH₂-O-tert.-C₄H₉, -C(CH₃)=N-O-(CH₂)₃-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-(4-Cl-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-C₆H₅, -C(CH₃)=N-OCH₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(3-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-CH₂-(4-CH₃O-C₆H₄), -C(CH₃)=N-OCH₂-CH=C(CH₃)-C₆H₅, -C(CH₃)=N-O-(CH₂)₂-CH=CH-(3,4-Cl₂-C₆H₃), -C(CH₃)=N-O-(CH₂)₃-C≡C-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-OCH₃, -C(CH₃)=N-OCH₂CH₂-OCH₃, -C(CH₃)=N-OCH₂-OC₂H₅, -C(CH₃)=N-OCH(CH₃)-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=N-NH₂, -C(CH₃)=N-NH-CH₃, -C(CH₃)=N-NH-C₂H₅, -C(CH₃)=N-NH-n-C₃H₇, -C(CH₃)=N-NH-i-C₃H₇, -C(CH₃)=N-NH-n-C₄H₉, -C(CH₃)=N-NH-i-C₄H₉, -C(CH₃)=N-NH-s-C₄H₉, -C(CH₃)=N-NH-tert.-C₄H₉, -C(CH₃)=N-NH-cyclopropyl, -C(CH₃)=N-NH-cyclobutyl, -C(CH₃)=N-NH-cyclopentyl, -C(CH₃)=N-NH-cyclohexyl, -C(CH₃)=N-NH-cycloheptyl, -C(CH₃)=N-N(CH₃)₂, -C(CH₃)=N-N(C₂H₅)₂, -C(CH₃)=N-N(n-C₃H₇)₂, -C(CH₃)=N-N(i-C₃H₇)₂, -C(CH₃)=N-NH-CH₂-C=CH, -C(CH₃)=N-NH-CH₂-C≡CH, -C(CH₃)=N-N(CH₃)-CH₂-C≡CH, -C(CH₃)=N-NH-CH₂CF₃, -C(CH₃)=N-NH-CO-CH₃, -C(CH₃)=N-NH-CO-C₂H₅, -C(CH₃)=N-NH-CO-OCH₃, -C(CH₃)=N-NH-CO-OC₂H₅, -C(CH₃)=N-NH-CO-O-tert.-C₄H₉, -C(CH₃)=N-pyrrolidin-1-yl, -C(CH₃)=N-piperidin-1-yl, -C(CH₃)=N-morpholin-4-yl, -C(CH₃)=N-NH-C₆H₅, -C(CH₃)=N-NH-(4-Cl-C₆H₄), -C(CH₃)=N-NH-(4-NO₂-C₆H₄), -C(CH₃)=N-NH-(4-F-C₆H₄), -C(CH₃)=N-NH-(4-CH₃O-C₆H₄), -C(CH₃)=N-NH-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-NH-(2,4-(NO₂)₂-C₆H₃), -C(CH₃)=N-NH-CO-NH₂, -C(CH₃)=N-NH-CO-NHCH₃, -C(CH₃)=N-NH-CO-NHC₂H₅, -C(CH₃)=N-NH-CO-N(CH₃)₂, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=CH-CO-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-O-n-C₄H₉, -C(CH₃)=CH-CO-O-tert.-C₄H₉, -C(CH₃)=CH-CO-O-cyclopropyl, -C(CH₃)=CH-CO-O-cyclobutyl, -C(CH₃)=CH-CO-O-cyclopentyl, -C(CH₃)=CH-CO-O-cyclohexyl, -C(CH₃)=CH-CO-O-cycloheptyl, -C(CH₃)=C(CH₃)-COOH, -C(CH₃)=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-cyclopropyl, -C(CH₃)=C(CH₃)-CO-O-cyclobutyl, -C(CH₃)=C(CH₃)-CO-O-cyclopentyl, -C(CH₃)=C(CH₃)-CO-O-cyclohexyl, -C(CH₃)=C(CH₃)-CO-O-cycloheptyl, -C(CH₃)=C(C₂H₅)-COOH, -C(CH₃)=C(C₂H₅)-CO-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-cyclo­ propyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-O- cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-O-cycloheptyl, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=C(Cl)-CO-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-O-n-C₄H₉, -C(CH₃)=C(Cl)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-O-cyclopropyl, -C(CH₃)=C(Cl)-CO-O-cyclobutyl, -C(CH₃)=C(Cl)-CO-O-cyclopentyl, -C(CH₃)=C(Cl)-CO-O-cyclohexyl, -C(CH₃)=C(Cl)-CO-O-cycloheptyl, -C(CH₃)=C(Br)-COOH, -C(CH₃)=C(Br)-CO-OCH₃, -C(CH₃)=C(Br)-CO-OC₂H₅, -C(CH₃)=C(Br)-CO-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-O-n-C₄H₉, -C(CH₃)=C(Br)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-O-cyclopropyl, -C(CH₃)=C(Br)-CO-O-cyclobutyl, -C(CH₃)=C(Br)-CO-O-cyclopentyl, -C(CH₃)=C(Br)-CO-O-cyclohexyl, -C(CH₃)=C(Br)-CO-O-cycloheptyl, -C(CH₃)=C(CN)-COOH, -C(CH₃)=C(CN)-CO-OCH₃, -C(CH₃)=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CN)-CO-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-O-n-C₄H₉, -C(CH₃)=C(CN)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-O-cyclopropyl, -C(CH₃)=C(CN)-CO-O-cyclobutyl, -C(CH₃)=C(CN)-CO-O-cyclopentyl, -C(CH₃)=C(CN)-CO-O-cyclohexyl, -C(CH₃)=C(CN)-CO-O-cycloheptyl, -C(CH₃)=CH-CO-OCH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=CH-CO-O-i-C₃H₇, -C(CH₃)=CH-CO-OCH(CH₃)-OCH₃, -C(CH₃)=CH-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=CH-CO-OCH₂CH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-O-i-C₃H₇, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-O-i-C₃H₇, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-O-i-C₃H₇, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-CF₃, -C(CH₃)=CH-CO-OCH₂-CCl₃, -C(CH₃)=CH-CO-OCH₂-oxiranyl, -C(CH₃)=CH-CO-(CH₂)₃-Br,-C(CH₃)=CH-CO-OCH₂-CH=CH₂, -C(CH₃)=CH-CO-OCH₂-C≡CH, -C(CH₃)=CH-CO-OCH₂-CN, -C(CH₃)=CH-CO-OCH₂CH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CF₃, -C(CH₃)=C(CH₃)-CO-OCH₂-CCl₃, -C(CH₃)=C(CH₃)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CH₃)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(CH₃)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CH₃)-CO-OCH₂-C≡CH, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CF₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CCl₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-oxiranyl, -C(CH₃)=C(C₂H₅)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(C₂H₅)-CO-OCH₂-C≡CH, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂-CF₃, -C(CH₃)=C(Cl)-CO-OCH₂-CCl₃, -C(CH₃)=C(Cl)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Cl)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Cl)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Cl)-CO-OCH₂-C≡CH, -C(CH₃)=C(Cl)-CO-OCH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂-CF₃, -C(CH₃)=C(Br)-CO-OCH₂-CCl₃, -C(CH₃)=C(Br)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Br)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Br)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Br)-CO-OCH₂-C≡CH, -C(CH₃)=C(Br)-CO-OCH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂CH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂-CF₃, -C(CH₃)=C(CN)-CO-OCH₂-CCl₃, -C(CH₃)=C(CN)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CN)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(CN)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CN)-CO-OCH₂-C≡CH, -C(CH₃)=C(CN)-CO-OCH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂CH₂-CN, -C(CH₃)=CH-CO-CH₃, -C(CH₃)=CH-CO-C₂H₅, -C(CH₃)=CH-CO-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-n-C₄H₉, -C(CH₃)=CH-CO-tert.-C₄H₉, -C(CH₃)=CH-CO-CH₂Cl, -C(CH₃)=CH-CO-CH₂Br, -C(CH₃)=CH-CO-CHCl₂, -C(CH₃)=CH-CO-CH₂-OCH₃, -C(CH₃)=CH-CO-CH(OCH₃)₂, -C(CH₃)=CH-CO-CH₂-SCH₃, -C(CH₃)=C(CH₃)-CO-CH₃, -C(CH₃)=C(CH₃)-CO-C₂H₅, -C(CH₃)=C(CH₃)-CO-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-CH₂Cl -C(CH₃)=C(CH₃)-CO-CH₂Br, -C(CH₃)=C(CH₃)-CO-CHCl₂, -C(CH₃)=C(CH₃)-CO-CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-CH(OCH₃)₂, -C(CH₃)=C(CH₃)-CO-CH₂-SCH₃, -C(CH₃)=C(C₂H₅)-CO-CH₃, -C(CH₃)=C(C₂H₅)-CO-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-CHCl, -C(CH₃)=C(C₂H₅)-CO-CH₂Br, -C(CH₃)=C(C₂H₅)-CO-CH₂Cl₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-CH(OCH₃)₂ -C(CH₃)=C(C₂H₅)-CO-CH₂-SCH₃, -C(CH₃)=C(Cl)-CO-CH₃, -C(CH₃)=C(Cl)-CO-C₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-n-C₄H₉, -C(CH₃)=C(Cl)-CO-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-CH₂Cl, -C(CH₃)=C(Cl)-CO-CHCl₂, -C(CH₃)=C(Cl)-CO-CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-CH(OCH₃)₂, -C(CH₃)=C(Cl)-CO-CH₂-SCH₃, -C(CH₃)=C(Br)-CO-CH₃, -C(CH₃)=C(Br)-CO-C₂H₅, -C(CH₃)=C(Br)-CO-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-n-C₄H₉, -C(CH₃)=C(Br)-CO-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-CH₂Cl, -C(CH₃)=C(Br)-CO-CH₂Br, -C(CH₃)=C(Br)-CO-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-CH(OCH₃)₂, -C(CH₃)=C(Br)-CO-CH₂-SCH₃, -C(CH₃)=C(CN)-CO-CH₃, -C(CH₃)=C(CN)-CO-C₂H₅, -C(CH₃)=C(CN)-CO-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-n-C₄H₉, -C(CH₃)=C(CN)-CO-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-CH₂Cl, -C(CH₃)=C(CN)-CO-CH₂Br, -C(CH₃)=C(CN)-CO-CHCl₂, -C(CH₃)=C(CN)-CO-CH₂-OCH₃, -C(CH₃)=C(CN)-CO-CH(OCH₃)₂, -C(CH₃)=C(CN)-CO-CH₂-SCH₃, -C(CH₃)=CH-CO-C₆H₅, -C(CH₃)=CH-CO-(4-Cl-C₆H₄), -C(CH₃)=C(CH₃)-CO-C₆H₅, -C(CH₃)=C(CH₃)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(C₂H₅)-CO-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(Cl)-CO-C₆H₅, -C(CH₃)=C(Br)-CO-C₆H₅, -C(CH₃)=C(CN)-CO-C₆H₅, -C(CH₃)=CH-CO-NH₂, -C(CH₃)=CH-CO-NHCH₃, -C(CH₃)=CH-CO-N(CH₃)₂, -C(CH₃)=CH-CO-NH-C₂H₅, -C(CH₃)=CH-CO-N(C₂H₅)₂, -C(CH₃)=CH-CO-NH-n-C₃H₇, -C(CH₃)=CH-CO-NH-i-C₃H₇, -C(CH₃)=CH-CO-NH-tert.-C₄H₉, -C(CH₃)=CH-CO-NH-cyclopropyl, -C(CH₃)=CH-CO-NH-cyclobutyl, -C(CH₃)=CH-CO-NH-cyclopentyl, -C(CH₃)=CH-CO-NH-cyclohexyl, -C(CH₃)=CH-CO-NH-cycloheptyl, -C(CH₃)=CH-CO-NH-cyclooctyl, -C(CH₃)=CH-CO-pyrrolidin-1-yl, -C(CH₃)=CH-CO-piperidin-1-yl, -C(CH₃)=CH-CO-morpholin-4-yl, -C(CH₃)=CH-CO-NH-CH₂CH=CH₂, -C(CH₃)=CH-CO-NH-CH₂C≡CH, -C(CH₃)=CH-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=CH-CO-NH-(CH₂)₂Cl, -C(CH₃)=CH-CO-NH-C₆H₅, -C(CH₃)=C(CH₃)-CO-NH₂, -C(CH₃)=C(CH₃)-CO-NHCH₃, -C(CH₃)=C(CH₃)-CO-N(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-C₂H₅, -C(CH₃)=C(CH₃)-CO-N(C₂H₅)₂, -C(CH₃)=C(CH₃)-CO-NH-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-NH- cyclopropyl, -C(CH₃)=C(CH₃)-CO-NH-cyclobutyl, -C(CH₃)=C(CH₃)-CO-NH-cyclopentyl, -C(CH₃)=C(CH₃)-CO-NH- cyclohexyl, -C(CH₃)=C(CH₃)-CO-NH-cycloheptyl, -C(CH₃)=C(CH₃)-CO-NH-cyclooctyl, -C(CH₃)=C(CH₃)-CO- pyrrolidin-1-yl, -C(CH₃)=C(CH₃)-CO-piperidin-1-yl, -C(CH₃)=C(CH₃)-CO-morpholin-4-yl, -C(CH₃)=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CH₃)-CO-NH-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-NH₂, -C(CH₃)=C(C₂H₅)-CO-NHCH₃, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)₂, -C(CH₃)=C(C₂H₅)-CO-NH-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-N(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-NH- cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-NH-cycloheptyl, -C(CH₃)=C(C₂H₅)-CO-NH- cyclooctyl, -C(CH₃)=C(C₂H₅)-CO-pyrrolidin-1-yl, -C(CH₃)=C(C₂H₅)-CO-piperidin-1-yl, -C(CH₃)=C(C₂H₅)-CO- morpholin-4-yl, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(C₂H₅)-CO-NH-C₆H₅, -C(CH₃)=C(Cl)-CO-NH₂, -C(CH₃)=C(Cl)-CO-NHCH₃, -C(CH₃)=C(Cl)-CO-N(CH₃)₂, -C(CH₃)=C(Cl)-CO-NH-C₂H₅, -C(CH₃)=C(Cl)-CO-N(C₂H₅)₂, -C(CH₃)=C(Cl)-CO-NH-n-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-i-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-NH-cyclopropyl, -C(CH₃)=C(Cl)-CO-NH-cyclobutyl, -C(CH₃)=C(Cl)-CO-NH-cyclopentyl, -C(CH₃)=C(Cl)-CO-NH-cyclohexyl, -C(CH₃)=C(Cl)-CO-NH-cycloheptyl, -C(CH₃)=C(Cl)-CO-NH-cyclooctyl, -C(CH₃)=C(Cl)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Cl)-CO-piperidin-1- yl, -C(CH₃)=C(Cl)-CO-morpholin-4-yl, -C(CH₃)=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -C(CH₃)=C(Cl)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Cl)-CO-NH-C₆H₅, -C(CH₃)=C(Br)-CO-NH₂, -C(CH₃)=C(Br)-CO-NHCH₃, -C(CH₃)=C(Br)-CO-N(CH₃)₂, -C(CH₃)=C(Br)-CO-NH-C₂H₅, -C(CH₃)=C(Br)-CO-N(C₂H₅)₂, -C(CH₃)=C(Br)-CO-NH-n-C₃H₇, -C(CH₃)=C(Br)-CO-NH-i-C₃H₇, -C(CH₃)=C(Br)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-NH-cyclopropyl, -C(CH₃)=C(Br)-CO-NH-cyclobutyl, -C(CH₃)=C(Br)-CO-NH-cyclopentyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cycloheptyl, -C(CH₃)=C(Br)-CO-NH-cyclooctyl, -C(CH₃)=C(Br)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Br)-CO-piperidin-1-yl, -C(CH₃)=C(Br)-CO-morpholin-4-yl, -C(CH₃)=C(Br)-CO-NH-CH₂CH=C(Br)₂, -C(CH₃)=C(Br)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Br)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Br)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Br)-CO-NH-C₆H₅, -C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CN)-CO-NHCH₃, -C(CH₃)=C(CN)-CO-N(CH₃)₂, -C(CH₃)=C(CN)-CO-NH-C₂H₅, -C(CH₃)=C(CN)-CO-N(C₂H₅)₂, -C(CH₃)=C(CN)-CO-NH-n-C₃H₇, -C(CH₃)=C(CN)-CO-NH-i-C₃H₇, -C(CH₃)=C(CN)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-NH-cyclopropyl, -C(CH₃)=C(CN)-CO-NH-cyclobutyl, -C(CH₃)=C(CN)-CO-NH-cyclopentyl, -C(CH₃)=C(CN)-CO-NH-cyclohexyl, -C(CH₃)=C(CN)-CO-NH-cycloheptyl, -C(CH₃)=C(CN)-CO-NH-cyclooctyl, -C(CH₃)=C(CN)-CO-pyrrolidin-1-yl, -C(CH₃)=C(CN)-CO-piperidin-1-yl, -C(CH₃)=C(CN)-CO-morpholin-4-yl, -C(CH₃)=C(CN)-CO-NH-CH₂CH=C(CN)₂, -C(CH₃)=C(CN)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CN)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CN)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CN)-CO-NH-C₆H₅, -C(CH₃)=CH-CO-SCH₃, -C(CH₃)=CH-CO-SC₂H₅, -C(CH₃)=CH-CO-S-n-C₃H₇, -C(CH₃)=CH-CO-S-i-C₃H₇, -C(CH₃)=CH-CO-S-n-C₄H₉, -C(CH₃)=CH-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-SCH₃, -C(CH₃)=C(CH₃)-CO-SC₂H₅, -C(CH₃)=C(CH₃)-CO-S-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-S-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-SCH₃, -C(CH₃)=C(C₂H₅)-CO-SC₂H₅, -C(CH₃)=C(C₂H₅)-CO-S-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-SCH₃, -C(CH₃)=C(Cl)-CO-SC₂H₅, -C(CH₃)=C(Cl)-CO-S-n-C₃H₇, -C(CH₃)=C(Cl)-CO-S-i-C₃H₇, -C(CH₃)=C(Cl)-CO-S-n-C₄H₉, -C(CH₃)=C(Cl)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-SCH₃, -C(CH₃)=C(Br)-CO-SC₂H₅, -C(CH₃)=C(Br)-CO-S-n-C₃H₇, -C(CH₃)=C(Br)-CO-S-i-C₃H₇, -C(CH₃)=C(Br)-CO-S-n-C₄H₉, -C(CH₃)=C(Br)-CO-S-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-SCH₃, -C(CH₃)=C(CN)-CO-SC₂H₅, -C(CH₃)=C(CN)-CO-S-n-C₃H₇, -C(CH₃)=C(CN)-CO-S-i-C₃H₇, -C(CH₃)=C(CN)-CO-S-n-C₄H₉ -C(CH₃)=C(CN)-CO-S-tert.-C₄H₉, -C(CH₃)=C(COCH₃)-CO-OCH₃, -C(CH₃)=C(COC₂H₅)-CO-OCH₃, -C(CH₃)=C(CO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COCH₃)-CO-OC₂H₅, -C(CH₃)=C(COC₂H₅)-CO-OC₂H₅, -C(CH₃)=C(CO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COCH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(COC₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-OCH₃, -C(CH₃)=C(CF₃)-CO-OC₂H₅, -C(CH₃)=C(CF₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CF₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(COOCH₃)₂, -C(CH₃)=C(COOC₂H₅)₂, -C(CH₃)=C(COOCH₃)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)₂, -C(CH₃)=CH-CH=CH-COOH, -C(CH₃)=CH-CH=CH-CO-OCH₃, -C(CH₃)=CH-CH=CH-CO-OC₂H₅, -C(CH₃)=CH-CH=C(COOCH)₃)₂, -C(CH₃)=CH-CH=C(CN)-CO-OCH₃, -C(CH₃)=CH-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH₂, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -C(CH₃)=CH-(CH₂)₂-COOH, -C(CH₃)=CH(CH₂)₂-CO-OCH₃, -C(CH₃)=CH-(CH₂)₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(COOCH₃)₂, -C(CH₃)=CH-CH₂-CH(COOC₂H₅)₂, -C(CH₃)=CH-CH₂-CH(CN)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CN)-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -C(CH₃)=CH-(CH₂)₂-CO-NH₂, -C(CH₃)=CH-(CH₂)₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-COOH, -C(CH₃)=CH-CH₂-CO-OCH₃, -C(CH₃)=CH-CH₂-CO-OC₂H₅, -C(CH₃)=C(COOCH₃)-CH₂-CO-OCH₃, -C(CH₃)=CH-(COOCH₃)-CH₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CO-NH₂, -C(CH₃)=CH-CH₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-CO-N(CH₃)₂.
wobei W für eine der folgenden Bedeutungen steht:
-CHO, -COCH₃, -COC₂H₅, -CO-n-C₃H₇, -CO-i-C₃H₇, -CO-n-C₄H₉, -CO-i-C₄H₉, -CO-s-C₄H₉, -CO-tert.-C₄H₉, -CO-CH₂CH=CH₂, -CO-CF₃, -COCCl₃, -COCH₂C≡CH, -CO-cyclopropyl, -CO-cyclobutyl, -CO-cyclopentyl, -CO-cyclohexyl, -CO-CN, -CO-COOCH₃, -CO-COOC₂H₅, -CH=NH, -CH=NCH₃, -CH=NC₂H₅, -CH=N-n-C₃H₅, -CH=N-i-C₃H₅, -CH=N-n-C₄H₉, -CH=NCH₂CH=CH₂, -CH=NCH₂CH=CH₂-CH₃, -CH=NCH₂C≡CH, -CH=NCH₂C≡C-CH₃, -CH=N-cyclopropyl, -CH=N-cyclobutyl, -CH=N-cyclopentyl, -CH=N-cyclohexyl, -CH=N-cycloheptyl, -CH=N-CH₂-CH₂Cl, -CH=N-CH₂Cl, -CH=N-C₆H₅, -CH=N-4-Br-C₆H₄, -CH=N-3-F-C₆H₄, -CH=N-4-F-C₆H₄, -CH=N-2-Cl-C₆H₄, -CH=N-3-Cl-C₆H₄, -CH=N-4-Cl-C₆H₄, -CH=N-2-Br-C₆H₄, -CH=N-2-F-C₆H₄, -CH=N-2-CH₃-C₆H₄, -CH=N-3-CH₃-C₆H₄, -CH=N-4-CH₃-C₆H₄, -CH=N-2-CF₃-C₆H₄, -CH=N-3-CF₃-C₆H₄, -CH=N-4-CF₃-C₆H₄, -CH=N-2-OCH₃-C₆H₄, -CH=N-3-OCH₃-C₆H₄, -CH=N-4-OCH₃-C₆H₄, -CH=N-4-NO₂-C₆H₄, -CH=N-4-CN-C₆H₄, -CH=N-2,4-(Cl,Cl)-C₆H₄, -CH=N-2,4-(CH₃,CH₃)-C₆H₄, -CH=N-CH₂OCH₃ -CH=N-CH₂OC₂H₅, -CH=N-CH₂CH₂OCH₃, -CH=N-CH₂CH₂OC₂H₅, -CH=N-OH, -CH=N-OCH₃, -CH=N-OC₂H₅, -CH=N-O-n-C₃H₇, -CH=N-O-i-C₃H₇, -CH=N-O-n-C₄H₉, -CH=N-O-i-C₄H₉, -CH=N-O-s-C₄H₉, -CH=N-O-tert.-C₄H₉, -CH=N-O-CH₂CH=CH₂, -CH=N-O-CH(CH₃)CH=CH₂, -CH=N-O-CH₂C≡CH, -CH=N-O-CH(CH₃)-C≡CH, -CH=N-O-CH₂-CH=CH-CH₃, -CH=N-O-CH₂-CH₂-Cl, -CH=N-O-CH₂-CH₂-F, -CH=N-O-CH₂-CF₃, -CH=N-O-CH₂-CH=CHCl, -CH=N-O-CH₂-CCl=CH₂, -CH=N-O-CH₂-CBr=CH₂, -CH=N-O-CH₂-CH=CCl-CH₃, -CH=N-OC(O)CH₃, -CH=N-OC(O)C₂H₅, -CH=N-O-CH₂-CN, -CH=N-O-CH₂-CH=CH-CH₂-O-CH₃, -CH=N-O-CH₂-CH=CH-CH₂-O-tert.-C₄H₉, -CH=N-O-(CH₂)₃-C₆H₅, -CH=N-O-(CH₂)₄-C₆H₅, -CH=N-O-(CH₂)₄-4-Cl-C₆H₄, -CH=N-O-(CH₂)₄-4-OCH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-CH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-C₆H₅, -CH=N-O-CH₂CH=CH-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CH-3-OCH₃-C₆H₄, -CH=N-O-(CH₂)₂CH=CH-4-F-C₆H₄, -CH=N-O-(CH₂)CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CHCH₂-4-OCH₃-C₆H₄, -CH=N-O-CH₂-CH=C(CH₃)-C₆H₅, -CH=N-O-(CH₂)₂CH=CH-3,4(Cl,Cl)-C₆H₃, -CH=N-O-(CH₂)₃C≡C-4-F-C₆H₄, -CH₂=N-OCHOCH₃, -CH=N-OC₂H₄OCH₃, -CH=N-OCH₂OC₂H₅, -CH=N-OCH(CH₃)OCH₃, -CH=N-OCH(CH₃)COOCH₃, -CH=N-OCH(CH₃)COO-n-C₄H₉, -CH=N-NH₂, -CH=N-NHCH₃, -CH=N-NHC₂H₅, -CH=N-NH-n-C₃H₇, -CH=N-NH-i-C₃H₇, -CH=N-NH-n-C₄H₉, -CH=N-NH-i-C₄H₉, -CH=N-NH-s-C₄H₈, -CH=N-NH-tert.-C₄H₉, -CH=N-NH-cyclopropyl, -CH=N-NH-cyclobutyl, -CH=N-NH-cyclopentyl, -CH=N-NH-cyclohexyl, -CH=N-NH-cycloheptyl, -CH=N-N(CH₃)₂, -CH=N-N(C₂H₅)₂, -CH=N-N(C₃H₇)₂, -CH=N-N(i-C₃H₇)(CH₃), -CH=N-NHCH₂-C=CH, -CH=N-NHCH₂-C≡CH, -CH=N-N(CH₃)-CH₂-C≡CH, -CH=N-NHCH₂CF₃, -CH=N-NH-CO-CH₃, -CH=N-NH-CO-CH₂H₅, -CH=N-NH-COOCH₃, -CH=N-NH-COOC₂H₅, -CH=N-NH-COO-tert.-C₄H₉, -CH=N-pyrrolidin-1-yl, -CH=N-piperidin-1-yl, -CH=N-morpholin-4-yl, -CH=N-NH-C₆H₅, -CH=N-NH-(4-Cl-C₆H₄), -CH=N-NH-(4-NO₂-C₆H₄), -CH=N-NH-(4-F-C₆H₄), -CH=N-NH-(4-CH₃O-C₆H₄), -CH=N-NH-(2,4-Cl₂-C₆H₃), -CH=N-NH-(2,4-(NO₂)₂-C₆H₃), -CH=N-NH-CO-NH₂, -CH=N-NH-CO-NHCH₃, -CH=N-NH-CO-NHC₂H₅, -CH=N-NH-CO-N(CH₃)₂, -CH=CH-COOH, -CH=CH-CO-OCH₃, -CH=CH-CO-OC₂H₅, -CH=CH-CO-O-n-C₃H₇, -CH=CH-CO-O-i-C₃H₇, -CH=CH-CO-O-n-C₄H₉, -CH=CH-CO-O-tert.-C₄H₉, -CH=CH-CO-O-cyclopropyl, -CH=CH-CO-O-cyclobutyl, -CH=CH-CO-O-cyclopentyl, -CH=CH-CO-O-cyclohexyl, -CH=CH-CO-O-cycloheptyl, -CH=C(CH₃)-COOH, -CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CO-O-n-C₃H₇, -CH=C(CH₃)-CO-O-i-C₃H₇, -CH=C(CH₃)-CO-O-n-C₄H₉, -CH=C(CH₃)-CO-O-tert.-C₄H₉, -CH=C(CH₃)-CO-O-cyclopropyl, -CH=C(CH₃)-CO-O-cyclobutyl, -CH=C(CH₃)-CO-O-cyclopentyl, -CH=C(CH₃)-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cycloheptyl, -CH=C(C₂H₅)-COOH, -CH=C(C₂H₅)-CO-OCH₃, -CH=C(C₂H₅)-CO-OC₂H₅, -CH=C(C₂H₅)-CO-O-n-C₃H₇, -CH=C(C₂H₅)-CO-O-i-C₃H₇, -CH=C(C₂H₅)-CO-O-n-C₄H₉, -CH=C(C₂H₅)-CO-O-tert.-C₄H₉, -CH=C(C₂H₅)-CO-O-cyclopropyl, -CH=C(C₂H₅)-CO-O-cyclobutyl, -CH=C(C₂H₅)-CO-O-cyclopentyl, -CH=C(C₂H₅)-CO-O-cyclohexyl, -CH=C(C₂H₅)-CO-O-cycloheptyl, -CH=C(Cl)-COOH, -CH=C(Cl)-CO-OCH₃, -CH=C(Cl)-CO-OC₂H₅, -CH=C(Cl)-CO-O-n-C₃H₇, -CH=C(Cl)-CO-O-i-C₃H₇, -CH=C(Cl)-CO-O-n-C₄H₉, -CH=C(Cl)-CO-O-tert.-C₄H₉, -CH=C(Cl)-CO-O-cyclopropyl, -CH=C(Cl)-CO-O-cyclobutyl, -CH=C(Cl)-CO-O-cyclopentyl, -CH=C(Cl)-CO-O-cyclohexyl, -CH=C(Cl)-CO-O-cycloheptyl, -CH=C(Br)-COOH, -CH=C(Br)-CO-OCH₃, -CH=C(Br)-CO-OC₂H₅, -CH=C(Br)-CO-O-n-C₃H₇, -CH=C(Br)-CO-O-i-C₃H₇, -CH=C(Br)-CO-O-n-C₄H₉, -CH=C(Br)-CO-O-tert.-C₄H₉, -CH=C(Br)-CO-O-cyclopropyl, -CH=C(Br)-CO-O-cyclobutyl, -CH=C(Br)-CO-O-cyclopentyl, -CH=C(Br)-CO-O-cyclohexyl, -CH=C(Br)-CO-O-cycloheptyl, -CH=C(CN)-COOH, -CH=C(CN)-CO-OCH₃, -CH=C(CN)-CO-OC₂H₅, -CH=C(CN)-CO-O-n-C₃H₇, -CH=C(CN)-CO-O-i-C₃H₇, -CH=C(CN)-CO-O-n-C₄H₉, -CH=C(CN)-CO-O-tert.-C₄H₉, -CH=C(CN)-CO-O-cyclopropyl, -CH=C(CN)-CO-O-cyclobutyl, -CH=C(CN)-CO-O-cyclopentyl, -CH=C(CN)-CO-O-cyclohexyl, -CH=C(CN)-CO-O-cycloheptyl, -CH=CH-CO-OCH₂-OCH₃, -CH=CH-CO-OCH₂-OC₂H₅, -CH=CH-CO-OCH₂-O-n-C₃H₅, -CH=CH-CO-OCH₂-O-i-C₃H₅, -CH=CH-CO-OCH(CH₃)-OCH₃, -CH=CH-CO-OCH(CH₃)-OC₂H₅, -CH=CH-CO-O-CH₂CH₂-OCH₃, -CH=CH-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-OCH₃, -CH=C(CH₃)-CO-OCH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-O-n-C₃H₅, -CH=C(CH₃)-CO-OCH₂-O-i-C₃H₅, -CH=C(CH₃)-CO-OCH(CH₃)-OCH₃, -CH=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CH₃)-CO-O-CH₂CH₂-OCH₃, -CH=C(CH₃)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-OCH₃, -CH=C(C₂H₅)-CO-OCH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-O-n-C₃H₅, -CH=C(C₂H₅)-CO-OCH₂-O-i-C₃H₅, -CH=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -CH=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OCH₃, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-OCH₃, -CH=C(Cl)-CO-OCH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-O-n-C₃H₅, -CH=C(Cl)-CO-OCH₂-O-i-C₃H₅, -CH=C(Cl)-CO-OCH(CH₃)-OCH₃, -CH=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Cl)-CO-O-CH₂CH₂-OCH₃, -CH=C(Cl)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-OCH₃, -CH=C(Br)-CO-OCH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-O-n-C₃H₅, -CH=C(Br)-CO-OCH₂-O-i-C₃H₅, -CH=C(Br)-CO-OCH(CH₃)-OCH₃, -CH=C(Br)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Br)-CO-O-CH₂CH₂-OCH₃, -CH=C(Br)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-OCH₃, -CH=C(CN)-CO-OCH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-O-n-C₃H₅, -CH=C(CN)-CO-OCH₂-O-i-C₃H₅, -CH=C(CN)-CO-OCH(CH₃)-OCH₃, -CH=C(CN)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CN)-CO-O-CH₂CH₂-OCH₃, -CH=C(CN)-CO-O-CH₂CH₂-OC₂H₅, -CH=CH-CO-OCH₂-CF₃, -CH=CH-CO-OCH₂-CCl₃, -CH=CH-CO-OCH₂-oxiranyl, -CH=CH-CO-O(CH₂)₃-Br, -CH=CH-CO-OCH₂-CH=CH₂, -CH=CH-CO-OCH₂-C≡CH, -CH=CH-CO-OCH₂-CN, -CH=CH-CO-O(CH₂)₂-CN, -CH=C(CH₃)-CO-OCH₂-CF₃, -CH=C(CH₃)-CO-OCH₂-CCl₃, -CH=C(CH₃)-CO-OCH₂-oxiranyl, -CH=C(CH₃)-CO-O(CH₂)₃-Br, -CH=C(CH₃)-CO-OCH₂-CH=CH₂, -CH=C(CH₃)-CO-OCH₂-C≡CH, -CH=C(CH₃)-CO-OCH₂-CN, -CH=C(CH₃)-CO-O(CH₂)₂-CN, -CH=C(C₂H₅)-CO-OCH₂-CF₃, -CH=C(C₂H₅)-CO-OCH₂-CCl₃, -CH=C(C₂H₅)-CO-OCH₂-oxiranyl, -CH=C(C₂H₅)-CO-O(CH₂)₃-Br, -CH=C(C₂H₅)-CO-OCH₂-CH=CH₂, -CH=C(C₂H₅)-CO-OCH₂-C≡CH, -CH=C(C₂H₅)-CO-OCH₂-CN, -CH=C(C₂H₅)-CO-O(CH₂)₂-CN, -CH=C(Cl)-CO-OCH₂-CF₃, -CH=C(Cl)-CO-OCH₂-CCl₃, -CH=C(Cl)-CO-OCH₂-oxiranyl, -CH=C(Cl)-CO-O(CH₂)₃-Br, -CH=C(Cl)-CO-OCH₂-CH=CH₂, -CH=C(Cl)-CO-OCH₂-C≡CH, -CH=C(Cl)-CO-OCH₂-CN, -CH=C(Cl)-CO-O(CH₂)₂-CN, -CH=C(Br)-CO-OCH₂-CF₃, -CH=C(Br)-CO-OCH₂-CCl₃, -CH=C(Br)-CO-OCH₂-oxiranyl, -CH=C(Br)-CO-O(CH₂)₃-Br, -CH=C(Br)-CO-OCH₂-CH=CH₂, -CH=C(Br)-CO-OCH₂-C≡CH, -CH=C(Br)-CO-OCH₂-CN, -CH=C(Br)-CO-O(CH₂)₂-CN, -CH=C(CN)-CO-OCH₂-CF₃, -CH=C(CN)-CO-OCH₂-CCl₃, -CH=C(CN)-CO-OCH₂-oxiranyl -CH=C(CN)-CO-O(CH₂)₃-Br, -CH=C(CN)-CO-OCH₂-CH=CH₂, -CH=C(CN)-CO-OCH₂-C≡CH, -CH=C(CN)-CO-OCH₂-CN, -CH=C(CN)-CO-O(CH₂)₂-CN, -CH=CH-CO-CH₃, -CH=CH-CO-C₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-i-C₃H₇, -CH=CH-CO-n-C₄H₉, -CH=CH-CO-tert.-C₄H₉, -CH=CH-CO-CH₂Cl, -CH=CH-CO-CH₂Br, -CH=CH-CO-CHCl₂, -CH=CH-CO-CH₂-OCH₃, -CH=CH-CO-CH(OCH₃)₂, -CH=CH-CO-CH₂-SCH₃, -CH=C(CH₃)-CO-CH₃, -CH=C(CH₃)-CO-C₂H₅, -CH=C(CH₃)-CO-n-C₃H₇, -CH=C(CH₃)-CO-i-C₃H₇, -CH=C(CH₃)-CO-n-C₄H₉, -CH=C(CH₃)-CO-tert.-C₄H₉, -CH=C(CH₃)-CO-CH₂Cl, -CH=C(CH₃)-CO-CH₂Br, -CH=C(CH₃)-CO-CHCl₂, -CH=C(CH₃)-CO-CH₂-OCH₃, -CH=C(CH₃)-CO-CH(OCH₃)₂, -CH=C(CH₃)-CO-CH₂-SCH₃, -CH=C(C₂H₅)-CO-CH₃, -CH=C(C₂H₅)-CO-C₂H₅, -CH=C(C₂H₅)-CO-n-C₃H₇, -CH=C(C₂H₅)-CO-i-C₃H₇, -CH=C(C₂H₅)-CO-n-C₄H₉, -CH=C(C₂H₅)-CO-tert.-C₄H₉, -CH=C(C₂H₅)-CO-CH₂Cl, -CH=C(C₂H₅)-CO-CH₂Br, -CH=C(C₂H₅)-CO-CHCl₂, -CH=C(C₂H₅)-CO-CH₂-OCH₃, -CH=C(C₂H₅)-CO-CH(OCH₃)₂, -CH=C(C₂H₅)-CO-CH₂-SCH₃, -CH=C(Cl)-CO-CH₃, -CH=C(Cl)-CO-C₂H₅, -CH=C(Cl)-CO-n-C₃H₇, -CH=C(Cl)-CO-i-C₃H₇, -CH=C(Cl)-CO-n-C₄H₉, -CH=C(Cl)-CO-tert.-C₄H₉, -CH=C(Cl)-CO-CH₂Cl, -CH=C(Cl)-CO-CH₂Br, -CH=C(Cl)-CO-CHCl₂, -CH=C(Cl)-CO-CH₂-OCH₃, -CH=C(Cl)-CO-CH(OCH₃)₂, -CH=C(Cl)-CO-CH₂-SCH₃, -CH=C(Br)-CO-CH₃, -CH=C(Br)-CO-C₂H₅, -CH=C(Br)-CO-n-C₃H₇, -CH=C(Br)-CO-i-C₃H₇, -CH=C(Br)-CO-n-C₄H₉, -CH=C(Br)-CO-tert.-C₄H₉, -CH=C(Br)-CO-CH₂Cl, -CH=C(Br)-CO-CH₂Br, -CH=C(Br)-CO-CHCl₂, -CH=C(Br)-CO-CH₂-OCH₃, -CH=C(Br)-CO-CH(OCH₃)₂, -CH=C(Br)-CO-CH₂-SCH₃, -CH=C(CN)-CO-CH₃, -CH=C(CN)-CO-C₂H₅, -CH=C(CN)-CO-n-C₃H₇, -CH=C(CN)-CO-i-C₃H₇, -CH=C(CN)-CO-n-C₄H₉, -CH=C(CN)-CO-tert.-C₄H₉, -CH=C(CN)-CO-CH₂Cl, -CH=C(CN)-CO-CH₂Br, -CH=C(CN)-CO-CHCl₂, -CH=C(CN)-CO-CH₂-OCH₃, -CH=C(CN)-CO-CH(OCH₃)₂, -CH=C(CN)-CO-CH₂-SCH₃, -CH=CH-CO-C₆H₅, -CH=CH-CO-(4-Cl-C₆H₄), -CH=C(CH₃)-CO-C₆H₅, -CH=C(CH₃)-CO-(4-Cl-C₆H₄), -CH=C(C₂H₅)-CO-C₆H₅, -CH=C(C₂H₅)-CO-(4-Cl-C₆H₄), -CH=C(Cl)-CO-C₆H₅, -CH=C(Br)-CO-C₆H₅, -CH=C(CN)-CO-C₆H₅, -CH=CH-CO-NH₂, -CH=CH-CO-NHCH₃, -CH=CH-CO-N(CH₃)₂, -CH=CH-CO-NH-C₂H₅, -CH=CH-CO-N(C₂H₅)₂, -CH=CH-CO-NH-n-C₃H₇, -CH=CH-CO-NH-i-C₃H₇, -CH=CH-CO-NH-tert.-C₄H₉, -CH=CH-CO-NH-cyclopropyl, -CH=CH-CO-NH-cyclobutyl, -CH=CH-CO-NH-cyclopentyl, -CH=CH-CO-NH-cyclohexyl, -CH=CH-CO-NH-cycloheptyl, -CH=CH-CO-NH-cyclooctyl, -CH=CH-CO-pyrrolidin-1-yl, -CH=CH-CO-piperidin-1-yl, -CH=CH-CO-morpholin-4-yl, -CH=CH-CO-NH-CH₂CH=CH₂, -CH=CH-CO-NH-CH₂C≡CH, -CH=CH-CO-N(CH₃)-CH₂C≡CH, -CH=CH-CO-NH-(CH₂)₂Cl, -CH=CH-CO-NH-C₆H₅, -CH=C(CH₃)-CO-NH₂, -CH=C(CH₃)-CO-NHCH₃, -CH=C(CH₃)-CO-N(CH₃)₂, -CH=C(CH₃)-CO-NH-C₂H₅, -CH=C(CH₃)-CO-N(C₂H₅)₂, -CH=C(CH₃)-CO-NH-n-C₃H₇, -CH=C(CH₃)-CO-NH-i-C₃H₇, -CH=C(CH₃)-CO-NH-tert.-C₄H₉, -CH=C(CH₃)-CO-NH-cyclopropyl, -CH=C(CH₃)-CO-NH-cyclobutyl, -CH=C(CH₃)-CO-NH-cyclopentyl, -CH=C(CH₃)-CO-NH-cyclohexyl, -CH=C(CH₃)-CO-NH-cycloheptyl, -CH=C(CH₃)-CO-NH-cyclooctyl, -CH=C(CH₃)-CO-pyrrolidin-1-yl, -CH=C(CH₃)-CO-piperidin-1-yl, -CH=C(CH₃)-CO-morpholin-4-yl, -CH=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -CH=C(CH₃)-CO-NH-CH₂C≡CH, -CH=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CH₃)-CO-NH-(CH₂)₂Cl, -CH=C(CH₃)-CO-NH-C₆H₅, -CH=C(C₂H₅)-CO-NH₂, -CH=C(C₂H₅)-CO-NHCH₃, -CH=C(C₂H₅)-CO-N(CH₃)₂, -CH=C(C₂H₅)-CO-NH-C₂H₅, -CH=C(C₂H₅)-CO-N(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-n-C₃H₇, -CH=C(C₂H₅)-CO-NH-i-C₃H₇, -CH=C(C₂H₅)-CO-NH-tert.-C₄H₉, -CH=C(C₂H₅)-CO-NH-cyclopropyl, -CH=C(C₂H₅)-CO-NH-cyclobutyl, -CH=C(C₂H₅)-CO-NH-cyclopentyl, -CH=C(C₂H₅)-CO-NH-cyclohexyl, -CH=C(C₂H₅)-CO-NH-cycloheptyl, -CH=C(C₂H₅)-CO-NH-cyclooctyl, -CH=C(C₂H₅)-CO-pyrrolidin-1-yl, -CH=C(C₂H₅)-CO-piperidin-1-yl, -CH=C(C₂H₅)-CO-morpholin-4-yl, -CH=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-CH₂C≡CH, -CH=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -CH=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -CH=C(C₂H₅)-CO-NH-C₆H₅, -CH=C(Cl)-CO-NH₂, -CH=C(Cl)-CO-NHCH₃, -CH=C(Cl)-CO-N(CH₃)₂, -CH=C(Cl)-CO-NH-C₂H₅, -CH=C(Cl)-CO-N(C₂H₅)₂, -CH=C(Cl)-CO-NH-n-C₃H₇, -CH=C(Cl)-CO-NH-i-C₃H₇, -CH=C(Cl)-CO-NH-tert.-C₄H₉, -CH=C(Cl)-CO-NH-cyclopropyl, -CH=C(Cl)-CO-NH-cyclobutyl, -CH=C(Cl)-CO-NH-cyclopentyl, -CH=C(Cl)-CO-NH-cyclohexyl, -CH=C(Cl)-CO-NH-cycloheptyl, -CH=C(Cl)-CO-NH-cyclooctyl, -CH=C(Cl)-CO-pyrrolidin-1-yl, -CH=C(Cl)-CO-piperidin-1-yl, -CH=C(Cl)-CO-morpholin-4-yl, -CH=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -CH=C(Cl)-CO-NH-CH₂C≡CH, -CH=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Cl)-CO-NH-(CH₂)₂Cl, -CH=C(Cl)-CO-NH-C₆H₅, -CH=C(Br)-CO-NH₂, -CH=C(Br)-CO-NHCH₃, -CH=C(Br)-CO-N(CH₃)₂, -CH=C(Br)-CO-NH-C₂H₅, -CH=C(Br)-CO-N(C₂H₅)₂, -CH=C(Br)-CO-NH-n-C₃H₇, -CH=C(Br)-CO-NH-i-C₃H₇, -CH=C(Br)-CO-NH-tert.-C₄H₉, -CH=C(Br)-CO-NH-cyclopropyl, -CH=C(Br)-CO-NH-cyclobutyl, -CH=C(Br)-CO-NH-cyclopentyl, -CH=C(Br)-CO-NH-cyclohexyl, -CH=C(Br)-CO-NH-cycloheptyl, -CH=C(Br)-CO-NH-cyclooctyl, -CH=C(Br)-CO-pyrrolidin-1-yl, -CH=C(Br)-CO-piperidin-1-yl, -CH=C(Br)-CO-morpholin-4-yl, -CH=C(Br)-CO-NH-CH₂CH=C(Br)₂, -CH=C(Br)-CO-NH-CH₂C≡CH, -CH=C(Br)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Br)-CO-NH-(CH₂)₂Cl, -CH=C(Br)-CO-NH-C₆H₅, -CH=C(CN)-CO-NH₂, -CH=C(CN)-CO-NHCH₃, -CH=C(CN)-CO-N(CH₃)₂, -CH=C(CN)-CO-NH-C₂H₅, -CH=C(CN)-CO-N(C₂H₅)₂, -CH=C(CN)-CO-NH-n-C₃H₇, -CH=C(CN)-CO-NH-i-C₃H₇, -CH=C(CN)-CO-NH-tert.-C₄H₉, -CH=C(CN)-CO-NH-cyclopropyl, -CH=C(CN)-CO-NH-cyclobutyl, -CH=C(CN)-CO-NH-cyclopentyl, -CH=C(CN)-CO-NH-cyclohexyl, -CH=C(CN)-CO-NH-cycloheptyl, -CH=C(CN)-CO-NH-cyclooctyl, -CH=C(CN)-CO-pyrrolidin-1-yl, -CH=C(CN)-CO-piperidin-1-yl, -CH=C(CN)-CO-morpholin-4-yl, -CH=C(CN)-CO-NH-CH₂CH=C(CN)₂, -CH=C(CN)-CO-NH-CH₂C≡CH, -CH=C(CN)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CN)-CO-NH-(CH₂)₂Cl, -CH=C(CN)-CO-NH-C₆H₅, -CH=CH-CO-SCH₃, -CH=CH-CO-SC₂H₅, -CH=CH-CO-S-n-C₃H₇, -CH=CH-CO-S-i-C₃H₇, -CH=CH-CO-S-n-C₄H₉, -CH=CH-CO-S-tert.-C₄H₉, -CH=C(CH₃)-CO-SCH₃, -CH=C(CH₃)-CO-SC₂H₅, -CH=C(CH₃)-CO-S-n-C₃H₇, -CH=C(CH₃)-CO-S-i-C₃H₇, -CH=C(CH₃)-CO-S-n-C₄H₉, -CH=C(CH₃)-CO-S-tert.-C₄H₉, -CH=C(C₂H₅)-CO-SCH₃, -CH=C(C₂H₅)-CO-SC₂H₅, -CH=C(C₂H₅)-CO-S-n-C₃H₇, -CH=C(C₂H₅)-CO-S-i-C₃H₇, -CH=C(C₂H₅)-CO-S-n-C₄H₉, -CH=C(C₂H₅)-CO-S-tert.-C₄H₉, -CH=C(Cl)-CO-SCH₃, -CH=C(Cl)-CO-SC₂H₅, -CH=C(Cl)-CO-S-n-C₃H₇, -CH=C(Cl)-CO-S-i-C₃H₇, -CH=C(Cl)-CO-S-n-C₄H₉, -CH=C(Cl)-CO-S-tert.-C₄H₉, -CH=C(Br)-CO-SCH₃, -CH=C(Br)-CO-SC₂H₅, -CH=C(Br)-CO-S-n-C₃H₇, -CH=C(Br)-CO-S-i-C₃H₇, -CH=C(Br)-CO-S-n-C₄H₉, -CH=C(Br)-CO-S-tert.-C₄H₉, -CH=C(CN)-CO-SCH₃, -CH=C(CN)-CO-SC₂H₅, -CH=C(CN)-CO-S-n-C₃H₇, -CH=C(CN)-CO-S-i-C₃H₇, -CH=C(CN)-CO-S-n-C₄H₉, -CH=C(CN)-CO-S-tert.-C₄H₉, -CH=C(COCH₃)-CO-OCH₃, -CH=C(COC₂H₅)-CO-OCH₃, -CH=C(CO-n-C₃H₇)-CO-OCH₃, -CH=C(COCH₃)-CO-OC₂H₅, -CH=C(COC₂H₅)-CO-OC₂H₅, -CH=C(CO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COCH₃)-CO-O-n-C₃H₇, -CH=C(COC₂H₅)-CO-O-n-C₃H₇, -CH=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-OCH₃, -CH=C(CF₃)-CO-OC₂H₅, -CH=C(CF₃)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-O-i-C₃H₇, -CH=C(CF₃)-CO-O-n-C₄H₉, -CH=C(CF₃)-CO-O-tert.-C₄H₉, -CH=C(COOCH₃)₂, -CH=C(COOC₂H₅)₂, -CH=C(COOCH₃)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)-CO-OCH₃, -CH=C(COO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)₂, -CH=CH-CH=CH-COOH, -CH=CH-CH=CH-CO-OCH₃, -CH=CH-CH=CH-CO-OC₂H₅, -CH=CH-CH=C(COOCH₃)₂, -CH=CH-CH=C(CN)-CO-OCH₃, -CH=CH-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-OCH₃, -CH=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CH=C(Cl)-CO-OCH₃, -CH=C(CH₃)-CH=C(Br)-CO-OCH₃, -CH=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-NH₂, -CH=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -CH=CH-(CH₂)₂-COOH, -CH=CH-(CH₂)₂-CO-OCH₃, -CH=CH-(CH₂)₂-CO-OC₂H₅, -CH=CH-CH₂-CH(COOCH₃)₂, -CH=CH-CH₂-CH(COOC₂H₅)₂, -CH=CH-CH₂-CH(CN)-CO-OCH₃, -CH=CH-CH₂-CH(CN)-CO-OC₂H₅, -CH=CH-CH₂-CH(CH₃)-CO-OCH₃, -CH=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -CH=CH-(CH₂)₂-CO-NH₂, -CH=CH-(CH₂)₂-CO-NH-CH₃, -CH=CH-CH₂-COOH, -CH=CH-CH₂-CO-OCH₃, -CH=CH-CH₂-CO-OC₂H₅, -CH=C(COOCH₃)-CH₂-CO-OCH₃, -CH=C(COOCH₃)-CH₂-CO-OC₂H₅, -CH=CH-CH₂-CO-NH₂, -CH=CH-CH₂-CO-NH-CH₃, -CH=CH-CH₂-CO-N(CH₃)₂, -CH(OCH₃)₂, -CH(SCH₃)₂, -CH(OC₂H₅)₂, -CH(SC₂H₅)₂, -CH(O-n-C₃H₇)₂, -CH(O-i-C₃H₇)₂, -CH(S-n-C₃H₇)₂, -CH(S-i-C₃H₇)₂, -CH(O-n-C₄H₉)₂, -CH(O-i-C₄H₉)₂, -CH(O-s-C₄H₉)₂, -CH(O-tert.-C₄H₉)₂, -CH(S-n-C₄H₉)₂, -CH(S-i-C₄H₉)₂, -CH(S-s-C₄H₉)₂, -CH(S-tert.-C₄H₉)₂, -CH(OC₅H₁₁)₂, 1,3-Dioxolan-2-yl, 1,3-Dithio­ lan-2-yl, 1,3-Oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 5-Methyl-1,3-oxathiolan-2-yl, 4-Ethyl-1,3-dioxolan-2-yl, 4-Ethyl- 1,4-dithiolan-2-yl, 4-Ethyl-1,3-oxathiolan-2-yl, 5-Ethyl-1,3-oxa­ thiolan-2-yl, 4,5-Dimethyl-1,3-dioxolan-2-yl, 4,4-Dimethyl-1,3- dioxolan-2-yl, 4,5-Dimethyl-1,3-dithiolan-2-yl, 5,5-Dimethyl-1,3- dithiolan-2-yl, 4,5-Dimethyl-1,3-oxathiolan-2-yl, 5,5-Dimethyl- 1,3-oxathiolan-2-yl, 4,4-Dimethyl-1,3-oxathiolan-2-yl, 4-Vinyl- 1,3-dioxolan-2-yl, 4-Vinyl-1,3-dithiolan-2-yl, 4-Vinyl-1,3-oxa­ thiolan-2-yl, 5-Vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3- dioxolan-2-yl, 4-Chlormethyl-1,3-dithiolan-2-yl, 4-Chlormethyl- 1,3-oxathiolan-2-yl, 5-Chlormethyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-1,3-dithio­ lan-2-yl, 4-Hydroxymethyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl- 1,3-oxathiolan-2-yl, 4-Methoxymethyl-1,3-dioxolan-2-yl, 4-Allyl­ oxymethyl-1,3-dioxolan-2-yl, 4-Propargyloxymethyl-1,3-dioxolan- 2-yl, 4-Acetoxymethyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-1,3-dithiolan-2-yl, 4-Propargyl­ oxymethyl-1,3-dithiolan-2-yl, 4-Acetoxymethyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-1,3-oxathiolan- 2-yl, 4-Allyloxymethyl-1,3-oxathiolan-2-yl, 5-Allyloxymethyl- 1,3-oxathiolan-2-yl, 4-Propargyloxymethyl-1,3-oxathiolan- 2-yl, 5-Propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxymethyl- 1,3-oxathiolan-2-yl, 5-Acetoxymethyl-1,3-oxathiolan-2-yl, 4-Methylthiomethyl-1,3-dioxolan-2-yl, 4-Methylthiomethyl-1,3- dithiolan-2-yl, 4-Carboxy-1,3-dioxolan-2-yl, 4-Carboxy-1,3- dithiolan-2-yl, 4-Methoxycarbonyl-1,3-dioxolan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-1,3-dithiolan- 2-yl, 4-n-Butoxycarbonyl-1,3-dithiolan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-4-methyl- 1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-di­ thiolan-2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-1,3- dithiolan-2-yl, 1,3-Dioxan-2-yl, 1,3-Dithian-2-yl, 1,3-Oxathian- 2-yl, 5-Methyl-1,3-dioxan-2-yl, 5-Methyl-1,3-dithian-2-yl, 5-Methyl-1,3-oxathian-2-yl, 5,5-Dimethyl-1,3-dioxan-2-yl, 4,6-Dimethyl- 1,3-dioxan-2-yl, 4,4-Dimethyl-1,3-dioxan-2-yl, 5,5-Dimethyl- 1,3-dithian-2-yl, 4,6-Dimethyl-1,3-dithian-2-yl, 4,4-Dimethyl- 1,3-dithian-2-yl, 5,5-Dimethyl-1,3-oxathian-2-yl, 4,4-Dimethyl- 1,3-oxathian-2-yl, 6,6-Dimethyl-1,3-oxathian-2-yl, 4-Hydroxymethyl-1,3-dioxan-2-yl, 4-Methoxymethyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-1,3-dioxan-2- yl, 4-Hydroxymethyl-1,3-dithian-2-yl, 4-Methoxymethyl-1,3-dithian- 2-yl, 4-Allyloxymethyl-1,3-dithian-2-yl, 4-Acetoxymethyl- 1,3-dithian-2-yl, 4-Chlormethyl-1,3-dioxan-2-yl, 4-Chlormethyl- 1,3-dithian-2-yl, 1,3-Dioxepan-2-yl, 1,3-Dithiepan-2-yl, 1,3-Dioxep- 5-en-2-yl, 4-Methoxycarbonyl-1,3-dioxan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-1,3-dithian- 2-yl, 4-n-Butoxycarbonyl-1,3-dithian-2-yl, 4-Methoxycarbonyl-4- methyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxan-2- yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-4-methyl- 1,3-dithian-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithian-2-yl, -C(CH₃)(OCH₃)₂, -C(CH₃)(SCH₃)₂, -C(CH₃)(OC₂H₅)₂, -C(CH₃)(SC₂H₅)₂, -C(CH₃)(O-n-C₃H₇)₂, -C(CH₃)(O-i-C₃H₇)₂, -C(CH₃)(S-n-C₃H₇)₂, -C(CH₃)(S-i-C₃H₇)₂, -C(CH₃)(O-n-C₄H₉)₂, -C(CH₃)(O-i-C₄H₉)₂, -C(CH₃)(O-s-C₄H₉)₂, -C(CH₃)(O-tert.-C₄H₉)₂, -C(CH₃)(S-n-C₄H₉)₂, -C(CH₃)(S-i-C₄H₉)₂, -C(CH₃)(S-s-C₄H₉)₂, -C(CH₃)(S-tert.-C₄H₉)₂, -C(CH₃)(O-n-C₅H₁₁)′′, 2-Methyl-1,3-dioxolan-2-yl, 2-Methyl-1,3-dithiolan- 2-yl, 2-Methyl-1,3-oxathiolan-2-yl, 2,4-Dimethyl-1,3- dioxolan-2-yl, 2,4-Dimethyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-1,3- oxathiolan-2-yl, 2,5-Dimethyl-1,3-oxathiolan-2-yl, 4-Ethyl-2- methyl-1,3-dioxolan-2-yl, 4-Ethyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Ethyl-2-methyl-1,3- oxathiolan-2-yl, 2,4,5-Trimethyl-1,3-dioxolan-2-yl, 2,4,4-Trimethyl- 1,3-dioxolan-2-yl, 2,4,5-Trimethyl-1,3-dithiolan-2-yl, 2,4,4-Trimethyl-1,3-dithiolan-2-yl, 2,4,5-Trimethyl-1,3-oxathiolan- 2-yl, 2,4,4-Trimethyl-1,3-oxathiolan-2-yl, 2-Methyl-4-vinyl- 1,3-dioxolan-2-yl, 2-Methyl-4-vinyl-1,3-dithiolan-2-yl, 2-Methyl- 4-vinyl-1,3-oxathiolan-2-yl, 2-Methyl-5-vinyl-1,3-oxathiolan-2- yl, 4-Chlormethyl-2-methyl-1,3-dioxolan-2-yl, 4-Chlormethyl-2- methyl-1,3-dithiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-oxathiolan- 2-yl, 5-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl- 2-methyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-2- methyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dioxolan- 2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxy- 2-methyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dithiolan-2-yl, 4-Acetoxy-2- methyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-oxathiolan- 2-yl, 5-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl- 2-methyl-1,3-oxathiolan-2-yl, 5-Allyloxymethyl-2- methyl-1,3-oxathiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3- oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3-oxathiolan-2- yl, 4-Acetoxy-2-methyl-1,3-oxathiolan-2-yl, 5-Acetoxy-2-methyl- 1,3-oxathiolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dioxolan-2- yl, 2-Methyl-4-methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-2- methyl-1,3-dioxolan-2-yl, 4-Carboxy-2-methyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-2- methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-2-methyl-1,3-dioxolan- 2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl- 2-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-2- methyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dioxolan- 2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-ethoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4- ethoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-n-butoxy­ carbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl-1,3- dithiolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-dioxan-2- yl, 2-Methyl-1,3-dithian-2-yl, 2-Methyl-1,3-oxathian-2-yl, 2,5- Dimethyl-1,3-dioxan-2-yl, 2,5-Dimethyl-1,3-dithian-2-yl, 2,5-Dimethyl- 1,3-oxathian-2-yl, 2,5,5-Trimethyl-1,3-dioxan-2-yl, 2,4,6- Trimethyl-1,3-dioxan-2-yl, 2,4,4-Trimethyl-1,3-dioxan-2-yl, 2,5,5-Trimethyl-1,3-dithian-2-yl, 2,4,6-Trimethyl-1,3-dithian-2- yl, 2,4,4-Trimethyl-1,3-dithian-2-yl, 2,5,5-Trimethyl-1,3-oxathian- 2-yl, 2,4,4-Trimethyl-1,3-oxathian-2-yl, 2,6,6-Trimethyl- 1,3-oxathian-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-2- methyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dithian-2-yl, 4-Methoxymethyl-2- methyl-1,3-dithian-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithian-2- yl, 4-Acetoxymethyl-2-methyl-1,3-dithian-2-yl, 4-Chlormethyl-2- methyl-1,3-dioxan-2-yl, 4-Chlormethyl-2-methyl-1,3-dithian-2-yl, -C(CH₃)=NH, -C(CH₃)=N-CH₃, -C(CH₃)=N-C₂H₅, -C(CH₃)=N-n-C₃H₇, -C(CH₃)=N-i-C₃H₇, -C(CH₃)=N-n-C₄H₉, -C(CH₃)=N-CH₂CH=CH₂, -C(CH₃)=N-CH₂CH=CH₂-CH₃, -C(CH₃)=N-CH₂C≡CH, -C(CH₃)=N-CH₂C≡C-CH₃, -C(CH₃)=N-cyclopropyl, -C(CH₃)=N-cyclobutyl, -C(CH₃)=N-cyclopentyl, -C(CH₃)=N-cyclohexyl, -C(CH₃)=N-cycloheptyl, -C(CH₃)=N-CH₂-CH₂Cl, -C(CH₃)=N-CH₂Cl, -C(CH₃)=N-C₆H₅, -C(CH₃)=N-(2-F-C₆H₄), -C(CH₃)=N-(3-F-C₆H₄), -C(CH₃)=N-(4-F-C₆H₄), -C(CH₃)=N-(2-Cl-C₆H₄), -C(CH₃)=N-(3-Cl-C₆H₄), -C(CH₃)=N-(4-Cl-C₆H₄), -C(CH₃)=N-(2-CH₃-C₆H₄), -C(CH₃)=N-(3-CH₃-C₆H₄), -C(CH₃)=N-(4-CH₃-C₆H₄), -C(CH₃)=N-(2-CF₃-C₆H₄), -C(CH₃)=N-(3-CF₃-C₆H₄), -C(CH₃)=N-(4-CF₃-C₆H₄), -C(CH₃)=N-(2-OCH₃-C₆H₄), -C(CH₃)=N-(3-OCH₃-C₆H₄), -C(CH₃)=N-(4-OCH₃-C₆H₄), -C(CH₃)=N-(4-NO₂-C₆H₄), -C(CH₃)=N-(4-CN-C₆H₄), -C(CH₃)=N-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-(2,4-(CH₃)₂-C₆H₃), -C(CH₃)=N-CH₂-OCH₃, -C(CH₃)=N-CH₂-OC₂H₅, -C(CH₃)=N-CH₂CH₂-OCH₃, -C(CH₃)=N-CH₂CH₂-OC₂H₅, -C(CH₃)=N-OH, -C(CH₃)=N-OCH₃, -C(CH₃)=N-OC₂H₅, -C(CH₃)=N-O-n-C₃H₇, -C(CH₃)=N-O-i-C₃H₇, -C(CH₃)=N-O-n-C₄H₉, -C(CH₃)=N-O-i-C₄H₉, -C(CH₃)=N-O-s-C₄H₉, -C(CH₃)=N-O-tert.-C₄H₉, -C(CH₃)=N-OCH₂-CH=CH₂, -C(CH₃)=N-OCH(CH₃)-CH=CH₂, -C(CH₃)=N-OCH₂-C≡CH, -C(CH₃)=N-CH(CH₃)-C≡CH, -C(CH₃)=N-OCH₂-CH=C-CH₃, -C(CH₃)=N-OCH₂CH₂-Cl, -C(CH₃)=N-OCH₂CH₂-F, -C(CH₃)=N-OCH₂-CF₃, -C(CH₃)=N-OCH₂-CH=CHCl, -C(CH₃)=N-OCH₂-C(Cl)=CH₂, -C(CH₃)=N-OCH₂-C(Br)=CH₂, -C(CH₃)=N-OCH₂-CH=C(Cl)-CH₃, -C(CH₃)=N-O-CO-CH₃, -C(CH₃)=N-O-CO-C₂H₅, -C(CH₃)=N-OCH₂-CN, -C(CH₃)=N-OCH₂-CH=CH-CH₂-OCH₃, -C(CH₃)=N-OCH₂-CH=CH-CH₂-O-tert.-C₄H₉, -C(CH₃)=N-O-(CH₂)₃-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-(4-Cl-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-C₆H₅, -C(CH₃)=N-OCH₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(3-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-CH₂-(4-CH₃O-C₆H₄), -C(CH₃)=N-OCH₂-CH=C(CH₃)-C₆H₅, -C(CH₃)=N-O-(CH₂)₂-CH=CH-(3,4-Cl₂-C₆H₃), -C(CH₃)=N-O-(CH₂)₃-C≡C-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-OCH₃, -C(CH₃)=N-OCH₂CH₂-OCH₃, -C(CH₃)=N-OCH₂-OC₂H₅, -C(CH₃)=N-OCH(CH₃)-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=N-NH₂, -C(CH₃)=N-NH-CH₃, -C(CH₃)=N-NH-C₂H₅, -C(CH₃)=N-NH-n-C₃H₇, -C(CH₃)=N-NH-i-C₃H₇, -C(CH₃)=N-NH-n-C₄H₉, -C(CH₃)=N-NH-i-C₄H₉, -C(CH₃)=N-NH-s-C₄H₉, -C(CH₃)=N-NH-tert.-C₄H₉, -C(CH₃)=N-NH-cyclopropyl, -C(CH₃)=N-NH- cyclobutyl, -C(CH₃)=N-NH-cyclopentyl, -C(CH₃)=N-NH-cyclohexyl, -C(CH₃)=N-NH-cycloheptyl, -C(CH₃)=N-N(CH₃)₂, -C(CH₃)=N-N(C₂H₅)₂, -C(CH₃)=N-N(n-C₃H₇)₂, -C(CH₃)=N-N(i-C₃H₇)₂, -C(CH₃)=N-NH-CH₂-C=CH, -C(CH₃)=N-NH-CH₂-C≡CH, -C(CH₃)=N-N(CH₃)-CH₂-C≡CH, -C(CH₃)=N-NH-CH₂CF₃, -C(CH₃)=N-NH-CO-CH₃, -C(CH₃)=N-NH-CO-C₂H₅, -C(CH₃)=N-NH-CO-OCH₃, -C(CH₃)=N-NH-CO-OC₂H₅, -C(CH₃)=N-NH-CO-O-tert.-C₄H₉, -C(CH₃)=N- pyrrolidin-1-yl, -C(CH₃)=N-piperidin-1-yl, -C(CH₃)=N-morpholin- 4-yl, -C(CH₃)=N-NH-C₆H₅, -C(CH₃)=N-NH-(4-Cl-C₆H₄), -C(CH₃)=N-NH-(4-NO₂-C₆H₄), -C(CH₃)=N-NH-(4-F-C₆H₄), -C(CH₃)=N-NH-(4-CH₃O-C₆H₄), -C(CH₃)=N-NH-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-NH-(2,4-(NO₂)₂-C₆H₃), -C(CH₃)=N-NH-CO-NH₂, -C(CH₃)=N-NH-CO-NHCH₃, -C(CH₃)=N-NH-CO-NHC₂H₅, -C(CH₃)=N-NH-CO-N(CH₃)₂, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=CH-CO-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-O-n-C₄H₉, -C(CH₃)=CH-CO-O-tert.-C₄H₉, -C(CH₃)=CH-CO-O-cyclopropyl, -C(CH₃)=CH-CO-O-cyclobutyl, -C(CH₃)=CH-CO-O-cyclopentyl, -C(CH₃)=CH-CO-O-cyclohexyl, -C(CH₃)=CH-CO-O-cycloheptyl, -C(CH₃)=C(CH₃)-COOH, -C(CH₃)=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-cyclopropyl, -C(CH₃)=C(CH₃)-CO-O-cyclobutyl, -C(CH₃)=C(CH₃)-CO-O-cyclopentyl, -C(CH₃)=C(CH₃)-CO-O-cyclohexyl, -C(CH₃)=C(CH₃)-CO-O-cycloheptyl, -C(CH₃)=C(C₂H₅)-COOH, -C(CH₃)=C(C₂H₅)-CO-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-cyclo­ propyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-O- cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-O-cycloheptyl, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-O-n-C₄H₉, -C(CH₃)=C(Cl)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-O-cyclopropyl, -C(CH₃)=C(Cl)-CO-O-cyclobutyl, -C(CH₃)=C(Cl)-CO-O-cyclopentyl, -C(CH₃)=C(Cl)-CO-O-cyclohexyl, -C(CH₃)=C(Cl)-CO-O-cycloheptyl, -C(CH₃)=C(Br)-COOH, -C(CH₃)=C(Br)-CO-OCH₃, -C(CH₃)=C(Br)-CO-OC₂H₅, -C(CH₃)=C(Br)-CO-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-O-n-C₄H₉, -C(CH₃)=C(Br)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-O-cyclopropyl, -C(CH₃)=C(Br)-CO-O-cyclobutyl, -C(CH₃)=C(Br)-CO-O-cyclopentyl, -C(CH₃)=C(Br)-CO-O-cyclohexyl, -C(CH₃)=C(Br)-CO-O-cycloheptyl, -C(CH₃)=C(CN)-COOH, -C(CH₃)=C(CN)-CO-OCH₃, -C(CH₃)=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CN)-CO-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-O-n-C₄H₉, -C(CH₃)=C(CN)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-O-cyclopropyl, -C(CH₃)=C(CN)-CO-O-cyclobutyl, -C(CH₃)=C(CN)-CO-O-cyclopentyl, -C(CH₃)=C(CN)-CO-O-cyclohexyl, -C(CH₃)=C(CN)-CO-O-cycloheptyl, -C(CH₃)=CH-CO-OCH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-OCH(CH₃)-OCH₃, -C(CH₃)=CH-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=CH-CO-OCH₂CH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-O-i-C₃H₇, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-O-i-C₃H₇, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-O-i-C₃H₇, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-CF₃, -C(CH₃)=CH-CO-OCH₂-CCl₃, -C(CH₃)=CH-CO-OCH₂-oxiranyl, -C(CH₃)=CH-CO-(CH₂)₃-Br,-C(CH₃)=CH-CO-OCH₂-CH=CH₂, -C(CH₃)=CH-CO-OCH₂-C≡CH, -C(CH₃)=CH-CO-OCH₂-CN, -C(CH₃)=CH-CO-OCH₂CH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CF₃, -C(CH₃)=C(CH₃)-CO-OCH₂-CCl₃, -C(CH₃)=C(CH₃)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CH₃)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CH₃)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CH₃)-CO-OCH₂-C≡CH, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CF₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CCl₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-oxiranyl, -C(CH₃)=C(C₂H₅)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(C₂H₅)-CO-OCH₂-C≡CH, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂-CF₃, -C(CH₃)=C(Cl)-CO-OCH₂-CCl₃, -C(CH₃)=C(Cl)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Cl)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Cl)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Cl)-CO-OCH₂-C≡CH, -C(CH₃)=C(Cl)-CO-OCH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂-CF₃, -C(CH₃)=C(Br)-CO-OCH₂-CCl₃, -C(CH₃)=C(Br)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Br)-CO-O(CH₂)₃-Br, -C(CH₃)=C(Br)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Br)-CO-OCH₂-C≡CH, -C(CH₃)=C(Br)-CO-OCH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂CH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂-CF₃, -C(CH₃)=C(CN)-CO-OCH₂-CCl₃, -C(CH₃)=C(CN)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CN)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CN)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CN)-CO-OCH₂-C≡CH, -C(CH₃)=C(CN)-CO-OCH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂CH₂-CN, -C(CH₃)=CH-CO-CH₃, -C(CH₃)=CH-CO-C₂H₅, -C(CH₃)=CH-CO-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-n-C₄H₉, -C(CH₃)=CH-CO-tert.-C₄H₉, -C(CH₃)=CH-CO-CH₂Cl, -C(CH₃)=CH-CO-CH₂Br, -C(CH₃)=CH-CO-CHCl₂, -C(CH₃)=CH-CO-CH₂-OCH₃, -C(CH₃)=CH-CO-CH(OCH₃)₂, -C(CH₃)=CH-CO-CH₂-SCH₃, -C(CH₃)=C(CH₃)-CO-CH₃, -C(CH₃)=C(CH₃)-CO-C₂H₅, -C(CH₃)=C(CH₃)-CO-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-CH₂Cl, -C(CH₃)=C(CH₃)-CO-CH₂Br, -C(CH₃)=C(CH₃)-CO-CHCl₂, -C(CH₃)=C(CH₃)-CO-CH₂-OCH₃, -C(CH₃)=C(CH₃)- ⁹⁹⁹⁹⁹ ⁰⁰⁰⁷⁰ ⁵⁵² ⁰⁰¹⁰⁰⁰²⁸⁰⁰⁰⁰⁰00200012000285919988800040 0002004131038 00004 99880CO-CH(OCH₃)₂, -C(CH₃)=C(CH₃)-CO-CH₂-SCH₃, -C(CH₃)=C(C₂H₅)-CO-CH₃, -C(CH₃)=C(C₂H₅)-CO-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-CH₂Cl, -C(CH₃)=C(C₂H₅)-CO-CH₂Br, -C(CH₃)=C(C₂H₅)-CO-CHCl₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-CH(OCH₃)₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-SCH₃, -C(CH₃)=C(Cl)-CO-CH₃, -C(CH₃)=C(Cl)-CO-C₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-n-C₄H₉, -C(CH₃)=C(Cl)-CO-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-CH₂Cl, -C(CH₃)=C(Cl)-CO-CHCl₂, -C(CH₃)=C(Cl)-CO-CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-CH(OCH₃)₂, -C(CH₃)=C(Cl)-CO-CH₂-SCH₃, -C(CH₃)=C(Br)-CO-CH₃, -C(CH₃)=C(Br)-CO-C₂H₅, -C(CH₃)=C(Br)-CO-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-n-C₄H₉, -C(CH₃)=C(Br)-CO-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-CH₂Cl, -C(CH₃)=C(Br)-CO-CH₂Br, -C(CH₃)=C(Br)-CO-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-CH(OCH₃)₂, -C(CH₃)=C(Br)-CO-CH₂-SCH₃, -C(CH₃)=C(CN)-CO-CH₃, -C(CH₃)=C(CN)-CO-C₂H₅, -C(CH₃)=C(CN)-CO-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-n-C₄H₉, -C(CH₃)=C(CN)-CO-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-CH₂Cl, -C(CH₃)=C(CN)-CO-CH₂Br, -C(CH₃)=C(CN)-CO-CHCl₂, -C(CH₃)=C(CN)-CO-CH₂-OCH₃, -C(CH₃)=C(CN)-CO-CH(OCH₃)₂, -C(CH₃)=C(CN)-CO-CH₂-SCH₃, -C(CH₃)=CH-CO-C₆H₅, -C(CH₃)=CH-CO-(4-Cl-C₆H₄), -C(CH₃)=C(CH₃)-CO-C₆H₅, -C(CH₃)=C(CH₃)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(C₂H₅)-CO-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(Cl)-CO-C₆H₅, -C(CH₃)=C(Br)-CO-C₆H₅, -C(CH₃)=C(CN)-CO-C₆H₅, -C(CH₃)=CH-CO-NH₂, -C(CH₃)=CH-CO-NHCH₃, -C(CH₃)=CH-CO-N(CH₃)₂, -C(CH₃)=CH-CO-NH-C₂H₅, -C(CH₃)=CH-CO-N(C₂H₅)₂, -C(CH₃)=CH-CO-NH-n-C₃H₇, -C(CH₃)=CH-CO-NH-i-C₃H₇, -C(CH₃)=CH-CO-NH-tert.-C₄H₉, -C(CH₃)=CH-CO-NH-cyclopropyl, -C(CH₃)=CH-CO-NH-cyclobutyl, -C(CH₃)=CH-CO-NH-cyclopentyl, -C(CH₃)=CH-CO-NH-cyclohexyl, -C(CH₃)=CH-CO-NH-cycloheptyl, -C(CH₃)=CH-CO-NH-cyclooctyl, -C(CH₃)=CH-CO-pyrrolidin-1-yl, -C(CH₃)=CH-CO-piperidin-1-yl, -C(CH₃)=CH-CO-morpholin-4-yl, -C(CH₃)=CH-CO-NH-CH₂CH=CH₂, -C(CH₃)=CH-CO-NH-CH₂C≡CH, -C(CH₃)=CH-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=CH-CO-NH-(CH₂)₂Cl, -C(CH₃)=CH-CO-NH-C₆H₅, -C(CH₃)=C(CH₃)-CO-NH₂, -C(CH₃)=C(CH₃)-CO-NHCH₃, -C(CH₃)=C(CH₃)-CO-N(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-C₂H₅, -C(CH₃)=C(CH₃)-CO-N(C₂H₅)₂, -C(CH₃)=C(CH₃)-CO-NH-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-NH- cyclopropyl, -C(CH₃)=C(CH₃)-CO-NH-cyclobutyl, -C(CH₃)=C(CH₃)-CO-NH-cyclopentyl, -C(CH₃)=C(CH₃)-CO-NH- cyclohexyl, -C(CH₃)=C(CH₃)-CO-NH-cycloheptyl, -C(CH₃)=C(CH₃)-CO-NH-cyclooctyl, -C(CH₃)=C(CH₃)-CO- pyrrolidin-1-yl, -C(CH₃)=C(CH₃)-CO-piperidin-1-yl, -C(CH₃)=C(CH₃)-CO-morpholin-4-yl, -C(CH₃)=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CH₃)-CO-NH-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-NH₂, -C(CH₃)=C(C₂H₅)-CO-NHCH₃, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)₂, -C(CH₃)=C(C₂H₅)-CO-NH-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-N(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-NH- cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclo­ hexyl, -C(CH₃)=C(C₂H₅)-CO-NH-cycloheptyl, -C(CH₃)=C(C₂H₅)-CO-NH- cyclooctyl, -C(CH₃)=C(C₂H₅)-CO-pyrrolidin-1-yl, -C(CH₃)=C(C₂H₅)-CO-piperidin-1-yl, -C(CH₃)=C(C₂H₅)-CO- morpholin-4-yl, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(C₂H₅)-CO-NH-C₆H₅, -C(CH₃)=C(Cl)-CO-NH₂, -C(CH₃)=C(Cl)-CO-NHCH₃, -C(CH₃)=C(Cl)-CO-N(CH₃)₂, -C(CH₃)=C(Cl)-CO-NH-C₂H₅, -C(CH₃)=C(Cl)-CO-N(C₂H₅)₂, -C(CH₃)=C(Cl)-CO-NH-n-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-i-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-NH-cyclopropyl, -C(CH₃)=C(Cl)-CO-NH-cyclobutyl, -C(CH₃)=C(Cl)-CO-NH-cyclopentyl, -C(CH₃)=C(Cl)-CO-NH-cyclohexyl, -C(CH₃)=C(Cl)-CO-NH-cycloheptyl, -C(CH₃)=C(Cl)-CO-NH-cyclooctyl, -C(CH₃)=C(Cl)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Cl)-CO-piperidin-1- yl, -C(CH₃)=C(Cl)-CO-morpholin-4-yl, -C(CH₃)=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -C(CH₃)=C(Cl)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Cl)-CO-NH-C₆H₅, -C(CH₃)=C(Br)-CO-NH₂, -C(CH₃)=C(Br)-CO-NHCH₃, -C(CH₃)=C(Br)-CO-N(CH₃)₂, -C(CH₃)=C(Br)-CO-NH-C₂H₅, -C(CH₃)=C(Br)-CO-N(C₂H₅)₂, -C(CH₃)=C(Br)-CO-NH-n-C₃H₇, -C(CH₃)=C(Br)-CO-NH-i-C₃H₇, -C(CH₃)=C(Br)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-NH-cyclopropyl, -C(CH₃)=C(Br)-CO-NH-cyclobutyl, -C(CH₃)=C(Br)-CO-NH-cyclopentyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cycloheptyl, -C(CH₃)=C(Br)-CO-NH-cyclooctyl, -C(CH₃)=C(Br)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Br)-CO-piperidin-1-yl, -C(CH₃)=C(Br)-CO-morpholin-4-yl, -C(CH₃)=C(Br)-CO-NH-CH₂CH=C(Br)₂, -C(CH₃)=C(Br)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Br)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Br)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Br)-CO-NH-C₆H₅, -C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CN)-CO-NHCH₃, -C(CH₃)=C(CN)-CO-N(CH₃)₂, -C(CH₃)=C(CN)-CO-NH-C₂H₅, -C(CH₃)=C(CN)-CO-N(C₂H₅)₂, -C(CH₃)=C(CN)-CO-NH-n-C₃H₇, -C(CH₃)=C(CN)-CO-NH-i-C₃H₇, -C(CH₃)=C(CN)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-NH-cyclopropyl, -C(CH₃)=C(CN)-CO-NH-cyclobutyl, -C(CH₃)=C(CN)-CO-NH-cyclopentyl, -C(CH₃)=C(CN)-CO-NH-cyclohexyl, -C(CH₃)=C(CN)-CO-NH-cycloheptyl, -C(CH₃)=C(CN)-CO-NH-cyclooctyl, -C(CH₃)=C(CN)-CO-pyrrolidin-1-yl, -C(CH₃)=C(CN)-CO-piperidin-1-yl, -C(CH₃)=C(CN)-CO-morpholin-4-yl, -C(CH₃)=C(CN)-CO-NH-CH₂CH=C(CN)₂, -C(CH₃)=C(CN)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CN)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CN)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CN)-CO-NH-C₆H₅, -C(CH₃)=CH-CO-SCH₃, -C(CH₃)=CH-CO-SC₂H₅, -C(CH₃)=CH-CO-S-n-C₃H₇, -C(CH₃)=CH-CO-S-i-C₃H₇, -C(CH₃)=CH-CO-S-n-C₄H₉, -C(CH₃)=CH-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-SCH₃, -C(CH₃)=C(CH₃)-CO-SC₂H₅, -C(CH₃)=C(CH₃)-CO-S-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-S-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-SCH₃, -C(CH₃)=C(C₂H₅)-CO-SC₂H₅, -C(CH₃)=C(C₂H₅)-CO-S-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-SCH₃, -C(CH₃)=C(Cl)-CO-SC₂H₅, -C(CH₃)=C(Cl)-CO-S-n-C₃H₇, -C(CH₃)=C(Cl)-CO-S-i-C₃H₇, -C(CH₃)=C(Cl)-CO-S-n-C₄H₉, -C(CH₃)=C(Cl)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-SCH₃, -C(CH₃)=C(Br)-CO-SC₂H₅, -C(CH₃)=C(Br)-CO-S-n-C₃H₇, -C(CH₃)=C(Br)-CO-S-i-C₃H₇, -C(CH₃)=C(Br)-CO-S-n-C₄H₉, -C(CH₃)=C(Br)-CO-S-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-SCH₃, -C(CH₃)=C(CN)-CO-SC₂H₅, -C(CH₃)=C(CN)-CO-S-n-C₃H₇, -C(CH₃)=C(CN)-CO-S-i-C₃H₇, -C(CH₃)=C(CN)-CO-S-N-C₄H₉, -C(CH₃)=C(CN)-CO-S-tert.-C₄H₉, -C(CH₃)=C(COCH₃)-CO-OCH₃, -C(CH₃)=C(COC₂H₅)-CO-OCH₃, -C(CH₃)=C(CO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COCH₃)-CO-OC₂H₅, -C(CH₃)=C(COC₂H₅)-CO-OC₂H₅, -C(CH₃)=C(CO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COCH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(COC₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-OCH₃, -C(CH₃)=C(CF₃)-CO-OC₂H₅, -C(CH₃)=C(CF₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CF₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(COOCH₃)₂, -C(CH₃)=C(COOC₂H₅)₂, -C(CH₃)=C(COOCH₃)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)₂, -C(CH₃)=CH-CH=CH-COOH, -C(CH₃)=CH-CH=CH-CO-OCH₃, -C(CH₃)=CH-CH=CH-CO-OC₂H₅, -C(CH₃)=CH-CH=C(COOCH₃)₂, -C(CH₃)=CH-CH=C(CN)-CO-OCH₃, -C(CH₃)=CH-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CN)CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH₂, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -C(CH₃)=CH-(CH₂)₂-COOH, -C(CH₃)=CH-(CH₂)₂-CO-OCH₃, -C(CH₃)=CH-(CH₂)₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(COOCH₃)₂, -C(CH₃)=CH-CH₂-CH(COOC₂H₅)₂, -C(CH₃)=CH-CH₂-CH(CN)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CN)-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -C(CH₃)=CH-(CH₂)₂-CO-NH₂, -C(CH₃)=CH-(CH₂)₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-COOH, -C(CH₃)=CH-CH₂-CO-OCH₃, -C(CH₃)=CH-CH₂-CO-OC₂H₅, -C(CH₃)=C(COOCH₃)-CH₂-CO-OCH₃, -C(CH₃)=C(COOCH₃)-CH₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CO-NH₂, -C(CH₃)=CH-CH₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-CO-N(CH₃)₂.
wobei W für eine der folgenden Bedeutungen steht:
-CHO, -COCH₃, -COC₂H₅, -CO-n-C₃H₇, -CO-i-C₃H₇, -CO-n-C₄H₉, -CO-i-C₄H₉, -CO-s-C₄H₉, -CO-tert.-C₄H₉, -CO-CH₂CH=CH₂, -CO-CF₃, -COCCl₃, -COCH₂C≡CH, -CO-cyclopropyl, -CO-cyclobutyl, -CO-cyclopentyl, -CO-cyclohexyl, -CO-CN, -CO-COOCH₃, -CO-COOC₂H₅, -CH=NH, -CH=NCH₃, -CH=NC₂H₅, -CH=N-n-C₃H₅, -CH=N-i-C₃H₅, -CH=N-n-C₄H₉, -CH=NCH₂CH=CH₂, -CH=NCH₂CH=CH₂-CH₃, -CH=NCH₂C≡CH, -CH=NCH₂C≡C-CH₃, -CH=N-cyclopropyl, -CH=N-cyclobutyl, -CH=N-cyclopentyl, -CH=N-cyclohexyl, -CH=N-cycloheptyl, -CH=N-CH₂-CH₂Cl, -CH=N-CH₂Cl, -CH=N-C₆H₅, -CH=N-4-Br-C₆H₄, -CH=N-3-F-C₆H₄, -CH=N-4-F-C₆H₄, -CH=N-2-Cl-C₆H₄, -CH=N-3-Cl-C₆H₄, -CH=N-4-Cl-C₆H₄, -CH=N-2-Br-C₆H₄, -CH=N-2-F-C₆H₄, -CH=N-2-CH₃-C₆H₄, -CH=N-3-CH₃-C₆H₄, -CH=N-4-CH₃-C₆H₄, -CH=N-2-CF₃-C₆H₄, -CH=N-3-CF₃-C₆H₄, -CH=N-4-CF₃-C₆H₄, -CH=N-2-OCH₃-C₆H₄, -CH=N-3-OCH₃-C₆H₄, -CH=N-4-OCH₃-C₆H₄, -CH=N-4-NO₂-C₆H₄, -CH=N-4-CN-C₆H₄, -CH=N-2,4-(Cl,Cl)-C₆H₄, -CH=N-2,4-(CH₃,CH₃)-C₆H₄, -CH=N-CH₂OCH₃ -CH=N-CH₂OC₂H₅, -CH=N-CH₂CH₂OCH₃, -CH=N-CH₂CH₂OC₂H₅, -CH=N-OH, -CH=N-OCH₃, -CH=N-OC₂H₅, -CH=N-O-n-C₃H₇, -CH=N-O-i-C₃H₇, -CH=N-O-n-C₄H₉, -CH=N-O-i-C₄H₉, -CH=N-O-s-C₄H₉, -CH=N-O-tert.-C₄H₉, -CH=N-O-CH₂CH=CH₂, -CH=N-O-CH(CH₃)CH=CH₂, -CH=N-O-CH₂C≡CH, -CH=N-O-CH(CH₃)-C≡CH, -CH=N-O-CH₂-CH=CH-CH₃, -CH=N-O-CH₂-CH₂-Cl, -CH=N-O-CH₂-CH₂-F, -CH=N-O-CH₂-CF₃, -CH=N-O-CH₂-CH=CHCl, -CH=N-O-CH₂-CCl=CH₂, -CH=N-O-CH₂-CBr=CH₂, -CH=N-O-CH₂-CH=CCl-CH₃, -CH=N-OC(O)CH₃, -CH=N-OC(O)C₂H₅, -CH=N-O-CH₂-CN, -CH=N-O-CH₂-CH=CH-CH₂-O-CH₃, -CH=N-O-CH₂-CH=CH-CH₂-O-tert.-C₄H₉, -CH=N-O-(CH₂)₃-C₆H₅, -CH=N-O-(CH₂)₄-C₆H₅, -CH=N-O-(CH₂)₄-4-Cl-C₆H₄, -CH=N-O-(CH₂)₄-4-OCH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-CH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-C₆H₅, -CH=N-O-CH₂CH=CH-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CH-3-OCH₃-C₆H₄, -CH=N-O-(CH₂)₂CH=CH-4-F-C₆H₄, -CH=N-O-(CH₂)CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CHCH₂-4-OCH₃-C₆H₄, -CH=N-O-CH₂-CH=C(CH₃)-C₆H₄ -CH=N-O-(CH₂)₂CH=CH-3,4(Cl,Cl)-C₆H₃, -CH=N-O-(CH₂)₃C≡C-4-F-C₆H₄, -CH₂=N-OCHOCH₃, -CH=N-OC₂H₄OCH₃, -CH=N-OCH₂OC₂H₅, -CH=N-OCH(CH₃)OCH₃, -CH=N-OCH(CH₃)COOCH₃, -CH=N-OCH(CH₃)COO-n-C₄H₉, -CH=N-NH₂, -CH=N-NHCH₃, -CH=N-NHC₂H₅, -CH=N-NH-n-C₃H₇, -CH=N-NH-i-C₃H₇, -CH=N-NH-n-C₄H₉, -CH=N-NH-i-C₄H₉, -CH=N-NH-s-C₄H₉, -CH=N-NH-tert.-C₄H₉, -CH=N-NH-cyclopropyl, -CH=N-NH-cyclobutyl, -CH=N-NH-cyclopentyl, -CH=N-NH-cyclohexyl, -CH=N-NH-cycloheptyl, -CH=N-N(CH₃)₂, -CH=N-N(C₂H₅)₂, -CH=N-N(C₃H₇)₂, -CH=N-N(i-C₃H₇)(CH₃), -CH=N-NHCH₂-C=CH, -CH=N-NHCH₂-C≡CH, -CH=N-N(CH₃)-CH₂-C≡CH, -CH=N-NHCH₂CF₃, -CH=N-NH-CO-CH₃, -CH=N-NH-CO-CH₂H₅, -CH=N-NH-COOCH₃, -CH=N-NH-COOC₂H₅, -CH=N-NH-COO-tert.-C₄H₉, -CH=N-pyrrolidin-1-yl, -CH=N-piperidin-1-yl, -CH=N-morpholin-4-yl, -CH=N-NH-C₆H₅, -CH=N-NH-(4-Cl-C₆H₄), -CH=N-NH-(4-NO₂-C₆H₄), -CH=N-NH-(4-F-C₆H₄), -CH=N-NH-(4-CH₃O-C₆H₄), -CH=N-NH-(2,4-Cl₂-C₆H₃), -CH=N-NH-(2,4-(NO₂)₂-C₆H₃), -CH=N-NH-CO-NH₂, -CH=N-NH-CO-NHCH₃, -CH=N-NH-CO-NHC₂H₅, -CH=N-NH-CO-N(CH₃)₂, -CH=CH-COOH, -CH=CH-CO-OCH₃, -CH=CH-CO-OC₂H₅, -CH=CH-CO-O-n-C₃H₇, -CH=CH-CO-O-i-C₃H₇, -CH=CH-CO-O-n-C₄H₉, -CH=CH-CO-O-tert.-C₄H₉, -CH=CH-CO-O-cyclopropyl, -CH=CH-CO-O-cyclobutyl, -CH=CH-CO-O-cyclopentyl, -CH=CH-CO-O-cyclohexyl, -CH=CH-CO-O-cycloheptyl, -CH=C(CH₃)-COOH, -CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CO-O-n-C₃H₇, -CH=C(CH₃)-CO-O-i-C₃H₇, -CH=C(CH₃)-CO-O-n-C₄H₉, -CH=C(CH₃)-CO-O-tert.-C₄H₉, -CH=C(CH₃)-CO-O-cyclopropyl, -CH=C(CH₃)-CO-O-cyclobutyl, -CH=C(CH₃)-CO-O-cyclopentyl, -CH=C(CH₃)-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cycloheptyl, -CH=C(C₂H₅)-COOH, -CH=C(C₂H₅)-CO-OCH₃, -CH=C(C₂H₅)-CO-OC₂H₅, -CH=C(C₂H₅)-CO-O-n-C₃H₇, -CH=C(C₂H₅)-CO-O-i-C₃H₇, -CH=C(C₂H₅)-CO-O-n-C₄H₉, -CH=C(C₂H₅)-CO-O-tert.-C₄H₉, -CH=C(C₂H₅)-CO-O-cyclopropyl, -CH=C(C₂H₅)-CO-O-cyclobutyl, -CH=C(C₂H₅)-CO-O-cyclopentyl, -CH=C(C₂H₅)-CO-O-cyclohexyl, -CH=C(C₂H₅)-CO-O-cycloheptyl, -CH=C(Cl)-COOH, -CH=C(Cl)-CO-OCH₃, -CH=C(Cl)-CO-OC₂H₅, -CH=C(Cl)-CO-O-n-C₃H₇, -CH=C(Cl)-CO-O-i-C₃H₇, -CH=C(Cl)-CO-O-n-C₄H₉, -CH=C(Cl)-CO-O-tert.-C₄H₉, -CH=C(Cl)-CO-O-cyclopropyl, -CH=C(Cl)-CO-O-cyclobutyl, -CH=C(Cl)-CO-O-cyclopentyl, -CH=C(Cl)-CO-O-cyclohexyl, -CH=C(Cl)-CO-O-cycloheptyl, -CH=C(Br)-COOH, -CH=C(Br)-CO-OCH₃, -CH=C(Br)-CO-OC₂H₅, -CH=C(Br)-CO-O-n-C₃H₇, -CH=C(Br)-CO-O-i-C₃H₇, -CH=C(Br)-CO-O-n-C₄H₉, -CH=C(Br)-CO-O-tert.-C₄H₉, -CH=C(Br)-CO-O-cyclopropyl, -CH=C(Br)-CO-O-cyclobutyl, -CH=C(Br)-CO-O-cyclopentyl, -CH=C(Br)-CO-O-cyclohexyl, -CH=C(Br)-CO-O-cycloheptyl, -CH=C(CN)-COOH, -CH=C(CN)-CO-OCH₃, -CH=C(CN)-CO-OC₂H₅, -CH=C(CN)-CO-O-n-C₃H₇, -CH=C(CN)-CO-O-i-C₃H₇, -CH=C(CN)-CO-O-n-C₄H₉, -CH=C(CN)-CO-O-tert.-C₄H₉, -CH=C(CN)-CO-O-cyclopropyl, -CH=C(CN)-CO-O-cyclobutyl, -CH=C(CN)-CO-O-cyclopentyl, -CH=C(CN)-CO-O-cyclohexyl, -CH=C(CN)-CO-O-cycloheptyl, -CH=CH-CO-OCH₂-OCH₃, -CH=CH-CO-OCH₂-OC₂H₅, -CH=CH-CO-OCH₂-O-n-C₃H₅, -CH=CH-CO-OCH₂-O-i-C₃H₅, -CH=CH-CO-OCH(CH₃)-OCH₃, -CH=CH-CO-OCH(CH₃)-OC₂H₅, -CH=CH-CO-O-CH₂CH₂-OCH₃, -CH=CH-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-OCH₃, -CH=C(CH₃)-CO-OCH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-O-n-C₃H₅, -CH=C(CH₃)-CO-OCH₂-O-i-C₃H₅, -CH=C(CH₃)-CO-OCH(CH₃)-OCH₃, -CH=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CH₃)-CO-O-CH₂CH₂-OCH₃, -CH=C(CH₃)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-OCH₃, -CH=C(C₂H₅)-CO-OCH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-O-n-C₃H₅, -CH=C(C₂H₅)-CO-OCH₂-O-i-C₃H₅, -CH=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -CH=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OCH₃, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-OCH₃, -CH=C(Cl)-CO-OCH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-O-n-C₃H₅, -CH=C(Cl)-CO-OCH₂-O-i-C₃H₅, -CH=C(Cl)-CO-OCH(CH₃)-OCH₃, -CH=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Cl)-CO-O-CH₂CH₂-OCH₃, -CH=C(Cl)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-OCH₃, -CH=C(Br)-CO-OCH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-O-n-C₃H₅, -CH=C(Br)-CO-OCH₂-O-i-C₃H₅, -CH=C(Br)-CO-OCH(CH₃)-OCH₃, -CH=C(Br)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Br)-CO-O-CH₂CH₂-OCH₃, -CH=C(Br)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-OCH₃, -CH=C(CN)-CO-OCH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-O-n-C₃H₅, -CH=C(CN)-CO-OCH₂-O-i-C₃H₅, -CH=C(CN)-CO-OCH(CH₃)-OCH₃, -CH=C(CN)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CN)-CO-O-CH₂CH₂-OCH₃, -CH=C(CN)-CO-O-CH₂CH₂-OC₂H₅, -CH=CH-CO-OCH₂-CF₃, -CH=CH-CO-OCH₂-CCl₃, -CH=CH-CO-OCH₂-oxiranyl, -CH=CH-CO-O(CH₂)₃-Br, -CH=CH-CO-OCH₂-CH=CH₂, -CH=CH-CO-OCH₂-C≡CH, -CH=CH-CO-OCH₂-CN, -CH=CH-CO-O(CH₂)₂-CN, -CH=C(CH₃)-CO-OCH₂-CF₃, -CH=C(CH₃)-CO-OCH₂-CCl₃, -CH=C(CH₃)-CO-OCH₂-oxiranyl, -CH=C(CH₃)-CO-O(CH₂)₃-Br, -CH=C(CH₃)-CO-OCH₂-CH=CH₂, -CH=C(CH₃)-CO-OCH₂-C≡CH, -CH=C(CH₃)-CO-OCH₂-CN, -CH=C(CH₃)-CO-O(CH₂)₂-CN, -CH=C(C₂H₅)-CO-OCH₂-CF₃, -CH=C(C₂H₅)-CO-OCH₂-CCl₃, -CH=C(C₂H₅)-CO-OCH₂-oxiranyl, -CH=C(C₂H₅)-CO-O(CH₂)₃-Br, -CH=C(C₂H₅)-CO-OCH₂-CH=CH₂, -CH=C(C₂H₅)-CO-OCH₂-C≡CH, -CH=C(C₂H₅)-CO-OCH₂-CN, -CH=C(C₂H₅)-CO-O(CH₂)₂-CN, -CH=C(Cl)-CO-OCH₂-CF₃, -CH=C(Cl)-CO-OCH₂-CCl₃, -CH=C(Cl)-CO-OCH₂-oxiranyl, -CH=C(Cl)-CO-O(CH₂)₃-Br, -CH=C(Cl)-CO-OCH₂-CH=CH₂, -CH=C(Cl)-CO-OCH₂-C≡CH, -CH=C(Cl)-CO-OCH₂-CN, -CH=C(Cl)-CO-O(CH₂)₂-CN, -CH=C(Br)-CO-OCH₂-CF₃, -CH=C(Br)-CO-OCH₂-CCl₃, -CH=C(Br)-CO-OCH₂-oxiranyl, -CH=C(Br)-CO-O(CH₂)₃-Br, -CH=C(Br)-CO-OCH₂-CH=CH₂, -CH=C(Br)-CO-OCH₂-C≡CH, -CH=C(Br)-CO-OCH₂-CN, -CH=C(Br)-CO-O(CH₂)₂-CN, -CH=C(CN)-CO-OCH₂-CF₃, -CH=C(CN)-CO-OCH₂-CCl₃, -CH=C(CN)-CO-OCH₂-oxiranyl -CH=C(CN)-CO-O(CH₂)₃-Br, -CH=C(CN)-CO-OCH₂-CH=CH₂, -CH=C(CN)-CO-OCH₂-C≡CH, -CH=C(CN)-CO-OCH₂-CN, -CH=C(CN)-CO-O(CH₂)₂-CN, -CH=CH-CO-CH₃, -CH=CH-CO-C₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-i-C₃H₇, -CH=CH-CO-n-C₄H₉, -CH=CH-CO-tert.-C₄H₉, -CH=CH-CO-CH₂Cl, -CH=CH-CO-CH₂Br, -CH=CH-CO-CHCl₂, -CH=CH-CO-CH₂-OCH₃, -CH=CH-CO-CH(OCH₃)₂, -CH=CH-CO-CH₂-SCH₃, -CH=C(CH₃)-CO-CH₃, -CH=C(CH₃)-CO-C₂H₅, -CH=C(CH₃)-CO-n-C₃H₇, -CH=C(CH₃)-CO-i-C₃H₇, -CH=C(CH₃)-CO-n-C₄H₉, -CH=C(CH₃)-CO-tert.-C₄H₉, -CH=C(CH₃)-CO-CH₂Cl, -CH=C(CH₃)-CO-CH₂Br, -CH=C(CH₃)-CO-CHCl₂, -CH=C(CH₃)-CO-CH₂-OCH₃, -CH=C(CH₃)-CO-CH(OCH₃)₂, -CH=C(CH₃)-CO-CH₂-SCH₃, -CH=C(C₂H₅)-CO-CH₃, -CH=C(C₂H₅)-CO-C₂H₅, -CH=C(C₂H₅)-CO-n-C₃H₇, -CH=C(C₂H₅)-CO-i-C₃H₇, -CH=C(C₂H₅)-CO-n-C₄H₉, -CH=C(C₂H₅)-CO-tert.-C₄H₉, -CH=C(C₂H₅)-CO-CH₂Cl, -CH=C(C₂H₅)-CO-CH₂Br, -CH=C(C₂H₅)-CO-CHCl₂, -CH=C(C₂H₅)-CO-CH₂-OCH₃, -CH=C(C₂H₅)-CO-CH(OCH₃)₂, -CH=C(C₂H₅)-CO-CH₂-SCH₃, -CH=C(Cl)-CO-CH₃, -CH=C(Cl)-CO-C₂H₅, -CH=C(Cl)-CO-n-C₃H₇, -CH=C(Cl)-CO-i-C₃H₇, -CH=C(Cl)-CO-n-C₄H₉, -CH=C(Cl)-CO-tert.-C₄H₉, -CH=C(Cl)-CO-CH₂Cl, -CH=C(Cl)-CO-CH₂Br, -CH=C(Cl)-CO-CHCl₂, -CH=C(Cl)-CO-CH₂-OCH₃, -CH=C(Cl)-CO-CH(OCH₃)₂, -CH=C(Cl)-CO-CH₂-SCH₃, -CH=C(Br)-CO-CH₃, -CH=C(Br)-CO-C₂H₅, -CH=C(Br)-CO-n-C₃H₇, -CH=C(Br)-CO-i-C₃H₇, -CH=C(Br)-CO-n-C₄H₉, -CH=C(Br)-CO-tert.-C₄H₉, -CH=C(Br)-CO-CH₂Cl, -CH=C(Br)-CO-CH₂Br, -CH=C(Br)-CO-CHCl₂, -CH=C(Br)-CO-CH₂-OCH₃, -CH=C(Br)-CO-CH(OCH₃)₂, -CH=C(Br)-CO-CH₂-SCH₃, -CH=C(CN)-CO-CH₃, -CH=C(CN)-CO-C₂H₅, -CH=C(CN)-CO-n-C₃H₇, -CH=C(CN)-CO-i-C₃H₇, -CH=C(CN)-CO-n-C₄H₉, -CH=C(CN)-CO-tert.-C₄H₉, -CH=C(CN)-CO-CH₂Cl, -CH=C(CN)-CO-CH₂Br, -CH=C(CN)-CO-CHCl₂, -CH=C(CN)-CO-CH₂-OCH₃, -CH=C(CN)-CO-CH(OCH₃)₂, -CH=C(CN)-CO-CH₂-SCH₃, -CH=CH-CO-C₆H₅, -CH=CH-CO-(4-Cl-C₆H₄), -CH=C(CH₃)-CO-C₆H₅, -CH=C(CH₃)-CO-(4-Cl-C₆H₄), -CH=C(C₂H₅)-CO-C₆H₅, -CH=C(C₂H₅)-CO-(4-Cl-C₆H₄), -CH=C(Cl)-CO-C₆H₅, -CH=C(Br)-CO-C₆H₅, -CH=C(CN)-CO-C₆H₅, -CH=CH-CO-NH₂, -CH=CH-CO-NHCH₃, -CH=CH-CO-N(CH₃)₂, -CH=CH-CO-NH-C₂H₅, -CH=CH-CO-N(C₂H₅)₂, -CH=CH-CO-NH-n-C₃H₇, -CH=CH-CO-NH-i-C₃H₇, -CH=CH-CO-NH-tert.-C₄H₉, -CH=CH-CO-NH-cyclopropyl, -CH=CH-CO-NH-cyclobutyl, -CH=CH-CO-NH-cyclopentyl, -CH=CH-CO-NH-cyclohexyl, -CH=CH-CO-NH-cycloheptyl, -CH=CH-CO-NH-cyclooctyl, -CH=CH-CO-pyrrolidin-1-yl, -CH=CH-CO-piperidin-1-yl, -CH=CH-CO-morpholin-4-yl, -CH=CH-CO-NH-CH₂CH=CH₂, -CH=CH-CO-NH-CH₂C≡CH, -CH=CH-CO-N(CH₃)-CH₂C≡CH, -CH=CH-CO-NH-(CH₂)₂Cl, -CH=CH-CO-NH-C₆H₅, -CH=C(CH₃)-CO-NH₂, -CH=C(CH₃)-CO-NHCH₃, -CH=C(CH₃)-CO-N(CH₃)₂, -CH=C(CH₃)-CO-NH-C₂H₅, -CH=C(CH₃)-CO-N(C₂H₅)₂, -CH=C(CH₃)-CO-NH-n-C₃H₇, -CH=C(CH₃)-CO-NH-i-C₃H₇, -CH=C(CH₃)-CO-NH-tert.-C₄H₉, -CH=C(CH₃)-CO-NH-cyclopropyl, -CH=C(CH₃)-CO-NH-cyclobutyl, -CH=C(CH₃)-CO-NH-cyclopentyl, -CH=C(CH₃)-CO-NH-cyclohexyl, -CH=C(CH₃)-CO-NH-cycloheptyl, -CH=C(CH₃)-CO-NH-cyclooctyl, -CH=C(CH₃)-CO-pyyrolidin-1-yl, -CH=C(CH₃)-CO-piperidin-1-yl, -CH=C(CH₃)-CO-morpholin-4-yl, -CH=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -CH=C(CH₃)-CO-NH-CH₂C≡CH, -CH=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CH₃)-CO-NH-(CH₂)₂Cl, -CH=C(CH₃)-CO-NH-C₆H₅, -CH=C(C₂H₅)-CO-NH₂, -CH=C(C₂H₅)-CO-NHCH₃, -CH=C(C₂H₅)-CO-N(CH₃)₂, -CH=C(C₂H₅)-CO-NH-C₂H₅, -CH=C(C₂H₅)-CO-N(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-n-C₃H₇, -CH=C(C₂H₅)-CO-NH-i-C₃H₇, -CH=C(C₂H₅)-CO-NH-tert.-C₄H₉, -CH=C(C₂H₅)-CO-NH-cyclopropyl, -CH=C(C₂H₅)-CO-NH-cyclobutyl, -CH=C(C₂H₅)-CO-NH-cyclopentyl, -CH=C(C₂H₅)-CO-NH-cyclohexyl, -CH=C(C₂H₅)-CO-NH-cycloheptyl, -CH=C(C₂H₅)-CO-NH-cyclooctyl, -CH=C(C₂H₅)-CO-pyrrolidin-1-yl, -CH=C(C₂H₅)-CO-piperidin-1-yl, -CH=C(C₂H₅)-CO-morpholin-4-yl, -CH=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-CH₂C≡CH, -CH=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -CH=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -CH=C(C₂H₅)-CO-NH-C₆H₅, -CH=C(Cl)-CO-NH₂, -CH=C(Cl)-CO-NHCH₃, -CH=C(Cl)-CO-N(CH₃)₂, -CH=C(Cl)-CO-NH-C₂H₅, -CH=C(Cl)-CO-N(C₂H₅)₂, -CH=C(Cl)-CO-NH-n-C₃H₇, -CH=C(Cl)-CO-NH-i-C₃H₇, -CH=C(Cl)-CO-NH-tert.-C₄H₉, -CH=C(Cl)-CO-NH-cyclopropyl, -CH=C(Cl)-CO-NH-cyclobutyl, -CH=C(Cl)-CO-NH-cyclopentyl, -CH=C(Cl)-CO-NH-cyclohexyl, -CH=C(Cl)-CO-NH-cycloheptyl, -CH=C(Cl)-CO-NH-cyclooctyl, -CH=C(Cl)-CO-pyrrolidin-1-yl, -CH=C(Cl)-CO-piperidin-1-yl, -CH=C(Cl)-CO-morpholin-4-yl, -CH=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -CH=C(Cl)-CO-NH-CH₂C≡CH, -CH=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Cl)-CO-NH-(CH₂)₂Cl, -CH=C(Cl)-CO-NH-C₆H₅, -CH=C(Br)-CO-NH₂, -CH=C(Br)-CO-NHCH₃, -CH=C(Br)-CO-N(CH₃)₂, -CH=C(Br)-CO-NH-C₂H₅, -CH=C(Br)-CO-N(C₂H₅)₂, -CH=C(Br)-CO-NH-n-C₃H₇, -CH=C(Br)-CO-NH-i-C₃H₇, -CH=C(Br)-CO-NH-tert.-C₄H₉, -CH=C(Br)-CO-NH-cyclopropyl, -CH=C(Br)-CO-NH-cyclobutyl, -CH=C(Br)-CO-NH-cyclopentyl, -CH=C(Br)-CO-NH-cyclohexyl, -CH=C(Br)-CO-NH-cycloheptyl, -CH=C(Br)-CO-NH-cyclooctyl, -CH=C(Br)-CO-pyrrolidin-1-yl, -CH=C(Br)-CO-piperidin-1-yl, -CH=C(Br)-CO-morpholin-4-yl, -CH=C(Br)-CO-NH-CH₂CH=C(Br)₂, -CH=C(Br)-CO-NH-CH₂C≡CH, -CH=C(Br)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Br)-CO-NH-(CH₂)₂Cl, -CH=C(Br)-CO-NH-C₆H₅, -CH=C(CN)-CO-NH₂, -CH=C(CN)-CO-NHCH₃, -CH=C(CN)-CO-N(CH₃)₂, -CH=C(CN)-CO-NH-C₂H₅, -CH=C(CN)-CO-N(C₂H₅)₂, -CH=C(CN)-CO-NH-n-C₃H₇, -CH=C(CN)-CO-NH-i-C₃H₇, -CH=C(CN)-CO-NH-tert.-C₄H₉, -CH=C(CN)-CO-NH-cyclopropyl, -CH=C(CN)-CO-NH-cyclobutyl, -CH=C(CN)-CO-NH-cyclopentyl, -CH=C(CN)-CO-NH-cyclohexyl, -CH=C(CN)-CO-NH-cycloheptyl, -CH=C(CN)-CO-NH-cyclooctyl, -CH=C(CN)-CO-pyrrolidin-1-yl, -CH=C(CN)-CO-piperidin-1-yl, -CH=C(CN)-CO-morpholin-4-yl, -CH=C(CN)-CO-NH-CH₂CH=C(CN)₂, -CH=C(CN)-CO-NH-CH₂C≡CH, -CH=C(CN)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CN)-CO-NH-(CH₂)₂Cl, -CH=C(CN)-CO-NH-C₆H₅, -CH=CH-CO-SCH₃, -CH=CH-CO-SC₂H₅, -CH=CH-CO-S-n-C₃H₇, -CH=CH-CO-S-i-C₃H₇, -CH=CH-CO-S-n-C₄H₉, -CH=CH-CO-S-tert.-C₄H₉, -CH=C(CH₃)-CO-SCH₃, -CH=C(CH₃)-CO-SC₂H₅, -CH=C(CH₃)-CO-S-n-C₃H₇, -CH=C(CH₃)-CO-S-i-C₃H₇, -CH=C(CH₃)-CO-S-n-C₄H₉, -CH=C(CH₃)-CO-S-tert.-C₄H₉, -CH=C(C₂H₅)-CO-SCH₃, -CH=C(C₂H₅)-CO-SC₂H₅, -CH=C(C₂H₅)-CO-S-n-C₃H₇, -CH=C(C₂H₅)-CO-S-i-C₃H₇, -CH=C(C₂H₅)-CO-S-n-C₄H₉, -CH=C(C₂H₅)-CO-S-tert.-C₄H₉, -CH=C(Cl)-CO-SCH₃, -CH=C(Cl)-CO-SC₂H₅, -CH=C(Cl)-CO-S-n-C₃H₇, -CH=C(Cl)-CO-S-i-C₃H₇, -CH=C(Cl)-CO-S-n-C₄H₉, -CH=C(Cl)-CO-S-tert.-C₄H₉, -CH=C(Br)-CO-SCH₃, -CH=C(Br)-CO-SC₂H₅, -CH=C(Br)-CO-S-n-C₃H₇, -CH=C(Br)-CO-S-i-C₃H₇, -CH=C(Br)-CO-S-n-C₄H₉, -CH=C(Br)-CO-S-tert.-C₄H₉, -CH=C(CN)-CO-SCH₃, -CH=C(CN)-CO-SC₂H₅, -CH=C(CN)-CO-S-n-C₃H₇, -CH=C(CN)-CO-S-i-C₃H₇, -CH=C(CN)-CO-S-n-C₄H₉, -CH=C(CN)-CO-S-tert.-C₄H₉, -CH=C(COCH₃)-CO-OCH₃, -CH=C(COC₂H₅)-CO-OCH₃, -CH=C(CO-n-C₃H₇)-CO-OCH₃, -CH=C(COCH₃)-CO-OC₂H₅, -CH=C(COC₂H₅)-CO-OC₂H₅, -CH=C(CO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COCH₃)-CO-O-n-C₃H₇, -CH=C(COC₂H₅)-CO-O-n-C₃H₇, -CH=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-OCH₃, -CH=C(CF₃)-CO-OC₂H₅, -CH=C(CF₃)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-O-i-C₃H₇, -CH=C(CF₃)-CO-O-n-C₄H₉, -CH=C(CF₃)-CO-O-tert.-C₄H₉, -CH=C(COOCH₃)₂, -CH=C(COOC₂H₅)₂, -CH=C(COOCH₃)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)-CO-OCH₃, -CH=C(COO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)₂, -CH=CH-CH=CH-COOH, -CH=CH-CH=CH-CO-OCH₃, -CH=CH-CH=CH-CO-OC₂H₅, -CH=CH-CH=C(COOCH₃)₂, -CH=CH-CH=C(CN)-CO-OCH₃, -CH=CH-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-OCH₃, -CH=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CH=C(Cl)-CO-OCH₃, -CH=C(CH₃)-CH=C(Br)-CO-OCH₃, -CH=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-NH₂, -CH=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -CH=CH-(CH₂)₂-COOH, -CH=CH-(CH₂)₂-CO-OCH₃, -CH=CH-(CH₂)₂-CO-OC₂H₅, -CH=CH-CH₂-CH(COOCH₃)₂, -CH=CH-CH₂-CH(COOC₂H₅)₂, -CH=CH-CH₂-CH(CN)-CO-OCH₃, -CH=CH-CH₂-CH(CN)-CO-OC₂H₅, -CH=CH-CH₂-CH(CH₃)-CO-OCH₃, -CH=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -CH=CH-(CH₂)₂-CO-NH₂, -CH=CH-(CH₂)₂-CO-NH-CH₃, -CH=CH-CH₂-COOH, -CH=CH-CH₂-CO-OCH₃, -CH=CH-CH₂-CO-OC₂H₅, -CH=C(COOCH₃)-CH₂-CO-OCH₃, -CH=C(COOCH₃)-CH₂-CO-OC₂H₅, -CH=CH-CH₂-CO-NH₂, -CH=CH-CH₂-CO-NH-CH₃, -CH=CH-CH₂-CO-N(CH₃)₂, -CH(OCH₃)₂, -CH(SCH₃)₂, -CH(OC₂H₅)₂, -CH(SC₂H₅)₂, -CH(O-n-C₃H₇)₂, -CH(O-i-C₃H₇)₂, -CH(S-n-C₃H₇)₂, -CH(S-i-C₃H₇)₂, -CH(O-n-C₄H₉)₂, -CH(O-i-C₄H₉)₂, -CH(O-s-C₄H₉)₂, -CH(O-tert.-C₄H₉)₂, -CH(S-n-C₄H₉)₂, -CH(S-i-C₄H₉)₂, -CH(S-s-C₄H₉)₂, -CH(S-tert.-C₄H₉)₂, -CH(OC₅H₁₁)₂, 1,3-Dioxolan-2-yl, 1,3-Dithio­ lan-2-yl, 1,3-Oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 5-Methyl-1,3-oxathiolan-2-yl, 4-Ethyl-1,3-dioxolan-2-yl, 4-Ethyl- 1,4-dithiolan-2-yl, 4-Ethyl-1,3-oxathiolan-2-yl, 5-Ethyl-1,3-oxa­ thiolan-2-yl, 4,5-Dimethyl-1,3-dioxolan-2-yl, 4,4-Dimethyl-1,3- dioxolan-2-yl, 4,5-Dimethyl-1,3-dithiolan-2-yl, 5,5-Dimethyl-1,3- dithiolan-2-yl, 4,5-Dimethyl-1,3-oxathiolan-2-yl, 5,5-Dimethyl- 1,3-oxathiolan-2-yl, 4,4-Dimethyl-1,3-oxathiolan-2-yl, 4-Vinyl- 1,3-dioxolan-2-yl, 4-Vinyl-1,3-dithiolan-2-yl, 4-Vinyl-1,3-oxa­ thiolan-2-yl, 5-Vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3- dioxolan-2-yl, 4-Chlormethyl-1,3-dithiolan-2-yl, 4-Chlormethyl- 1,3-oxathiolan-2-yl, 5-Chlormethyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-1,3-dithio­ lan-2-yl, 4-Hydroxymethyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl- 1,3-oxathiolan-2-yl, 4-Methoxymethyl-1,3-dioxolan-2-yl, 4-Allyl­ oxymethyl-1,3-dioxolan-2-yl, 4-Propargyloxymethyl-1,3-dioxolan- 2-yl, 4-Acetoxymethyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-1,3-dithiolan-2-yl, 4-Propargyl­ oxymethyl-1,3-dithiolan-2-yl, 4-Acetoxymethyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-1,3-oxathiolan- 2-yl, 4-Allyloxymethyl-1,3-oxathiolan-2-yl, 5-Allyloxy­ methyl-1,3-oxathiolan-2-yl, 4-Propargyloxymethyl-1,3-oxathiolan-2-yl, 5-Propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxymethyl- 1,3-oxathiolan-2-yl, 5-Acetoxymethyl-1,3-oxathiolan-2-yl, 4-Methylthiomethyl-1,3-dioxolan-2-yl, 4-Methylthiomethyl-1,3- dithiolan-2-yl, 4-Carboxy-1,3-dioxolan-2-yl, 4-Carboxy-1,3- dithiolan-2-yl, 4-Methoxycarbonyl-1,3-dioxolan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-1,3-dithiolan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-4-methyl- 1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-di­ thiolan-2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-1,3- dithiolan-2-yl, 1,3-Dioxan-2-yl, 1,3-Dithian-2-yl, 1,3-Oxathian- 2-yl, 5-Methyl-1,3-dioxan-2-yl, 5-Methyl-1,3-dithian-2-yl, 5-Methyl-1,3-oxathian-2-yl, 5,5-Dimethyl-1,3-dioxan-2-yl, 4,6-Dimethyl- 1,3-dioxan-2-yl, 4,4-Dimethyl-1,3-dioxan-2-yl, 5,5-Dimethyl- 1,3-dithian-2-yl, 4,6-Dimethyl-1,3-dithian-2-yl, 4,4-Dimethyl- 1,3-dithian-2-yl, 5,5-Dimethyl-1,3-oxathian-2-yl, 4,4-Dimethyl- 1,3-oxathian-2-yl, 6,6-Dimethyl-1,3-oxathian-2-yl, 4-Hydroxymethyl-1,3-dioxan-2-yl, 4-Methoxymethyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-1,3-dithian-2-yl, 4-Methoxymethyl-1,3-dithian-2-yl, 4-Allyloxymethyl-1,3-dithian-2-yl, 4-Acetoxymethyl- 1,3-dithian-2-yl, 4-Chlormethyl-1,3-dioxan-2-yl, 4-Chlormethyl- 1,3-dithian-2-yl, 1,3-Dioxepan-2-yl, 1,3-Dithiepan-2-yl, 1,3-Di­ oxep-5-en-2-yl, 4-Methoxycarbonyl-1,3-dioxan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-1,3-dithian- 2-yl, 4-n-Butoxycarbonyl-1,3-dithian-2-yl, 4-Methoxycarbonyl-4- methyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-4-methyl- 1,3-dithian-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithian-2-yl, -C(CH₃)(OCH₃)₂, -C(CH₃)(SCH₃)₂, -C(CH₃)(OC₂H₅)₂, -C(CH₃)(SC₂H₅)₂, -C(CH₃)(O-n-C₃H₇)₂, -C(CH₃)(O-i-C₃H₇)₂, -C(CH₃)(S-n-C₃H₇)₂, -C(CH₃)(S-i-C₃H₇)₂, -C(CH₃)(O-n-C₄H₉)₂, -C(CH₃)(O-i-C₄H₉)₂, -C(CH₃)(O-s-C₄H₉)₂, -C(CH₃)(O-tert.-C₄H₉)₂, -C(CH₃)(S-n-C₄H₉)₂, -C(CH₃)(S-i-C₄H₉)₂, -C(CH₃)(S-s-C₄H₉)₂, -C(CH₃)(S-tert.-C₄H₉)₂, -C(CH₃)(O-n-C₅H₁₁)′′, 2-Methyl-1,3-dioxolan-2-yl, 2-Methyl-1,3-di­ thiolan-2-yl, 2-Methyl-1,3-oxathiolan-2-yl, 2,4-Dimethyl-1,3- dioxolan-2-yl, 2,4-Dimethyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-1,3- oxathiolan-2-yl, 2,5-Dimethyl-1,3-oxathiolan-2-yl, 4-Ethyl-2- methyl-1,3-dioxolan-2-yl, 4-Ethyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Ethyl-2-methyl-1,3- oxathiolan-2-yl, 2,4,5-Trimethyl-1,3-dioxolan-2-yl, 2,4,4-Trimethyl- 1,3-dioxolan-2-yl, 2,4,5-Trimethyl-1,3-dithiolan-2-yl, 2,4,4-Trimethyl-1,3-dithiolan-2-yl, 2,4,5-Trimethyl-1,3-oxathiolan- 2-yl, 2,4,4-Trimethyl-1,3-oxathiolan-2-yl, 2-Methyl-4-vinyl- 1,3-dioxolan-2-yl, 2-Methyl-4-vinyl-1,3-dithiolan-2-yl, 2-Methyl- 4-vinyl-1,3-oxathiolan-2-yl, 2-Methyl-5-vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-dioxolan-2-yl, 4-Chlormethyl-2- methyl-1,3-dithiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl- 2-methyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-2- methyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dioxolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxy- 2-methyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dithiolan-2-yl, 4-Acetoxy-2- methyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl- 2-methyl-1,3-oxathiolan-2-yl, 5-Allyloxymethyl-2- methyl-1,3-oxathiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3- oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxy-2-methyl-1,3-oxathiolan-2-yl, 5-Acetoxy-2-methyl- 1,3-oxathiolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dioxolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-2- methyl-1,3-dioxolan-2-yl, 4-Carboxy-2-methyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-2- methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl- 2-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-2- methyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-di­ oxolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-ethoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4- ethoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-n-butoxy­ carbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl-1,3- dithiolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-dioxan-2-yl, 2-Methyl-1,3-dithian-2-yl, 2-Methyl-1,3-oxathian-2-yl, 2,5- Dimethyl-1,3-dioxan-2-yl, 2,5-Dimethyl-1,3-dithian-2-yl, 2,5-Dimethyl- 1,3-oxathian-2-yl, 2,5,5-Trimethyl-1,3-dioxan-2-yl, 2,4,6- Trimethyl-1,3-dioxan-2-yl, 2,2,4-Trimethyl-1,3-dioxan-2-yl, 2,5,5-Trimethyl-1,3-dithian-2-yl, 2,4,6-Trimethyl-1,3-dithian-2-yl, 2,4,4-Trimethyl-1,3-dithian-2-yl, 2,5,5-Trimethyl-1,3-oxathian-2-yl, 2,4,4-Trimethyl-1,3-oxathian-2-yl, 2,6,6-Trimethyl- 1,3-oxathian-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-2- methyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dithian-2-yl, 4-Methoxymethyl-2- methyl-1,3-dithian-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithian-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dithian-2-yl, 4-Chlormethyl-2- methyl-1,3-dioxan-2-yl, 4-Chlormethyl-2-methyl-1,3-dithian-2-yl, -C(CH₃)=NH, -C(CH₃)=N-CH₃, -C(CH₃)=N-C₂H₅, -C(CH₃)=N-n-C₃H₇, -(CH₃)=N-i-C₃H₇, -C(CH₃)=N-n-C₄H₉, -C(CH₃)=N-CH₂CH=CH₂, -C(CH₃)=N-CH₂CH=CH₂-CH₃, -C(CH₃)=N-CH₂C≡CH, -C(CH₃)=N-CH₂C≡C-CH₃, -C(CH₃)=N-cyclopropyl, -C(CH₃)=N-cyclobutyl, -C(CH₃)=N-cyclopentyl, -C(CH₃)=N-cyclohexyl, -C(CH₃)=N-cycloheptyl, -C(CH₃)=N-CH₂-CH₂Cl, -C(CH₃)=N-CH₂Cl, -C(CH₃)=N-C₆H₅, -C(CH₃)=N-(2-F-C₆H₄), -C(CH₃)=N-(3-F-C₆H₄), -C(CH₃)=N-(4-F-C₆H₄), -C(CH₃)=N-(2-Cl-C₆H₄), -C(CH₃)=N-(3-Cl-C₆H₄), -C(CH₃)=N-(4-Cl-C₆H₄), -C(CH₃)=N-(2-CH₃-C₆H₄), -C(CH₃)=N-(3-CH₃-C₆H₄), -C(CH₃)=N-(4-CH₃-C₆H₄), -C(CH₃)=N-(2-CF₃-C₆H₄), -C(CH₃)=N-(3-CF₃-C₆H₄), -C(CH₃)=N-(4-CF₃-C₆H₄), -C(CH₃)=N-(2-OCH₃-C₆H₄), -C(CH₃)=N-(3-OCH₃-C₆H₄), -C(CH₃)=N-(4-OCH₃-C₆H₄), -C(CH₃)=N-(4-NO₂-C₆H₄), -C(CH₃)=N-(4-CN-C₆H₄), -C(CH₃)=N-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-(2,4-(CH₃)₂-C₆H₃), -C(CH₃)=N-CH₂-OCH₃, -C(CH₃)=N-CH₂-OC₂H₅, -C(CH₃)=N-CH₂CH₂-OCH₃, -C(CH₃)=N-CH₂CH₂-OC₂H₅, -C(CH₃)=N-OH, -C(CH₃)=N-OCH₃, -C(CH₃)=N-OC₂H₅, -C(CH₃)=N-O-n-C₃H₇, -C(CH₃)=N-O-i-C₃H₇, -C(CH₃)=N-O-n-C₄H₉, -C(CH₃)=N-O-i-C₄H₉, -C(CH₃)=N-O-s-C₄H₉, -C(CH₃)=N-O-tert.-C₄H₉, -C(CH₃)=N-OCH₂-CH=CH₂, -C(CH₃)=N-OCH(CH₃)-CH=CH₂, -C(CH₃)=N-OCH₂-C≡CH, -C(CH₃)=N-CH(CH₃)-C≡CH, -C(CH₃)=N-OCH₂-CH=C-CH₃, -C(CH₃)=N-OCH₂CH₂-Cl, -C(CH₃)=N-OCH₂CH₂-F, -C(CH₃)=N-OCH₂-CF₃, -C(CH₃)=N-OCH₂-CH=CHCl, -C(CH₃)=N-OCH₂-C(Cl)=CH₂, -C(CH₃)=N-OCH₂-C(Br)=CH₂, -C(CH₃)=N-OCH₂-CH=C(Cl)-CH₃, -C(CH₃)=N-O-CO-CH₃, -C(CH₃)=N-O-CO-C₂H₅, -C(CH₃)=N-OCH₂-CN, -C(CH₃)=N-OCH₂-CH=CH-CH₂-OCH₃, -C(CH₃)=N-OCH₂-CH=CH-CH₂-O-tert.-C₄H₉, -C(CH₃)=N-O-(CH₂)₃-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-(4-Cl-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-C₆H₅, -C(CH₃)=N-OCH₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(3-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-CH₂-(4-CH₃O-C₆H₄), -C(CH₃)=N-OCH₂-CH=C(CH₃)-C₆H₅, -C(CH₃)=N-O-(CH₂)₂-CH=CH-(3,4-Cl₂-C₆H₃), -C(CH₃)=N-O-(CH₂)₃-C≡C-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-OCH₃, -C(CH₃)=N-OCH₂CH₂-OCH₃, -C(CH₃)=N-OCH₂-OC₂H₅, -C(CH₃)=N-OCH(CH₃)-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=N-NH₂, -C(CH₃)=N-NH-CH₃, -C(CH₃)=N-NH-C₂H₅, -C(CH₃)=N-NH-n-C₃H₇, -C(CH₃)=N-NH-i-C₃H₇, -C(CH₃)=N-NH-n-C₄H₉, -C(CH₃)=N-NH-i-C₄H₉, -C(CH₃)=N-NH-s-C₄H₉, -C(CH₃)=N-NH-tert.-C₄H₉, -C(CH₃)=N-NH-cyclopropyl, -C(CH₃)=N-NH- cyclobutyl, -C(CH₃)=N-NH-cyclopentyl, -C(CH₃)=N-NH-cyclohexyl, -C(CH₃)=N-NH-cycloheptyl, -C(CH₃)=N-N(CH₃)₂, -C(CH₃)=N-N(C₂H₅)₂, -C(CH₃)=N-N(n-C₃H₇)₂, -C(CH₃)=N-N(i-C₃H₇)₂, -C(CH₃)=N-NH-CH₂-C=CH, -C(CH₃)=N-NH-CH₂-C≡CH, -C(CH₃)=N-N(CH₃)-CH₂-C≡CH, -C(CH₃)=N-NH-CH₂CF₃, -C(CH₃)=N-NH-CO-CH₃, -C(CH₃)=N-NH-CO-C₂H₅, -C(CH₃)=N-NH-CO-OCH₃, -C(CH₃)=N-NH-CO-OC₂H₅, -C(CH₃)=N-NH-CO-O-tert.-C₄H₉, -C(CH₃)=N- pyrrolidin-1-yl, -C(CH₃)=N-piperidin-1-yl, -C(CH₃)=N-morpholin- 4-yl, -C(CH₃)=N-NH-C₆H₅, -C(CH₃)=N-NH-(4-Cl-C₆H₄), -C(CH₃)=N-NH-(4-NO₂-C₆H₄), -C(CH₃)=N-NH-(4-F-C₆H₄), -C(CH₃)=N-NH-(4-CH₃O-C₆H₄), -C(CH₃)=N-NH-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-NH-(2,4-(NO₂)₂-C₆H₃), -C(CH₃)=N-NH-CO-NH₂, -C(CH₃)=N-NH-CO-NHCH₃, -C(CH₃)=N-NH-CO-NHC₂H₅, -C(CH₃)=N-NH-CO-N(CH₃)₂, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=CH-CO-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -(CH₃)=CH-CO-O-n-C₄H₉, -C(CH₃)=CH-CO-O-tert.-C₄H₉, -C(CH₃)=CH-CO-O-cyclopropyl, -C(CH₃)=CH-CO-O-cyclobutyl, -C(CH₃)=CH-CO-O-cyclopentyl, -C(CH₃)=CH-CO-O-cyclohexyl, -C(CH₃)=CH-CO-O-cycloheptyl, -C(CH₃)=C(CH₃)-COOH, -C(CH₃)=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CH )-CO-O-cyclopropyl, -C(CH₃)=C(CH₃)-CO-O-cyclobutyl, -C(CH₃)=C(CH₃)-CO-O-cyclopentyl, -C(CH₃)=C(CH₃)-CO-O-cyclohexyl, -C(CH₃)=C(CH₃)-CO-O-cycloheptyl, -C(CH₃)=C(C₂H₅)-COOH, -C(CH₃)=C(C₂H₅)-CO-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-cyclo­ propyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-O- cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-O-cycloheptyl, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-O-n-C₄H₉, -C(CH₃)=C(Cl)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-O-cyclopropyl, -C(CH₃)=C(Cl)-CO-O-cyclobutyl, -C(CH₃)=C(Cl)-CO-O-cyclopentyl, -C(CH₃)=C(Cl)-CO-O-cyclohexyl, -C(CH₃)=C(Cl)-CO-O-cycloheptyl, -C(CH₃)=C(Br)-COOH, -C(CH₃)=C(Br)-CO-OCH₃, -C(CH₃)=C(Br)-CO-OC₂H₅, -C(CH₃)=C(Br)-CO-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-O-n-C₄H₉, -C(CH₃)=C(Br)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-O-cyclopropyl, -C(CH₃)=C(Br)-CO-O-cyclobutyl, -C(CH₃)=C(Br)-CO-O-cyclopentyl, -C(CH₃)=C(Br)-CO-O-cyclohexyl, -C(CH₃)=C(Br)-CO-O-cycloheptyl, -C(CH₃)=C(CN)-COOH, -C(CH₃)=C(CN)-CO-OCH₃, -C(CH₃)=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CN)-CO-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-O-n-C₄H₉, -C(CH₃)=C(CN)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-O-cyclopropyl, -C(CH₃)=C(CN)-CO-O-cyclobutyl, -C(CH₃)=C(CN)-CO-O-cyclopentyl, -C(CH₃)=C(CN)-CO-O-cyclohexyl, -C(CH₃)=C(CN)-CO-O-cycloheptyl, -C(CH₃)=CH-CO-OCH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-OCH(CH₃)-OCH₃, -C(CH₃)=CH-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=CH-CO-OCH₂CH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=(C₂H₅)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-O-i-C₃H₇, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -(CH₃)=C(Cl)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-O-i-C₃H₇, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-O-i-C₃H₇, -C(CH₃)=C(CN)-CO-OCH(CH₃)OCH₃, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-CF₃, -C(CH₃)=CH-CO-OCH₂-CCl₃, -C(CH₃)=CH-CO-OCH₂-oxiranyl, -C(CH₃)=CH-CO-(CH₂)₃-Br, -C(CH₃)=CH-CO-OCH₂-CH=CH₂, -C(CH₃)=CH-CO-OCH₂-C≡CH, -C(CH₃)=CH-CO-OCH₂-CN, -C(CH₃)=CH-CO-OCH₂CH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CF₃, -C(CH₃)=C(CH₃)-CO-OCH₂-CCl₃, -C(CH₃)=C(CH₃)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CH₃)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(CH₃)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CH₃)-CO-OCH₂-C≡CH, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CF₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CCl₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-oxiranyl, -C(CH₃)=C(C₂H₅)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(C₂H₅)-CO-OCH₂-C≡CH, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-C₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂-CF₃, -C(CH₃)=C(Cl)-CO-OCH₂-CCl₃, -C(CH₃)=C(Cl)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Cl)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Cl)-CO-OCH₂-CH≡CH₂, -C(CH₃)=C(Cl)-CO-OCH₂-C≡CH, -C(CH₃)=C(Cl)-CO-OCH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂-CF₃, -C(CH₃)=C(Br)-CO-OCH₂-CCl₃, -C(CH₃)=C(Br)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Br)-CO-O(CH₂)₃-Br, -C(CH₃)=C(Br)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Br)-CO-OCH₂-C≡CH, -C(CH₃)=C(Br)-CO-OCH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂CH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂-CF₃, -C(CH₃)=C(CN)-CO-OCH₂-CCl₃, -C(CH₃)=C(CN)-O-OCH₂-oxiranyl, -C(CH₃)=C(CN)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CN)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CN)-CO-OCH₂-C≡CH, -C(CH₃)=C(CN)-CO-OCH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂CH₂-CN, -C(CH₃)=CH-CO-CH₃, -C(CH₃)=CH-CO-C₂H₅, -C(CH₃)=CH-CO-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-n-C₄H₉, -C(CH₃)=CH-CO-tert.-C₄H₉, -C(CH₃)=CH-CO-CH₂Cl, -C(CH₃)=CH-CO-CH₂Br, -C(CH₃)=CH-CO-CHCl₂, -C(CH₃)=CH-CO-CH₂-OCH₃, -C(CH₃)=CH-CO-CH(OCH₃)₂, -C(CH₃)=CH-CO-CH₂-SCH₃, -C(CH₃)=C(CH₃)-CO-CH₃, -C(CH₃)=C(CH₃)-CO-C₂H₅, -C(CH₃)=C(CH₃)-CO-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-CH₂Cl, -C(CH₃)=C(CH₃)-CO-CH₂Br, -C(CH₃)=C(CH₃)-CO-CHCl₂, -C(CH₃)=C(CH₃)-CO-CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-CH(OCH₃)₂, -C(CH₃)=C(CH₃)-CO-CH₂-SCH₃, -C(CH₃)=C(C₂H₅)-CO-CH₃, -C(CH₃)=C(C₂H₅)-CO-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-CH₂Cl, -C(CH₃)=C(C₂H₅)-CO-CH₂Br, -C(CH₃)=C(C₂H₅)-CO-CHCl₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-CH(OCH₃)₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-SCH₃, -C(CH₃)=C(Cl)-CO-CH₃, -C(CH₃)=C(Cl)-CO-C₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-n-C₄H₉, -C(CH₃)=C(Cl)-CO-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-CH₂Cl, -C(CH₃)=C(Cl)-CO-CHCl₂, -C(CH₃)=C(Cl)-CO-CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-CH(OCH₃)₂, -C(CH₃)=C(Cl)-CO-CH₂-SCH₃, -C(CH₃)=C(Br)-CO-CH₃, -C(CH₃)=C(Br)-CO-C₂H₅, -C(CH₃)=C(Br)-CO-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-n-C₄H₉, -C(CH₃)=C(Br)-CO-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-CH₂Cl, -C(CH₃)=C(Br)-CO-CH₂Br, -C(CH₃)=C(Br)-CO-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-CH(OCH₃)₂, -C(CH₃)=C(Br)-CO-CH₂-SCH₃, -C(CH₃)=C(CN)-CO-CH₃, -C(CH₃)=C(CN)-CO-C₂H₅, -C(CH₃)=C(CN)-CO-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-n-C₄H₉, -C(CH₃)=C(CN)-CO-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-CH₂Cl, -C(CH₃)=C(CN)-CO-CH₂Br, -C(CH₃)=C(CN)-CO-CHCl₂, -C(CH₃)=C(CN)-CO-CH₂-OCH₃, -C(CH₃)=C(CN)-CO-CH(OCH₃)₂, -C(CH₃)=C(CN)-CO-CH₂-SCH₃, -C(CH₃)=CH-CO-C₆H₅, -C(CH₃)=CH-CO-(4-Cl-C₆H₄), -C(CH₃)=C(CH₃)-CO-C₆H₅, -C(CH₃)=C(CH₃)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(C₂H₅)-CO-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(Cl)-CO-C₆H₅, -C(CH₃)=C(Br)-CO-C₆H₅, -C(CH₃)=C(CN)-CO-C₆H₅, -C(CH₃)=CH-CO-NH₂, -C(CH₃)=CH-CO-NHCH₃, -C(CH₃)=CH-CO-N(CH₃)₂, -C(CH₃)=CH-CO-NH-C₂H₅, -C(CH₃)=CH-CO-N(C₂H₅)₂, -C(CH₃)=CH-CO-NH-n-C₃H₇, -C(CH₃)=CH-CO-NH-i-C₃H₇, -C(CH₃)=CH-CO-NH-tert.-C₄H₉, -C(CH₃)=CH-CO-NH-cyclopropyl, -C(CH₃)=CH-CO-NH-cyclobutyl, -C(CH₃)=CH-CO-NH-cyclopentyl, -C(CH₃)=CH-CO-NH-cyclohexyl, -C(CH₃)=CH-CO-NH-cycloheptyl, -C(CH₃)=CH-CO-NH-cyclooctyl, -C(CH₃)=CH-CO-pyrrolidin-1-yl, -C(CH₃)=CH-CO-piperidin-1-yl, -C(CH₃)=CH-CO-morpholin-4-yl, -C(CH₃)=CH-CO-NH-CH₂CH=CH₂, -C(CH₃)=CH-CO-NH-CH₂C≡CH, -C(CH₃)=CH-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=CH-CO-NH-(CH₂)₂Cl, -C(CH₃)=CH-CO-NH-C₆H₅, -C(CH₃)=C(CH₃)-CO-NH₂, -C(CH₃)=C(CH₃)-CO-NHCH₃, -C(CH₃)=C(CH₃)-CO-N(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-C₂H₅, -C(CH₃)=C(CH₃)-CO-N(C₂H₅)₂, -C(CH₃)=C(CH₃)-CO-NH-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-NH- cyclopropyl, -C(CH₃)=C(CH₃)-CO-NH-cyclobutyl, -C(CH₃)=C(CH₃)-CO-NH-cyclopentyl, -C(CH₃)=C(CH₃)-CO-NH- cyclohexyl, -C(CH₃)=C(CH₃)-CO-NH-cycloheptyl, -C(CH₃)=C(CH₃)-CO-NH-cyclooctyl, -C(CH₃)=C(CH₃)-CO- pyrrolidin-1-yl, -C(CH₃)=C(CH₃)-CO-piperidin-1-yl, -C(CH₃)=C(CH₃)-CO-morpholin-4-yl, -C(CH₃)=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CH₃)-CO-NH-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-NH₂, -C(CH₃)=C(C₂H₅)-CO-NHCH₃, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)₂, -C(CH₃)=C(C₂H₅)-CO-NH-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-N(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-NH- cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclo­ hexyl, -C(CH₃)=C(C₂H₅)-CO-NH-cycloheptyl, -C(CH₃)=C(C₂H₅)-CO-NH- cyclooctyl, -C(CH₃)=C(C₂H₅)-CO-pyrrolidin-1-yl, -C(CH₃)=C(C₂H₅)-CO-piperidin-1-yl, -C(CH₃)=C(C₂H₅)-CO- morpholin-4-yl, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(C₂H₅)-CO-NH-C₆H₅, -C(CH₃)=C(Cl)-CO-NH₂, -C(CH₃)=C(Cl)-CO-NHCH₃, -C(CH₃)=C(Cl)-CO-N(CH₃)₂, -C(CH₃)=C(Cl)-CO-NH-C₂H₅, -C(CH₃)=C(Cl)-CO-N(C₂H₅)₂, -C(CH₃)=C(Cl)-CO-NH-n-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-i-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-NH-cyclopropyl, -C(CH₃)=C(Cl)-CO-NH-cyclobutyl, -C(CH₃)=C(Cl)-CO-NH-cyclopentyl, -C(CH₃)=C(Cl)-CO-NH-cyclohexyl, -C(CH₃)=C(Cl)-CO-NH-cycloheptyl, -C(CH₃)=C(Cl)-CO-NH-cyclooctyl, -C(CH₃)=C(Cl)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Cl)-CO-piperidin-1- yl, -C(CH₃)=C(Cl)-CO-morpholin-4-yl, -C(CH₃)=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -C(CH₃)=C(Cl)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-N(CH₃)-CH₂≡CH, -C(CH₃)=C(Cl)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Cl)-CO-NH-C₆H₅, -C(CH₃)=C(Br)-CO-NH₂, -C(CH₃)=C(Br)-CO-NHCH₃, -C(CH₃)=C(Br)-CO-N(CH₃)₂, -C(CH₃)=C(Br)-CO-NH-C₂H₅, -C(CH₃)=C(Br)-CO-N(C₂H₅)₂, -C(CH₃)=C(Br)-CO-NH-n-C₃H₇, -C(CH₃)=C(Br)-CO-NH-i-C₃H₇, -C(CH₃)=C(Br)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-NH-cyclopropyl, -C(CH₃)=C(Br)-CO-NH-cyclobutyl, -C(CH₃)=C(Br)-CO-NH-cyclopentyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cycloheptyl, -C(CH₃)=C(Br)-CO-NH-cyclooctyl, -C(CH₃)=C(Br)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Br)-CO-piperidin-1-yl, -C(CH₃)=C(Br)-CO-morpholin-4-yl, -C(CH₃)=C(Br)-CO-NH-CH₂CH=C(Br)₂, -C(CH₃)=C(Br)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Br)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Br)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Br)-CO-NH-C₆H₅, -C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CN)-CO-NHCH₃, -C(CH₃)=C(CN)-CO-N(CH₃)₂, -C(CH₃)=C(CN)-CO-NH-C₂H₅, -C(CH₃)=C(CN)-CO-N(C₂H₅)₂, -C(CH₃)=C(CN)-CO-NH-n-C₃H₇, -C(CH₃)=C(CN)-CO-NH-i-C₃H₇, -C(CH₃)=C(CN)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-NH-cyclopropyl, -C(CH₃)=C(CN)-CO-NH-cyclobutyl, -C(CH₃)=C(CN)-CO-NH-cyclopentyl, -C(CH₃)=C(CN)-CO-NH-cyclohexyl, -C(CH₃)=C(CN)-CO-NH-cycloheptyl, -C(CH₃)=C(CN)-CO-NH-cyclooctyl, -C(CH₃)=C(CN)-CO-pyrrolidin-1-yl, -C(CH₃)=C(CN)-CO-piperidin-1-yl, -C(CH₃)=C(CN)-CO-morpholin-4-yl, -C(CH₃)=C(CN)-CO-NH-CH₂CH=C(CN)₂, -C(CH₃)=C(CN)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CN)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CN)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CN)-CO-NH-C₆H₅, -C(CH₃)=CH-SO-SCH₃, -C(CH₃)=CH-CO-SC₂H₅, -C(CH₃)=CH-CO-S-n-C₃H₇, -C(CH₃)=CH-CO-S-i-C₃H₇, -C(CH₃)=CH-CO äS-n-C₄H₉, -C(CH₃)=CH-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-SCH₃, -C(CH₃)=C(CH₃)-CO-SC₂H₅, -C(CH₃)=C(CH₃)-CO-S-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-S-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-SCH₃, -C(CH₃)=C(C₂H₅)-CO-SC₂H₅, -C(CH₃)=C(C₂H₅)-CO-S-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-SCH₃, -C(CH₃)=C(Cl)-CO-SC₂H₅, -C(CH₃)=C(Cl)-CO-S-n-C₃H₇, -C(CH₃)=C(Cl)-CO-S-i-C₃H₇, -C(CH₃)=C(Cl)-CO-S-n-C₄H₉, -C(CH₃)=C(Cl)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-SCH₃, -C(CH₃)=C(Br)-CO-SC₂H₅, -C(CH₃)=C(Br)-CO-S-n-C₃H₇, -C(CH₃)=C(Br)-CO-S-i-C₃H₇, -C(CH₃)=C(Br)-CO-S-n-C₄H₉, -C(CH₃)=C(Br)-CO-S-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-SCH₃, -C(CH₃)=C(CN)-CO-SC₂H₅, -C(CH₃)=C(CN)-CO-S-n-C₃H₇, -C(CH₃)=C(CN)-CO-S-i-C₃H₇, -C(CH₃)=C(CN)-CO-S-n-C₄H₉, -C(CH₃)=C(CN)-CO-S-tert.-C₄H₉, -C(CH₃)=C(COCH₃)-CO-OCH₃, -C(CH₃)=C(COC₂H₅)-CO-OCH₃, -C(CH₃)=C(CO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COCH₃)-CO-OC₂H₅, -C(CH₃)=C(COC₂H₅)-CO-OC₂H₅, -C(CH₃)=C(CO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COCH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(COC₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-OCH₃, -C(CH₃)=C(CF₃)-CO-OC₂H₅, -C(CH₃)=C(CF₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CF₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(COOCH₃)₂, -C(CH₃)=C(COOC₂H₅)₂, -C(CH₃)=C(COOCH₃)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)₂, -C(CH₃)=CH-CH=CH-COOH, -C(CH₃)=CH-CH=CH-CO-OCH₃, -C(CH₃)=CH-CH=CH-CO-OC₂H₅, -C(CH₃)=CH-CH=C(COOCH₃)₂, -C(CH₃)=CH-CH=C(CN)-CO-OCH₃, -C(CH₃)=CH-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH₂, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -C(CH₃)=CH-(CH₂)₂-COOH, -C(CH₃)=CH-(CH₂)₂-CO-OCH₃, -C(CH₃)=CH-(CH₂)₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(COOCH₃)₂, -C(CH₃)=CH-CH₂-CH(COOC₂H₅)₂, -C(CH₃)=CH-CH₂-CH(CN)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CN)-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -C(CH₃)=CH-(CH₂)₂-CO-NH₂, -C(CH₃)=CH-(CH₂)₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-COOH, -C(CH₃)=CH-CH₂-CO-OCH₃, -C(CH₃)=CH-CH₂-CO-OC₂H₅, -C(CH₃)=C(COOCH₃)-CH₂-CO-OCH₃, -C(CH₃)=C(COOCH₃)-CH₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CO-NH₂, -C(CH₃)=CH-CH₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-CO-N(CH₃)₂.
wobei W für eine der folgenden Bedeutungen steht:
-CHO, -COCH₃, -COC₂H₅, -CO-n-C₃H₇, -CO-i-C₃H₇, -CO-n-C₄H₉, -CO-i-C₄H₉, -CO-s-C₄H₉, -CO-tert.-C₄H₉, -CO-CH₂CH=CH₂, -CO-CF₃, -COCCl₃, -COCH₂C≡CH, -CO-cyclopropyl, -CO-cyclobutyl, -CO-cyclopentyl, -CO-cyclohexyl, -CO-CN, -CO-COOCH₃, -CO-COOC₂H₅, -CH=NH, -CH=NCH₃, -CH=NC₂H₅, -CH=N-n-C₃H₅, -CH=N-i-C₃H₅, -CH=N-n-C₄H₉, -CH=NCH₂CH=CH₂, -CH=NCH₂CH=CH₂-CH₃, -CH=NCH₂≡CH, -CH=NCH₂C≡C-CH₃, -CH=N-cyclopropyl, -CH=N-cyclobutyl, -CH=N-cyclopentyl, -CH=N-cyclohexyl, -CH=N-cycloheptyl, -CH=N-CH₂-CH₂Cl, -CH=N-CH₂Cl, -CH=N-₆H₅, -CH=N-4-Br-C₆H₄, -CH=N-3-F-C₆H₄, -CH=N-4-F-C₆H₄, -CH=N-2-Cl-C₆H₄, -CH=N-3-Cl-C₆H₄, -CH=N-4-Cl-C₆H₄, -CH=N-2-Br-C₆H₄, -CH=N-2-F-C₆H₄, -CH=N-2-CH₃-C₆H₄, -CH=N-3-CH₃-C₆H₄, -CH=N-4-CH₃-C₆H₄, -CH=N-2-CF₃-C₆H₄, -CH=N-3-CF₃-C₆H₄, -CH=N-4-CF₃-C₆H₄, -CH=N-2-OCH₃-C₆H₄, -CH=N-3-OCH₃-C₆H₄, -CH=N-4-OCH₃-C₆H₄, -CH=N-4-NO₂-C₆H₄, -CH=N-4-CN-C₆H₄, -CH=N-2,4-(Cl,Cl)-C₆H₄, -CH=N-2,4-(CH₃,CH₃)-C₆H₄, -CH=N-CH₂OCH₃ -CH=N-CH₂OC₂H₅, -CH=N-CH₂CH₂OCH₃, -CH=N-CH₂CH₂OC₂H₅, -CH=N-OH, -CH=N-OCH₃, -CH=N-OC₂H₅, -CH=N-O-n-C₃H₇, -CH=N-O-i-C₃H₇, -CH=N-O-n-C₄H₉, -CH=N-O-i-C₄H₉, -CH=N-O-s-C₄H₉, -CH=N-O-tert.-C₄H₉, -CH=N-O-CH₂CH=CH₂, -CH=N-O-CH(CH₃)CH=CH₂, -CH=N-O-CH₂C≡CH, -CH=N-O-CH(CH₃)-C≡CH, -CH=N-O-CH₂-CH=CH-CH₃, -CH=N-O-CH₂-CH₂-Cl, -CH=N-O-CH₂-CH₂-F, -CH=N-O-CH₂-CF₃, -CH=N-O-CH₂-CH=CHCl, -CH=N-O-CH₂-CCl=CH₂, -CH=N-O-CH₂-CBr=CH₂, -CH=N-O-CH₂-CH=CCl-CH₃, -CH=N-OC(O)CH₃, -CH=N-OC(O)C₂H₅, -CH=N-O-CH₂-CN, -CH=N-O-CH₂-CH=CH-CH₂-O-CH₃, -CH=N-O-CH₂-CH=CH-CH₂-O-tert.-C₄H₉, -CH=N-O-(CH₂)₃-C₆H₅, -CH=N-O-(CH₂)₄-C₆H₅, -CH=N-O-(CH₂)₄-4-Cl-C₆H₄, -CH=N-O-(CH₂)₄-4-OCH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-CH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-C₆H₅, -CH=N-O-CH₂CH=CH-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CH-3-OCH₃-C₆H₄, -CH=N-O-(CH₂)₂CH=CH-4-F-C₆H₄, -CH=N-O-(CH₂)CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CHCH₂-4-OCH₃-C₆H₄, -CH=N-O-CH₂-CH=C(CH₃)-C₆H₅, -CH=N-O-(CH₂)₂CH=CH-3,4(Cl,Cl)-C₆H₃, -CH=N-O-(CH₂)₃C≡C-4-F-C₆H₄, -CH₂=N-OCHOCH₃, -CH=N-OC₂H₄OCH₃, -CH=N-OCH₂OC₂H₅, -CH=N-OCH(CH₃)OCH₃, -CH=N-OCH(CH₃)COOCH₃, -CH=N-OCH(CH₃)COO-n-C₄H₉, -CH=N-NH₂, -CH=N-NHCH₃, -CH=N-NHC₂H₅, -CH=N-NH-n-C₃H₇, -CH=N-NH-i-C₃H₇, -CH=N-NH-n-C₄H₉, -CH=N-NH-cyclopropyl, -CH=N-NH-cyclobutyl, -CH=N-NH-cyclopentyl, -CH=N-NH-cyclohexyl, -CH=N-NH-cycloheptyl, -CH=N-N(CH₃)₂, -CH=N-N(C₂H₅)₂, -CH=N-N(C₃H₇)₂, -CH=N-N(i-C₃H₇)(CH₃), -CH=N-NHCH₂-C=CH, -CH=N-NHCH₂-C≡CH, -CH=N-N(CH₃)-CH₂-C≡CH, -CH=N-NHCH₂CF₃, -CH=N-NH-CO-CH₃, -CH=N-NH-CO-CH₂H₅, -CH=N-NH-COOCH₃, -CH=N-NH-COOC₂H₅, -CH=N-NH-COO-tert.-C₄H₉, -CH=N-pyrrolidin-1-yl, -CH=N-piperidin-1-yl, -CH=N-morpholin-4-yl, -CH=N-NH-C₆H₅, -CH=N-NH-(4-Cl-C₆H₄), -CH=N-NH-(4-NO₂-C₆H₄), -CH=N-NH-(4-F-C₆H₄), -CH=N-NH-(4-CH₃O-C₆H₄), -CH=N-NH-(2,4-Cl₂-C₆H₃), -CH=N-NH-(2,4-(NO₂)₂-C₆H₃), -CH=N-NH-CO-NH₂, -CH=N-NH-CO-NHCH₃, -CH=N-NH-CO-NHC₂H₅, -CH=N-NH-CO-N(CH₃)₂, -CH=CH-COOH, -CH=CH-CO-OCH₃, -CH=C-CO-OC₂H₅, -CH=CH-CO-O-n-C₃H₇, -CH=CH-CO-O-i-C₃H₇, -CH=CH-CO-O-n-C₄H₉, -CH=CH-CO-O-tert.-C₄H₉, -CH=CH-CO-O-cyclopropyl, -CH=CH-CO-O-cyclobutyl, -CH=CH-CO-O-cyclopentyl, -CH=CH-CO-O-cyclohexyl, -CH=CH-CO-O-cycloheptyl, -CH=C(CH₃)-COOH, -CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CO-O-n-C₃H₇, -CH=C(CH₃)-CO-O-i-C₃H₇, -CH=C(CH₃)-CO-O-n-C₄H₉, -CH=C(CH₃)-CO-O-tert.-C₄H₉, -CH=C(CH₃)-CO-O-cyclopropyl, -CH=C(CH₃)-CO-O-cyclobutyl, -CH=C(CH₃)-CO-O-cyclopentyl, -CH=C(CH₃)-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cycloheptyl, -CH=C(C₂H₅)-COOH, -CH=C(C₂H₅)-CO-OCH₃, -CH=C(C₂H₅)-CO-OC₂H₅, -CH=C(C₂H₅)-CO-O-n-C₃H₇, -CH=C(C₂H₅)-CO-O-i-C₃H₇, -CH=C(C₂H₅)-CO-O-n-C₄H₉, -CH=C(C₂H₅)-CO-O-tert.-C₄H₉, -CH=C(C₂H₅)-CO-O-cyclopropyl, -CH=C(C₂H₅)-CO-O-cyclobutyl, -CH=C(C₂H₅)-CO-O-cyclopentyl, -CH=C(C₂H₅)-CO-O-cyclohexyl, -CH=C(C₂H₅)-CO-O-cycloheptyl, -CH=C(Cl)-COOH, -CH=C(Cl)-CO-OCH₃, -CH=C(Cl)-CO-OC₂H₅, -CH=C(Cl)-CO-O-n-C₃H₇, -CH=C(Cl)-CO-O-i-C₃H₇, -CH=C(Cl)-CO-O-n-C₄H₉, -CH=C(Cl)-CO-O-tert.-C₄H₉, -CH=C(Cl)-CO-O-cyclopropyl, -CH=C(Cl)-CO-O-cyclobutyl, -CH=C(Cl)-CO-O-cyclopentyl, -CH=C(Cl)-CO-O-cyclohexyl, -CH=C(Cl)-CO-O-cycloheptyl, -CH=C(Br)-COOH, -CH=C(Br)-CO-OCH₃, -CH=C(Br)-CO-OC₂H₅, -CH=C(Br)-CO-O-n-C₃H₇, -CH=C(Br)-CO-O-i-C₃H₇, -CH=C(Br)-CO-O-n-C₄H₉, -CH=C(Br)-CO-O-tert.-C₄H₉, -CH=C(Br)-CO-O-cyclopropyl, -CH=C(Br)-CO-O-cyclobutyl, -CH=C(Br)-CO-O-cyclopentyl, -CH=C(Br)-CO-O-cyclohexyl, -CH=C(Br)-CO-O-cycloheptyl, -CH=C(CN)-COOH, -CH=C(CN)-CO-OCH₃, -CH=C(CN)-CO-OC₂H₅, -CH=C(CN)-CO-O-n-C₃H₇, -CH=C(CN)-CO-O-i-C₃H₇, -CH=C(CN)-CO-O-n-C₄H₉, -CH=C(CN)-CO-O-tert.-C₄H₉, -CH=C(CN)-CO-O-cyclopropyl, -CH=C(CN)-CO-O-cyclobutyl, -CH=C(CN)-CO-O-cyclopentyl, -CH=C(CN)-CO-O-cyclohexyl, -CH=C(CN)-CO-O-cycloheptyl, -CH=CH-CO-OCH₂-OCH₃, -CH=CH-CO-OCH₂-OC₂H₅, -CH=CH-CO-OCH₂-O-n-C₃H₅, -CH=CH-CO-OCH₂-O-i-C₃H₅, -CH=CH-CO-OCH(CH₃)-OCH₃, -CH=CH-CO-OCH(CH₃)-OC₂H₅, -CH=CH-CO-O-CH₂CH₂-OCH₃, -CH=CH-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-OCH₃, -CH=C(CH₃)-CO-OCH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-O-n-C₃H₅, -CH=C(CH₃)-CO-OCH₂-O-i-C₃H₅, -CH=C(CH₃)-CO-OCH(CH₃)-OCH₃, -CH=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CH₃)-CO-O-CH₂CH₂-OCH₃, -CH=C(CH₃)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-OCH₃, -CH=C(C₂H₅)-CO-OCH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-O-n-C₃H₅, -CH=C(C₂H₅)-CO-OCH₂-O-i-C₃H₅, -CH=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -CH=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OCH₃, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-OCH₃, -CH=C(Cl)-CO-OCH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-O-n-C₃H₅, -CH=C(Cl)-CO-OCH₂-O-i-C₃H₅, -CH=C(Cl)-CO-OCH(CH₃)-OCH₃, -CH=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Cl)-CO-O-CH₂CH₂-OCH₃, -CH=C(Cl)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-OCH₃, -CH=C(Br)-CO-OCH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-O-n-C₃H₅, -CH=C(Br)-CO-OCH₂-O-i-C₃H₅, -CH=C(Br)-CO-OCH(CH₃)-OCH₃, -CH=C(Br)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Br)-CO-O-CH₂CH₂-OCH₃, -CH=C(Br)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-OCH₃, -CH=C(CN)-CO-OCH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-O-n-C₃H₅, -CH=C(CN)-CO-OCH₂-O-i-C₃H₅, -CH=C(CN)-CO-OCH(CH₃)-OCH₃, -CH=C(CN)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CN)-CO-O-CH₂CH₂-OCH₃, -CH=C(CN)-CO-O-CH₂CH₂-OC₂H₅, -CH=CH-CO-OCH₂-CF₃, -CH=CH-CO-OCH₂-CCl₃, -CH=CH-CO-OCH₂-oxiranyl, -CH=CH-CO-O(CH₂)₃-Br, -CH=CH-CO-OCH₂-CH=CH₂, -CH=CH-CO-OCH₂-C≡CH, -CH=CH-CO-OCH₂-CN, -CH=CH-CO-O(CH₂)₂-CN, -CH=C(CH₃)-CO-OCH₂-CF₃, -CH=C(CH₃)-CO-OCH₂-CCl₃, -CH=C(CH₃)-CO-OCH₂-oxiranyl, -CH=C(CH₃)-CO-O(CH₂)₂-Br, -CH=C(CH₃)-CO-OCH₂-CH=CH₂, -CH=C(CH₃)-CO-OCH₂-C≡CH, -CH=C(CH₃)-CO-OCH₂-CN, -CH=C(CH₃)-CO-O(CH₂)₂-CN, -CH=C(C₂H₅)-CO-OCH₂-CF₃, -CH=C(C₂H₅)-CO-OCH₂-CCl₃, -CH=C(C₂H₅)-CO-OCH₂-oxiranyl, -CH=C(C₂H₅)-CO-O(CH₂)₃-Br, -CH=C(C₂H₅)-CO-OCH₂-CH=CH₂, -CH=C(C₂H₅)-CO-OCH₂-C≡CH, -CH=C(C₂H₅)-CO-OCH₂-CN, -CH=C(C₂H₅)-CO-O(CH₂)₂-CN, -CH=C(Cl)-CO-OCH₂-CF₃, -CH=C(Cl)-CO-OCH₂-CCl₃, -CH=C(Cl)-CO-OCH₂-oxiranyl, -CH=C(Cl)-CO-O(CH₂)₃-Br, -CH=C(Cl)-CO-OCH₂-CH=CH₂, -CH=C(Cl)-CO-OCH₂-C≡CH, -CH=C(Cl)-CO-OCH₂-CN, -CH=C(Cl)-CO-O(CH₂)₂-CN, -CH=C(Br)-CO-OCH₂-CF₃, -CH=C(Br)-CO-OCH₂-CCl₃, -CH=C(Br)-CO-OCH₂-oxiranyl, -CH=C(Br)-CO-O(CH₂)₃-Br, -CH=C(Br)-CO-OCH₂-CH=CH₂, -CH=C(Br)-CO-OCH₂-C≡CH, -CH=C(Br)-CO-OCH₂-CN, -CH=C(Br)-CO-O(CH₂)₂-CN, -CH=C(CN)-CO-OCH₂-CF₃, -CH=C(CN)-CO-OCH₂-CCl₃, -CH=C(CN)-CO-OCH₂-oxiranyl -CH=C(CN)-CO-O(CH₂)₃-Br, -CH=C(CN)-CO-OCH₂-CH=CH₂, -CH=C(CN)-CO-OCH₂-C≡CH, -CH=C(CN)-CO-OCH₂-CN, -CH=C(CN)-CO-O(CH₂)₂-CN, -CH=CH-CO-CH₃, -CH=CH-CO-C₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-i-C₃H₇, -CH=CH-CO-n-C₄H₉, -CH=CH-CO-tert.-C₄H₉, -CH=CH-CO-CH₂Cl, -CH=CH-CO-CH₂Br, -CH=CH-CO-CHCl₂, -CH=CH-CO-CH₂-OCH₃, -CH=CH-CO-CH(OCH₃)₂, -CH=CH-CO-CH₂-SCH₃, -CH=C(CH₃)-CO-CH₃, -CH=C(CH₃)-CO-C₂H₅, -CH=C(CH₃)-CO-n-C₃H₇, -CH=C(CH₃)-CO-i-C₃H₇, -CH=C(CH₃)-CO-n-C₄H₉, -CH=C(CH₃)-CO-tert.-C₄H₉, -CH=C(CH₃)-CO-CH₂Cl, -CH=C(CH₃)-CO-CH₂Br, -CH=C(CH₃)-CO-CHCl₂, -CH=C(CH₃)-CO-CH₂-OCH₃, -CH=C(CH₃)-CO-CH(OCH₃)₂, -CH=C(CH₃)-CO-CH₂-SCH₃, -CH=C(C₂H₅)-CO-CH₃, -CH=C(C₂H₅)-CO-C₂H₅, -CH=C(C₂H₅)-CO-n-C₃H₇, -CH=C(C₂H₅)-CO-i-C₃H₇, -CH=C(C₂H₅)-CO-n-C₄H₉, -CH=C(C₂H₅)-CO-tert.-C₄H₉, -CH=C(C₂H₅)-CO-CH₂Cl, -CH=C(C₂H₅)-CO-CH₂Br, -CH=C(C₂H₅)-CO-CHCl₂, -CH=C(C₂H₅)-CO-CH₂-OCH₃, -CH=C(C₂H₅)-CO-CH(OCH₃)₂, -CH=C(C₂H₅)-CO-CH₂-SCH₃, -CH=C(Cl)-CO-CH₃, -CH=C(Cl)-CO-C₂H₅, -CH=C(Cl)-CO-n-C₃H₇, -CH=C(Cl)-CO-i-C₃H₇, -CH=C(Cl)-CO-n-C₄H₉, -CH=C(Cl)-CO-tert.-C₄H₉, -CH=C(Cl)-CO-CH₂Cl, -CH=C(Cl)-CO-CH₂Br, -CH=C(Cl)-CO-CHCl₂, -CH=C(Cl)-CO-CH₂-OCH₃, -CH=C(Cl)-CO-CH(OCH₃)₂, -CH=C(Cl)-CO-CH₂-SCH₃, -CH=C(Br)-CO-CH₃, -CH=C(Br)-CO-C₂H₅, -CH=C(Br)-CO-n-C₃H₇, -CH=C(Br)-CO-i-C₃H₇, -CH=C(Br)-CO-n-C₄H₉, -CH=C 99999 00070 552 001000280000000200012000285919988800040 0002004131038 00004 99880(Br)-CO-tert.-C₄H₉, -CH=C(Br)-CO-CH₂Cl, -CH=C(Br)-CO-CH₂Br, -CH=C(Br)-CO-CHCl₂, -CH=C(Br)-CO-CH₂-OCH₃, -CH=C(Br)-CO-CH(OCH₃)₂, -CH=C(Br)-CO-CH₂-SCH₃, -CH=C(CN)-CO-CH₃, -CH=C(CN)-CO-C₂H₅, -CH=C(CN)-CO-n-C₃H₇, -CH=C(CN)-CO-i-C₃H₇, -CH=C(CN)-CO-n-C₄H₉, -CH=C(CN)-CO-tert.-C₄H₉, -CH=C(CN)-CO-CH₂Cl, -CH=C(CN)-CO-CH₂Br, -CH=C(CN)-CO-CHCl₂, -CH=C(CN)-CO-CH₂-OCH₃, -CH=C(CN)-CO-CH(OCH₃)₂, -CH=C(CN)-CO-CH₂-SCH₃, -CH=CH-CO-C₆H₅, -CH=CH-CO-(4-Cl-C₆H₄), -CH=C(CH₃)-CO-C₆H₅, -CH=C(CH₃)-CO-(4-Cl-C₆H₄), -CH=C(C₂H₅)-CO-C₆H₅, -CH=C(C₂H₅)-CO-(4-Cl-C₆H₄), -CH=C(Cl)-CO-C₆H₅, -CH=C(Br)-CO-C₆H₅, -CH=C(CN)-CO-C₆H₅, -CH=CH-CO-NH₂, -CH=CH-CO-NHCH₃, -CH=CH-CO-N(CH₃)₂, -CH=CH-CO-NH-C₂H₅, -CH=CH-CO-N(C₂H₅)₂, -CH=CH-CO-NH-n-C₃H₇, -CH=CH-CO-NH-i-C₃H₇, -CH=CH-CO-NH-tert.-C₄H₉, -CH=CH-CO-NH-cyclopropyl, -CH=CH-CO-NH-cyclobutyl, -CH=CH-CO-NH-cyclopentyl, -CH=CH-CO-NH-cyclohexyl, -CH=CH-CO-cycloheptyl, -CH=CH-CO-NH-cyclooctyl, -CH=CH-CO-pyrrolidin-1-yl, -CH=CH-CO-piperidin-1-yl, -CH=CH-CO-morpholin-4-yl, -CH=CH-CO-NH-CH₂CH=CH₂, -CH=CH-CO-NH-CH₂C≡CH, -CH=CH-CO-N(CH₃)-CH₂C≡CH, -CH=CH-CO-NH-(CH₂)₂Cl, -CH=CH-CO-NH-C₆H₅, -CH=C(CH₃)-CO-NH₂, -CH=C(CH₃)-CO-NHCH₃, -CH=C(CH₃)-CO-N(CH₃)₂, -CH=C(CH₃)-CO-NH-C₂H₅, -CH=C(CH₃)-CO-N(C₂H₅)₂, -CH=C(CH₃)-CO-NH-n-C₃H₇, -CH=C(CH₃)-CO-NH-i-C₃H₇, -CH=C(CH₃)-CO-NH-tert.-C₄H₉, -CH=C(CH₃)-CO-NH-cyclopropyl, -CH=C(CH₃)-CO-NH-cyclobutyl, -CH=C(CH₃)-CO-NH-cyclopentyl, -CH=C(CH₃)-CO-NH-cyclohexyl, -CH=C(CH₃)-CO-NH-cycloheptyl, -CH=C(CH₃)-CO-NH-cyclooctyl, -CH=C(CH₃)-CO-pyrolidin-1-yl, -CH=C(CH₃)-CO-piperidin-1-yl, -CH=C(CH₃)-CO-morpholin-4-yl, -CH=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -CH=C(CH₃)-CO-NH-CH₂C≡CH, -CH=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CH₃)-CO-NH-(CH₂)₂Cl, -CH=C(CH₃)-CO-NH-C₆H₅, -CH=C(C₂H₅)-CO-NH₂, -CH=C(C₂H₅)-CO-NHCH₃, -CH=C(C₂H₅)-CO-N(CH₃)₂, -CH=C(C₂H₅)-CO-NH-C₂H₅, -CH=C(C₂H₅)-CO-N(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-n-C₃H₇, -CH=C(C₂H₅)-CO-NH-i-C₃H₇, -CH=C(C₂H₅)-CO-NH-tert.-C₄H₉, -CH=C(C₂H₅)-CO-NH-cyclopropyl, -CH=C(C₂H₅)-CO-NH-cyclobutyl, -CH=C(C₂H₅)-CO-NH-cyclopentyl, -CH=C(C₂H₅)-CO-NH-cyclohexyl, -CH=C(C₂H₅)-CO-NH-cycloheptyl, -CH=C(C₂H₅)-CO-NH-cyclooctyl, -CH=C(C₂H₅)-CO-pyrrolidin-1-yl, -CH=C(C₂H₅)-CO-piperidin-1-yl, -CH=C(C₂H₅)-CO-morpholin-4-yl, -CH=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-CH₂C≡CH, -CH=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -CH=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -CH=C(C₂H₅)-CO-NH-C₆H₅, -CH=C(Cl)-CO-NH₂, -CH=C(Cl)-CO-NHCH₃, -CH=C(Cl)-CO-N(CH₃)₂, -CH=C(Cl)-CO-NH-C₂H₅, -CH=C(Cl)-CO-N(C₂H₅)₂, -CH=C(Cl)-CO-NH-n-C₃H₇, -CH=C(Cl)-CO-NH-i-C₃H₇, -CH=C(Cl)-CO-NH-tert.-C₄H₉, -CH=C(Cl)-CO-NH-cyclopropyl, -CH=C(Cl)-CO-NH-cyclobutyl, -CH=C(Cl)-CO-NH-cyclopentyl, -CH=C(Cl)-CO-NH-cyclohexyl, -CH=C(Cl)-CO-NH-cycloheptyl, -CH=C(Cl)-CO-NH-cyclooctyl, -CH=C(Cl)-CO-pyrrolidin-1-yl, -CH=C(Cl)-CO-piperidin-1-yl, -CH=C(Cl)-CO-morpholin-4-yl, -CH=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -CH=C(Cl)-CO-NH-CH₂C≡CH, -CH=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Cl)-CO-NH-(CH₂)₂Cl, -CH=C(Cl)-CO-NH-C₆H₅, -CH=C(Br)-CO-NH₂, -CH=C(Br)-CO-NHCH₃, -CH=C(Br)-CO-N(CH₃)₂, -CH=C(Br)-CO-NH-C₂H₅, -CH=C(Br)-CO-N(C₂H₅)₂, -CH=C(Br)-CO-NH-n-C₃H₇, -CH=C(Br)-CO-NH-i-C₃H₇, -CH=C(Br)-CO-NH-tert.-C₄H₉, -CH=C(Br)-CO-NH-cyclopropyl, -CH=C(Br)-CO-NH-cyclobutyl, -CH=C(Br)-CO-NH-cyclopentyl, -CH=C(Br)-CO-NH-cyclohexyl, -CH=C(Br)-CO-NH-cycloheptyl, -CH=C(Br)-CO-NH-cyclooctyl, -CH=C(Br)-CO-pyrrolidin-1-yl, -CH=C(Br)-CO-piperidin-1-yl, -CH=C(Br)-CO-morpholin-4-yl, -CH=C(Br)-CO-NH-CH₂CH=C(Br)₂, -CH=C(Br)-CO-NH-CH₂C≡CH, -CH=C(Br)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Br)-CO-NH-(CH₂)₂Cl, -CH=C(Br)-CO-NH-C₆H₅, -CH=C(CN)-CO-NH₂, -CH=C(CN)-CO-NHCH₃, -CH=C(CN)-CO-N(CH₃)₂, -CH=C(CN)-CO-NH-C₂H₅, -CH=C(CN)-CO-N(C₂H₅)₂, -CH=C(CN)-CO-NH-n-C₃H₇, -CH=C(CN)-CO-NH-i-C₃H₇, -CH=C(CN)-CO-NH-tert.-C₄H₉, -CH=C(CN)-CO-NH-cyclopropyl, -CH=C(CN)-CO-NH-cyclobutyl, -CH=C(CN)-CO-NH-cyclopentyl, -CH=C(CN)-CO-NH-cyclohexyl, -CH=C(CN)-CO-NH-cycloheptyl, -CH=C(CN)-CO-NH-cyclooctyl, -CH=C(CN)-CO-pyrrolidin-1-yl, -CH=C(CN)-CO-piperidin-1-yl, -CH=C(CN)-CO-morpholin-4-yl, -CH=C(CN)-CO-NH-CH₂CH=C(CN)₂, -CH=C(CN)-CO-NH-CH₂C≡CH, -CH=C(CN)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CN)-CO-NH-(CH₂)₂Cl, -CH=C(CN)-CO-NH-C₆H₅, -CH=CH-CO-SCH₃, -CH=CH-CO-SC₂H₅, -CH=CH-CO-S-n-C₃H₇, -CH=CH-CO-S-i-C₃H₇, -CH=CH-CO-S-n-C₄H₉, -CH=CH-CO-S-tert.-C₄H₉, -CH=C(CH₃)-CO-SCH₃, -CH=C(CH₃)-CO-SC₂H₅, -CH=C(CH₃)-CO-S-n-C₃H₇, -CH=C(CH₃)-CO-S-i-C₃H₇, -CH=C(CH₃)-CO-S-n-C₄H₉, -CH=C(CH₃)-CO-S-tert.-C₄H₉, -CH=C(C₂H₅)-CO-SCH₃, -CH=C(C₂H₅)-CO-SC₂H₅, -CH=C(C₂H₅)-CO-S-n-C₃H₇, -CH=C(C₂H₅)-CO-S-i-C₃H₇, -CH=C(C₂H₅)-CO-S-n-C₄H₉, -CH=C(C₂H₅)-CO-S-tert.-C₄H₉, -CH=C(Cl)-CO-SCH₃, -CH=C(Cl)-CO-SC₂H₅, -CH=C(Cl)-CO-S-n-C₃H₇, -CH=C(Cl)-CO-S-i-C₃H₇, -CH=C(Cl)-CO-S-n-C₄H₉, -CH=C(Cl)-CO-S-tert.-C₄H₉, -CH=C(Br)-CO-SCH₃, -CH=C(Br)-CO-SC₂H₅, -CH=C(Br)-CO-S-n-C₃H₇, -CH=C(Br)-CO-S-i-C₃H₇, -CH=C(Br)-CO-S-n-C₄H₉, -CH=C(Br)-CO-S-tert.-C₄H₉, -CH=C(CN)-CO-SCH₃, -CH=C(CN)-CO-SC₂H₅, -CH=C(CN)-CO-S-n-C₃H₇, -CH=C(CN)-CO-S-i-C₃H₇, -CH=C(CN)-CO-S-n-C₄H₉, -CH=C(CN)-CO-S-tert.-C₄H₉, -CH=C(COCH₃)-CO-OCH₃, -CH=C(COC₂H₅)-CO-OCH₃, -CH=C(CO-n-C₃H₇)-CO-OCH₃, -CH=C(COCH₃)-CO-OC₂H₅, -CH=C(COC₂H₅)-CO-OC₂H₅, -CH=C(CO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COCH₃)-CO-O-n-C₃H₇, -CH=C(COC₂H₅)-CO-O-n-C₃H₇, -CH=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-OCH₃, -CH=C(CF₃)-CO-OC₂H₅, -CH=C(CF₃)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-O-i-C₃H₇, -CH=C(CF₃)-CO-O-n-C₄H₉, -CH=C(CF₃)-CO-O-tert.-C₄H₉, -CH=C(COOCH₃)₂, -CH=C(COOC₂H₅)₂, -CH=C(COOCH₃)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)-CO-OCH₃, -CH=C(COO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)₂, -CH=CH-CH=CH-COOH, -CH=CH-CH=CH-CO-OCH₃, -CH=CH-CH=CH-CO-OC₂H₅, -CH=CH-CH=C(COOCH₃)₂, -CH=CH-CH=C(CN)-CO-OCH₃, -CH=CH-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-OCH₃, -CH=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CH=C(Cl)-CO-OCH₃, -CH=C(CH₃)-CH=C(Br)-CO-OCH₃, -CH=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-NH₂, -CH=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -CH=CH-(CH₂)₂-COOH, -CH=CH-(CH₂)₂-CO-OCH₃, -CH=CH-(CH₂)₂-CO-OC₂H₅, -CH=CH-CH₂-CH(COOCH₃)₂, -CH=CH-CH₂-CH(COOC₂H₅)₂, -CH=CH-CH₂-CH(CN)-CO-OCH₃, -CH=CH-CH₂-CH(CN)-CO-OC₂H₅, -CH=CH-CH₂-CH(CH₃)-CO-OCH₃, -CH=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -CH=CH-(CH₂)₂-CO-NH₂, -CH=CH-(CH₂)₂-CO-NH-CH₃, -CH=CH-CH₂-COOH, -CH=CH-CH₂-CO-OCH₃, -CH=CH-CH₂-CO-OC₂H₅, -CH=C(COOCH₃)-CH₂-CO-OCH₃, -CH=C(COOCH₃)-CH₂-CO-OC₂H₅, -CH=CH-CH₂-CO-NH₂, -CH=CH-CH₂-CO-NH-CH₃, -CH=CH-CH₂-CO-N(CH₃)₂, -CH(OCH₃)₂, -CH(SCH₃)₂, -CH(OC₂H₅)₂, -CH(SC₂H₅)₂, -CH(O-n-C₃H₇)₂, -CH(O-i-C₃H₇)₂, -CH(S-n-C₃H₇)₂, -CH(S-i-C₃H₇)₂, -CH(O-n-C₄H₉)₂, -CH(O-i-C₄H₉)₂, -CH(O-s-C₄H₉)₂, -CH(O-tert.-C₄H₉)₂, -CH(S-n-C₄H₉)₂, -CH(S-i-C₄H₉)₂, -CH(S-s-C₄H₉)₂, -CH(S-tert.-C₄H₉)₂, -CH(OC₅H₁₁)₂, 1,3-Dioxolan-2-yl, 1,3-Dithio­ lan-2-yl, 1,3-Oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 5-Methyl-1,3-oxathiolan-2-yl, 4-Ethyl-1,3-dioxolan-2-yl, 4-Ethyl- 1,4-dithiolan-2-yl, 4-Ethyl-1,3-oxathiolan-2-yl, 5-Ethyl-1,3-oxa­ thiolan-2-yl, 4,5-Dimethyl-1,3-dioxolan-2-yl, 4,4-Dimethyl-1,3- dioxolan-2-yl, 4,5-Dimethyl-1,3-dithiolan-2-yl, 5,5-Dimethyl-1,3- dithiolan-2-yl, 4,5-Dimethyl-1,3-oxathiolan-2-yl, 5,5-Dimethyl- 1,3-oxathiolan-2-yl, 4,4-Dimethyl-1,3-oxathiolan-2-yl, 4-Vinyl- 1,3-dioxolan-2-yl, 4-Vinyl-1,3-dithiolan-2-yl, 4-Vinyl-1,3-oxa­ thiolan-2-yl, 5-Vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3- dioxolan-2-yl, 4-Chlormethyl-1,3-dithiolan-2-yl, 4-Chlormethyl- 1,3-oxathiolan-2-yl, 5-Chlormethyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-1,3-dithio­ lan-2-yl, 4-Hydroxymethyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl- 1,3-oxathiolan-2-yl, 4-Methoxymethyl-1,3-dioxolan-2-yl, 4-Allyl­ oxymethyl-1,3-dioxolan-2-yl, 4-Propargyloxymethyl-1,3-dioxolan- 2-yl, 4-Acetoxymethyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-1,3-dithiolan-2-yl, 4-Propargyl­ oxymethyl-1,3-dithiolan-2-yl, 4-Acetoxymethyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl-1,3-oxathiolan-2-yl, 5-Allyloxy­ methyl-1,3-oxathiolan-2-yl, 4-Propargyloxymethyl-1,3-oxathiolan-2-yl, 5-Propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxymethyl- 1,3-oxathiolan-2-yl, 5-Acetoxymethyl-1,3-oxathiolan-2-yl, 4-Methylthiomethyl-1,3-dioxolan-2-yl, 4-Methylthiomethyl-1,3- dithiolan-2-yl, 4-Carboxy-1,3-dioxolan-2-yl, 4-Carboxy-1,3- dithiolan-2-yl, 4-Methoxycarbonyl-1,3-dioxolan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-1,3-dithiolan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-4-methyl- 1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-di­ thiolan-2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-1,3- dithiolan-2-yl, 1,3-Dioxan-2-yl, 1,3-Dithian-2-yl, 1,3-Oxathian- 2-yl, 5-Methyl-1,3-dioxan-2-yl, 5-Methyl-1,3-dithian-2-yl, 5-Methyl-1,3-oxathian-2-yl, 5,5-Dimethyl-1,3-dioxan-2-yl, 4,6-Dimethyl- 1,3-dioxan-2-yl, 4,4-Dimethyl-1,3-dioxan-2-yl, 5,5-Dimethyl- 1,3-dithian-2-yl, 4,6-Dimethyl-1,3-dithian-2-yl, 4,4-Dimethyl- 1,3-dithian-2-yl, 5,5-Dimethyl-1,3-oxathian-2-yl, 4,4-Dimethyl- 1,3-oxathian-2-yl, 6,6-Dimethyl-1,3-oxathian-2-yl, 4-Hydroxymethyl-1,3-dioxan-2-yl, 4-Methoxymethyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-1,3-dithian-2-yl, 4-Methoxymethyl-1,3-dithian-2-yl, 4-Allyloxymethyl-1,3-dithian-2-yl, 4-Acetoxymethyl- 1,3-dithian-2-yl, 4-Chlormethyl-1,3-dioxan-2-yl, 4-Chlormethyl- 1,3-dithian-2-yl, 1,3-Dioxepan-2-yl, 1,3-Dithiepan-2-yl, 1,3-Dioxep-5-en-2-yl, 4-Methoxycarbonyl-1,3-dioxan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-1,3-dithian-2-yl, 4-n-Butoxycarbonyl-1,3-dithian-2-yl, 4-Methoxycarbonyl-4- methyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-4-methyl- 1,3-dithian-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithian-2-yl, -C(CH₃)(OCH₃)₂, -C(CH₃)(SCH₃)₂, -C(CH₃)(OC₂H₅)₂, -C(CH₃)(SC₂H₅)₂, -C(CH₃)(O-n-C₃H₇)₂, -C(CH₃)(O-i-C₃H₇)₂, -C(CH₃)(S-n-C₃H₇)₂, -C(CH₃)(S-i-C₃H₇)₂, -C(CH₃)(O-n-C₄H₉)₂, -C(CH₃)(O-i-C₄H₉)₂, -C(CH₃)(O-s-C₄H₉)₂, -C(CH₃)(O-tert.-C₄H₉)₂, -C(CH₃)(S-n-C₄H₉)₂, -C(CH₃)(S-i-C₄H₉)₂, -C(CH₃)(S-s-C₄H₉)₂, -C(CH₃)(S-tert.-C₄H₉)₂, -C(CH₃)(O-n-C₅H₁₁)′′, 2-Methyl-1,3-dioxolan-2-yl, 2-Methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-oxathiolan-2-yl, 2,4-Dimethyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-1,3- oxathiolan-2-yl, 2,5-Dimethyl-1,3-oxathiolan-2-yl, 4-Ethyl-2- methyl-1,3-dioxolan-2-yl, 4-Ethyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Ethyl-2-methyl-1,3- oxathiolan-2-yl, 2,4,5-Trimethyl-1,3-dioxolan-2-yl, 2,4,4-Trimethyl- 1,3-dioxolan-2-yl, 2,4,5-Trimethyl-1,3-dithiolan-2-yl, 2,4,4-Trimethyl-1,3-dithiolan-2-yl, 2,4,5-Trimethyl-1,3-oxathiolan-2-yl, 2,4,4-Trimethyl-1,3-oxathiolan-2-yl, 2-Methyl-4-vinyl- 1,3-dioxolan-2-yl, 2-Methyl-4-vinyl-1,3-dithiolan-2-yl, 2-Methyl- 4-vinyl-1,3-oxathiolan-2-yl, 2-Methyl-5-vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-dioxolan-2-yl, 4-Chlormethyl-2- methyl-1,3-dithiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl- 2-methyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-2- methyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dioxolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxy- 2-methyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dithiolan-2-yl, 4-Acetoxy-2- methyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl- 2-methyl-1,3-oxathiolan-2-yl, 5-Allyloxymethyl-2- methyl-1,3-oxathiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3- oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxy-2-methyl-1,3-oxathiolan-2-yl, 5-Acetoxy-2-methyl- 1,3-oxathiolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dioxolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-2- methyl-1,3-dioxolan-2-yl, 4-Carboxy-2-methyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-2- methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl- 2-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-2- methyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-ethoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4- ethoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-n-butoxy- carbony-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl-1,3- dithiolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-dioxan-2-yl, 2-Methyl-1,3-dithian-2-yl, 2-Methyl-1,3-oxathian-2-yl, 2,5- Dimethyl-1,3-dioxan-2-yl, 2,5-Dimethyl-1,3-dithian-2-yl, 2,5-Dimethyl- 1,3-oxathian-2-yl, 2,5,5-Trimethyl-1,3-dioxan-2-yl, 2,4,6- Trimethyl-1,3-dioxan-2-yl, 2,2,4-Trimethyl-1,3-dioxan-2-yl, 2,5,5-Trimethyl-1,3-dithian-2-yl, 2,4,6-Trimethyl-1,3-dithian-2-yl, 2,4,4-Trimethyl-1,3-dithian-2-yl, 2,5,5-Trimethyl-1,3-oxathian-2-yl, 2,4,4-Trimethyl-1,3-oxathian-2-yl, 2,6,6-Trimethyl- 1,3-oxathian-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-2- methyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dithian-2-yl, 4-Methoxymethyl-2- methyl-1,3-dithian-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithian-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dithian-2-yl, 4-Chlormethyl-2- methyl-1,3-dioxan-2-yl, 4-Chlormethyl-2-methyl-1,3-dithian-2-yl, -C(CH₃)=NH, -C(CH₃)=N-CH₃, -C(CH₃)=N-C₂H₅, -C(CH₃)=N-n-C₃H₇, -C(CH₃)=N-i-C₃H₇, -C(CH₃)=N-n-C₄H₉, -C(CH₃)=N-CH₂CH=CH₂, -C(CH₃)=N-CH₂CH=CH₂-CH₃, -C(CH₃)=N-CH₂C≡CH, -C(CH₃)=N-CH₂C≡C-CH₃, -C(CH₃)=N-cyclopropyl, -C(CH₃)=N-cyclobutyl, -C(CH₃)=N-cyclopentyl, -C(CH₃)=N-cyclohexyl, -C(CH₃)=N-cycloheptyl, -C(CH₃)=N-CH₂-CH₂Cl, -C(CH₃)=N-CH₂Cl, -C(CH₃)=N-C₆H₅, -C(CH₃)=N-(2-F-C₆H₄), -C(CH₃)=N-(3-F-C₆H₄), -C(CH₃)=N-(4-F-C₆H₄), -C(CH₃)=N-(2-Cl-C₆H₄), -C(CH₃)=N-(3-Cl-C₆H₄), -C(CH₃)=N-(4-Cl-C₆H₄), -C(CH₃)=N-(2-CH₃-C₆H₄), -C(CH₃)=N-(3-CH₃-C₆H₄), -C(CH₃)=N-(4-CH₃-C₆H₄), -C(CH₃)=N-(2-CF₃-C₆H₄), -C(CH₃)=N-(3-CF₃-C₆H₄), -C(CH₃)=N-(4-CF₃-C₆H₄), -C(CH₃)=N-(2-OCH₃-C₆H₄), -C(CH₃)=N-(3-OCH₃-C₆H₄), -C(CH₃)=N-(4-OCH₃-C₆H₄), -C(CH₃)=N-(4-NO₂-C₆H₄), -C(CH₃)=N-(4-CN-C₆H₄), -C(CH₃)=N-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-(2,4-(CH₃)₂-C₆H₃), -C(CH₃)=N-CH₂-OCH₃, -C(CH₃)=N-CH₂-OC₂H₅, -C(CH₃)=N-CH₂CH₂-OCH₃, -C(CH₃)=N-CH₂CH-OC₂H₅, -C(CH₃)=N-OH, -C(CH₃)=N-OCH₃, -C(CH₃)=N-OC₂H₅, -C(CH₃)=N-O-n-C₃H₇, -C(CH₃)=N-O-i-C₃H₇, -C(CH₃)=N-O-n-C₄H₉, -C(CH₃)=N-O-i-C₄H₉, -C(CH₃)=N-O-s-C₄H₉, -C(CH₃)=N-O-tert.-C₄H₉, -C(CH₃)=N-OCH₂-CH=CH₂, -C(CH₃)=N-OCH(CH₃)-CH=CH₂, -C(CH₃)=N-OCH₂-C≡CH, -C(CH₃)=N-CH(CH₃)-C≡CH, -C(CH₃)=N-OCH₂-CH=C-CH₃, -C(CH₃)=N-OCH₂CH₂-Cl, -C(CH₃)=N-OCH₂CH₂-F, -C(CH₃)=N-OCH₂-CF₃, -C(CH₃)=N-OCH₂-CH=CHCl, -C(CH₃)=N-OCH₂-C(Cl)=CH₂, -C(CH₃)=N-OCH₂-C(Br)=CH₂, -C(CH₃)=N-OCH₂-CH=C(Cl)-CH₃, -C(CH₃)=N-O-CO-CH₃, -C(CH₃)=N-O-CO-C₂H₅, -C(CH₃)=N-OCH₂-CN, -C(CH₃)=N-OCH₂-CH=CH-CH₂-OCH₃, -C(CH₃)=N-OCH₂-CH=CH-CH₂-O-tert.-C₄H₉, -C(CH₃)=N-O-(CH₂)₃-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-(4-Cl-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-C₆H₅, -C(CH₃)=N-OCH₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(3-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-CH₂-(4-CH₃O-C₆H₄), -C(CH₃)=N-OCH₂-CH=C(CH₃)-C₆H₅, -C(CH₃)=N-O-(CH₂)₂-CH=CH-(3,4-Cl₂-C₆H₃), -C(CH₃)=N-O-(CH₂)₃-C≡-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-OCH₃, -C(CH₃)=N-OCH₂CH₂-OCH₃, -C(CH₃)=N-OCH₂-OC₂H₅, -C(CH₃)=N-OCH(CH₃)-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=N-NH₂, -C(CH₃)=N-NH-CH₃, -C(CH₃)=N-NH-C₂H₅, -C(CH₃)=N-NH-n-C₃H₇, -C(CH₃)=N-NH-i-C₃H₇, -C(CH₃)=N-NH-n-C₄H₉, -C(CH₃)=N-NH-i-C₄H₉, -C(CH₃)=N-NH-s-C₄H₉, -C(CH₃)=N-NH-tert.-C₄H₉, -C(CH₃)=N-NH-cyclopropyl, -C(CH₃)=N-NH-cyclobutyl, -C(CH₃)=N-NH-cyclopentyl, -C(CH₃)=N-NH-cyclohexyl, -C(CH₃)=N-NH-cycloheptyl, -C(CH₃)=N-N(CH₃)₂, -C(CH₃)=N-N(C₂H₅)₂, -C(CH₃)=N-N(n-C₃H₇)₂, -C(CH₃)=N-N(i-C₃H₇)₂, -C(CH₃)=N-NH-CH₂-C=CH, -C(CH₃)=N-NH-CH₂-C≡CH, -C(CH₃)=N-N(CH₃)-CH₂-C≡CH, -C(CH₃)=N-NH-CH₂CF₃, -C(CH₃)=N-NH-CO-CH₃, -C(CH₃)=N-NH-CO-C₂H₅, -C(CH₃)=N-NH-CO-OCH₃, -C(CH₃)=N-NH-CO-OC₂H₅, -C(CH₃)=N-NH-CO-O-tert.-C₄H₉, -C(CH₃)=N-pyrrolidin-1-yl, -C(CH₃)=N-piperidin-1-yl, -C(CH₃)=N-morpholin-4-yl, -C(CH₃)=N-NH-C₆H₅, -C(CH₃)=N-NH-(4-Cl-C₆H₄), -C(CH₃)=N-NH-(4-NO₂-C₆H₄), -C(CH₃)=N-NH-(4-F-C₆H₄), -C(CH₃)=N-NH-(4-CH₃O-C₆H₄), -C(CH₃)=N-NH-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-NH-(2,4-(NO₂)₂-C₆H₃), -C(CH₃)=N-NH-CO-NH₂, -C(CH₃)=N-NH-CO-NHCH₃, -C(CH₃)=N-NH-CO-NHC₂H₅, -C(CH₃)=N-NH-CO-N(CH₃)₂, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=CH-CO-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-O-n-C₄H₉, -C(CH₃)=CH-CO-O-tert.-C₄H₉, -C(CH₃)=CH-CO-O-cyclopropyl, -C(CH₃)=CH-CO-O-cyclobutyl, -C(CH₃)=CH-CO-O-cyclopentyl, -C(CH₃)=CH-CO-O-cyclohexyl, -C(CH₃)=CH-CO-O-cycloheptyl, -C(CH₃)=C(CH₃)-COOH, -C(CH₃)=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-cyclopropyl, -C(CH₃)=C(CH₃)-CO-O-cyclobutyl, -C(CH₃)=C(CH₃)-CO-O-cyclopentyl, -C(CH₃)=C(CH₃)-CO-O-cyclohexyl, -C(CH₃)=C(CH₃)-CO-O-cycloheptyl, -C(CH₃)=C(C₂H₅)-COOH, -C(CH₃)=C(C₂H₅)-CO-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-cyclo­ propyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-O- cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-O-cycloheptyl, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=C(Cl)-CO-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-O-n-C₄H₉, -C(CH₃)=C(Cl)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-O-cyclopropyl, -C(CH₃)=C(Cl)-CO-O-cyclobutyl, -C(CH₃)=C(Cl)-CO-O-cyclopentyl, -C(CH₃)=C(Cl)-CO-O-cyclohexyl, -C(CH₃)=C(Cl)-CO-O-cycloheptyl, -C(CH₃)=C(Br)-COOH, -C(CH₃)=C(Br)-CO-OCH₃, -C(CH₃)=C(Br)-CO-OC₂H₅, -C(CH₃)=C(Br)-CO-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-O-n-C₄H₉, -C(CH₃)=C(Br)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-O-cyclopropyl, -C(CH₃)=C(Br)-CO-O-cyclobutyl, -C(CH₃)=C(Br)-CO-O-cyclopentyl, -C(CH₃)=C(Br)-CO-O-cyclohexyl, -C(CH₃)=C(Br)-CO-O-cycloheptyl, -C(CH₃)=C(CN)-COOH, -C(CH₃)=C(CN)-CO-OCH₃, -C(CH₃)=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CN)-CO-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-O-n-C₄H₉, -C(CH₃)=C(CN)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-O-cyclopropyl, -C(CH₃)=C(CN)-CO-O-cyclobutyl, -C(CH₃)=C(CN)-CO-O-cyclopentyl, -C(CH₃)=C(CN)-CO-O-cyclohexyl, -C(CH₃)=C(CN)-CO-O-cycloheptyl, -C(CH₃)=CH-CO-OCH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=CH-CO-O-i-C₃H₇, -C(CH₃)=CH-CO-OCH(CH₃)-OCH₃, -C(CH₃)=CH-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=CH-CO-OCH₂CH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-O-i-C₃H₇, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -(CH₃)=C(Cl)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-O-i-C₃H₇, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-O-i-C₃H₇, -C(CH₃)=C(CN)-CO-OCH(CH₃)OCH₃, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-CF₃, -C(CH₃)=CH-CO-OCH₂-CCl₃, -C(CH₃)=CH-CO-OCH₂-oxiranyl, -C(CH₃)=CH-CO-(CH₂)₃-Br,-C(CH₃)=CH-CO-OCH₂-CH=CH₂, -C(CH₃)=CH-CO-OCH₂-C≡CH, -C(CH₃)=CH-CO-OCH₂-CN, -C(CH₃)=CH-CO-OCH₂CH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CF₃, -C(CH₃)=C(CH₃)-CO-OCH₂-CCl₃, -C(CH₃)=C(CH₃)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CH₃)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CH₃)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CH₃)-CO-OCH₂-C≡CH, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CF₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CCl₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-oxiranyl, -C(CH₃)=C(C₂H₅)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(C₂H₅)-CO-OCH₂-C≡CH, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂-CF₃, -C(CH₃)=C(Cl)-CO-OCH₂-CCl₃, -C(CH₃)=C(Cl)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Cl)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Cl)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Cl)-CO-OCH₂-C≡CH, -C(CH₃)=C(Cl)-CO-OCH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂-CF₃, -C(CH₃)=C(Br)-CO-OCH₂-CCl₃, -C(CH₃)=C(Br)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Br)-CO-O(CH₂)₃-Br, -C(CH₃)=C(Br)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Br)-CO-OCH₂-C≡CH, -C(CH₃)=C(Br)-CO-OCH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂CH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂-CF₃, -C(CH₃)=C(CN)-CO-OCH₂-CCl₃, -C(CH₃)=C(CN)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CN)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(CN)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CN)-CO-OCH₂-C≡CH, -C(CH₃)=C(CN)-CO-OCH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂CH₂-CN, -C(CH₃)=CH-CO-CH₃, -C(CH₃)=CH-CO-C₂H₅, -C(CH₃)=CH-CO-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-n-C₄H₉, -C(CH₃)=CH-CO-tert.-C₄H₉, -C(CH₃)=CH-CO-CH₂Cl, -C(CH₃)=CH-CO-CH₂Br, -C(CH₃)=CH-CO-CHCl₂, -C(CH₃)=CH-CO-CH₂-OCH₃, -C(CH₃)=CH-CO-CH(OCH₃)₂, -C(CH₃)=CH-CO-CH₂-SCH₃, -C(CH₃)=C(CH₃)-CO-CH₃, -C(CH₃)=C(CH₃)-CO-C₂H₅, -C(CH₃)=C(CH₃)-CO-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-CH₂Cl, -C(CH₃)=C(CH₃)-CO-CH₂Br, -C(CH₃)=C(CH₃)-CO-CHCl₂, -C(CH₃)=C(CH₃)-CO-CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-CH(OCH₃)₂, -C(CH₃)=C(CH₃)-CO-CH₂-SCH₃, -C(CH₃)=C(C₂H₅)-CO-CH₃, -C(CH₃)=C(C₂H₅)-CO-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-CH₂Cl, -C(CH₃)=C(C₂H₅)-CO-CH₂Br, -C(CH₃)=C(C₂H₅)-CO-CHCl₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-CH(OCH₃)₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-SCH₃, -C(CH₃)=C(Cl)-CO-CH₃, -C(CH₃)=C(Cl)-CO-C₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-n-C₄H₉, -C(CH₃)=C(Cl)-CO-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-CH₂Cl, -C(CH₃)=C(Cl)-CO-CHCl₂, -C(CH₃)=C(Cl)-CO-CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-CH(OCH₃)₂, -C(CH₃)=C(Cl)-CO-CH₂-SCH₃, -C(CH₃)=C(Br)-CO-CH₃, -C(CH₃)=C(Br)-CO-C₂H₅, -C(CH₃)=C(Br)-CO-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-n-C₄H₉, -C(CH₃)=C(Br)-CO-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-CH₂Cl, -C(CH₃)=C(Br)-CO-CH₂Br, -C(CH₃)=C(Br)-CO-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-CH(OCH₃)₂, -C(CH₃)=C(Br)-CO-CH₂-SCH₃, -C(CH₃)=C(CN)-CO-CH₃, -C(CH₃)=C(CN)-CO-C₂H₅, -C(CH₃)=C(CN)-CO-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-n-C₄H₉, -C(CH₃)=C(CN)-CO-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-CH₂Cl, -C(CH₃)=C(CN)-CO-CH₂Br, -C(CH₃)=C(CN)-CO-CHCl₂, -C(CH₃)=C(CN)-CO-CH₂-OCH₃, -C(CH₃)=C(CN)-CO-CH(OCH₃ )₂, -C(CH₃)=C(CN)-CO-CH₂-SCH₃, -C(CH₃)=CH-CO-C₆H₅, -C(CH₃)=CH-CO-(4-Cl-C₆H₄), -C(CH₃)=C(CH₃)-CO-C₆H₅, -C(CH₃)=C(CH₃)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(C₂H₅)-CO-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(Cl)-CO-C₆H₅, -C(CH₃)=C(Br)-CO-C₆H₅, -C(CH₃)=C(CN)-CO-C₆H₅, -C(CH₃)=CH-CO-NH₂, -C(CH₃)=CH-CO-NHCH₃, -C(CH₃)=CH-CO-N(CH₃)₂, -C(CH₃)=CH-CO-NH-C₂H₅, -C(CH₃)=CH-CO-N(C₂H₅)₂, -C(CH₃)=CH-CO-NH-n-C₃H₇, -C(CH₃)=CH-CO-NH-i-C₃H₇, -C(CH₃)=CH-CO-NH-tert.-C₄H₉, -C(CH₃)=CH-CO-NH-cyclopropyl, -C(CH₃)=CH-CO-NH-cyclobutyl, -C(CH₃)=CH-CO-NH-cyclopentyl, -C(CH₃)=CH-CO-NH-cyclohexyl, -C(CH₃)=CH-CO-NH-cycloheptyl, -C(CH₃)=CH-CO-NH-cyclooctyl, -C(CH₃)=CH-CO-pyrrolidin-1-yl, -C(CH₃)=CH-CO-piperidin-1-yl, -C(CH₃)=CH-CO-morpholin-4-yl, -C(CH₃)=CH-CO-NH-CH₂CH=CH₂, -C(CH₃)=CH-CO-NH-CH₂C≡CH, -C(CH₃)=CH-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=CH-CO-NH-(CH₂)₂Cl, -C(CH₃)=CH-CO-NH-C₆H₅, -C(CH₃)=C(CH₃)-CO-NH₂, -C(CH₃)=C(CH₃)-CO-NHCH₃, -C(CH₃)=C(CH₃)-CO-N(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-C₂H₅, -C(CH₃)=C(CH₃)-CO-N(C₂H₅)₂, -C(CH₃)=C(CH₃)-CO-NH-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-NH- cyclopropyl, -C(CH₃)=C(CH₃)-CO-NH-cyclobutyl, -C(CH₃)=C(CH₃)-CO-NH-cyclopentyl, -C(CH₃)=C(CH₃)-CO-NH- cyclehexyl, -C(CH₃)=C(CH₃)-CO-NH-cycloheptyl, -C(CH₃)=C(CH₃)-CO-NH-cyclooctyl, -C(CH₃)=C(CH₃)-CO- pyrrolidin-1-yl, -C(CH₃)=C(CH₃)-CO-piperidin-1-yl, -C(CH₃)=C(CH₃)-CO-morpholin-4-yl, -C(CH₃)=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-NH(CH₂)₂Cl, -C(CH₃)=C(CH₃)-CO-NH-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-NH₂, -C(CH₃)=C(C₂H₅)-CO-NHCH₃, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)₂, -C(CH₃)=C(C₂H₅)-CO-NH-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-N(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-NH- cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclo­ hexyl, -C(CH₃)=C(C₂H₅)-CO-NH-cycloheptyl, -C(CH₃)=C(C₂H₅)-CO-NH- cyclooctyl, -C(CH₃)=C(C₂H₅)-CO-pyrrolidin-1-yl, -C(CH₃)=C(C₂H₅)-CO-piperidin-1-yl, -C(CH₃)=C(C₂H₅)-CO- morpholin-4-yl, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(C₂H₅)-CO-NH-C₆H₅, -C(CH₃)=C(Cl)-CO-NH₂, -C(CH₃)=C(CH₃)=C(Cl)-CO-NHCH₃, -C(CH₃)=C(Cl)-CO-N(CH₃)₂, -C(CH₃)=C(Cl)-CO-NH-C₂H₅, -C(CH₃)=C(Cl)-CO-N(C₂H₅)₂, -C(CH₃)=C(Cl)-CO-NH-n-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-i-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-NH-cyclopropyl, -C(CH₃)=C(Cl)-CO-NH-cyclobutyl, -C(CH₃)=C(Cl)-CO-NH-cyclopentyl, -C(CH₃)=C(Cl)-CO-NH-cyclohexyl, -C(CH₃)=C(Cl)-CO-NH-cycloheptyl, -C(CH₃)=C(Cl)-CO-NH-cyclooctyl, -C(CH₃)=C(Cl)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Cl)-CO-piperidin-1- yl, -C(CH₃)=C(Cl)-CO-morpholin-4-yl, -C(CH₃)=C(Cl)-CO-NH-CH₂CH=C(Cl)₂-CO-NH-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Cl)-CO-NH-C₆H₅, -C(CH₃)=C(Br)-CO-NH₂, -C(CH₃)=C(Br)-CO-NHCH₃, -C(CH₃)=C(Br)-CO-N(CH₃)₂, -C(CH₃)=C(Br)-CO-NH-C₂H₅, -C(CH₃)=C(Br)-CO-N(C₂H₅)₂, -C(CH₃)=C(Br)-CO-NH-n-C₃H₇, -C(CH₃)=C(Br)-CO-NH-i-C₃H₇, -C(CH₃)=C(Br)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-NH-cyclopropyl, -C(CH₃)=C(Br)-CO-NH-cyclobutyl, -C(CH₃)=C(Br)-CO-NH-cyclopentyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cycloheptyl, -C(CH₃)=C(Br)-CO-NH-cyclooctyl, -C(CH₃)=C(Br)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Br)-CO-piperidin-1-yl, -C(CH₃)=C(Br)-CO-morpholin-4-yl, -C(CH₃)=C(Br)-CO-NH-CH₂CH=C(Br)₂, -C(CH₃)=C(Br)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Br)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Br)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Br)-CO-NH-C₆H₅, -C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CN)-CO-NHCH₃, -C(CH₃)=C(CN)-CO-N(CH₃)₂, -C(CH₃)=C(CN)-CO-NH-C₂H₅, -C(CH₃)=C(CN)-CO-N(C₂H₅)₂, -C(CH₃)=C(CN)-CO-NH-n-C₃H₇, -C(CH₃)=C(CN)-CO-NH-i-C₃H₇, -C(CH₃)=C(CN)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-NH-cyclopropyl, -C(CH₃)=C(CN)-CO-NH-cyclobutyl, -C(CH₃)=C(CN)-CO-NH-cyclopentyl, -C(CH₃)=C(CN)-CO-NH-cyclohexyl, -C(CH₃)=C(CN)-CO-NH-cycloheptyl, -C(CH₃)=C(CN)-CO-NH-cyclooctyl, -C(CH₃)=C(CN)-CO-pyrrolidin-1-yl, -C(CH₃)=C(CN)-CO-piperidin-1-yl, -C(CH₃)=C(CN)-CO-morpholin-4-yl, -C(CH₃)=C(CN)-CO-NH-CH₂CH=C(CN)₂, -C(CH₃)=C(CN)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CN)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CN)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CN)-CO-NH-C₆H₅, -C(CH₃)=CH-SO-SCH₃, -C(CH₃)=CH-CO-SC₂H₅, -C(CH₃)=CH-CO-S-n-C₃H₇, -C(CH₃)=CH-CO-S-i-C₃H₇, -C(CH₃)=CH-CO-S-n-C₄H₉, -C(CH₃)=CH-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-SCH₃, -C(CH₃)=C(CH₃)-CO-SC₂H₅, -C(CH₃)=C(CH₃)-CO-S-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-S-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-SCH₃, -C(CH₃)=C(C₂H₅)-CO-SC₂H₅, -C(CH₃)=C(C₂H₅)-CO-S-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-SCH₃, -C(CH₃)=C(Cl)-CO-SC₂H₅, -C(CH₃)=C(Cl)-CO-S-n-C₃H₇, -C(CH₃)=C(Cl)-CO-S-i-C₃H₇, -C(CH₃)=C(Cl)-CO-S-n-C₄H₉, -C(CH₃)=C(Cl)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-SCH₃, -C(CH₃)=C(Br)-CO-SC₂H₅, -C(CH₃)=C(Br)-CO-S-n-C₃H₇, -C(CH₃)=C(Br)-CO-S-i-C₃H₇, -C(CH₃)=C(Br)-CO-S-n-C₄H₉, -C(CH₃)=C(Br)-CO-S-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-SCH₃, -C(CH₃)=C(CN)-CO-SC₂H₅, -C(CH₃)=C(CN)-CO-S-n-C₃H₇, -C(CH₃)=C(CN)-CO-S-i-C₃H₇, -C(CH₃)=C(CN)-CO-S-n-C₄H₉, -C(CH₃)=C(CN)-CO-S-tert.-C₄H₉, -C(CH₃)=C(COCH₃)-CO-OCH₃, -C(CH₃)=C(COC₂H₅)-CO-OCH₃, -C(CH₃)=C(CO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COCH₃)-CO-OC₂H₅, -C(CH₃)=C(COC₂H₅)-CO-OC₂H₅, -C(CH₃)=C(CO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COCH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(COC₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-OCH₃, -C(CH₃)=C(CF₃)-CO-OC₂H₅, -C(CH₃)=C(CF₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CF₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(COOCH₃)₂, -C(CH₃)=C(COOC₂H₅)₂, -C(CH₃)=C(COOCH₃)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)₂, -C(CH₃)=CH-CH=CH-COOH, -C(CH₃)=CH-CH=CH-CO-OCH₃, -C(CH₃)=CH-CH=CH-CO-OC₂H₅, -C(CH₃)=CH-CH=C(COOCH₃)₂, -C(CH₃)=CH-CH=C(CN)-CO-OCH₃, -C(CH₃)=CH-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH₂, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -C(CH₃)=CH-(CH₂)₂-COOH, -C(CH₃)=CH-(CH₂)₂-CO-OCH₃, -C(CH₃)=CH-(CH₂)₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(COOCH₃)₂, -C(CH₃)=CH-CH₂-CH(COOC₂H₅)₂, -C(CH₃)=CH-CH₂-CH(CN)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CN)-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -C(CH₃)=CH-(CH₂)₂-CO-NH₂, -C(CH₃)=CH-(CH₂)₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-COOH, -C(CH₃)=CH-CH₂-CO-OCH₃, -C(CH₃)=CH-CH₂-CO-OC₂H₅, -C(CH₃)=C(COOCH₃)-CH₂-CO-OCH₃, -C(CH₃)=C(COOCH₃)-CH₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CO-NH₂, -C(CH₃)=CH-CH₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-CO-N(CH₃)₂.
wobei W für eine der folgenden Bedeutungen steht:
-CHO, -COCH₃, -COC₂H₅, -CO-n-C₃H₇, -CO-i-C₃H₇, -CO-n-C₄H₉, -CO-i-C₄H₉, -CO-s-C₄H₉, -CO-tert.-C₄H₉, -CO-CH₂CH=CH₂, -CO-CF₃, -COCCl₃, -COCH₂C≡CH, -CO-cyclopropyl, -CO-cyclobutyl, -CO-cyclopentyl, -CO-cyclohexyl, -CO-CN, -CO-COOCH₃, -CO-COOC₂H₅, -CH=NH, -CH=NCH₃, -CH=NC₂H₅, -CH=N-n-C₃H₅, -CH=N-i-C₃H₅, -CH=N-n-C₄H₉, -CH=NCH₂CH=CH₂, -CH=NCH₂CH=CH₂-CH₃, -CH=NCH₂≡CH, -CH=NCH₂C≡C-CH₃, -CH=N-cyclopropyl, -CH=N-cyclobutyl, -CH=N-cyclopentyl, -CH=N-cyclohexyl, -CH=N-cycloheptyl, -CH=N-CH₂-CH₂Cl, -CH=N-CH₂Cl, -CH=N-C₆H₅, -CH=N-(4-Br-C₆H₄), -CH=N-3-F-C₆H₄, -CH=N-4-F-C₆H₄, -CH=N-2-Cl-C₆H₄, -CH=N-3-Cl-C₆H₄, -CH=N-4-Cl-C₆H₄, -CH=N-2-Br-C₆H₄, -CH=N-2-F-C₆H₄, -CH=N-2-CH₃-C₆H₄, -CH=N-3-CH₃-C₆H₄, -CH=N-4-CH₃-C₆H₄, -CH=N-2-CF₃-C₆H₄, -CH=N-3-CF₃-C₆H₄, -CH=N-4-CF₃-C₆H₄, -CH=N-2-OCH₃-C₆H₄, -CH=N-3-OCH₃-C₆H₄, -CH=N-4-OCH₃-C₆H₄, -CH=N-4-NO₂-C₆H₄, -CH=N-4-CN-C₆H₄, -CH=N-2,4-(Cl,Cl)-C₆H₄, -CH=N-2,4-(CH₃,CH₃)-C₆H₄, -CH=N-CH₂OCH₃ -CH=N-CH₂OC₂H₅, -CH=N-CH₂CH₂OCH₃, -CH=N-CH₂CH₂OC₂H₅, -CH=N-OH, -CH=N-OCH₃, -CH=N-OC₂H₅, -CH=N-O-n-C₃H₇, -CH=N-O-i-C₃H₇, -CH=N-O-n-C₄H₉, -CH=N-O-i-C₄H₉, -CH=N-O-s-C₄H₉, -CH=N-O-tert.-C₄H₉, -CH=N-O-CH₂CH=CH₂, -CH=N-O-CH(CH₃)CH=CH₂, -CH=N-O-CH₂C≡CH, -CH=N-O-CH(CH₃)-C≡CH, -CH=N-O-CH₂-CH=CH-CH₃, -CH=N-O-CH₂-CH₂-Cl, -CH=N-O-CH₂-CH₂-F, -CH=N-O-CH₂-CF₃, -CH=N-O-CH₂-CH=CHCl, -CH=N-O-CH₂-CCl=CH₂, -CH=N-O-CH₂-CBr=CH₂, -CH=N-O-CH₂-CH=CCl-CH₃, -CH=N-OC(O)CH₃, -CH=N-OC(O)C₂H₅, -CH=N-O-CH₂-CN, -CH=N-O-CH₂-CH=CH-CH₂-O-CH₃, -CH=N-O-CH₂-CH=CH-CH₂-O-tert.-C₄H₉, -CH=N-O-(CH₂)₃-C₆H₅, -CH=N-O-(CH₂)₄-C₆H₅, -CH=N-O-(CH₂)₄-4-Cl-C₆H₄, -CH=N-O-(CH₂)₄-4-OCH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-CH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-C₆H₅, -CH=N-O-CH₂CH=CH-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CH-3-OCH₃-C₆H₄, -CH=N-O-(CH₂)₂CH=CH-4-F-C₆H₄, -CH=N-O-(CH₂)CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CHCH₂-4-OCH₃-C₆H₄, -CH=N-O-CH₂-CH=C(CH₃)-C₆H₅ -CH=N-O-(CH₂)₂CH=CH-3,4(Cl,Cl)-C₆H₃, -CH=N-O-(CH₂)₃C≡C-4-F-C₆H₄, -CH₂=N-OCHOCH₃, -CH=N-OC₂H₄OCH₃, -CH=N-OCH₂OC₂H₅, -CH=N-OCH(CH₃)OCH₃, -CH=N-OCH(CH₃)COOCH₃, -CH=N-OCH(CH₃)COO-n-C₄H₉, -CH=N-NH₂, -CH=N-NHCH₃, -CH=N-NHC₂H₅, -CH=N-NH-n-C₃H₇, -CH=N-NH-i-C₃H₇, -CH=N-NH-n-C₄H₉, -CH=N-NH-i-C₄H₉, -CH=N-NH-s-C₄H₉, -CH=N-NH-tert.-C₄H₉, -CH=N-NH-cyclopropyl, -CH=N-NH-cyclobutyl, -CH=N-NH-cyclopentyl, -CH=N-NH-cyclohexyl, -CH=N-NH-cycloheptyl, -CH=N-N(CH₃)₂, -CH=N-N(C₂H₅)₂, -CH=N-N(C₃H₇)₂, -CH=N-N(i-C₃H₇)(CH₃), -CH=N-NHCH₂-C=CH, -CH=N-NHCH₂-C≡CH, -CH=N-N(CH₃)-CH₂-C≡CH, -CH=N-NHCH₂CF₃, -CH=N-NH-CO-CH₃, -CH=N-NH-CO-CH₂H₅, -CH=N-NH-COOCH₃, -CH=N-NH-COOC₂H₅, -CH=N-NH-COO-tert.-C₄H₉, -CH=N-pyrrolidin-1-yl, -CH=N-piperidin-1-yl, -CH=N-morpholin-4-yl, -CH=N-NH-C₆H₅, -CH=N-NH-(4-Cl-C₆H₄), -CH=N-NH-(4-NO₂-C₆H₄), -CH=N-NH-(4-F-C₆H₄), -CH=N-NH-(4-CH₃O-C₆H₄), -CH=N-NH-(2,4-Cl₂-C₆H₃), -CH=N-NH-(2,4-(NO₂)₂-C₆H₃), -CH=N-NH-CO-NH₂, -CH=N-NH-CO-NHCH₃, -CH=N-NH-CO-NHC₂H₅, -CH=N-NH-CO-N(CH₃)₂, -CH=CH-COOH, -CH=CH-CO-OCH₃, -CH=C-CO-OC₂H₅, -CH=CH-CO-O-n-C₃H₇, -CH=CH-CO-O-i-C₃H₇, -CH=CH-CO-O-n-C₄H₉, -CH=CH-CO-O-tert.-C₄H₉, -CH=CH-CO-O-cyclopropyl, -CH=CH-CO-O-cyclobutyl, -CH=CH-CO-O-cyclopentyl, -CH=CH-CO-O-cyclohexyl, -CH=CH-CO-O-cycloheptyl, -CH=C(CH₃)-COOH, -CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CO-O-n-C₃H₇, -CH=C(CH₃)-CO-O-i-C₃H₇, -CH=C(CH₃)-CO-O-n-C₄H₉, -CH=C(CH₃)-CO-O-tert.-C₄H₉, -CH=C(CH₃)-CO-O-cyclopropyl, -CH=C(CH₃)-CO-O-cyclobutyl, -CH=C(CH₃)-CO-O-cyclopentyl, -CH=C(CH₃)-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cycloheptyl, -CH=C(C₂H₅)-COOH, -CH=C(C₂H₅)-CO-OCH₃, -CH=C(C₂H₅)-CO-OC₂H₅, -CH=C(C₂H₅)-CO-O-n-C₃H₇, -CH=C(C₂H₅)-CO-O-i-C₃H₇, -CH=C(C₂H₅)-CO-O-n-C₄H₉, -CH=C(C₂H₅)-CO-O-tert.-C₄H₉, -CH=C(C₂H₅)-CO-O-cyclopropyl, -CH=C(C₂H₅)-CO-O-cyclobutyl, -CH=C(C₂H₅)-CO-O-cyclopentyl, -CH=C(C₂H₅)-CO-O-cyclohexyl, -CH=C(C₂H₅)-CO-O-cycloheptyl, -CH=C(Cl)-COOH, -CH=C(Cl)-CO-OCH₃, -CH=C(Cl)-CO-OC₂H₅, -CH=C(Cl)-CO-O-n-C₃H₇, -CH=C(Cl)-CO-O-i-C₃H₇, -CH=C(Cl)-CO-O-n-C₄H₉, -CH=C(Cl)-CO-O-tert.-C₄H₉, -CH=C(Cl)-CO-O-cyclopropyl, -CH=C(Cl)-CO-O-cyclobutyl, -CH=C(Cl)-CO-O-cyclopentyl, -CH=C(Cl)-CO-O-cyclohexyl, -CH=C(Cl)-CO-O-cycloheptyl, -CH=C(Br)-COOH, -CH=C(Br)-CO-OCH₃, -CH=C(Br)-CO-OC₂H₅, -CH=C(Br)-CO-O-n-C₃H₇, -CH=C(Br)-CO-O-i-C₃H₇, -CH=C(Br)-CO-O-n-C₄H₉, -CH=C(Br)-CO-O-tert.-C₄H₉, -CH=C(Br)-CO-O-cyclopropyl, -CH=C(Br)-CO-O-cyclobutyl, -CH=C(Br)-CO-O-cyclopentyl, -CH=C(Br)-CO-O-cyclohexyl, -CH=C(Br)-CO-O-cycloheptyl, -CH=C(CN)-COOH, -CH=C(CN)-CO-OCH₃, -CH=C(CN)-CO-OC₂H₅, -CH=C(CN)-CO-O-n-C₃H₇, -CH=C(CN)-CO-O-i-C₃H₇, -CH=C(CN)-CO-O-n-C₄H₉, -CH=C(CN)-CO-O-tert.-C₄H₉, -CH=C(CN)-CO-O-cyclopropyl, -CH=C(CN)-CO-O-cyclobutyl, -CH=C(CN)-CO-O-cyclopentyl, -CH=C(CN)-CO-O-cyclohexyl, -CH=C(CN)-CO-O-cycloheptyl, -CH=CH-CO-OCH₂-OCH₃, -CH=CH-CO-OCH₂-OC₂H₅, -CH=CH-CO-OCH₂-O-n-C₃H₅, -CH=CH-CO-OCH₂-O-i-C₃H₅, -CH=CH-CO-OCH(CH₃)-OCH₃, -CH=CH-CO-OCH(CH₃)-OC₂H₅, -CH=CH-CO-O-CH₂CH₂-OCH₃, -CH=CH-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-OCH₃, -CH=C(CH₃)-CO-OCH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-O-n-C₃H₅, -CH=C(CH₃)-CO-OCH₂-O-i-C₃H₅, -CH=C(CH₃)-CO-OCH(CH₃)-OCH₃, -CH=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CH₃)-CO-O-CH₂CH₂-OCH₃, -CH=C(CH₃)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-OCH₃, -CH=C(C₂H₅)-CO-OCH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-O-n-C₃H₅, -CH=C(C₂H₅)-CO-OCH₂-O-i-C₃H₅, -CH=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -CH=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OCH₃, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-OCH₃, -CH=C(Cl)-CO-OCH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-O-n-C₃H₅, -CH=C(Cl)-CO-OCH₂-O-i-C₃H₅, -CH=C(Cl)-CO-OCH(CH₃)-OCH₃, -CH=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Cl)-CO-O-CH₂CH₂-OCH₃, -CH=C(Cl)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-OCH₃, -CH=C(Br)-CO-OCH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-O-n-C₃H₅, -CH=C(Br)-CO-OCH₂-O-i-C₃H₅, -CH=C(Br)-CO-OCH(CH₃)-OCH₃, -CH=C(Br)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Br)-CO-O-CH₂CH₂-OCH₃, -CH=C(Br)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-OCH₃, -CH=C(CN)-CO-OCH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-O-n-C₃H₅, -CH=C(CN)-CO-OCH₂-O-i-C₃H₅, -CH=C(CN)-CO-OCH(CH₃)-OCH₃, -CH=C(CN)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CN)-CO-O-CH₂CH₂-OCH₃, -CH=C(CN)-CO-O-CH₂CH₂-OC₂H₅, -CH=CH-CO-OCH₂-CF₃, -CH=CH-CO-OCH₂-CCl₃, -CH=CH-CO-OCH₂-oxiranyl, -CH=CH-CO-O(CH₂)₃-Br, -CH=CH-CO-OCH₂-CH=CH₂, -CH=CH-CO-OCH₂-C≡CH, -CH=CH-CO-OCH₂-CN, -CH=CH-CO-O(CH₂)₂-CN, -CH=C(CH₃)-CO-OCH₂-CF₃, -CH=C(CH₃)-CO-OCH₂-CCl₃, -CH=C(CH₃)-CO-OCH₂-oxiranyl, -CH=C(CH₃)-CO-O(CH₂)₃-Br, -CH=C(CH₃)-CO-OCH₂-CH=CH₂, -CH=C(CH₃)-CO-OCH₂-C≡CH, -CH=C(CH₃)-CO-OCH₂-CN, -CH=C(CH₃)-CO-O(CH₂)₂-CN, -CH=C(C₂H₅)-CO-OCH₂-CF₃, -CH=C(C₂H₅)-CO-OCH₂-CCl₃, -CH=C(C₂H₅)-CO-OCH₂-oxiranyl, -CH=C(C₂H₅)-CO-O(CH₂)₃-Br, -CH=C(C₂H₅)-CO-OCH₂-CH=CH₂, -CH=C(C₂H₅)-CO-OCH₂-C≡CH, -CH=C(C₂H₅)-CO-OCH₂-CN, -CH=C(C₂H₅)-CO-O(CH₂)₂-CN, -CH=C(Cl)-CO-OCH₂-CF₃, -CH=C(Cl)-CO-OCH₂-CCl₃, -CH=C(Cl)-CO-OCH₂-oxiranyl, -CH=C(Cl)-CO-O(CH₂)₃-Br, -CH=C(Cl)-CO-OCH₂-CH=CH₂, -CH=C(Cl)-CO-OCH₂-C≡CH, -CH=C(Cl)-CO-OCH₂-CN, -CH=C(Cl)-CO-O(CH₂)₂-CN, -CH=C(Br)-CO-OCH₂-CF₃, -CH=C(Br)-CO-OCH₂-CCl₃, -CH=C(Br)-CO-OCH₂-oxiranyl, -CH=C(Br)-CO-O(CH₂)₃-Br, -CH=C(Br)-CO-OCH₂-CH=CH₂, -CH=C(Br)-CO-OCH₂-C≡CH, -CH=C(Br)-CO-OCH₂-CN, -CH=C(Br)-CO-O(CH₂)₂-CN, -CH=C(CN)-CO-OCH₂-CF₃, -CH=C(CN)-CO-OCH₂-CCl₃, -CH=C(CN)-CO-OCH₂-oxiranyl -CH=C(CN)-CO-O(CH₂)₃-Br, -CH=C(CN)-CO-OCH₂-CH=CH₂, -CH=C(CN)-CO-OCH₂-C≡CH, -CH=C(CN)-CO-OCH₂-CN, -CH=C(CN)-CO-O(CH₂)₂-CN, -CH=CH-CO-CH₃, -CH=CH-CO-C₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-i-C₃H₇, -CH=CH-CO-n-C₄H₉, -CH=CH-CO-tert.-C₄H₉, -CH=CH-CO-CH₂Cl, -CH=CH-CO-CH₂Br, -CH=CH-CO-CHCl₂, -CH=CH-CO-CH₂-OCH₃, -CH=CH-CO-CH(OCH₃)₂, -CH=CH-CO-CH₂-SCH₃, -CH=C(CH₃)-CO-CH₃, -CH=C(CH₃)-CO-C₂H₅, -CH=C(CH₃)-CO-n-C₃H₇, -CH=C(CH₃)-CO-i-C₃H₇, -CH=C(CH₃)-CO-n-C₄H₉, -CH=C(CH₃)-CO-tert.-C₄H₉, -CH=C(CH₃)-CO-CH₂Cl, -CH=C(CH₃)-CO-CH₂Br, -CH=C(CH₃)-CO-CHCl₂, -CH=C(CH₃)-CO-CH₂-OCH₃, -CH=C(CH₃)-CO-CH(OCH₃)₂, -CH=C(CH₃)-CO-CH₂-SCH₃, -CH=C(C₂H₅)-CO-CH₃, -CH=C(C₂H₅)-CO-C₂H₅, -CH=C(C₂H₅)-CO-n-C₃H₇, -CH=C(C₂H₅)-CO-i-C₃H₇, -CH=C(C₂H₅)-CO-n-C₄H₉, -CH=C(C₂H₅)-CO-tert.-C₄H₉, -CH=C(C₂H₅)-CO-CH₂Cl, -CH=C(C₂H₅)-CO-CH₂Br, -CH=C(C₂H₅)-CO-CHCl₂, -CH=C(C₂H₅)-CO-CH₂-OCH₃, -CH=C(C₂H₅)-CO-CH(OCH₃)₂, -CH=C(C₂H₅)-CO-CH₂-SCH₃, -CH=C(Cl)-CO-CH₃, -CH=C(Cl)-CO-C₂H₅, -CH=C(Cl)-CO-n-C₃H₇, -CH=C(Cl)-CO-i-C₃H₇, -CH=C(Cl)-CO-n-C₄H₉, -CH=C(Cl)-CO-tert.-C₄H₉, -CH=C(Cl)-CO-CH₂Cl, -CH=C(Cl)-CO-CH₂Br, -CH=C(Cl)-CO-CHCl₂, -CH=C(Cl)-CO-CH₂-OCH₃, -CH=C(Cl)-CO-CH(OCH₃)₂, -CH=C(Cl)-CO-CH₂-SCH₃, -CH=C(Br)-CO-CH₃, -CH=C(Br)-CO-C₂H₅, -CH=C(Br)-CO-n-C₃H₇, -CH=C(Br)-CO-i-C₃H₇, -CH=C(Br)-CO-n-C₄H₉, -CH=C(Br)-CO-tert.-C₄H₉, -CH=C(Br)-CO-CH₂Cl, -CH=C(Br)-CO-CH₂Br, -CH=C(Br)-CO-CHCl₂, -CH=C(Br)-CO-CH₂-OCH₃, -CH=C(Br)-CO-CH(OCH₃)₂, -CH=C(Br)-CO-CH₂-SCH₃, -CH=C(CN)-CO-CH₃, -CH=C(CN)-CO-C₂H₅, -CH=C(CN)-CO-n-C₃H₇, -CH=C(CN)-CO-i-C₃H₇, -CH=C(CN)-CO-n-C₄H₉, -CH=C(CN)-CO-tert.-C₄H₉, -CH=C(CN)-CO-CH₂Cl, -CH=C(CN)-CO-CH₂Br, -CH=C(CN)-CO-CHCl₂, -CH=C(CN)-CO-CH₂-OCH₃, -CH=C(CN)-CO-CH(OCH₃)₂, -CH=C(CN)-CO-CH₂-SCH₃, -CH=CH-CO-C₆H₅, -CH=CH-CO-(4-Cl-C₆H₄), -CH=C(CH₃)-CO-C₆H₅, -CH=C(CH₃)-CO-(4-Cl-C₆H₄), -CH=C(C₂H₅)-CO-C₆H₅, -CH=C(C₂H₅)-CO-(4-Cl-C₆H₄), -CH=C(Cl)-CO-C₆H₅, -CH=C(Br)-CO-C₆H₅, -CH=C(CN)-CO-C₆H₅, -CH=CH-CO-NH₂, -CH=CH-CO-NHCH₃, -CH=CH-CO-N(CH₃)₂, -CH=CH-CO-NH-C₂H₅, -CH=CH-CO-N(C₂H₅)₂, -CH=CH-CO-NH-n-C₃H₇, -CH=CH-CO-NH-i-C₃H₇, -CH=CH-CO-NH-tert.-C₄H₉, -CH=CH-CO-NH-cyclopropyl, -CH=CH-CO-NH-cyclobutyl, -CH=CH-CO-NH-cyclopentyl, -CH=CH-CO-NH-cyclohexyl, -CH=CH-CO-cycloheptyl, -CH=CH-CO-NH-cyclooctyl, -CH=CH-CO-pyrrolidin-1-yl, -CH=CH-CO-piperidin-1-yl, -CH=CH-CO-morpholin-4-yl, -CH=CH-CO-NH-CH₂CH=CH₂, -CH=CH-CO-NH-CH₂C≡CH, -CH=CH-CO-N(CH₃)-CH₂C≡CH, -CH=CH-CO-NH-(CH₂)₂Cl, -CH=CH-CO-NH-C₆H₅, -CH=C(CH₃)-CO-NH₂, -CH=C(CH₃)-CO-NHCH₃, -CH=C(CH₃)-CO-N(CH₃)₂, -CH=C(CH₃)-CO-NH-C₂H₅, -CH=C(CH₃)-CO-N(C₂H₅)₂, -CH=C(CH₃)-CO-NH-n-C₃H₇, -CH=C(CH₃)-CO-NH-i-C₃H₇, -CH=C(CH₃)-CO-NH-tert.-C₄H₉, -CH=C(CH₃)-CO-NH-cyclopropyl, -CH=C(CH₃)-CO-NH-cyclobutyl, -CH=C(CH₃)-CO-NH-cyclopentyl, -CH=C(CH₃)-CO-NH-cyclohexyl, -CH=C(CH₃)-CO-NH-cycloheptyl, -CH=C(CH₃)-CO-NH-cyclooctyl, -CH=C(CH₃)-CO-pyrrolidin-1-yl, -CH=C(CH₃)-CO-piperidin-1-yl, -CH=C(CH₃)-CO-morpholin-4-yl, -CH=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -CH=C(CH₃)-CO-NH-CH₂C≡CH, -CH=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CH₃)-CO-NH-(CH₂)₂Cl, -CH=C(CH₃)-CO-NH-C₆H₅, -CH=C(C₂H₅)-CO-NH₂, -CH=C(C₂H₅)-CO-NHCH₃, -CH=C(C₂H₅)-CO-N(CH₃)₂, -CH=C(C₂H₅)-CO-NH-C₂H₅, -CH=C(C₂H₅)-CO-N(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-n-C₃H₇, -CH=C(C₂H₅)-CO-NH-i-C₃H₇, -CH=C(C₂H₅)-CO-NH-tert.-C₄H₉, -CH=C(C₂H₅)-CO-NH-cyclopropyl, -CH=C(C₂H₅)-CO-NH-cyclobutyl, -CH=C(C₂H₅)-CO-NH-cyclopentyl, -CH=C(C₂H₅)-CO-NH-cyclohexyl, -CH=C(C₂H₅)-CO-NH-cycloheptyl, -CH=C(C₂H₅)-CO-NH-cyclooctyl, -CH=C(C₂H₅)-CO-pyrrolidin-1-yl, -CH=C(C₂H₅)-CO-piperidin-1-yl, -CH=C(C₂H₅)-CO-morpholin-4-yl, -CH=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-CH₂C≡CH, -CH=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -CH=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -CH=C(C₂H₅)-CO-NH-C₆H₅, -CH=C(Cl)-CO-NH₂, -CH=C(Cl)-CO-NHCH₃, -CH=C(Cl)-CO-N(CH₃)₂, -CH=C(Cl)-CO-NH-C₂H₅, -CH=C(Cl)-CO-N(C₂H₅)₂, -CH=C(Cl)-CO-NH-n-C₃H₇, -CH=C(Cl)-CO-NH-i-C₃H₇, -CH=C(Cl)-CO-NH-tert.-C₄H₉, -CH=C(Cl)-CO-NH-cyclopropyl, -CH=C(Cl)-CO-NH-cyclobutyl, -CH=C(Cl)-CO-NH-cyclopentyl, -CH=C(Cl)-CO-NH-cyclohexyl, -CH=C(Cl)-CO-NH-cycloheptyl, -CH=C(Cl)-CO-NH-cyclooctyl, -CH=C(Cl)-CO-pyrrolidin-1-yl, -CH=C(Cl)-CO-piperidin-1-yl, -CH=C(Cl)-CO-morpholin-4-yl, -CH=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -CH=C(Cl)-CO-NH-CH₂C≡CH, -CH=C(Cl)-CO-N(CH₃)-CH₂C-≡CH, -CH=C(Cl)-CO-NH-(CH₂)₂Cl, -CH=C(Cl)-CO-NH-C₆H₅, -CH=C(Br)-CO-NH₂, -CH=C(Br)-CO-NHCH₃, -CH=C(Br)-CO-N(CH₃)₂, -CH=C(Br)-CO-NH-C₂H₅, -CH=C(Br)-CO-N(C₂H₅)₂, -CH=C(Br)-CO-NH-n-C₃H₇, -CH=C(Br)-CO-NH-i-C₃H₇, -CH=C(Br)-CO-NH-tert.-C₄H₉, -CH=C(Br)-CO-NH-cyclopropyl, -CH=C(Br)-CO-NH-cyclobutyl, -CH=C(Br)-CO-NH-cyclopentyl, -CH=C(Br)-CO-NH-cyclohexyl, -CH=C(Br)-CO-NH-cycloheptyl, -CH=C(Br)-CO-NH-cyclooctyl, -CH=C(Br)-CO-pyrrolidin-1-yl, -CH=C(Br)-CO-piperidin-1-yl, -CH=C(Br)-CO-morpholin-4-yl, -CH=C(Br)-CO-NH-CH₂CH=C(Br)₂, -CH=C(Br)-CO-NH-CH₂C≡CH, -CH=C(Br)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Br)-CO-NH-(CH₂)₂Cl, -CH=C(Br)-CO-NH-C₆H₅, -CH=C(CN)-CO-NH₂, -CH=C(CN)-CO-NHCH₃, -CH=C(CN)-CO-N(CH₃)₂, -CH=C(CN)-CO-NH-C₂H₅, -CH=C(CN)-CO-N(C₂H₅)₂, -CH=C(CN)-CO-NH-n-C₃H₇, -CH=C(CN)-CO-NH-i-C₃H₇, -CH=C(CN)-CO-NH-tert.-C₄H₉, -CH=C(CN)-CO-NH-cyclopropyl, -CH=C(CN)-CO-NH-cyclobutyl, -CH=C(CN)-CO-NH-cyclopentyl, -CH=C(CN)-CO-NH-cyclohexyl, -CH=C(CN)-CO-NH-cycloheptyl, -CH=C(CN)-CO-NH-cyclooctyl, -CH=C(CN)-CO-pyrrolidin-1-yl, -CH=C(CN)-CO-piperidin-1-yl, -CH=C(CN)-CO-morpholin-4-yl, -CH=C(CN)-CO-NH-CH₂CH=C(CN)₂, -CH=C(CN)-CO-NH-CH₂C≡CH, -CH=C(CN)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CN)-CO-NH-(CH₂)₂Cl, -CH=C(CN)-CO-NH-C₆H₅, -CH=CH-CO-SCH₃, -CH=CH-CO-SC₂H₅, -CH=CH-CO-S-n-C₃H₇, -CH=CH-CO-S-i-C₃H₇, -CH=CH-CO-S-n-C₄H₉, -CH=CH-CO-S-tert.-C₄H₉, -CH=C(CH₃)-CO-SCH₃, -CH=C(CH₃)-CO-SC₂H₅, -CH=C(CH₃)-CO-S-n-C₃H₇, -CH=C(CH₃)-CO-S-i-C₃H₇, -CH=C(CH₃)-CO-S-n-C₄H₉, -CH=C(CH₃)-CO-S-tert.-C₄H₉, -CH=C(C₂H₅)-CO-SCH₃, -CH=C(C₂H₅)-CO-SC₂H₅, -CH=C(C₂H₅)-CO-S-n-C₃H₇, -CH=C(C₂H₅)-CO-S-i-C₃H₇, -CH=C(C₂H₅)-CO-S-n-C₄H₉, -CH=C(C₂H₅)-CO-S-tert.-C₄H₉, -CH=C(Cl)-CO-SCH₃, -CH=C(Cl)-CO-SC₂H₅, -CH=C(Cl)-CO-S-n-C₃H₇, -CH=C(Cl)-CO-S-i-C₃H₇, -CH=C(Cl)-CO-S-n-C₄H₉, -CH=C(Cl)-CO-S-tert.-C₄H₉, -CH=C(Br)-CO-SCH₃, -CH=C(Br)-CO-SC₂H₅, -CH=C(Br)-CO-S-n-C₃H₇, -CH=C(Br)-CO-S-i-C₃H₇, -CH=C(Br)-CO-S-n-C₄H₉, -CH=C(Br)-CO-S-tert.-C₄H₉, -CH=C(CN)-CO-SCH₃, -CH=C(CN)-CO-SC₂H₅, -CH=C(CN)-CO-S-n-C₃H₇, -CH=C(CN)-CO-S-i-C₃H₇, -CH=C(CN)-CO-S-n-C₄H₉, -CH=C(CN)-CO-S-tert.-C₄H₉, -CH=C(COCH₃)-CO-OCH₃, -CH=C(COC₂H₅)-CO-OCH₃, -CH=C(CO-n-C₃H₇)-CO-OCH₃, -CH=C(COCH₃)-CO-OC₂H₅, -CH=C(COC₂H₅)-CO-OC₂H₅, -CH=C(CO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COCH₃)-CO-O-n-C₃H₇, -CH=C(COC₂H₅)-CO-O-n-C₃H₇, -CH=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-OCH₃, -CH=C(CF₃)-CO-OC₂H₅, -CH=C(CF₃)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-O-i-C₃H₇, -CH=C(CF₃)-CO-O-n-C₄H₉, -CH=C(CF₃)-CO-O-tert.-C₄H₉, -CH=C(COOCH₃)₂, -CH=C(COOC₂H₅)₂, -CH=C(COOCH₃)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)-CO-OCH₃, -CH=C(COO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)₂, -CH=CH-CH=CH-COOH, -CH=CH-CH=CH-CO-OCH₃, -CH=CH-CH=CH-CO-OC₂H₅, -CH=CH-CH=C(COOCH₃)₂, -CH=CH-CH=C(CN)-CO-OCH₃, -CH=CH-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-OCH₃, -CH=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CH=C(Cl)-CO-OCH₃, -CH=C(CH₃)-CH=C(Br)-CO-OCH₃, -CH=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-NH₂, -CH=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -CH=CH-(CH₂)₂-COOH, -CH=CH-(CH₂)₂-CO-OCH₃, -CH=CH-(CH₂)₂-CO-OC₂H₅, -CH=CH-CH₂-CH(COOCH₃)₂, -CH=CH-CH₂-CH(COOC₂H₅)₂, -CH=CH-CH₂-CH(CN)-CO-OCH₃, -CH=CH-CH₂-CH(CN)-CO-OC₂H₅, -CH=CH-CH₂-CH(CH₃)-CO-OCH₃, -CH=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -CH=CH-(CH₂)₂-CO-NH₂, -CH=CH-(CH₂)₂-CO-NH-CH₃, -CH=CH-CH₂-COOH, -CH=CH-CH₂-CO-OCH₃, -CH=CH-CH₂-CO-OC₂H₅, -CH=C(COOCH₃)-CH₂-CO-OCH₃, -CH=C(COOCH₃)-CH₂-CO-OC₂H₅, -CH=CH-CH₂-CO-NH₂, -CH=CH-CH₂-CO-NH-CH₃, -CH=CH-CH₂-CO-N(CH₃)₂, -CH(OCH₃)₂, -CH(SCH₃)₂, -CH(OC₂H₅)₂, -CH(SC₂H₅)₂, -CH(O-n-C₃H₇)₂, -CH(O-i-C₃H₇)₂, -CH(S-n-C₃H₇)₂, -CH(S-i-C₃H₇)₂, -CH(O-n-C₄H₉)₂, -CH(O-i-C₄H₉)₂, -CH(O-s-C₄H₉)₂, -CH(O-tert.-C₄H₉)₂, -CH(S-n-C₄H₉)₂, -CH(S-i-C₄H₉)₂, -CH(S-s-C₄H₉)₂, -CH(S-tert.-C₄H₉)₂, -CH(OC₅H₁₁)₂, 1,3-Dioxolan-2-yl, 1,3-Dithio­ lan-2-yl, 1,3-Oxathiolan-2-yl, 4-Methyl-1,3-dioxolan-2-yl, 4-Methyl-1,3-dithiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 5-Methyl-1,3-oxathiolan-2-yl, 4-Ethyl-1,3-dioxolan-2-yl, 4-Ethyl- 1,4-dithiolan-2-yl, 4-Ethyl-1,3-oxathiolan-2-yl, 5-Ethyl-1,3-oxa­ thiolan-2-yl, 4,5-Dimethyl-1,3-dioxolan-2-yl, 4,4-Dimethyl-1,3- dioxolan-2-yl, 4,5-Dimethyl-1,3-dithiolan-2-yl, 5,5-Dimethyl-1,3- dithiolan-2-yl, 4,5-Dimethyl-1,3-oxathiolan-2-yl, 5,5-Dimethyl- 1,3-oxathiolan-2-yl, 4,4-Dimethyl-1,3-oxathiolan-2-yl, 4-Vinyl- 1,3-dioxolan-2-yl, 4-Vinyl-1,3-dithiolan-2-yl, 4-Vinyl-1,3-oxa­ thiolan-2-yl, 5-Vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3- dioxolan-2-yl, 4-Chlormethyl-1,3-dithiolan-2-yl, 4-Chlormethyl- 1,3-oxathiolan-2-yl, 5-Chlormethyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-1,3-dithio­ lan-2-yl, 4-Hydroxymethyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl- 1,3-oxathiolan-2-yl, 4-Methoxymethyl-1,3-dioxolan-2-yl, 4-Allyl­ oxymethyl-1,3-dioxolan-2-yl, 4-Propargyloxymethyl-1,3-dioxolan- 2-yl, 4-Acetoxymethyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-1,3-dithiolan-2-yl, 4-Propargyl­ oxymethyl-1,3-dithiolan-2-yl, 4-Acetoxymethyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-1,3-oxa­ thiolan-2-yl, 4-Allyloxymethyl-1,3-oxathiolan-2-yl, 5-Allyloxy­ methyl-1,3-oxathiolan-2-yl, 4-Propargyloxymethyl-1,3-oxathiolan- 2-yl, 5-Propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxymethyl- 1,3-oxathiolan-2-yl, 5-Acetoxymethyl-1,3-oxathiolan-2-yl, 4-Methylthiomethyl-1,3-dioxolan-2-yl, 4-Methylthiomethyl-1,3- dithiolan-2-yl, 4-Carboxy-1,3-dioxolan-2-yl, 4-Carboxy-1,3- dithiolan-2-yl, 4-Methoxycarbonyl-1,3-dioxolan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-1,3-di­ thiolan-2-yl, 4-n-Butoxycarbonyl-1,3-dithiolan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-4-methyl- 1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-di­ thiolan-2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-1,3- dithiolan-2-yl, 1,3-Dioxan-2-yl, 1,3-Dithian-2-yl, 1,3-Oxathian- 2-yl, 5-Methyl-1,3-dioxan-2-yl, 5-Methyl-1,3-dithian-2-yl, 5-Methyl-1,3-oxathian-2-yl, 5,5-Dimethyl-1,3-dioxan-2-yl, 4,6-Di­ methyl-1,3-dioxan-2-yl, 4,4-Dimethyl-1,3-dioxan-2-yl, 5,5-Di­ methyl-1,3-dithian-2-yl, 4,6-Dimethyl-1,3-dithian-2-yl, 4,4-Di­ methyl-1,3-dithian-2-yl, 5,5-Dimethyl-1,3-oxathian-2-yl, 4,4-Di­ methyl-1,3-oxathian-2-yl, 6,6-Dimethyl-1,3-oxathian-2-yl, 4-Hydroxymethyl-1,3-dioxan-2-yl, 4-Methoxymethyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-1,3-dioxan-2- yl, 4-Hydroxymethyl-1,3-dithian-2-yl, 4-Methoxymethyl-1,3-di­ thian-2-yl, 4-Allyloxymethyl-1,3-dithian-2-yl, 4-Acetoxymethyl- 1,3-dithian-2-yl, 4-Chlormethyl-1,3-dioxan-2-yl, 4-Chlormethyl- 1,3-dithian-2-yl, 1,3-Dioxepan-2-yl, 1,3-Dithiepan-2-yl, 1,3-Di­ oxep-5-en-2-yl, 4-Methoxycarbonyl-1,3-dioxan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-1,3-dithian- 2-yl, 4-n-Butoxycarbonyl-1,3-dithian-2-yl, 4-Methoxycarbonyl-4- methyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxan-2- yl, 4-n-Butoxyvarbonyl-4-methyl-1,3-dioxan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-4-methyl- 1,3-dithian-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithian-2-yl, -C(CH₃)(OCH₃)₂, -C(CH₃)(SCH₃)₂, -C(CH₃)(OC₂H₅)₂, -C(CH₃)(SC₂H₅)₂, -C(CH₃)(O-n-C₃H₇)₂, -C(CH₃)(O-i-C₃H₇)₂, -C(CH₃)(S-n-C₃H₇)₂, -C(CH₃)(S-i-C₃H₇)₂, -C(CH₃)(O-n-C₄H₉)₂, -C(CH₃)(O-i-C₄H₉)₂, -C(CH₃)(O-s-C₄H₉)₂, -C(CH₃)(O-tert.-C₄H₉)₂, -C(CH₃)(S-n-C₄H₉)₂, -C(CH₃)(S-i-C₄H₉)₂, -C(CH₃)(S-s-C₄H₉)₂, -C(CH₃)(S-tert.-C₄H₉)₂, -C(CH₃)(O-n-C₅H₁₁)′′, 2-Methyl-1,3-dixolan-2-yl, 2-Methyl-1,3-di­ thiolan-2-yl, 2-Methyl-1,3-oxathiolan-2-yl, 2,4-Dimethyl-1,3- dixolan-2-yl, 2,4-Dimethyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-1,3- oxathiolan-2-yl, 2,5-Dimethyl-1,3-oxathiolan-2-yl, 4-Ethyl-2- methyl-1,3-dioxolan-2-yl, 4-Ethyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Ethyl-2-methyl-1,3- oxathiolan-2-yl, 2,4,5-Trimethyl-1,3-dioxolan-2-yl, 2,4,4-Tri­ methyl-1,3-dioxolan-2-yl, 2,4,5-Trimethyl-1,3-dithiolan-2-yl, 2,4,4-Trimethyl-1,3-dithiolan-2-yl, 2,4,5-Trimethyl-1,3-oxathio­ lan-2-yl, 2,4,4-Trimethyl-1,3-oxathiolan-2-yl, 2-Methyl-4-vinyl- 1,3-dioxolan-2-yl, 2-Methyl-4-vinyl-1,3-dithiolan-2-yl, 2-Methyl- 4-vinyl-1,3-oxathiolan-2-yl, 2-Methyl-5-vinyl-1,3-oxathiolan-2- yl, 4-Chlormethyl-2-methyl-1,3-dioxolan-2-yl, 4-Chlormethyl-2- methyl-1,3-dithiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-oxathio­ lan-2-yl, 5-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Hydroxy­ methyl-2-methyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-2- methyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dioxolan- 2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxy- 2-methyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dithiolan-2-yl, 4-Acetoxy-2- methyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-oxathio­ lan-2-yl, 5-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Allyl­ oxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Allyloxymethyl-2- methyl-1,3-oxathiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3- oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3-oxathiolan-2- yl, 4-Acetoxy-2-methyl-1,3-oxathiolan-2-yl, 5-Acetoxy-2-methyl- 1,3-oxathiolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dioxolan-2- yl, 2-Methyl-4-methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-2- methyl-1,3-dioxolan-2-yl, 4-Carboxy-2-methyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-2- methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-2-methyl-1,3-dioxo­ lan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethoxy­ carbonyl-2-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-2- methyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-di­ oxolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-ethoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4- ethoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-n-butoxy­ carbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl-1,3- dithiolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-dioxan-2- yl, 2-Methyl-1,3-dithian-2-yl, 2-Methyl-1,3-oxathian-2-yl, 2,5- Dimethyl-1,3-dioxan-2-yl, 2,5-Dimethyl-1,3-dithian-2-yl, 2,5-Di­ methyl-1,3-oxathian-2-yl, 2,5,5-Trimethyl-1,3-dioxan-2-yl, 2,4,6- Trimethyl-1,3-dioxan-2-yl, 2,4,4-Trimethyl-1,3-dioxan-2-yl, 2,5,5-Trimethyl-1,3-dithian-2-yl, 2,4,6-Trimethyl-1,3-dithian-2- yl, 2,4,4-Trimethyl-1,3-dithian-2-yl, 2,5,5-Trimethyl-1,3-oxa­ thian-2-yl, 2,4,4-Trimethyl-1,3-oxathian-2-yl, 2,6,6-Trimethyl- 1,3-oxathian-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-2- methyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dithian-2-yl, 4-Methoxymethyl-2- methyl-1,3-dithian-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithian-2- yl, 4-Acetoxymethyl-2-methyl-1,3-dithian-2-yl, 4-Chlormethyl-2- methyl-1,3-dioxan-2-yl, 4-Chlormethyl-2-methyl-1,3-dithian-2-yl, -C(CH₃)=NH, -C(CH₃)=N-CH₃, -C(CH₃)=N-C₂H₅, -C(CH₃)=N-n-C₃H₇, -C(CH₃)=N-i-C₃H₇, -C(CH₃)=N-n-C₄H₉, -C(CH₃)=N-CH₂CH=CH₂, -C(CH₃)=N-CH₂CH=CH₂-CH₃, -C(CH₃)=N-CH₂C≡CH, -C(CH₃)=N-CH₂C≡C-CH₃, -C(CH₃)=N-cyclopropyl, -C(CH₃)=N-cyclobutyl, -C(CH₃)=N-cyclo­ pentyl, -C(CH₃)=N-cyclohexyl, -C(CH₃)=N-cycloheptyl, -C(CH₃)=N-CH₂-CH₂Cl, -C(CH₃)=N-CH₂Cl, -C(CH₃)=N-C₆H₅, -C(CH₃)=N-(2-F-C₆H₄), -C(CH₃)=N-(3-F-C₆H₄), -C(CH₃)=N-(4-F-C₆H₄), -C(CH₃)=N-(2-Cl-C₆H₄), -C(CH₃)=N-(3-Cl-C₆H₄), -C(CH₃)=N-(4-Cl-C₆H₄), -C(CH₃)=N-(2-CH₃-C₆H₄), -C(CH₃)=N-(3-CH₃-C₆H₄), -C(CH₃)=N-(4-CH₃-C₆H₄), -C(CH₃)=N-(2-CF₃-C₆H₄), -C(CH₃)=N-(3-CF₃-C₆H₄), -C(CH₃)=N-(4-CF₃-C₆H₄), -C(CH₃)=N-(2-OCH₃-C₆H₄), -C(CH₃)=N-(3-OCH₃-C₆H₄), -C(CH₃)=N-(4-OCH₃-C₆H₄), -C(CH₃)=N-(4-NO₂-C₆H₄), -C(CH₃)=N-(4-CN-C₆H₄), -C(CH₃)=N-(2,4-Cl₂-C₆H₄), -C(CH₃)=N-(2,4-(CH₃)₂-C₆H₃), -C(CH₃)=N-CH₂-OCH₃, -C(CH₃)=N-CH₂-OC₂H₅, -C(CH₃)=N-CH₂CH₂-OCH₃, -C(CH₃)=N-CH₂CH₂-OC₂H₅, -C(CH₃)=N-OH, -C(CH₃)=N-OCH₃, -C(CH₃)=N-OC₂H₅, -C(CH₃)=N-O-n-C₃H₇, -C(CH₃)=N-O-i-C₃H₇, -C(CH₃)=N-O-n-C₄H₉, -C(CH₃)=N-O-i-C₄H₉, -C(CH₃)=N-O-s-C₄H₉, -C(CH₃)=N-O-tert.-C₄H₉, -C(CH₃)=N-OCH₂-CH=CH₂, -C(CH₃)=N-OCH(CH₃)-CH=CH₂, -C(CH₃)=N-OCH₂-C≡CH, -C(CH₃)=N-CH(CH₃)-C≡CH, -C(CH₃)=N-OCH₂-CH=C-CH₃, -C(CH₃)=N-OCH₂CH₂-Cl, -C(CH₃)=N-OCH₂CH₂-F, -C(CH₃)=N-OCH₂-CF₃, -C(CH₃)=N-OCH₂-CH=CHCl, -C(CH₃)=N-OCH₂-C(Cl)=CH₂, -C(CH₃)=N-OCH₂-C(Br)=CH₂, -C(CH₃)=N-OCH₂-CH=C(Cl)-CH₃, -C(CH₃)=N-O-CO-CH₃, -C(CH₃)=N-O-CO-C₂H₅, -C(CH₃)=N-OCH₂-CN, -C(CH₃)=N-OCH₂-CH=CH-CH₂-OCH₃, -C(CH₃)=N-OCH₂-CH=CH-CH₂-O-tert.-C₄H₉, -C(CH₃)=N-O-(CH₂)₃-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-(4-Cl-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₂O-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-C₆H₅, -C(CH₃)=N-OCH₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(3-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-CH₂-(4-CH₃O-C₆H₄), -C(CH₃)=N-OCH₂-CH=C(CH₃)-C₆H₅, -C(CH₃)=N-O-(CH₂)₂-CH=CH-(3,4-Cl₂-C₆H₃), -C(CH₃)=N-O-(CH₂)₃-C≡C-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-OCH₃, -C(CH₃)=N-OCH₂CH₂-OCH₃, -C(CH₃)=N-OCH₂-OC₂H₅, -C(CH₃)=N-OCH(CH₃)-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=N-NH₂, -C(CH₃)=N-NH-CH₃, -C(CH₃)=N-NH-C₂H₅, -C(CH₃)=N-NH-n-C₃H₇, -C(CH₃)=N-NH-i-C₃H₇, -C(CH₃)=N-NH-n-C₄H₉, -C(CH₃)=N-NH-i-C₄H₉, -C(CH₃)=N-NH-s-C₄H₉, -C(CH₃)=N-NH-tert.-C₄H₉, -C(CH₃)=N-NH-cyclopropyl, -C(CH₃)=N-NH- cyclobutyl, -C(CH₃)=N-NH-cyclopentyl, -C(CH₃)=N-NH-cyclohexyl, -C(CH₃)=N-NH-cycloheptyl, -C(CH₃)=N-N(CH₃)₂, -C(CH₃)=N-N(C₂H₅)₂, -C(CH₃)=N-N(n-C₃H₇)₂, -C(CH₃)=N-N(i-C₃H₇)₂, -C(CH₃)=N-NH-CH₂-C=CH, -C(CH₃)=N-NH-CH₂-C≡CH, -C(CH₃)=N-N(CH₃)-CH₂-C≡CH, -C(CH₃)=N-NH-CH₂CF₃, -C(CH₃)=N-NH-CO-CH₃, -C(CH₃)=N-NH-CO-C₂H₅, -C(CH₃)=N-NH-CO-OCH₃, -C(CH₃)=N-NH-CO-OC₂H₅, -C(CH₃)=N-NH-CO-O-tert.-C₄H₉, -C(CH₃)=N- pyrrolidin-1-yl, -C(CH₃)=N-piperidin-1-yl, -C(CH₃)=N-morpholin- 4-yl, -C(CH₃)=N-NHC₆H₅, -C(CH₃)=N-NH-(4-Cl-C₆H₄), -C(CH₃)=N-NH-(4-NO₂-C₆H₄), -C(CH₃)=N-NH-(4-F-C₆H₄), -C(CH₃)=N-NH-(4-CH₃O-C₆H₄), -C(CH₃)=N-NH-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-NH-(2,4-(NO₂)₂-C₆H₃), -C(CH₃)=N-NH-CO-NH₂, -C(CH₃)=N-NH-CO-NHCH₃, -C(CH₃)=N-NH-CO-NHC₂H₅, -C(CH₃)=N-NH-CO-N(CH₃)₂, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=CH-CO-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-O-n-C₄H₉, -C(CH₃)=CH-CO-O-tert.-C₄H₉, -C(CH₃)=CH-CO-O-cyclopropyl, -C(CH₃)=CH-CO-O-cyclobutyl, -C(CH₃)=CH-CO-O-cyclopentyl, -C(CH₃)=CH-CO-O-cyclohexyl, -C(CH₃)=CH-CO-O-cycloheptyl, -C(CH₃)=C(CH₃)-COOH, -C(CH₃)=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-cyclopropyl, -C(CH₃)=C(CH₃)-CO-O-cyclobutyl, -C(CH₃)=C(CH₃)-CO-O-cyclopentyl, -C(CH₃)=C(CH₃)-CO-O-cyclohexyl, -C(CH₃)=C(CH₃)-CO-O-cycloheptyl, -C(CH₃)=C(C₂H₅)-COOH, -C(CH₃)=C(C₂H₅)-CO-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-cyclo­ propyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-O- cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-O-cycloheptyl, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=C(Cl)-CO-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-O-n-C₄H₉, -C(CH₃)=C(Cl)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-O-cyclopropyl, -C(CH₃)=C(Cl)-CO-O-cyclobutyl, -C(CH₃)=C(Cl)-CO-O-cyclopentyl, -C(CH₃)=C(Cl)-CO-O-cyclohexyl, -C(CH₃)=C(Cl)-CO-O-cycloheptyl, -C(CH₃)=C(Br)-COOH, -C(CH₃)=C(Br)-CO-OCH₃, -C(CH₃)=C(Br)-CO-OC₂H₅, -C(CH₃)=C(Br)-CO-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-O-n-C₄H₉, -C(CH₃)=C(Br)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-O-cyclopropyl, -C(CH₃)=C(Br)-CO-O-cyclobutyl, -C(CH₃)=C(Br)-CO-O-cyclopentyl, -C(CH₃)=C(Br)-CO-O-cyclohexyl, -C(CH₃)=C(Br)-CO-O-cycloheptyl, -C(CH₃)=C(CN)-COOH, -C(CH₃)=C(CN)-CO-OCH₃, -C(CH₃)=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CN)-CO-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-O-n-C₄H₉, -C(CH₃)=C(CN)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-O-cyclopropyl, -C(CH₃)=C(CN)-CO-O-cyclobutyl, -C(CH₃)=C(CN)-CO-O-cyclopentyl, -C(CH₃)=C(CN)-CO-O-cyclohexyl, -C(CH₃)=C(CN)-CO-O-cycloheptyl, -C(CH₃)=CH-CO-OCH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-OCH(CH₃)-OCH₃, -C(CH₃)=CH-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=CH-CO-OCH₂CH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(C 99999 00070 552 001000280000000200012000285919988800040 0002004131038 00004 99880₂H₅)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-O-i-C₃H₇, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -(CH₃)=C(Cl)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-O-i-C₃H₇, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-O-i-C₃H₇, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-CF₃, -C(CH₃)=CH-CO-OCH₂-CCl₃, -C(CH₃)=CH-CO-OCH₂-oxiranyl, -C(CH₃)=CH-CO-(CH₂)₃-Br, -C(CH₃)=CH-CO-OCH₂-CH=CH₂, -C(CH₃)=CH-CO-OCH₂-C≡CH, -C(CH₃)=CH-CO-OCH₂-CN, -C(CH₃)=CH-CO-OCH₂CH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CF₃, -C(CH₃)=C(CH₃)-CO-OCH₂-CCl₃, -C(CH₃)=C(CH₃)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CH₃)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CH₃)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CH₃)-CO-OCH₂-C≡CH, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CF₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CCl₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-oxiranyl, -C(CH₃)=C(C₂H₅)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(C₂H₅)-CO-OCH₂-C≡CH, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-C₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂-CF₃, -C(CH₃)=C(Cl)-CO-OCH₂-CCl₃, -C(CH₃)=C(Cl)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Cl)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Cl)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Cl)-CO-OCH₂-C≡CH, -C(CH₃)=C(Cl)-CO-OCH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂-CF₃, -C(CH₃)=C(Br)-CO-OCH₂-CCl₃, -C(CH₃)=C(Br)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Br)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Br)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Br)-CO-OCH₂-C≡CH, -C(CH₃)=C(Br)-CO-OCH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂CH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂-CF₃, -C(CH₃)=C(CN)-CO-OCH₂-CCl₃, -C(CH₃)=C(CN)-OCH₂-oxiranyl, -C(CH₃)=C(CN)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CN)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CN)-CO-OCH₂-C≡CH, -C(CH₃)=C(CN)-CO-OCH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂CH₂-CN, -C(CH₃)=CH-CO-CH₃, -C(CH₃)=CH-CO-C₂H₅, -C(CH₃)=CH-CO-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-n-C₄H₉, -C(CH₃)=CH-CO-tert.-C₄H₉, -C(CH₃)=CH-CO-CH₂Cl, -C(CH₃)=CH-CO-CH₂Br, -C(CH₃)=CH-CO-CHCl₂, -C(CH₃)=CH-CO-CH₂-OCH₃, -C(CH₃)=CH-CO-CH(OCH₃)₂, -C(CH₃)=CH-CO-CH₂-SCH₃, -C(CH₃)=C(CH₃)-CO-CH₃, -C(CH₃)=C(CH₃)-CO-C₂H₅, -C(CH₃)=C(CH₃)-CO-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-CH₂Cl, -C(CH₃)=C(CH₃)-CO-CH₂Br, -C(CH₃)=C(CH₃)-CO-CHCl₂, -C(CH₃)=C(CH₃)-CO-CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-CH(OCH₃)₂, -C(CH₃)=C(CH₃)-CO-CH₂-SCH₃, -C(CH₃)=C(C₂H₅)-CO-CH₃, -C(CH₃)=C(C₂H₅)-CO-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-CH₂Cl, -C(CH₃)=C(C₂H₅)-CO-CH₂Br, -C(CH₃)=C(C₂H₅)-CO-CHCl₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-CH(OCH₃)₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-SCH₃, -C(CH₃)=C(Cl)-CO-CH₃, -C(CH₃)=C(Cl)-CO-C₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-n-C₄H₉, -C(CH₃)=C(Cl)-CO-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-CH₂Cl, -C(CH₃)=C(Cl)-CO-CHCl₂, -C(CH₃)=C(Cl)-CO-CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-CH(OCH₃)₂, -C(CH₃)=C(Cl)-CO-CH₂-SCH₃, -C(CH₃)=C(Br)-CO-CH₃, -C(CH₃)=C(Br)-CO-C₂H₅, -C(CH₃)=C(Br)-CO-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-n-C₄H₉, -C(CH₃)=C(Br)-CO-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-CH₂Cl, -C(CH₃)=C(Br)-CO-CH₂Br, -C(CH₃)=C(Br)-CO-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-CH(OCH₃)₂, -C(CH₃)=C(Br)-CO-CH₂-SCH₃, -C(CH₃)=C(CN)-CO-CH₃, -C(CH₃)=C(CN)-CO-C₂H₅, -C(CH₃)=C(CN)-CO-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-n-C₄H₉, -C(CH₃)=C(CN)-CO-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-CH₂Cl, -C(CH₃)=C(CN)-CO-CH₂Br, -C(CH₃)=C(CN)-CO-CHCl₂, -C(CH₃)=C(CN)-CO-CH₂-OCH₃, -C(CH₃)=C(CN)-CO-CH(OCH₃)₂, -C(CH₃)=C(CN)-CO-CH₂-SCH₃, -C(CH₃)=CH-CO-C₆H₅, -C(CH₃)=CH-CO-(4-Cl-C₆H₄), -C(CH₃)=C(CH₃)-CO-C₆H₅, -C(CH₃)=C(CH₃)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(C₂H₅)-CO-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(Cl)-CO-C₆H₅, -C(CH₃)=C(Br)-CO-C₆H₅, -C(CH₃)=C(CN)-CO-C₆H₅, -C(CH₃)=CH-CO-NH₂, -C(CH₃)=CH-CO-NHCH₃, -C(CH₃)=CH-CO-N(CH₃)₂, -C(CH₃)=CH-CO-NH-C₂H₅, -C(CH₃)=CH-CO-N(C₂H₅)₂, -C(CH₃)=CH-CO-NH-n-C₃H₇, -C(CH₃)=CH-CO-NH-i-C₃H₇, -C(CH₃)=CH-CO-NH-tert.-C₄H₉, -C(CH₃)=CH-CO-NH-cyclopropyl, -C(CH₃)=CH-CO-NH-cyclobutyl, -C(CH₃)=CH-CO-NH-cyclopentyl, -C(CH₃)=CH-CO-NH-cyclohexyl, -C(CH₃)=CH-CO-NH-cycloheptyl, -C(CH₃)=CH-CO-NH-cyclooctyl, -C(CH₃)=CH-CO-pyrrolidin-1-yl, -C(CH₃)=CH-CO-piperidin-1-yl, -C(CH₃)=CH-CO-morpholin-4-yl, -C(CH₃)=CH-CO-NH-CH₂CH=CH₂, -C(CH₃)=CH-CO-NH-CH₂C≡CH, -C(CH₃)=CH-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=CCH-CO-NH-(CH₂)₂Cl, -C(CH₃)=CH-CO-NH-C₆H₅, -C(CH₃)=C(CH₃)-CO-NH₂, -C(CH₃)=C(CH₃)-CO-NHCH₃, -C(CH₃)=C(CH₃)-CO-N(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-C₂H₅, -C(CH₃)=C(CH₃)-CO-N(C₂H₅)₂, -C(CH₃)=C(CH₃)-CO-NH-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-NH- cyclopropyl, -C(CH₃)=C(CH₃)-CO-NH-cyclobutyl, -C(CH₃)=C(CH₃)-CO-NH-cyclopentyl, -C(CH₃)=C(CH₃)-CO-NH- cyclehexyl, -C(CH₃)=C(CH₃)-CO-NH-cycloheptyl, -C(CH₃)=C(CH₃)-CO-NH-cyclooctyl, -C(CH₃)=C(CH₃)-CO- pyrrolidin-1-yl, -C(CH₃)=C(CH₃)-CO-piperidin-1-yl, -C(CH₃)=C(CH₃)-CO-morpholin-4-yl, -C(CH₃)=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-NH(CH₂)₂Cl, -C(CH₃)=C(CH₃)-CO-NH-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-NH₂, -C(CH₃)=C(C₂H₅)-CO-NHCH₃, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)₂, -C(CH₃)=C(C₂H₅)-CO-NH-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-N(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-NH- cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclo­ hexyl, -C(CH₃)=C(C₂H₅)-CO-NH-cycloheptyl, -C(CH₃)=C(C₂H₅)-CO-NH- cyclooctyl, -C(CH₃)=C(C₂H₅)-CO-pyrrolidin-1-yl, -C(CH₃)=C(C₂H₅)-CO-piperidin-1-yl, -C(CH₃)=C(C₂H₅)-CO- morpholin-4-yl, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(C₂H₅)-CO-NH-C₆H₅, -C(CH₃)=C(Cl)-CO-NH₂, -C(CH₃)=C(Cl)-CO-NHCH₃, -C(CH₃)=C(Cl)-CO-N(CH₃)₂, -C(CH₃)=C(Cl)-CO-NH-C₂H₅, -C(CH₃)=C(Cl)-CO-N(C₂H₅)₂, -C(CH₃)=C(Cl)-CO-NH-n-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-i-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-NH-cyclopropyl, -C(CH₃)=C(Cl)-CO-NH-cyclobutyl, -C(CH₃)=C(Cl)-CO-NH-cyclopentyl, -C(CH₃)=C(Cl)-CO-NH-cyclohexyl, -C(CH₃)=C(Cl)-CO-NH-cycloheptyl, -C(CH₃)=C(Cl)-CO-NH-cyclooctyl, -C(CH₃)=C(Cl)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Cl)-CO-piperidin-1- yl, -C(CH₃)=C(Cl)-CO-morpholin-4-yl, -C(CH₃)=C(Cl)-CO-NH-CH₂CH=C(Cl)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-N(CH₃)-CH₂≡CH, -C(CH₃)=C(Cl)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Cl)-NO-NH-C₆H₅, -C(CH₃)=C(Br)-CO-NH₂, -C(CH₃)=C(Br)-CO-NHCH₃, -C(CH₃)=C(Br)-CO-N(CH₃)₂, -C(CH₃)=C(Br)-CO-NH-C₂H₅, -C(CH₃)=C(Br)-CO-N(C₂H₅)₂, -C(CH₃)=C(Br)-CO-NH-n-C₃H₇, -C(CH₃)=C(Br)-CO-NH-i-C₃H₇, -C(CH₃)=C(Br)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-NH-cyclopropyl, -C(CH₃)=C(Br)-CO-NH-cyclobutyl, -C(CH₃)=C(Br)-CO-NH-cyclopentyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cycloheptyl, -C(CH₃)=C(Br)-CO-NH-cyclooctyl, -C(CH₃)=C(Br)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Br)-CO-piperidin-1-yl, -C(CH₃)=C(Br)-CO-morpholin-4-yl, -C(CH₃)=C(Br)-CO-NH-CH₂CH=C(Br)₂, -C(CH₃)=C(Br)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Br)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Br)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Br)-CO-NH-C₆H₅, -C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CN)-CO-NHCH₃, -C(CH₃)=C(CN)-CO-N(CH₃)₂, -C(CH₃)=C(CN)-CO-NH-C₂H₅, -C(CH₃)=C(CN)-CO-N(C₂H₅)₂, -C(CH₃)=C(CN)-CO-NH-n-C₃H₇, -C(CH₃)=C(CN)-CO-NH-i-C₃H₇, -C(CH₃)=C(CN)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-NH-cyclopropyl, -C(CH₃)=C(CN)-CO-NH-cyclobutyl, -C(CH₃)=C(CN)-CO-NH-cyclopentyl, -C(CH₃)=C(CN)-CO-NH-cyclohexyl, -C(CH₃)=C(CN)-CO-NH-cycloheptyl, -C(CH₃)=C(CN)-CO-NH-cyclooctyl, -C(CH₃)=C(CN)-CO-pyrrolidin-1-yl, -C(CH₃)=C(CN)-CO-piperidin-1-yl, -C(CH₃)=C(CN)-CO-morpholin-4-yl, -C(CH₃)=C(CN)-CO-NH-CH₂CH=C(CN)₂, -C(CH₃)=C(CN)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CN)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=(CN)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CN)-CO-NH-C₆H₅, -C(CH₃)=CH-CO-SCH₃, -C(CH₃)=CH-CO-SC₂H₅, -C(CH₃)=CH-CO-S-n-C₃H₇, -C(CH₃)=CH-CO-S-i-C₃H₇, -C(CH₃)=CH-CO-S-n-C₄H₉, -C(CH₃)=CH-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-SCH₃, -C(CH₃)=C(CH₃)-CO-SC₂H₅, -C(CH₃)=C(CH₃)CO-S-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-S-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-SCH₃, -C(CH₃)=C(C₂H₅)-CO-SC₂H₅, -C(CH₃)=C(C₂H₅)-CO-S-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-SCH₃, -C(CH₃)=C(Cl)-CO-SC₂H₅, -C(CH₃)=C(Cl)-CO-S-n-C₃H₇, -C(CH₃)=C(Cl)-CO-S-i-C₃H₇, -C(CH₃)=C(Cl)-CO-S-n-C₄H₉, -C(CH₃)=C(Cl)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-SCH₃, -C(CH₃)=C(Br)-CO-SC₂H₅, -C(CH₃)=C(Br)-CO-S-n-C₃H₇, -C(CH₃)=C(Br)-CO-S-i-C₃H₇, -C(CH₃)=C(Br)-CO-S-n-C₄H₉, -C(CH₃)=C(Br)-CO-S-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-SCH₃, -C(CH₃)=C(CN)-CO-SC₂H₅, -C(CH₃)=C(CN)-CO-S-n-C₃H₇, -C(CH₃)=C(CN)-CO-S-i-C₃H₇, -C(CH₃)=C(CN)-CO-S-n-C₄H₉, -C(CH₃)=C(CN)-CO-S-tert.-C₄H₉, -C(CH₃)=C(COCH₃)-CO-OCH₃, -C(CH₃)=C(COC₂H₅)-CO-OCH₃, -C(CH₃)=C(CO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COCH₃)-CO-OC₂H₅, -C(CH₃)=C(COC₂H₅)-CO-OC₂H₅, -C(CH₃)=C(CO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COCH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(COC₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-OCH₃, -C(CH₃)=C(CF₃)-CO-OC₂H₅, -C(CH₃)=C(CF₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CF₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(COOCH₃)₂, -C(CH₃)=C(COOC₂H₅)₂, -C(CH₃)=C(COOCH₃)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)₂, -C(CH₃)=CH-CH=CH-COOH, -C(CH₃)=CH-CH=CH-CO-OCH₃, -C(CH₃)=CH-CH=CH-CO-OC₂H₅, -C(CH₃)=CH-CH=C(COOCH₃)₂, -C(CH₃)=CH-CH=C(CN)-CO-OCH₃, -C(CH₃)=CH-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH₂, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -C(CH₃)=CH-(CH₂)₂-COOH, -C(CH₃)=CH-(CH₂)₂-CO-OCH₃, -C(CH₃)=CH-(CH₂)₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(COOCH₃)₂, -C(CH₃)=CH-CH₂-CH(COOC₂H₅)₂, -C(CH₃)=CH-CH₂-CH(CN)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CN)-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -C(CH₃)=CH-(CH₂)₂-CO-NH₂, -C(CH₃)=CH-(CH₂)₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-COOH, -C(CH₃)=CH-CH₂-CO-OCH₃, -C(CH₃)=CH-CH₂-CO-OC₂H₅, -C(CH₃)=C(COOCH₃)-CH₂-CO-OCH₃, -C(CH₃)=C(COOCH₃)-CH₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CO-NH₂, -C(CH₃)=CH-CH₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-CO-N(CH₃)₂.
wobei W für eine der folgenden Bedeutungen steht:
-CHO, -COCH₃, -COC₂H₅, -CO-n-C₃H₇, -CO-i-C₃H₇, -CO-n-C₄H₉, -CO-i-C₄H₉, -CO-s-C₄H₉, -CO-tert.-C₄H₉, -CO-CH₂CH=CH₂, -CO-CF₃, -COCCl₃, -COCH₂C≡CH, -CO-cyclopropyl, -CO-cyclobutyl, -CO-cyclo­ pentyl, -CO-cyclohexyl, -CO-CN, -CO-COOCH₃, -CO-COOC₂H₅, -CH=NH, -CH=NCH₃, -CH=NC₂H₅, -CH=N-n-C₃H₅, -CH=N-i-C₃H₅, -CH=N-n-C₄H₉, -CH=NCH₂CH=CH₂, -CH=NCH₂CH=CH₂-CH₃, -CH=NCH₂≡CH, -CH=NCH₂C≡C-CH₃, -CH=N-cyclopropyl, -CH=N-cyclobutyl, -CH=N-cyclopentyl, -CH=N-cyclohexyl, -CH=N-cycloheptyl, -CH=N-CH₂-CH₂Cl, -CH=N-CH₂Cl, -CH=N-C₆H₅, -CH=N-4-Br-C₆H₄, -CH=N-3-F-C₆H₄, -CH=N-4-F-C₆H₄, -CH=N-2-Cl-C₆H₄, -CH=N-3-Cl-C₆H₄, -CH=N-4-Cl-C₆H₄, -CH=N-2-Br-C₆H₄, -CH=N-2-F-C₆H₄, -CH=N-2-CH₃-C₆H₄, -CH=N-3-CH₃-C₆H₄, -CH=N-4-CH₃-C₆H₄, -CH=N-2-CF₃-C₆H₄, -CH=N-3-CF₃-C₆H₄, -CH=N-4-CF₃-C₆H₄, -CH=N-2-OCH₃-C₆H₄, -CH=N-3-OCH₃-C₆H₄, -CH=N-4-OCH₃-C₆H₄, -CH=N-4-NO₂-C₆H₄, -CH=N-4-CN-C₆H₄, -CH=N-2,4-(Cl,Cl)-C₆H₄, -CH=N-2,4-(CH₃,CH₃)-C₆H₄, -CH=N-CH₂OCH₃ -CH=N-CH₂OC₂H₅, -CH=N-CH₂CH₂OCH₃, -CH=N-CH₂CH₂OC₂H₅, -CH=N-OH, -CH=N-OCH₃, -CH=N-OC₂H₅, -CH=N-O-n-C₃H₇, -CH=N-O-i-C₃H₇, -CH=N-O-n-C₄H₉, -CH=N-O-i-C₄H₉, -CH=N-O-s-C₄H₉, -CH=N-O-tert.-C₄H₉, -CH=N-O-CH₂CH=CH₂, -CH=N-O-CH(CH₃)CH=CH₂, -CH=N-O-CH₂C≡CH, -CH=N-O-CH(CH₃)-C≡CH, -CH=N-O-CH₂-CH=CH-CH₃, -CH=N-O-CH₂-CH₂-Cl, -CH=N-O-CH₂-CH₂-F, -CH=N-O-CH₂-CF₃, -CH=N-O-CH₂-CH=CHCl, -CH=N-O-CH₂-CCl=CH₂, -CH=N-O-CH₂-CBr=CH₂, -CH=N-O-CH₂-CH=CCl-CH₃, -CH=N-OC(O)CH₃, -CH=N-OC(O)C₂H₅, -CH=N-O-CH₂-CN, -CH=N-O-CH₂-CH=CH-CH₂-O-CH₃, -CH=N-O-CH₂-CH=CH-CH₂-O-tert.-C₄H₉, -CH=N-O-(CH₂)₃-C₆H₅, -CH=N-O-(CH₂)₄-C₆H₅, -CH=N-O-(CH₂)₄-4-Cl-C₆H₄, -CH=N-O-(CH₂)₄-4-OCH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-CH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-C₆H₅, -CH=N-O-CH₂CH=CH-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CH-3-OCH₃-C₆H₄, -CH=N-O-(CH₂)₂CH=CH-4-F-C₆H₄, -CH=N-O-(CH₂)CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CHCH₂-4-OCH₃-C₆H₄, -CH=N-O-CH₂-CH=C(CH₃)-C₆H₅ -CH=N-O-(CH₂)₂CH=CH-3,4(Cl,Cl)-C₆H₃, -CH=N-O-(CH₂)₃C≡C-4-F-C₆H₄, -CH₂=N-OCHOCH₃, -CH=N-OC₂H₄OCH₃, -CH=N-OCH₂OC₂H₅, -CH=N-OCH(CH₃)OCH₃, -CH=N-OCH(CH₃)COOCH₃, -CH=N-OCH(CH₃)COO-n-C₄H₉, -CH=N-NH₂, -CH=N-NHCH₃, -CH=N-NHC₂H₅, -CH=N-NH-n-C₃H₇, -CH=N-NH-i-C₃H₇, -CH=N-NH-n-C₄H₉, -CH=N-NH-i-C₄H₉, -CH=N-NH-s-C₄H₉, -CH=N-NH-tert.-C₄H₉, -CH=N-NH-cyclopropyl, -CH=N-NH-cyclobutyl, -CH=N-NH-cyclopentyl, -CH=N-NH-cyclohexyl, -CH=N-NH-cycloheptyl, -CH=N-N(CH₃)₂, -CH=N-N(C₂H₅)₂, -CH=N-N(C₃H₇)₂, -CH=N-N(i-C₃H₇)(CH₃), -CH=N-NHCH₂-C=CH, -CH=N-NHCH₂-C≡CH, -CH=N-N(CH₃)-CH₂-C≡CH, -CH=N-NHCH₂CF₃, -CH=N-NH-CO-CH₃, -CH=N-NH-CO-CH₂H₅, -CH=N-NH-COOCH₃, -CH=N-NH-COOC₂H₅, -CH=N-NH-COO-tert.-C₄H₉, -CH=N-pyrrolidin-1-yl, -CH=N-piperidin-1-yl, -CH=N-morpholin-4-yl, -CH=N-NH-C₆H₅, -CH=N-NH-(4-Cl-C₆H₄), -CH=N-NH-(4-NO₂-C₆H₄), -CH=N-NH-(4-F-C₆H₄), -CH=N-NH-(4-CH₃O-C₆H₄), -CH=N-NH-(2,4-Cl₂-C₆H₃), -CH=N-NH-(2,4-(NO₂)₂-C₆H₃), -CH=N-NH-CO-NH₂, -CH=N-NH-CO-NHCH₃, -CH=N-NH-CO-NHC₂H₅, -CH=N-NH-CO-N(CH₃)₂, -CH=CH-COOH, -CH=CH-CO-OCH₃, -CH=C-CO-OC₂H₅, -CH=CH-CO-O-n-C₃H₇, -CH=CH-CO-O-i-C₃H₇, -CH=CH-CO-O-n-C₄H₉, -CH=CH-CO-O-tert.-C₄H₉, -CH=CH-CO-O-cyclopropyl, -CH=CH-CO-O-cyclobutyl, -CH=CH-CO-O-cyclopentyl, -CH=CH-CO-O-cyclohexyl, -CH=CH-CO-O-cycloheptyl, -CH=C(CH₃)-COOH, -CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CO-O-n-C₃H₇, -CH=C(CH₃)-CO-O-i-C₃H₇, -CH=C(CH₃)-CO-O-n-C₄H₉, -CH=C(CH₃)-CO-O-tert.-C₄H₉, -CH=C(CH₃)-CO-O-cyclopropyl, -CH=C(CH₃)-CO-O-cyclobutyl, -CH=C(CH₃)-CO-O-cyclopentyl, -CH=C(CH₃)-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cycloheptyl, -CH=C(C₂H₅)-COOH, -CH=C(C₂H₅)-CO-OCH₃, -CH=C(C₂H₅)-CO-OC₂H₅, -CH=C(C₂H₅)-CO-O-n-C₃H₇, -CH=C(C₂H₅)-CO-O-i-C₃H₇, -CH=C(C₂H₅)-CO-O-n-C₄H₉, -CH=C(C₂H₅)-CO-O-tert.-C₄H₉, -CH=C(C₂H₅)-CO-O-cyclopropyl, -CH=C(C₂H₅)-CO-O-cyclobutyl, -CH=C(C₂H₅)-CO-O-cyclopentyl, -CH=C(C₂H₅)-CO-O-cyclohexyl, -CH=C(C₂H₅)-CO-O-cycloheptyl, -CH=C(Cl)-COOH, -CH=C(Cl)-CO-OCH₃, -CH=C(Cl)-CO-OC₂H₅, -CH=C(Cl)-CO-O-n-C₃H₇, -CH=C(Cl)-CO-O-i-C₃H₇, -CH=C(Cl)-CO-O-n-C₄H₉, -CH=C(Cl)-CO-O-tert.-C₄H₉, -CH=C(Cl)-CO-O-cyclopropyl, -CH=C(Cl)-CO-O-cyclobutyl, -CH=C(Cl)-CO-O-cyclopentyl, -CH=C(Cl)-CO-O-cyclohexyl, -CH=C(Cl)-CO-O-cycloheptyl, -CH=C(Br)-COOH, -CH=C(Br)-CO-OCH₃, -CH=C(Br)-CO-OC₂H₅, -CH=C(Br)-CO-O-n-C₃H₇, -CH=C(Br)-CO-O-i-C₃H₇, -CH=C(Br)-CO-O-n-C₄H₉, -CH=C(Br)-CO-O-tert.-C₄H₉, -CH=C(Br)-CO-O-cyclopropyl, -CH=C(Br)-CO-O-cyclobutyl, -CH=C(Br)-CO-O-cyclopentyl, -CH=C(Br)-CO-O-cyclohexyl, -CH=C(Br)-CO-O-cycloheptyl, -CH=C(CN)-COOH, -CH=C(CN)-CO-OCH₃, -CH=C(CN)-CO-OC₂H₅, -CH=C(CN)-CO-O-n-C₃H₇, -CH=C(CN)-CO-O-i-C₃H₇, -CH=C(CN)-CO-O-n-C₄H₉, -CH=C(CN)-CO-O-tert.-C₄H₉, -CH=C(CN)-CO-O-cyclopropyl, -CH=C(CN)-CO-O-cyclobutyl, -CH=C(CN)-CO-O-cyclopentyl, -CH=C(CN)-CO-O-cyclohexyl, -CH=C(CN)-CO-O-cycloheptyl, -CH=CH-CO-OCH₂-OCH₃, -CH=CH-CO-OCH₂-OC₂H₅, -CH=CH-CO-OCH₂-O-n-C₃H₅, -CH=CH-CO-OCH₂-O-i-C₃H₅, -CH=CH-CO-OCH(CH₃)-OCH₃, -CH=CH-CO-OCH(CH₃)-OC₂H₅, -CH=CH-CO-O-CH₂CH₂-OCH₃, -CH=CH-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-OCH₃, -CH=C(CH₃)-CO-OCH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-O-n-C₃H₅, -CH=C(CH₃)-CO-OCH₂-O-i-C₃H₅, -CH=C(CH₃)-CO-OCH(CH₃)-OCH₃, -CH=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CH₃)-CO-O-CH₂CH₂-OCH₃, -CH=C(CH₃)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-OCH₃, -CH=C(C₂H₅)-CO-OCH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-O-n-C₃H₅, -CH=C(C₂H₅)-CO-OCH₂-O-i-C₃H₅, -CH=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-OCH₃, -CH=C(Cl)-CO-OCH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-O-n-C₃H₅, -CH=C(Cl)-CO-OCH₂-O-i-C₃H₅, -CH=C(Cl)-CO-OCH(CH₃)-OCH₃, -CH=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Cl)-CO-O-CH₂CH₂-OCH₃, -CH=C(Cl)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-OCH₃, -CH=C(Br)-CO-OCH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-O-n-C₃H₅, -CH=C(Br)-CO-OCH₂-O-i-C₃H₅, -CH=C(Br)-CO-OCH(CH₃)-OCH₃, -CH=C(Br)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Br)-CO-O-CH₂CH₂-OCH₃, -CH=C(Br)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-OCH₃, -CH=C(CN)-CO-OCH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-O-n-C₃H₅, -CH=C(CN)-CO-OCH₂-O-i-C₃H₅, -CH=C(CN)-CO-OCH(CH₃)-OCH₃, -CH=C(CN)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CN)-CO-O-CH₂CH₂-OCH₃, -CH=C(CN)-CO-O-CH₂CH₂-OC₂H₅, -CH=CH-CO-OCH₂-CF₃, -CH=CH-CO-OCH₂-CCl₃, -CH=CH-CO-OCH₂-oxiranyl, -CH=CH-CO-O(CH₂)₃-Br, -CH=CH-CO-OCH₂-CH=CH₂, -CH=CH-CO-OCH₂-C≡CH, -CH=CH-CO-OCH₂-CN, -CH=CH-CO-O(CH₂)₂-CN, -CH=C(CH₃)-CO-OCH₂-CF₃, -CH=C(CH₃)-CO-OCH₂-CCl₃, -CH=C(CH₃)-CO-OCH₂-oxiranyl, -CH=C(CH₃)-CO-O(CH₂)₃-Br, -CH=C(CH₃)-CO-OCH₂-CH=CH₂, -CH=C(CH₃)-CO-OCH₂-C≡CH, -CH=C(CH₃)-CO-OCH₂-CN, -CH=C(CH₃)-CO-O(CH₂)₂-CN, -CH=C(C₂H₅)-CO-OCH₂-CF₃, -CH=C(C₂H₅)-CO-OCH₂-CCl₃, -CH=C(C₂H₅)-CO-OCH₂-oxiranyl, -CH=C(C₂H₅)-CO-O(CH₂)₃-Br, -CH=C(C₂H₅)-CO-OCH₂-CH=CH₂, -CH=C(C₂H₅)-CO-OCH₂-C≡CH, -CH=C(C₂H₅)-CO-OCH₂-CN, -CH=C(C₂H₅)-CO-O(CH₂)₂-CN, -CH=C(Cl)-CO-OCH₂-CF₃, -CH=C(Cl)-CO-OCH₂-CCl₃, -CH=C(Cl)-CO-OCH₂-oxiranyl, -CH=C(Cl)-CO-O(CH₂)₃-Br, -CH=C(Cl)-CO-OCH₂-CH=CH₂, -CH=C(Cl)-CO-OCH₂-C≡CH, -CH=C(Cl)-CO-OCH₂-CN, -CH=C(Cl)-CO-O(CH₂)₂-CN, -CH=C(Br)-CO-OCH₂-CF₃, -CH=C(Br)-CO-OCH₂-CCl₃, -CH=C(Br)-CO-OCH₂-oxiranyl, -CH=C(Br)-CO-O(CH₂)₃-Br, -CH=C(Br)-CO-OCH₂-CH=CH₂, -CH=C(Br)-CO-OCH₂-C≡CH, -CH=C(Br)-CO-OCH₂-CN, -CH=C(Br)-CO-O(CH₂)₂-CN, -CH=C(CN)-CO-OCH₂-CF₃, -CH=C(CN)-CO-OCH₂-CCl₃, -CH=C(CN)-CO-OCH₂-oxiranyl -CH=C(CN)-CO-O(CH₂)₃-Br, -CH=C(CN)-CO-OCH₂-CH=CH₂, -CH=C(CN)-CO-OCH₂-C≡CH, -CH=C(CN)-CO-OCH₂-CN, -CH=C(CN)-CO-O(CH₂)₂-CN, -CH=CH-CO-CH₃, -CH=CH-CO-C₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-i-C₃H₇, -CH=CH-CO-n-C₄H₉, -CH=CH-CO-tert.-C₄H₉, -CH=CH-CO-CH₂Cl, -CH=CH-CO-CH₂Br, -CH=CH-CO-CHCl₂, -CH=CH-CO-CH₂-OCH₃, -CH=CH-CO-CH(OCH₃)₂, -CH=CH-CO-CH₂-SCH₃, -CH=C(CH₃)-CO-CH₃, -CH=C(CH₃)-CO-C₂H₅, -CH=C(CH₃)-CO-n-C₃H₇, -CH=C(CH₃)-CO-i-C₃H₇, -CH=C(CH₃)-CO-n-C₄H₉, -CH=C(CH₃)-CO-tert.-C₄H₉, -CH=C(CH₃)-CO-CH₂Cl, -CH=C(CH₃)-CO-CH₂Br, -CH=C(CH₃)-CO-CHCl₂, -CH=C(CH₃)-CO-CH₂-OCH₃, -CH=C(CH₃)-CO-CH(OCH₃)₂, -CH=C(CH₃)-CO-CH₂-SCH₃, -CH=C(C₂H₅)-CO-CH₃, -CH=C(C₂H₅)-CO-C₂H₅, -CH=C(C₂H₅)-CO-n-C₃H₇, -CH=C(C₂H₅)-CO-i-C₃H₇, -CH=C(C₂H₅)-CO-n-C₄H₉, -CH=C(C₂H₅)-CO-tert.-C₄H₉, -CH=C(C₂H₅)-CO-CH₂Cl, -CH=C(C₂H₅)-CO-CH₂Br, -CH=C(C₂H₅)-CO-CHCl₂, -CH=C(C₂H₅)-CO-CH₂-OCH₃, -CH=C(C₂H₅)-CO-CH(OCH₃)₂, -CH=C(C₂H₅)-CO-CH₂-SCH₃, -CH=C(Cl)-CO-CH₃, -CH=C(Cl)-CO-C₂H₅, -CH=C(Cl)-CO-n-C₃H₇, -CH=C(Cl)-CO-i-C₃H₇, -CH=C(Cl)-CO-n-C₄H₉, -CH=C(Cl)-CO-tert.-C₄H₉, -CH=C(Cl)-CO-CH₂Cl, -CH=C(Cl)-CO-CH₂Br, -CH=C(Cl)-CO-CHCl₂, -CH=C(Cl)-CO-CH₂-OCH₃, -CH=C(Cl)-CO-CH(OCH₃)₂, -CH=C(Cl)-CO-CH₂-SCH₃, -CH=C(Br)-CO-CH₃, -CH=C(Br)-CO-C₂H₅, -CH=C(Br)-CO-n-C₃H₇, -CH=C(Br)-CO-i-C₃H₇, -CH=C(Br)-CO-n-C₄H₉, -CH=C(Br)-CO-tert.-C₄H₉, -CH=C(Br)-CO-CH₂Cl, -CH=C(Br)-CO-CH₂Br, -CH=C(Br)-CO-CHCl₂, -CH=C(Br)-CO-CH₂-OCH₃, -CH=C(Br)-CO-CH(OCH₃)₂, -CH=C(Br)-CO-CH₂-SCH₃, -CH=C(CN)-CO-CH₃, -CH=C(CN)-CO-C₂H₅, -CH=C(CN)-CO-n-C₃H₇, -CH=C(CN)-CO-i-C₃H₇, -CH=C(CN)-CO-n-C₄H₉, -CH=C(CN)-CO-tert.-C₄H₉, -CH=C(CN)-CO-CH₂Cl, -CH=C(CN)-CO-CH₂Br, -CH=C(CN)-CO-CHCl₂, -CH=C(CN)-CO-CH₂-OCH₃, -CH=C(CN)-CO-CH(OCH₃)₂, -CH=C(CN)-CO-CH₂-SCH₃, -CH=CH-CO-C₆H₅, -CH=CH-CO-(4-Cl-C₆H₄), -CH=C(CH₃)-CO-C₆H₅, -CH=C(CH₃)-CO-(4-Cl-C₆H₄), -CH=C(C₂H₅)-CO-C₆H₅, -CH=C(C₂H₅)-CO-(4-Cl-C₆H₄), -CH=C(Cl)-CO-C₆H₅, -CH=C(Br)-CO-C₆H₅, -CH=C(CN)-CO-C₆H₅, -CH=CH-CO-NH₂, -CH=CH-CO-NHCH₃, -CH=CH-CO-N(CH₃)₂, -CH=CH-CO-NH-C₂H₅, -CH=CH-CO-N(C₂H₅)₂, -CH=CH-CO-NH-n-C₃H₇, -CH=CH-CO-NH-i-C₃H₇, -CH=CH-CO-NH-tert.-C₄H₉, -CH=CH-CO-NH-cyclopropyl, -CH=CH-CO-NH-cyclobutyl, -CH=CH-CO-NH-cyclopentyl, -CH=CH-CO-NH-cyclohexyl, -CH=CH-CO-cycloheptyl, -CH=CH-CO-NH-cyclooctyl, -CH=CH-CO-pyrrolidin-1-yl, -CH=CH-CO-piperidin-1-yl, -CH=CH-CO-morpholin-4-yl, -CH=CH-CO-NH-CH₂CH=CH₂, -CH=CH-CO-NH-CH₂C≡CH, -CH=CH-CO-N(CH₃)-CH₂C≡CH, -CH=CH-CO-NH-(CH₂)₂Cl, -CH=CH-CO-NH-C₆H₅, -CH=C(CH₃)-CO-NH₂, -CH=C(CH₃)-CO-NHCH₃, -CH=C(CH₃)-CO-N(CH₃)₂, -CH=C(CH₃)-CO-NH-C₂H₅, -CH=C(CH₃)-CO-N(C₂H₅)₂, -CH=C(CH₃)-CO-NH-n-C₃H₇, -CH=C(CH₃)-CO-NH-i-C₃H₇, -CH=C(CH₃)-CO-NH-tert.-C₄H₉, -CH=C(CH₃)-CO-NH-cyclopropyl, -CH=C(CH₃)-CO-NH-cyclobutyl, -CH=C(CH₃)-CO-NH-cyclopentyl, -CH=C(CH₃)-CO-NH-cyclohexyl, -CH=C(CH₃)-CO-NH-cycloheptyl, -CH=C(CH₃)-CO-NH-cyclooctyl, -CH=C(CH₃)-CO-pyrrolidin-1-yl, -CH=C(CH₃)-CO-piperidin-1-yl, -CH=C(CH₃)-CO-morpholin-4-yl, -CH=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -CH=C(CH₃)-CO-NH-CH₂C≡CH, -CH=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CH₃)-CO-NH-(CH₂)₂Cl, -CH=C(CH₃)-CO-NH-C₆H₅, -CH=C(C₂H₅)-CO-NH₂, -CH=C(C₂H₅)-CO-NHCH₃, -CH=C(C₂H₅)-CO-N(CH₃)₂, -CH=C(C₂H₅)-CO-NH-C₂H₅, -CH=C(C₂H₅)-CO-N(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-n-C₃H₇, -CH=C(C₂H₅)-CO-NH-i-C₃H₇, -CH=C(C₂H₅)-CO-NH-tert.-C₄H₉, -CH=C(C₂H₅)-CO-NH-cyclopropyl, -CH=C(C₂H₅)-CO-NH-cyclobutyl, -CH=C(C₂H₅)-CO-NH-cyclopentyl, -CH=C(C₂H₅)-CO-NH-cyclohexyl, -CH=C(C₂H₅)-CO-NH-cycloheptyl, -CH=C(C₂H₅)-CO-NH-cyclooctyl, -CH=C(C₂H₅)-CO-pyrrolidin-1-yl, -CH=C(C₂H₅)-CO-piperidin-1-yl, -CH=C(C₂H₅)-CO-morpholin-4-yl, -CH=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-CH₂C≡CH, -CH=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -CH=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -CH=C(C₂H₅)-CO-NH-C₆H₅, -CH=C(Cl)-CO-NH₂, -CH=C(Cl)-CO-NHCH₃, -CH=C(Cl)-CO-N(CH₃)₂, -CH=C(Cl)-CO-NH-C₂H₅, -CH=C(Cl)-CO-N(C₂H₅)₂, -CH=C(Cl)-CO-NH-n-C₃H₇, -CH=C(Cl)-CO-NH-i-C₃H₇, -CH=C(Cl)-CO-NH-tert.-C₄H₉, -CH=C(Cl)-CO-NH-cyclopropyl, -CH=C(Cl)-CO-NH-cyclobutyl, -CH=C(Cl)-CO-NH-cyclopentyl, -CH=C(Cl)-CO-NH-cyclohexyl, -CH=C(Cl)-CO-NH-cycloheptyl, -CH=C(Cl)-CO-NH-cyclooctyl, -CH=C(Cl)-CO-pyrrolidin-1-yl, -CH=C(Cl)-CO-piperidin-1-yl, -CH=C(Cl)-CO-morpholin-4-yl, -CH=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -CH=C(Cl)-CO-NH-CH₂C≡CH, -CH=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Cl)-CO-NH-(CH₂)₂Cl, -CH=C(Cl)-CO-NH-C₆H₅, -CH=C(Br)-CO-NH₂, -CH=C(Br)-CO-NHCH₃, -CH=C(Br)-CO-N(CH₃)₂, -CH=C(Br)-CO-NH-C₂H₅, -CH=C(Br)-CO-N(C₂H₅)₂, -CH=C(Br)-CO-NH-n-C₃H₇, -CH=C(Br)-CO-NH-i-C₃H₇, -CH=C(Br)-CO-NH-tert.-C₄H₉, -CH=C(Br)-CO-NH-cyclopropyl, -CH=C(Br)-CO-NH-cyclobutyl, -CH=C(Br)-CO-NH-cyclopentyl, -CH=C(Br)-CO-NH-cyclohexyl, -CH=C(Br)-CO-NH-cycloheptyl, -CH=C(Br)-CO-NH-cyclooctyl, -CH=C(Br)-CO-pyrrolidin-1-yl, -CH=C(Br)-CO-piperidin-1-yl, -CH=C(Br)-CO-morpholin-4-yl, -CH=C(Br)-CO-NH-CH₂CH=C(Br)₂, -CH=C(Br)-CO-NH-CH₂C≡CH, -CH=C(Br)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Br)-CO-NH-(CH₂)₂Cl, -CH=C(Br)-CO-NH-C₆H₅, -CH=C(CN)-CO-NH₂, -CH=C(CN)-CO-NHCH₃, -CH=C(CN)-CO-N(CH₃)₂, -CH=C(CN)-CO-NH-C₂H₅, -CH=C(CN)-CO-N(C₂H₅)₂, -CH=C(CN)-CO-NH-n-C₃H₇, -CH=C(CN)-CO-NH-i-C₃H₇, -CH=C(CN)-CO-NH-tert.-C₄H₉, -CH=C(CN)-CO-NH-cyclopropyl, -CH=C(CN)-CO-NH-cyclobutyl, -CH=C(CN)-CO-NH-cyclopentyl, -CH=C(CN)-CO-NH-cyclohexyl, -CH=C(CN)-CO-NH-cycloheptyl, -CH=C(CN)-CO-NH-cyclooctyl, -CH=C(CN)-CO-pyrrolidin-1-yl, -CH=C(CN)-CO-piperidin-1-yl, -CH=C(CN)-CO-morpholin-4-yl, -CH=C(CN)-CO-NH-CH₂CH=C(CN)₂, -CH=C(CN)-CO-NH-CH₂C≡CH, -CH=C(CN)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CN)-CO-NH-(CH₂)₂Cl, -CH=C(CN)-CO-NH-C₆H₅, -CH=CH-CO-SCH₃, -CH=CH-CO-SC₂H₅, -CH=CH-CO-S-n-C₃H₇, -CH=CH-CO-S-i-C₃H₇, -CH=CH-CO-S-n-C₄H₉, -CH=CH-CO-S-tert.-C₄H₉, -CH=C(CH₃)-CO-SCH₃, -CH=C(CH₃)-CO-SC₂H₅, -CH=C(CH₃)-CO-S-n-C₃H₇, -CH=C(CH₃)-CO-S-i-C₃H₇, -CH=C(CH₃)-CO-S-n-C₄H₉, -CH=C(CH₃)-CO-S-tert.-C₄H₉, -CH=C(C₂H₅)-CO-SCH₃, -CH=C(C₂H₅)-CO-SC₂H₅, -CH=C(C₂H₅)-CO-S-n-C₃H₇, -CH=C(C₂H₅)-CO-S-i-C₃H₇, -CH=C(C₂H₅)-CO-S-n-C₄H₉, -CH=C(C₂H₅)-CO-S-tert.-C₄H₉, -CH=C(Cl)-CO-SCH₃, -CH=C(Cl)-CO-SC₂H₅, -CH=C(Cl)-CO-S-n-C₃H₇, -CH=C(Cl)-CO-S-i-C₃H₇, -CH=C(Cl)-CO-S-n-C₄H₉, -CH=C(Cl)-CO-S-tert.-C₄H₉, -CH=C(Br)-CO-SCH₃, -CH=C(Br)-CO-SC₂H₅, -CH=C(Br)-CO-S-n-C₃H₇, -CH=C(Br)-CO-S-i-C₃H₇, -CH=C(Br)-CO-S-n-C₄H₉, -CH=C(Br)-CO-S-tert.-C₄H₉, -CH=C(CN)-CO-SCH₃, -CH=C(CN)-CO-SC₂H₅, -CH=C(CN)-CO-S-n-C₃H₇, -CH=C(CN)-CO-S-i-C₃H₇, -CH=C(CN)-CO-S-n-C₄H₉, -CH=C(CN)-CO-S-tert.-C₄H₉, -CH=C(COCH₃)-CO-OCH₃, -CH=C(COC₂H₅)-CO-OCH₃, -CH=C(CO-n-C₃H₇)-CO-OCH₃, -CH=C(COCH₃)-CO-OC₂H₅, -CH=C(COC₂H₅)-CO-OC₂H₅, -CH=C(CO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COCH₃)-CO-O-n-C₃H₇, -CH=C(COC₂H₅)-CO-O-n-C₃H₇, -CH=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-OCH₃, -CH=C(CF₃)-CO-OC₂H₅, -CH=C(CF₃)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-O-i-C₃H₇, -CH=C(CF₃)-CO-O-n-C₄H₉, -CH=C(CF₃)-CO-O-tert.-C₄H₉, -CH=C(COOCH₃)₂, -CH=C(COOC₂H₅)₂, -CH=C(COOCH₃)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)-CO-OCH₃, -CH=C(COO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)₂, -CH=CH-CH=CH-COOH, -CH=CH-CH=CH-CO-OCH₃, -CH=CH-CH=CH-CO-OC₂H₅, -CH=CH-CH=C(COOCH₃)₂, -CH=CH-CH=C(CN)-CO-OCH₃, -CH=CH-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-OCH₃, -CH=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CH=C(Cl)-CO-OCH₃, -CH=C(CH₃)-CH=C(Br)-CO-OCH₃, -CH=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-NH₂, -CH=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -CH=CH-(CH₂)₂-COOH, -CH=CH-(CH₂)₂-CO-OCH₃, -CH=CH-(CH₂)₂-CO-OC₂H₅, -CH=CH-CH₂-CH(COOCH₃)₂, -CH=CH-CH₂-CH(COOC₂H₅)₂, -CH=CH-CH₂-CH(CN)-CO-OCH₃, -CH=CH-CH₂-CH(CN)-CO-OC₂H₅, -CH=CH-CH₂-CH(CH₃)-CO-OCH₃, -CH=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -CH=CH-(CH₂)₂-CO-NH₂, -CH=CH-(CH₂)₂-CO-NH-CH₃, -CH=CH-CH₂-COOH, -CH=CH-CH₂-CO-OCH₃, -CH=CH-CH₂-CO-OC₂H₅, -CH=C(COOCH₃)-CH₂-CO-OCH₃, -CH=C(COOCH₃)-CH₂-CO-OC₂H₅, -CH=CH-CH₂-CO-NH₂, -CH=CH-CH₂-CO-NH-CH₃, -CH=CH-CH₂-CO-N(CH₃)₂, -CH(OCH₃)₂, -CH(SCH₃)₂, -CH(OC₂H₅)₂, -CH(SC₂H₅)₂, -CH(O-n-C₃H₇)₂, -CH(O-i-C₃H₇)₂, -CH(S-n-C₃H₇)₂, -CH(S-i-C₃H₇)₂, -CH(O-n-C₄H₉)₂, -CH(O-i-C₄H₉)₂, -CH(O-s-C₄H₉)₂, -CH(O-tert.-C₄H₉)₂, -CH(S-n-C₄H₉)₂, -CH(S-i-C₄H₉)₂, -CH(S-s-C₄H₉)₂, -CH(S-tert.-C₄H₉)₂, -CH(OC₅H₁₁)₂, 1,3-Dioxolan-2-yl, 1,3-Dithio­ lan-2-yl, 1,3-Oxathiolan-2-yl, 4-Methyl-1,3-dioxalan-2-yl, 4-Methyl-1,3-dithiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 5-Methyl-1,3-oxathiolan-2-yl, 4-Ethyl-1,3-dioxolan-2-yl, 4-Ethyl- 1,4-dithiolan-2-yl, 4-Ethyl-1,3-oxathiolan-2-yl, 5-Ethyl-1,3-oxa­ thiolan-2-yl, 4,5-Dimethyl-1,3-dioxolan-2-yl, 4,4-Dimethyl-1,3- dioxolan-2-yl, 4,5-Dimethyl-1,3-dithiolan-2-yl, 5,5-Dimethyl-1,3- dithiolan-2-yl, 4,5-Dimethyl-1,3-oxathiolan-2-yl, 5,5-Dimethyl- 1,3-oxathiolan-2-yl, 4,4-Dimethyl-1,3-oxathiolan-2-yl, 4-Vinyl- 1,3-dioxolan-2-yl, 4-Vinyl-1,3-dithiolan-2-yl, 4-Vinyl-1,3-oxa­ thiolan-2-yl, 5-Vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3- dioxolan-2-yl, 4-Chlormethyl-1,3-dithiolan-2-yl, 4-Chlormethyl- 1,3-oxathiolan-2-yl, 5-Chlormethyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-1,3-dithio­ lan-2-yl, 4-Hydroxymethyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl- 1,3-oxathiolan-2-yl, 4-Methoxymethyl-1,3-dioxolan-2-yl, 4-Allyl­ oxymethyl-1,3-dioxolan-2-yl, 4-Propargyloxymethyl-1,3-dioxolan- 2-yl, 4-Acetoxymethyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-1,3-dithiolan-2-yl, 4-Propargyl- oxymethyl-1,3-dithiolan-2-yl, 4-Acetoxymethyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-1,3-oxa­ thiolan-2-yl, 4-Allyloxymethyl-1,3-oxathiolan-2-yl, 5-Allyloxy­ methyl-1,3-oxathiolan-2-yl, 4-Propargyloxymethyl-1,3-oxathiolan-2-yl, 5-Propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxymethyl- 1,3-oxathiolan-2-yl, 5-Acetoxymethyl-1,3-oxathiolan-2-yl, 4-Methylthiomethyl-1,3-dioxolan-2-yl, 4-Methylthiomethyl-1,3- dithiolan-2-yl, 4-Carboxy-1,3-dioxolan-2-yl, 4-Carboxy-1,3- dithiolan-2-yl, 4-Methoxycarbonyl-1,3-dioxolan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-1,3-dithiolan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-4-methyl- 1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-di­ thiolan-2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-1,3- dithiolan-2-yl, 1,3-Dioxan-2-yl, 1,3-Dithian-2-yl, 1,3-Oxathian- 2-yl, 5-Methyl-1,3-dioxan-2-yl, 5-Methyl-1,3-dithian-2-yl, 5-Methyl-1,3-oxathian-2-yl, 5,5-Dimethyl-1,3-dioxan-2-yl, 4,6-Dimethyl- 1,3-dioxan-2-yl, 4,4-Dimethyl-1,3-dioxan-2-yl, 5,5-Dimethyl- 1,3-dithian-2-yl, 4,6-Dimethyl-1,3-dithian-2-yl, 4,4-Dimethyl- 1,3-dithian-2-yl, 5,5-Dimethyl-1,3-oxathian-2-yl, 4,4-Dimethyl- 1,3-oxathian-2-yl, 6,6-Dimethyl-1,3-oxathian-2-yl, 4-Hydroxymethyl-1,3-dioxan-2-yl, 4-Methoxymethyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-1,3-dithian-2-yl, 4-Methoxymethyl-1,3-dithian-2-yl, 4-Allyloxymethyl-1,3-dithian-2-yl, 4-Acetoxymethyl- 1,3-dithian-2-yl, 4-Chlormethyl-1,3-dioxan-2-yl, 4-Chlormethyl- 1,3-dithian-2-yl, 1,3-Dioxepan-2-yl, 1,3-Dithiepan-2-yl, 1,3-Di­ oxep-5-en-2-yl, 4-Methoxycarbonyl-1,3-dioxan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-1,3-dithian- 2-yl, 4-n-Butoxycarbonyl-1,3-dithian-2-yl, 4-Methoxycarbonyl-4- methyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-Methoxy- carbonyl-4-methyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-4-methyl- 1,3-dithian-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithian-2-yl, -C(CH₃)(OCH₃)₂, -C(CH₃)(SCH₃)₂, -C(CH₃)(OC₂H₅)₂, -C(CH₃)(SC₂H₅)₂, -C(CH₃)(O-n-C₃H₇)₂, -C(CH₃)(O-i-C₃H₇)₂, -C(CH₃)(S-n-C₃H₇)₂, -C(CH₃)(S-i-C₃H₇)₂, -C(CH₃)(O-n-C₄H₉)₂, -C(CH₃)(O-i-C₄H₉)₂, -C(CH₃)(O-s-C₄H₉)₂, -C(CH₃)(O-tert.-C₄H₉)₂, -C(CH₃)(S-n-C₄H₉)₂, -C(CH₃)(S-i-C₄H₉)₂, -C(CH₃)(S-s-C₄H₉)₂, -C(CH₃)(S-tert.-C₄H₉)₂, -C(CH₃)(O-n-C₅H₁₁)′′, 2-Methyl-1,3-dioxolan-2-yl, 2-Methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-oxathiolan-2-yl, 2,4-Dimethyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-1,3- oxathiolan-2-yl, 2,5-Dimethyl-1,3-oxathiolan-2-yl, 4-Ethyl-2- methyl-1,3-dioxolan-2-yl, 4-Ethyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Ethyl-2-methyl-1,3- oxathiolan-2-yl, 2,4,5-Trimethyl-1,3-dioxolan-2-yl, 2,4,4-Trimethyl- 1,3-dioxolan-2-yl, 2,4,5-Trimethyl-1,3-dithiolan-2-yl, 2,4,4-Trimethyl-1,3-dithiolan-2-yl, 2,4,5-Trimethyl-1,3-oxathiolan-2-yl, 2,4,4-Trimethyl-1,3-oxathiolan-2-yl, 2-Methyl-4-vinyl- 1,3-dioxolan-2-yl, 2-Methyl-4-vinyl-1,3-dithiolan-2-yl, 2-Methyl- 4-vinyl-1,3-oxathiolan-2-yl, 2-Methyl-5-vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-dioxolan-2-yl, 4-Chlormethyl-2- methyl-1,3-dithiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl- 2-methyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-2- methyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dioxolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxy- 2-methyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dithiolan-2-yl, 4-Acetoxy-2- methyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl- 2-methyl-1,3-oxathiolan-2-yl, 5-Allyloxymethyl-2- methyl-1,3-oxathiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3- oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxy-2-methyl-1,3-oxathiolan-2-yl, 5-Acetoxy-2-methyl- 1,3-oxathiolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dioxolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-2- methyl-1,3-dioxolan-2-yl, 4-Carboxy-2-methyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-2- methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl- 2-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-2- methyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-ethoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4- ethoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-n-butoxy- carbony-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl-1,3- dithiolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-dioxan-2-yl, 2-Methyl-1,3-dithian-2-yl, 2-Methyl-1,3-oxathian-2-yl, 2,5- Dimethyl-1,3-dioxan-2-yl, 2,5-Dimethyl-1,3-dithian-2-yl, 2,5-Dimethyl- 1,3-oxathian-2-yl, 2,5,5-Trimethyl-1,3-dioxan-2-yl, 2,4,6- Trimethyl-1,3-dioxan-2-yl, 2,2,4-Trimethyl-1,3-dioxan-2-yl, 2,5,5-Trimethyl-1,3-dithian-2-yl, 2,4,6-Trimethyl-1,3-dithian-2-yl, 2,4,4-Trimethyl-1,3-dithian-2-yl, 2,5,5-Trimethyl-1,3-oxathian-2-yl, 2,4,4-Trimethyl-1,3-oxathian-2-yl, 2,6,6-Trimethyl- 1,3-oxathian-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-2- methyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dithian-2-yl, 4-Methoxymethyl-2- methyl-1,3-dithian-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithian-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dithian-2-yl, 4-Chlormethyl-2- methyl-1,3-dioxan-2-yl, 4-Chlormethyl-2-methyl-1,3-dithian-2-yl, -C(CH₃)=NH, -C(CH₃)=N-CH₃, -C(CH₃)=N-C₂H₅, -C(CH₃)=N-n-C₃H₇, -C(CH₃)=N-i-C₃H₇, -C(CH₃)=N-n-C₄H₉, -C(CH₃)=N-CH₂CH=CH₂, -C(CH₃)=N-CH₂CH=CH₂-CH₃, -C(CH₃)=N-CH₂C≡CH, -C(CH₃)=N-CH₂C≡C-CH₃, -C(CH₃)=N-cyclopropyl, -C(CH₃)=N-cyclobutyl, -C(CH₃)=N-cyclopentyl, -C(CH₃)=N-cyclohexyl, -C(CH₃)=N-cycloheptyl, -C(CH₃)=N-CH₂-CH₂Cl, -C(CH₃)=N-CH₂Cl, -C(CH₃)=N-C₆H₅, -C(CH₃)=N-(2-F-C₆H₄), -C(CH₃)=N-(3-F-C₆H₄), -C(CH₃)=N-(4-F-C₆H₄), -C(CH₃)=N-(2-Cl-C₆H₄), -C(CH₃)=N-(3-Cl-C₆H₄), -C(CH₃)=N-(4-Cl-C₆H₄), -C(CH₃)=N-(2-CH₃-C₆H₄), -C(CH₃)=N-(3-CH₃-C₆H₄), -C(CH₃)=N-(4-CH₃-C₆H₄), -C(CH₃)=N-(2-CF₃-C₆H₄), -C(CH₃)=N-(3-CF₃-C₆H₄), -C(CH₃)=N-(4-CF₃-C₆H₄), -C(CH₃)=N-(2-OCH₃-C₆H₄), -C(CH₃)=N-(3-OCH₃-C₆H₄), -C(CH₃)=N-(4-OCH₃-C₆H₄), -C(CH₃)=N-(4-NO₂-C₆H₄), -C(CH₃)=N-(4-CN-C₆H₄), -C(CH₃)=N-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-(2,4-(CH₃)₂-C₆H₃), -C(CH₃)=N-CH₂-OCH₃, -C(CH₃)=N-CH₂-OC₂H₅, -C(CH₃)=N-CH₂CH₂-OCH₃, -C(CH₃)=N-CH₂CH-OC₂H₅, -C(CH₃)=N-OH, -C(CH₃)=N-OCH₃, äC(CH₃)=N-OC₂H₅, -C(CH₃)=N-O-n-C₃H₇, -C(CH₃)=N-O-i-C₃H₇, -C(CH₃)=N-O-n-C₄H₉, -C(CH₃)=N-O-i-C₄H₉, -C(CH₃)=N-O-s-C₄H₉, -C(CH₃)=N-O-tert.-C₄H₉, -C(CH₃)=N-OCH₂-CH=CH₂, -C(CH₃)=N-OCH(CH₃)-CH=CH₂, -C(CH₃)=N-OCH₂-C≡CH, -C(CH₃)=N-CH(CH₃)-C≡CH, -C(CH₃)=N-OCH₂-CH=C-CH₃, -C(CH₃)=N-OCH₂CH₂-Cl, -C(CH₃)=N-OCH₂CH₂-F, -C(CH₃)=N-OCH₂-CF₃, -C(CH₃)=N-OCH₂-CH=CHCl, -C(CH₃)=N-OCH₂-C(Cl)=CH₂, -C(CH₃)=N-OCH₂-C(Br)=CH₂, -C(CH₃)=N-OCH₂-CH=C(Cl)-CH₃, -C(CH₃)=N-O-CO-CH₃, -C(CH₃)=N-O-CO-C₂H₅, -C(CH₃)=N-OCH₂-CN, -C(CH₃)=N-OCH₂-CH=CH-CH₂-OCH₃, -C(CH₃)=N-OCH₂-CH=CH-CH₂-O-tert.-C₄H₉, -C(CH₃)=N-O-(CH₂)₃-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-(4-Cl-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-C₆H₅, -C(CH₃)=N-OCH₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(3-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-CH₂-(4-CH₃O-C₆H₄), -C(CH₃)=N-OCH₂-CH=C(CH₃)-C₆H₅, -C(CH₃)=N-O-(CH₂)₂-CH=CH-(3,4-Cl₂-C₆H₃), -C(CH₃)=N-O-(CH₂)₃-C≡-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-OCH₃, -C(CH₃)=N-OCH₂CH₂-OCH₃, -C(CH₃)=N-OCH₂-OC₂H₅, -C(CH₃)=N-OCH(CH₃)-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=N-NH₂, -C(CH₃)=N-NH-CH₃, -C(CH₃)=N-NH-C₂H₅, -C(CH₃)=N-NH-n-C₃H₇, -C(CH₃)=N-NH-i-C₃H₇, -C(CH₃)=N-NH-n-C₄H₉, -C(CH₃)=N-NH-i-C₄H₉, -C(CH₃)=N-NH-s-C₄H₉, -C(CH₃)=N-NH-tert.-C₄H₉, -C(CH₃)=N-NH-cyclopropyl, -C(CH₃)=N-NH-cyclobutyl, -C(CH₃)=N-NH-cyclopentyl, -C(CH₃)=N-NH-cyclohexyl, -C(CH₃)=N-NH-cycloheptyl, -C(CH₃)=N-N(CH₃)₂, -C(CH₃)=N-N(C₂H₅)₂, -C(CH₃)=N-N(n-C₃H₇)₂, -C(CH₃)=N-N(i-C₃H₇)₂, -C(CH₃)=N-NH-CH₂-C=CH, -C(CH₃)=N-NH-CH₂-C≡CH, -C(CH₃)=N-N(CH₃)-CH₂-C≡CH, -C(CH₃)=N-NH-CH₂CF₃, -C(CH₃)=N-NH-CO-CH₃, -C(CH₃)=N-NH-CO-C₂H₅, -C(CH₃)=N-NH-CO-OCH₃, -C(CH₃)=N-NH-CO-OC₂H₅, -C(CH₃)=N-NH-CO-O-tert.-C₄H₉, -C(CH₃)=N-pyrrolidin-1-yl, -C(CH₃)=N-piperidin-1-yl, -C(CH₃)=N-morpholin-4-yl, -C(CH₃)=N-NH-C₆H₅, -C(CH₃)=N-NH-(4-Cl-C₆H₄), -C(CH₃)=N-NH-(4-NO₂-C₆H₄), -C(CH₃)=N-NH-(4-F-C₆H₄), -C(CH₃)=N-NH-(4-CH₃O-C₆H₄), -C(CH₃)=N-NH-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-NH-(2,4-(NO₂)₂-C₆H₃), -C(CH₃)=N-NH-CO-NH₂, -C(CH₃)=N-NH-CO-NHCH₃, -C(CH₃)=N-NH-CO-NHC₂H₅, -C(CH₃)=N-NH-CO-N(CH₃)₂, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=CH-CO-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -(CH₃)=CH-CO-O-n-C₄H₉, -C(CH₃)=CH-CO-O-tert.-C₄H₉, -C(CH₃)=CH-CO-O-cyclopropyl, -C(CH₃)=CH-CO-O-cyclobutyl, -C(CH₃)=CH-CO-O-cyclopentyl, -C(CH₃)=CH-CO-O-cyclohexyl, -C(CH₃)=CH-CO-O-cycloheptyl, -C(CH₃)=C(CH₃)-COOH, -C(CH₃)=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-cyclopropyl, -C(CH₃)=C(CH₃)-CO-O-cyclobutyl, -C(CH₃)=C(CH₃)-CO-O-cyclopentyl, -C(CH₃)=C(CH₃)-CO-O-cyclohexyl, -C(CH₃)=C(CH₃)-CO-O-cycloheptyl, -C(CH₃)=C(C₂H₅)-COOH, -C(CH₃)=C(C₂H₅)-CO-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-cyclo­ propyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-O- cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-O-cycloheptyl, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-O-n-C₄H₉, -C(CH₃)=C(Cl)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-O-cyclopropyl, -C(CH₃)=C(Cl)-CO-O-cyclobutyl, -C(CH₃)=C(Cl)-CO-O-cyclopentyl, -C(CH₃)=C(Cl)-CO-O-cyclohexyl, -C(CH₃)=C(Cl)-CO-O-cycloheptyl, -C(CH₃)=C(Br)-COOH, -C(CH₃)=C(Br)-CO-OCH₃, -C(CH₃)=C(Br)-CO-OC₂H₅, -C(CH₃)=C(Br)-CO-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-O-n-C₄H₉, -C(CH₃)=C(Br)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-O-cyclopropyl, -C(CH₃)=C(Br)-CO-O-cyclobutyl, -C(CH₃)=C(Br)-CO-O-cyclopentyl, -C(CH₃)=C(Br)-CO-O-cyclohexyl, -C(CH₃)=C(Br)-CO-O-cycloheptyl, -C(CH₃)=C(CN)-COOH, -C(CH₃)=C(CN)-CO-OCH₃, -C(CH₃)=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CN)-CO-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-O-n-C₄H₉, -C(CH₃)=C(CN)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-O-cyclopropyl, -C(CH₃)=C(CN)-CO-O-cyclobutyl, -C(CH₃)=C(CN)-CO-O-cyclopentyl, -C(CH₃)=C(CN)-CO-O-cyclohexyl, -C(CH₃)=C(CN)-CO-O-cycloheptyl, -C(CH₃)=CH-CO-OCH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-OCH(CH₃)-OCH₃, -C(CH₃)=CH-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=CH-CO-OCH₂CH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-O-i-C₃H₇, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-O-i-C₃H₇, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-O-i-C₃H₇, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-CF₃, -C(CH₃)=CH-CO-OCH₂-CCl₃, -C(CH₃)=CH-CO-OCH₂-oxiranyl, -C(CH₃)=CH-CO-(CH₂)₃-Br,-C(CH₃)=CH-CO-OCH₂-CH=CH₂, -C(CH₃)=CH-CO-OCH₂-C≡CH, -C(CH₃)=CH-CO-OCH₂-CN, -C(CH₃)=CH-CO-OCH₂CH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CF₃, -C(CH₃)=C(CH₃)-CO-OCH₂-CCl₃, -C(CH₃)=C(CH₃)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CH₃)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CH₃)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CH₃)-CO-OCH₂-C≡CH, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CF₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CCl₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-oxiranyl, -C(CH₃)=C(C₂H₅)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(C₂H₅)CO-OCH₂-C≡CH, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-C₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂-CF₃, -C(CH₃)=C(Cl)-CO-OCH₂-CCl₃, -C(CH₃)=C(Cl)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Cl)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Cl)-CO-OCH₂-CH≡CH₂, -C(CH₃)=C(Cl)-CO-OCH₂-C≡CH, -C(CH₃)=C(Cl)-CO-OCH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂-CF₃, -C(CH₃)=C(Br)-CO-OCH₂-CCl₃, -C(CH₃)=C(Br)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Br)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Br)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Br)-CO-OCH₂-C≡CH, -C(CH₃)=C(Br)-CO-OCH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂CH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂-CF₃, -C(CH₃)=C(CN)-CO-OCH₂-CCl₃, -C(CH₃)=C(CN)-OCH₂-oxiranyl, -C(CH₃)=C(CN)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CN)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CN)-CO-OCH₂-C≡CH, -C(CH₃)=C(CN)-CO-OCH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂CH₂-CN, -C(CH₃)=CH-CO-CH₃, -C(CH₃)=CH-CO-C₂H₅, -C(CH₃)=CH-CO-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-n-C₄H₉, -C(CH₃)=CH-CO-tert.-C₄H₉, -C(CH₃)=CH-CO-CH₂Cl, -C(CH₃)=CH-CO-CH₂Br, -C(CH₃)=CH-CO-CHCl₂, -C(CH₃)=CH-CO-CH₂-OCH₃, -C(CH₃)=CH-CO-CH(OCH₃)₂, -C(CH₃)=CH-CO-CH₂-SCH₃, -C(CH₃)=C(CH₃)-CO-CH₃, -C(CH₃)=C(CH₃)-CO-C₂H₅, -C(CH₃)=C(CH₃)-CO-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-CH₂Cl, -C(CH₃)=C(CH₃)-CO-CH₂Br, -C(CH₃)=C(CH₃)-CO-CHCl₂, -C(CH₃)=C(CH₃)-CO-CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-CH(OCH₃)₂, -C(CH₃)=C(CH₃)-CO-CH₂-SCH₃, -C(CH₃)=C(C₂H₅)-CO-CH₃, -C(CH₃)=C(C₂H₅)-CO-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-CH₂Cl, -C(CH₃)=C(C₂H₅)-CO-CH₂Br, -C(CH₃)=C(C₂H₅)-CO-CHCl₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-CH(OCH₃)₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-SCH₃, -C(CH₃)=C(Cl)-CO-CH₃, -C(CH₃)=C(Cl)-CO-C₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-n-C₄H₉, -C(CH₃)=C(Cl)-CO-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-CH₂Cl, -C(CH₃)=C(Cl)-CO-CHCl₂, -C(CH₃)=C(Cl)-CO-CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-CH(OCH₃)₂, -C(CH₃)=C(Cl)-CO-CH₂-SCH₃, -C(CH₃)=C(Br)-CO-CH₃, -C(CH₃)=C(Br)-CO-C₂H₅, -C(CH₃)=C(Br)-CO-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-n-C₄H₉, -C(CH₃)=C(Br)-CO-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-CH₂Cl, -C(CH₃)=C(Br)-CO-CH₂Br, -C(CH₃)=C(Br)-CO-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-CH(OCH₃)₂, -C(CH₃)=C(Br)-CO-CH₂-SCH₃, -C(CH₃)=C(CN)-CO-CH₃, -C(CH₃)=C(CN)-CO-C₂H₅, -C(CH₃)=C(CN)-CO-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-n-C₄H₉, -C(CH₃)=C(CN)-CO-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-CH₂Cl, -C(CH₃)=C(CN)-CO-CH₂Br, -C(CH₃)=C(CN)-CO-CHCl₂, -C(CH₃)=C(CN)-CO-CH₂-OCH₃, -C(CH₃)=C(CN)-CO-CH(OCH₃)₂, -C(CH₃)=C(CN)-CO-CH₂-SCH₃, -C(CH₃)=CH-CO-C₆H₅, -C(CH₃)=CH-CO-(4-Cl-C₆H₄), -C(CH₃)=C(CH₃)-CO-C₆H₅, -C(CH₃)=C(CH₃)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(C₂H₅)-CO-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(Cl)-CO-C₆H₅, -C(CH₃)=C(Br)-CO-C₆H₅, -C(CH₃)=C(CN)-CO-C₆H₅, -C(CH₃)=CH-CO-NH₂, -C(CH₃)=CH-CO-NHCH₃, -C(CH₃)=CH-CO-N(CH₃)₂, -C(CH₃)=CH-CO-NH-C₂H₅, -C(CH₃)=CH-CO-N(C₂H₅)₂, -C(CH₃)=CH-CO-NH-n-C₃H₇, -C(CH₃)=CH-CO-NH-i-C₃H₇, -C(CH₃)=CH-CO-NH-tert.-C₄H₉, -C(CH₃)=CH-CO-NH-cyclopropyl, -C(CH₃)=CH-CO-NH-cyclobutyl, -C(CH₃)=CH-CO-NH-cyclopentyl, -C(CH₃)=CH-CO-NH-cyclohexyl, -C(CH₃)=CH-CO-NH-cycloheptyl, -C(CH₃)=CH-CO-NH-cyclooctyl, -C(CH₃)=CH-CO-pyrrolidin-1-yl, -C(CH₃)=CH-CO-piperidin-1-yl, -C(CH₃)=CH-CO-morpholin-4-yl, -C(CH₃)=CH-CO-NH-CH₂CH=CH₂, -C(CH₃)=CH-CO-NH-CH₂C≡CH, -C(CH₃)=CH-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=CH-CO-NH-(CH₂)₂Cl, -C(CH₃)=CH-CO-NH-C₆H₅, -C(CH₃)=C(CH₃)-CO-NH₂, -C(CH₃)=C(CH₃)-CO-NHCH₃, -C(CH₃)=C(CH₃)-CO-N(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-C₂H₅, -C(CH₃)=C(CH₃)-CO-N(C₂H₅)₂, -C(CH₃)=C(CH₃)-CO-NH-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-NH- cyclopropyl, -C(CH₃)=C(CH₃)-CO-NH-cyclobutyl, -C(CH₃)=C(CH₃)-CO-NH-cyclopentyl, -C(CH₃)=C(CH₃)-CO-NH- cyclehexyl, -C(CH₃)=C(CH₃)-CO-NH-cycloheptyl, -C(CH₃)=C(CH₃)-CO-NH-cyclooctyl, -C(CH₃)=C(CH₃)-CO- pyrrolidin-1-yl, -C(CH₃)=C(CH₃)-CO-piperidin-1-yl, -C(CH₃)=C(CH₃)-CO-morpholin-4-yl, -C(CH₃)=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-NH(CH₂)₂Cl, -C(CH₃)=C(CH₃)-CO-NH-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-NH₂, -C(CH₃)=C(C₂H₅)-CO-NHCH₃, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)₂, -C(CH₃)=C(C₂H₅)-CO-NH-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-N(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-NH- cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclo­ hexyl, -C(CH₃)=C(C₂H₅)-CO-NH-cycloheptyl, -C(CH₃)=C(C₂H₅)-CO-NH- cyclooctyl, -C(CH₃)=C(C₂H₅)-CO-pyrrolidin-1-yl, -C(CH₃)=C(C₂H₅)-CO-piperidin-1-yl, -C(CH₃)=C(C₂H₅)-CO- morpholin-4-yl, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(C₂H₅)-CO-NH-C₆H₅, -C(CH₃)=C(Cl)-CO-NH₂, -C(CH₃)=C(CH₃)=C(Cl)-CO-NHCH₃, -C(CH₃)=C(Cl)-CO-N(CH₃)₂, -C(CH₃)=C(Cl)-CO-NH-C₂H₅, -C(CH₃)=C(Cl)-CO-N(C₂H₅)₂, -C(CH₃)=C(Cl)-CO-NH-n-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-i-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-NH-cyclopropyl, -C(CH₃)=C(Cl)-CO-NH-cyclobutyl, -C(CH₃)=C(Cl)-CO-NH-cyclopentyl, -C(CH₃)=C(Cl)-CO-NH-cyclohexyl, -C(CH₃)=C(Cl)-CO-NH-cycloheptyl, -C(CH₃)=C(Cl)-CO-NH-cyclooctyl, -C(CH₃)=C(Cl)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Cl)-CO-piperidin-1- yl, -C(CH₃)=C(Cl)-CO-morpholin-4-yl, -C(CH₃)=C(Cl)-CO-NH-CH₂CH=C(Cl)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-N(CH₃)-CH₂≡CH, -C(CH₃)=C(Cl)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Cl)-NO-NH-C₆H₅, -C(CH₃)=C(Br)-CO-NH₂, -C(CH₃)=C(Br)-CO-NHCH₃, -C(CH₃)=C(Br)-CO-N(CH₃)₂, -C(CH₃)=C(Br)-CO-NH-C₂H₅, -C(CH₃)=C(Br)-CO-N(C₂H₅)₂, -C(CH₃)=C(Br)-CO-NH-n-C₃H₇, -C(CH₃)=C(Br)-CO-NH-i-C₃H₇, -C(CH₃)=C(Br)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-NH-cyclopropyl, -C(CH₃)=C(Br)-CO-NH-cyclobutyl, -C(CH₃)=C(Br)-CO-NH-cyclopentyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cycloheptyl, -C(CH₃)=C(Br)-CO-NH-cyclooctyl, -C(CH₃)=C(Br)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Br)-CO-piperidin-1-yl, -C(CH₃)=C(Br)-CO-morpholin-4-yl, -C(CH₃)=C(Br)-CO-NH-CH₂CH=C(CH₃)=C(Br)₂, C(Br)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Br)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Br)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Br)-CO-NH-C₆H₅, -C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CN)-CO-NHCH₃, -C(CH₃)=C(CN)-CO-N(CH₃)₂, -C(CH₃)=C(CN)-CO-NH-C₂H₅, -C(CH₃)=C(CN)-CO-N(C₂H₅)₂, -C(CH₃)=C(CN)-CO-NH-n-C₃H₇, -C(CH₃)=C(CN)-CO-NH-i-C₃H₇, -C(CH₃)=C(CN)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-NH-cyclopropyl, -C(CH₃)=C(CN)-CO-NH-cyclobutyl, -C(CH₃)=C(CN)-CO-NH-cyclopentyl, -C(CH₃)=C(CN)-CO-NH-cyclohexyl, -C(CH₃)=C(CN)-CO-NH-cycloheptyl, -C(CH₃)=C(CN)-CO-NH-cyclooctyl, -C(CH₃)=C(CN)-CO-pyrrolidin-1-yl, -C(CH₃)=C(CN)-CO-piperidin-1-yl, -C(CH₃)=C(CN)-CO-morpholin-4-yl, -C(CH₃)=C(CN)-CO-NH-CH₂CH=C(CN)₂, -C(CH₃)=C(CN)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CN)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CN)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CN)-CO-NH-C₆H₅, -C(CH₃)=CH-SO-SCH₃, -C(CH₃)=CH-CO-SC₂H₅, -C(CH₃)=CH-CO-S-n-C₃H₇, -C(CH₃)=CH-CO-S-i-C₃H₇, -C(CH₃)=CH-CO-S-n-C₄H₉, -C(CH₃)=CH-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-SCH₃, -C(CH₃)=C(CH₃)-CO-SC₂H₅, -C(CH₃)=C(CH₃)CO-S-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-S-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-SCH₃, -C(CH₃)=C(C₂H₅)-CO-SC₂H₅, -C(CH₃)=C(C₂H₅)-CO-S-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-SCH₃, -C(CH₃)=C(Cl)-CO-SC₂H₅, -C(CH₃)=C(Cl)-CO-S-n-C₃H₇, -C(CH₃)=C(Cl)-CO-S-i-C₃H₇, -C(CH₃)=C(Cl)-CO-S-n-C₄H₉, -C(CH₃)=C(Cl)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-SCH₃, -C(CH₃)=C(Br)-CO-SC₂H₅, -C(CH₃)=C(Br)-CO-S-n-C₃H₇, -C(CH₃)=C(Br)-CO-S-i-C₃H₇, -C(CH₃)=C(Br)-CO-S-n-C₄H₉, -C(CH₃)=C(Br)-CO-S-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-SCH₃, -C(CH₃)=C(CN)-CO-SC₂H₅, -C(CH₃)=C(CN)-CO-S-n-C₃H₇, -C(CH₃)=C(CN)-CO-S-i-C₃H₇, -C(CH₃)=C(CN)-CO-S-N-C₄H₉, -C(CH₃)=C(CN)-CO-S-tert.-C₄H₉, -C(CH₃)=C(COCH₃)-CO-OCH₃, -C(CH₃)=C(COC₂H₅)-CO-OCH₃, -C(CH₃)=C(CO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COCH₃)-CO-OC₂H₅, -C(CH₃)=C(COC₂H₅)-CO-OC₂H₅, -C(CH₃)=C(CO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COCH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(COC₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-OCH₃, -C(CH₃)=C(CF₃)-CO-OC₂H₅, -C(CH₃)=C(CF₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CF₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(COOCH₃)₂, -C(CH₃)=C(COOC₂H₅)₂, -C(CH₃)=C(COOCH₃)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)₂, -C(CH₃)=CH-CH=CH-COOH, -C(CH₃)=CH-CH=CH-CO-OCH₃, -C(CH₃)=CH-CH=CH-CO-OC₂H₅, -C(CH₃)=CH-CH=C(COOCH₃)₂, -C(CH₃)=CH-CH=C(CN)-CO-OCH₃, -C(CH₃)=CH-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CN)CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH₂, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -C(CH₃)=CH-(CH₂)₂-COOH, -C(CH₃)=CH-(CH₂)₂-CO-OCH₃, -C(CH₃)=CH-(CH₂)₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(COOCH₃)₂, -C(CH₃)=CH-CH₂-CH(COOC₂H₅)₂, -C(CH₃)=CH-CH₂-CH(CN)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CN)-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -C(CH₃)=CH-(CH₂)₂-CO-NH₂, -C(CH₃)=CH-(CH₂)₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-COOH, -C(CH₃)=CH-CH₂-CO-OCH₃, -C(CH₃)=CH-CH₂-CO-OC₂H₅, -C(CH₃)=C(COOCH₃)-CH₂-CO-OCH₃, -C(CH₃)=C(COOCH₃)-CH₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CO-NH₂, -C(CH₃)=CH-CH₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-CO-N(CH₃)₂.
wobei W für eine der folgenden Bedeutungen steht:
-CHO, -COCH₃, -COC₂H₅, -CO-n-C₃H₇, -CO-i-C₃H₇, -CO-n-C₄H₉, -CO-i-C₄H₉, -CO-s-C₄H₉, -CO-tert.-C₄H₉, -CO-CH₂CH=CH₂, -CO-CF₃, -COCCl₃, -COCH₂C≡CH, -CO-cyclopropyl, -CO-cyclobutyl, -CO-cyclopentyl, -CO-cyclohexyl, -CO-CN, -CO-COOCH₃, -CO-COOC₂H₅, -CH=NH, -CH=NCH₃, -CH=NC₂H₅, -CH=N-n-C₃H₅, -CH=N-i-C₃H₅, -CH=N-n-C₄H₉, -CH=NCH₂CH=CH₂, -CH=NCH₂CH=CH₂-CH₃, -CH=NCH₂C≡CH, -CH=NCH₂C≡C-CH₃, -CH=N-cyclopropyl, -CH=N-cyclobutyl, -CH=N-cyclopentyl, -CH=N-cyclohexyl, -CH=N-cycloheptyl, -CH=N-CH₂-CH₂Cl, -CH=N-CH₂Cl, -CH=N-C₆H₅, -CH=N-4-Br-C₆H₄, -CH=N-3-F-C₆H₄, -CH=N-4-F-C₆H₄, -CH=N-2-Cl-C₆H₄, -CH=N-3-Cl-C₆H₄, -CH=N-4-Cl-C₆H₄, -CH=N-2-Br-C₆H₄, -CH=N-2-F-C₆H₄, -CH=N-2-CH₃-C₆H₄, -CH=N-3-CH₃-C₆H₄, -CH=N-4-CH₃-C₆H₄, -CH=N-2-CF₃-C₆H₄, -CH=N-3-CF₃-C₆H₄, -CH=N-4-CF₃-C₆H₄, -CH=N-2-OCH₃-C₆H₄, -CH=N-3-OCH₃-C₆H₄, -CH=N-4-OCH₃-C₆H₄, -CH=N-4-NO₂-C₆H₄, -CH=N-4-CN-C₆H₄, -CH=N-2,4-(Cl,Cl)-C₆H₄, -CH=N-2,4-(CH₃,CH₃)-C₆H₄, -CH=N-CH₂OCH₃ -CH=N-CH₂OC₂H₅, -CH=N-CH₂CH₂OCH₃, -CH=N-CH₂CH₂OC₂H₅, -CH=N-OH, -CH=N-OCH₃, -CH=N-OC₂H₅, -CH=N-O-n-C₃H₇, -CH=N-O-i-C₃H₇, -CH=N-O-n-C₄H₉, -CH=N-O-i-C₄H₉, -CH=N-O-s-C₄H₉, -CH=N-O-tert.-C₄H₉, -CH=N-O-CH₂CH=CH₂, -CH=N-O-CH(CH₃)CH=CH₂, -CH=N-O-CH₂C≡CH, -CH=N-O-CH(CH₃)-C≡CH, -CH=N-O-CH₂-CH=CH-CH₃, -CH=N-O-CH₂-CH₂-Cl, -CH=N-O-CH₂-CH₂-F, -CH=N-O-CH₂-CF₃, -CH=N-O-CH₂-CH=CHCl, -CH=N-O-CH₂-CCl=CH₂, -CH=N-O-CH₂-CBr=CH₂, -CH=N-O-CH₂-CH=CCl-CH₃, -CH=N-OC(O)CH₃, -CH=N-OC(O)C₂H₅, -CH=N-O-CH₂-CN, -CH=N-O-CH₂-CH=CH-CH₂-O-CH₃, -CH=N-O-CH₂-CH=CH-CH₂-O-tert.-C₄H₉, -CH=N-O-(CH₂)₃-C₆H₅, -CH=N-O-(CH₂)₄-C₆H₅, -CH=N-O-(CH₂)₄-4-Cl-C₆H₄, -CH=N-O-(CH₂)₄-4-OCH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-CH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-C₆H₅, -CH=N-O-CH₂CH=CH-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CH-3-OCH₃-C₆H₄, -CH=N-O-(CH₂)₂CH=CH-4-F-C₆H₄, -CH=N-O-(CH₂)CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CHCH₂-4-OCH₃-C₆H₄, -CH=N-O-CH₂-CH=C(CH₃)-C₆H₅ -CH=N-O-(CH₂)₂CH=CH-3,4(Cl,Cl)-C₆H₃, -CH=N-O-(CH₂)₃C≡C-4-F-C₆H₄, -CH₂=N-OCHOCH₃, -CH=N-OC₂H₄OCH₃, -CH=N-OCH₂OC₂H₅, -CH=N-OCH(CH₃)OCH₃, -CH=N-OCH(CH₃)COOCH₃, -CH=N-OCH(CH₃)COO-n-C₄H₉, -CH=N-NH₂, -CH=N-NHCH₃, -CH=N-NHC₂H₅, -CH=N-NH-n-C₃H₇, -CH=N-NH-i-C₃H₇, -CH=N-NH-n-C₄H₉, -CH=N-NH-i-C₄H₉, -CH=N-NH-s-C₄H₉, -CH=N-NH-tert.-C₄H₉, -CH=N-NH-cyclopropyl, -CH=N-NH-cyclobutyl, -CH=N-NH-cyclopentyl, -CH=N-NH-cyclohexyl, -CH=N-NH-cycloheptyl, -CH=N-N(CH₃)₂, -CH=N-N(C₂H₅)₂, -CH=N-N(C₃H₇)₂, -CH=N-N(i-C₃H₇)(CH₃), -CH=N-NHCH₂-C=CH, -CH=N-NHCH₂-C≡CH, -CH=N-N(CH₃)-CH₂-C≡CH, -CH=N-NHCH₂CF₃, -CH=N-NH-CO-CH₃, -CH=N-NH-CO-CH₂H₅, -CH=N-NH-COOCH₃, -CH=N-NH-COOC₂H₅, -CH=N-NH-COO-tert.-C₄H₉, -CH=N-pyrrolidin-1-yl, -CH=N-piperidin-1-yl, -CH=N-morpholin-4-yl, -CH=N-NH-C₆H₅, -CH=N-NH-(4-Cl-C₆H₄), -CH=N-NH-(4-NO₂-C₆H₄), -CH=N-NH-(4-F-C₆H₄), -CH=N-NH-(4-CH₃O-C₆H₄), -CH=N-NH-(2,4-Cl₂-C₆H₃), -CH=N-NH-(2,4-(NO₂)₂-C₆H₃), -CH=N-NH-CO-NH₂, -CH=N-NH-CO-NHCH₃, -CH=N-NH-CO-NHC₂H₅, -CH=N-NH-CO-N(CH₃)₂, -CH=CH-COOH, -CH=CH-CO-OCH₃, -CH=CH-CO-OC₂H₅, -CH=CH-CO-O-n-C₃H₇, -CH=CH-CO-O-i-C₃H₇, -CH=CH-CO-O-n-C₄H₉, -CH=CH-CO-O-tert.-C₄H₉, -CH=CH-CO-O-cyclopropyl, -CH=CH-CO-O-cyclobutyl, -CH=CH-CO-O-cyclopentyl, -CH=CH-CO-O-cyclohexyl, -CH=CH-CO-O-cycloheptyl, -CH=C(CH₃)-COOH, -CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CO-O-n-C₃H₇, -CH=C(CH₃)-CO-O-i-C₃H₇, -CH=C(CH₃)-CO-O-n-C₄H₉, -CH=C(CH₃)-CO-O-tert.-C₄H₉, -CH=C(CH₃)-CO-O-cyclopropyl, -CH=C(CH₃)-CO-O-cyclobutyl, -CH=C(CH₃)-CO-O-cyclopentyl, -CH=C(CH₃)-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cycloheptyl, -CH=C(C₂H₅)-COOH, -CH=C(C₂H₅)-CO-OCH₃, -CH=C(C₂H₅)-CO-OC₂H₅, -CH=C(C₂H₅)-CO-O-n-C₃H₇, -CH=C(C₂H₅)-CO-O-i-C₃H₇, -CH=C(C₂H₅)-CO-O-n-C₄H₉, -CH=C(C₂H₅)-CO-O-tert.-C₄H₉, -CH=C(C₂H₅)-CO-O-cyclopropyl, -CH=C(C₂H₅)-CO-O-cyclobutyl, -CH=C(C₂H₅)-CO-O-cyclopentyl, -CH=C(C₂H₅)-CO-O-cyclohexyl, -CH=C(C₂H₅)-CO-O-cycloheptyl, -CH=C(Cl)-COOH, -CH=C(Cl)-CO-OCH₃, -CH=C(Cl)-CO-OC₂H₅, -CH=C(Cl)-CO-O-n-C₃H₇, -CH=C(Cl)-CO-O-i-C₃H₇, -CH=C(Cl)-CO-O-n-C₄H₉, -CH=C(Cl)-CO-O-tert.-C₄H₉, -CH=C(Cl)-CO-O-cyclopropyl, -CH=C(Cl)-CO-O-cyclobutyl, -CH=C(Cl)-CO-O-cyclopentyl, -CH=C(Cl)-CO-O-cyclohexyl, -CH=C(Cl)-CO-O-cycloheptyl, -CH=C(Br)-COOH, -CH=C(Br)-CO-OCH₃, -CH=C(Br)-CO-OC₂H₅, -CH=C(Br)-CO-O-n-C₃H₇, -CH=C(Br)-CO-O-i-C₃H₇, -CH=C(Br)-CO-O-n-C₄H₉, -CH=C(Br)-CO-O-tert.-C₄H₉, -CH=C(Br)-CO-O-cyclopropyl, -CH=C(Br)-CO-O-cyclobutyl, -CH=C(Br)-CO-O-cyclopentyl, -CH=C(Br)-CO-O-cyclohexyl, -CH=C(Br)-CO-O-cycloheptyl, -CH=C(CN)-COOH, -CH=C(CN)-CO-OCH₃, -CH=C(CN)-CO-OC₂H₅, -CH=C(CN)-CO-O-n-C₃H₇, -CH=C(CN)-CO-O-i-C₃H₇, -CH=C(CN)-CO-O-n-C₄H₉, -CH=C(CN)-CO-O-tert.-C₄H₉, -CH=C(CN)-CO-O-cyclopropyl, -CH=C(CN)-CO-O-cyclobutyl, -CH=C(CN)-CO-O-cyclopentyl, -CH=C(CN)-CO-O-cyclohexyl, -CH=C(CN)-CO-O-cycloheptyl, -CH=CH-CO-OCH₂-OCH₃, -CH=CH-CO-OCH₂-OC₂H₅, -CH=CH-CO-OCH₂-O-n-C₃H₅, -CH=CH-CO-OCH₂-O-i-C₃H₅, -CH=CH-CO-OCH(CH₃)-OCH₃, -CH=CH-CO-OCH(CH₃)-OC₂H₅, -CH=CH-CO-O-CH₂CH₂-OCH₃, -CH=CH-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-OCH₃, -CH=C(CH₃)-CO-OCH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-O-n-C₃H₅, -CH=C(CH₃)-CO-OCH₂-O-i-C₃H₅, -CH=C(CH₃)-CO-OCH(CH₃)-OCH₃, -CH=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CH₃)-CO-O-CH₂CH₂-OCH₃, -CH=C(CH₃)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-OCH₃, -CH=C(C₂H₅)-CO-OCH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-O-n-C₃H₅, -CH=C(C₂H₅)-CO-OCH₂-O-i-C₃H₅, -CH=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-OCH₃, -CH=C(Cl)-CO-OCH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-O-n-C₃H₅, -CH=C(Cl)-CO-OCH₂-O-i-C₃H₅, -CH=C(Cl)-CO-OCH(CH₃)-OCH₃, -CH=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Cl)-CO-O-CH₂CH₂-OCH₃, -CH=C(Cl)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Br)- ⁹⁹⁹⁹⁹ ⁰⁰⁰⁷⁰ ⁵⁵² ⁰⁰¹⁰⁰⁰²⁸⁰⁰⁰⁰⁰00200012000285919988800040 0002004131038 00004 99880 CO-OCH₂-OCH₃, -CH=C(Br)-CO-OCH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-O-n-C₃H₅, -CH=C(Br)-CO-OCH₂-O-i-C₃H₅, -CH=C(Br)-CO-OCH(CH₃)-OCH₃, -CH=C(Br)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Br)-CO-O-CH₂CH₂-OCH₃, -CH=C(Br)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-OCH₃, -CH=C(CN)-CO-OCH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-O-n-C₃H₅, -CH=C(CN)-CO-OCH₂-O-i-C₃H₅, -CH=C(CN)-CO-OCH(CH₃)-OCH₃, -CH=C(CN)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CN)-CO-O-CH₂CH₂-OCH₃, -CH=C(CN)-CO-O-CH₂CH₂-OC₂H₅, -CH=CH-CO-OCH₂-CF₃, -CH=CH-CO-OCH₂-CCl₃, -CH=CH-CO-OCH₂-oxiranyl, -CH=CH-CO-O(CH₂)₃-Br, -CH=CH-CO-OCH₂-CH=CH₂, -CH=CH-CO-OCH₂-C≡CH, -CH=CH-CO-OCH₂-CN, -CH=CH-CO-O(CH₂)₂-CN, -CH=C(CH₃)-CO-OCH₂-CF₃, -CH=C(CH₃)-CO-OCH₂-CCl₃, -CH=C(CH₃)-CO-OCH₂-oxiranyl, -CH=C(CH₃)-CO-O(CH₂)₃-Br, -CH=C(CH₃)-CO-OCH₂-CH=CH₂, -CH=C(CH₃)-CO-OCH₂-C≡CH, -CH=C(CH₃)-CO-OCH₂-CN, -CH=C(CH₃)-CO-O(CH₂)₂-CN, -CH=C(C₂H₅)-CO-OCH₂-CF₃, -CH=C(C₂H₅)-CO-OCH₂-CCl₃, -CH=C(C₂H₅)-CO-OCH₂-oxiranyl, -CH=C(C₂H₅)-CO-O(CH₂)₃-Br, -CH=C(C₂H₅)-CO-OCH₂-CH=CH₂, -CH=C(C₂H₅)-CO-OCH₂-C≡CH, -CH=C(C₂H₅)-CO-OCH₂-CN, -CH=C(C₂H₅)-CO-O(CH₂)₂-CN, -CH=C(Cl)-CO-OCH₂-CF₃, -CH=C(Cl)-CO-OCH₂-CCl₃, -CH=C(Cl)-CO-OCH₂-oxiranyl, -CH=C(Cl)-CO-O(CH₂)₃-Br, -CH=C(Cl)-CO-OCH₂-CH=CH₂, -CH=C(Cl)-CO-OCH₂-C≡CH, -CH=C(Cl)-CO-OCH₂-CN, -CH=C(Cl)-CO-O(CH₂)₂-CN, -CH=C(Br)-CO-OCH₂-CF₃, -CH=C(Br)-CO-OCH₂-CCl₃, -CH=C(Br)-CO-OCH₂-oxiranyl, -CH=C(Br)-CO-O(CH₂)₃-Br, -CH=C(Br)-CO-OCH₂-CH=CH₂, -CH=C(Br)-CO-OCH₂-C≡CH, -CH=C(Br)-CO-OCH₂-CN, -CH=C(Br)-CO-O(CH₂)₂-CN, -CH=C(CN)-CO-OCH₂-CF₃, -CH=C(CN)-CO-OCH₂-CCl₃, -CH=C(CN)-CO-OCH₂-oxiranyl -CH=C(CN)-CO-O(CH₂)₃-Br, -CH=C(CN)-CO-OCH₂-CH=CH₂, -CH=C(CN)-CO-OCH₂-C≡CH, -CH=C(CN)-CO-OCH₂-CN, -CH=C(CN)-CO-O(CH₂)₂-CN, -CH=CH-CO-CH₃, -CH=CH-CO-C₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-i-C₃H₇, -CH=CH-CO-n-C₄H₉, -CH=CH-CO-tert.-C₄H₉, -CH=CH-CO-CH₂Cl, -CH=CH-CO-CH₂Br, -CH=CH-CO-CHCl₂, -CH=CH-CO-CH₂-OCH₃, -CH=CH-CO-CH(OCH₃)₂, -CH=CH-CO-CH₂-SCH₃, -CH=C(CH₃)-CO-CH₃, -CH=C(CH₃)-CO-C₂H₅, -CH=C(CH₃)-CO-n-C₃H₇, -CH=C(CH₃)-CO-i-C₃H₇, -CH=C(CH₃)-CO-n-C₄H₉, -CH=C(CH₃)-CO-tert.-C₄H₉, -CH=C(CH₃)-CO-CH₂Cl, -CH=C(CH₃)-CO-CH₂Br, -CH=C(CH₃)-CO-CHCl₂, -CH=C(CH₃)-CO-CH₂-OCH₃, -CH=C(CH₃)-CO-CH(OCH₃)₂, -CH=C(CH₃)-CO-CH₂-SCH₃, -CH=C(C₂H₅)-CO-CH₃, -CH=C(C₂H₅)-CO-C₂H₅, -CH=C(C₂H₅)-CO-n-C₃H₇, -CH=C(C₂H₅)-CO-i-C₃H₇, -CH=C(C₂H₅)-CO-n-C₄H₉, -CH=C(C₂H₅)-CO-tert.-C₄H₉, -CH=C(C₂H₅)-CO-CH₂Cl, -CH=C(C₂H₅)-CO-CH₂Br, -CH=C(C₂H₅)-CO-CHCl₂, -CH=C(C₂H₅)-CO-CH₂-OCH₃, -CH=C(C₂H₅)-CO-CH(OCH₃)₂, -CH=C(C₂H₅)-CO-CH₂-SCH₃, -CH=C(Cl)-CO-CH₃, -CH=C(Cl)-CO-C₂H₅, -CH=C(Cl)-CO-n-C₃H₇, -CH=C(Cl)-CO-i-C₃H₇, -CH=C(Cl)-CO-n-C₄H₉, -CH=C(Cl)-CO-tert.-C₄H₉, -CH=C(Cl)-CO-CH₂Cl, -CH=C(Cl)-CO-CH₂Br, -CH=C(Cl)-CO-CHCl₂, -CH=C(Cl)-CO-CH₂-OCH₃, -CH=C(Cl)-CO-CH(OCH₃)₂, -CH=C(Cl)-CO-CH₂-SCH₃, -CH=C(Br)-CO-CH₃, -CH=C(Br)-CO-C₂H₅, -CH=C(Br)-CO-n-C₃H₇, -CH=C(Br)-CO-i-C₃H₇, -CH=C(Br)-CO-n-C₄H₉, -CH=C(Br)-CO-tert.-C₄H₉, -CH=C(Br)-CO-CH₂Cl, -CH=C(Br)-CO-CH₂Br, -CH=C(Br)-CO-CHCl₂, -CH=C(Br)-CO-CH₂-OCH₃, -CH=C(Br)-CO-CH(OCH₃)₂, -CH=C(Br)-CO-CH₂-SCH₃, -CH=C(CN)-CO-CH₃, -CH=C(CN)-CO-C₂H₅, -CH=C(CN)-CO-n-C₃H₇, -CH=C(CN)-CO-i-C₃H₇, -CH=C(CN)-CO-n-C₄H₉, -CH=C(CN)-CO-tert.-C₄H₉, -CH=C(CN)-CO-CH₂Cl, -CH=C(CN)-CO-CH₂Br, -CH=C(CN)-CO-CHCl₂, -CH=C(CN)-CO-CH₂-OCH₃, -CH=C(CN)-CO-CH(OCH₃)₂, -CH=C(CN)-CO-CH₂-SCH₃, -CH=CH-CO-C₆H₅, -CH=CH-CO-(4-Cl-C₆H₄), -CH=C(CH₃)-CO-C₆H₅, -CH=C(CH₃)-CO-(4-Cl-C₆H₄), -CH=C(C₂H₅)-CO-C₆H₅, -CH=C(C₂H₅)-CO-(4-Cl-C₆H₄), -CH=C(Cl)-CO-C₆H₅, -CH=C(Br)-CO-C₆H₅, -CH=C(CN)-CO-C₆H₅, -CH=CH-CO-NH₂, -CH=CH-CO-NHCH₃, -CH=CH-CO-N(CH₃)₂, -CH=CH-CO-NH-C₂H₅, -CH=CH-CO-N(C₂H₅)₂, -CH=CH-CO-NH-n-C₃H₇, -CH=CH-CO-NH-i-C₃H₇, -CH=CH-CO-NH-tert.-C₄H₉, -CH=CH-CO-NH-cyclopropyl, -CH=CH-CO-NH-cyclobutyl, -CH=CH-CO-NH-cyclopentyl, -CH=CH-CO-NH-cyclohexyl, -CH=CH-CO-NH-cycloheptyl, -CH=CH-CO-NH-cyclooctyl, -CH=CH-CO-pyrrolidin-1-yl, -CH=CH-CO-piperidin-1-yl, -CH=CH-CO-morpholin-4-yl, -CH=CH-CO-NH-CH₂CH=CH₂, -CH=CH-CO-NH-CH₂C≡CH, -CH=CH-CO-N(CH₃)-CH₂C≡CH, -CH=CH-CO-NH-(CH₂)₂Cl, -CH=CH-CO-NH-C₆H₅, -CH=C(CH₃)-CO-NH₂, -CH=C(CH₃)-CO-NHCH₃, -CH=C(CH₃)-CO-N(CH₃)₂, -CH=C(CH₃)-CO-NH-C₂H₅, -CH=C(CH₃)-CO-N(C₂H₅)₂, -CH=C(CH₃)-CO-NH-n-C₃H₇, -CH=C(CH₃)-CO-NH-i-C₃H₇, -CH=C(CH₃)-CO-NH-tert.-C₄H₉, -CH=C(CH₃)-CO-NH-cyclopropyl, -CH=C(CH₃)-CO-NH-cyclobutyl, -CH=C(CH₃)-CO-NH-cyclopentyl, -CH=C(CH₃)-CO-NH-cyclohexyl, -CH=C(CH₃)-CO-NH-cycloheptyl, -CH=C(CH₃)-CO-NH-cyclooctyl, -CH=C(CH₃)-CO-pyrrolidin-1-yl, -CH=C(CH₃)-CO-piperidin-1-yl, -CH=C(CH₃)-CO-morpholin-4-yl, -CH=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -CH=C(CH₃)-CO-NH-CH₂C≡CH, -CH=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CH₃)-CO-NH-(CH₂)₂Cl, -CH=C(CH₃)-CO-NH-C₆H₅, -CH=C(C₂H₅)-CO-NH₂, -CH=C(C₂H₅)-CO-NHCH₃, -CH=C(C₂H₅)-CO-N(CH₃)₂, -CH=C(C₂H₅)-CO-NH-C₂H₅, -CH=C(C₂H₅)-CO-N(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-n-C₃H₇, -CH=C(C₂H₅)-CO-NH-i-C₃H₇, -CH=C(C₂H₅)-CO-NH-tert.-C₄H₉, -CH=C(C₂H₅)-CO-NH-cyclopropyl, -CH=C(C₂H₅)-CO-NH-cyclobutyl, -CH=C(C₂H₅)-CO-NH-cyclopentyl, -CH=C(C₂H₅)-CO-NH-cyclohexyl, -CH=C(C₂H₅)-CO-NH-cycloheptyl, -CH=C(C₂H₅)-CO-NH-cyclooctyl, -CH=C(C₂H₅)-CO-pyrrolidin-1-yl, -CH=C(C₂H₅)-CO-piperidin-1-yl, -CH=C(C₂H₅)-CO-morpholin-4-yl, -CH=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-CH₂C≡CH, -CH=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -CH=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -CH=C(C₂H₅)-CO-NH-C₆H₅, -CH=C(Cl)-CO-NH₂, -CH=C(Cl)-CO-NHCH₃, -CH=C(Cl)-CO-N(CH₃)₂, -CH=C(Cl)-CO-NH-C₂H₅, -CH=C(Cl)-CO-N(C₂H₅)₂, -CH=C(Cl)-CO-NH-n-C₃H₇, -CH=C(Cl)-CO-NH-i-C₃H₇, -CH=C(Cl)-CO-NH-tert.-C₄H₉, -CH=C(Cl)-CO-NH-cyclopropyl, -CH=C(Cl)-CO-NH-cyclobutyl, -CH=C(Cl)-CO-NH-cyclopentyl, -CH=C(Cl)-CO-NH-cyclohexyl, -CH=C(Cl)-CO-NH-cycloheptyl, -CH=C(Cl)-CO-NH-cyclooctyl, -CH=C(Cl)-CO-pyrrolidin-1-yl, -CH=C(Cl)-CO-piperidin-1-yl, -CH=C(Cl)-CO-morpholin-4-yl, -CH=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -CH=C(Cl)-CO-NH-CH₂C≡CH, -CH=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Cl)-CO-NH-(CH₂)₂Cl, -CH=C(Cl)-CO-NH-C₆H₅, -CH=C(Br)-CO-NH₂, -CH=C(Br)-CO-NHCH₃, -CH=C(Br)-CO-N(CH₃)₂, -CH=C(Br)-CO-NH-C₂H₅, -CH=C(Br)-CO-N(C₂H₅)₂, -CH=C(Br)-CO-NH-n-C₃H₇, -CH=C(Br)-CO-NH-i-C₃H₇, -CH=C(Br)-CO-NH-tert.-C₄H₉, -CH=C(Br)-CO-NH-cyclopropyl, -CH=C(Br)-CO-NH-cyclobutyl, -CH=C(Br)-CO-NH-cyclopentyl, -CH=C(Br)-CO-NH-cyclohexyl, -CH=C(Br)-CO-NH-cycloheptyl, -CH=C(Br)-CO-NH-cyclooctyl, -CH=C(Br)-CO-pyrrolidin-1-yl, -CH=C(Br)-CO-piperidin-1-yl, -CH=C(Br)-CO-morpholin-4-yl, -CH=C(Br)-CO-NH-CH₂CH=C(Br)₂, -CH=C(Br)-CO-NH-CH₂C≡CH, -CH=C(Br)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Br)-CO-NH-(CH₂)₂Cl, -CH=C(Br)-CO-NH-C₆H₅, -CH=C(CN)-CO-NH₂, -CH=C(CN)-CO-NHCH₃, -CH=C(CN)-CO-N(CH₃)₂, -CH=C(CN)-CO-NH-C₂H₅, -CH=C(CN)-CO-N(C₂H₅)₂, -CH=C(CN)-CO-NH-n-C₃H₇, -CH=C(CN)-CO-NH-i-C₃H₇, -CH=C(CN)-CO-NH-tert.-C₄H₉, -CH=C(CN)-CO-NH-cyclopropyl, -CH=C(CN)-CO-NH-cyclobutyl, -CH=C(CN)-CO-NH-cyclopentyl, -CH=C(CN)-CO-NH-cyclohexyl, -CH=C(CN)-CO-NH-cycloheptyl, -CH=C(CN)-CO-NH-cyclooctyl, -CH=C(CN)-CO-pyrrolidin-1-yl, -CH=C(CN)-CO-piperidin-1-yl, -CH=C(CN)-CO-morpholin-4-yl, -CH=C(CN)-CO-NH-CH₂CH=C(CN)₂, -CH=C(CN)-CO-NH-CH₂C≡CH, -CH=C(CN)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CN)-CO-NH-(CH₂)₂Cl, -CH=C(CN)-CO-NH-C₆H₅, -CH=CH-CO-SCH₃, -CH=CH-CO-SC₂H₅, -CH=CH-CO-S-n-C₃H₇, -CH=CH-CO-S-i-C₃H₇, -CH=CH-CO-S-n-C₄H₉, -CH=CH-CO-S-tert.-C₄H₉, -CH=C(CH₃)-CO-SCH₃, -CH=C(CH₃)-CO-SC₂H₅, -CH=C(CH₃)-CO-S-n-C₃H₇, -CH=C(CH₃)-CO-S-i-C₃H₇, -CH=C(CH₃)-CO-S-n-C₄H₉, -CH=C(CH₃)-CO-S-tert.-C₄H₉, -CH=C(C₂H₅)-CO-SCH₃, -CH=C(C₂H₅)-CO-SC₂H₅, -CH=C(C₂H₅)-CO-S-n-C₃H₇, -CH=C(C₂H₅)-CO-S-i-C₃H₇, -CH=C(C₂H₅)-CO-S-n-C₄H₉, -CH=C(C₂H₅)-CO-S-tert.-C₄H₉, -CH=C(Cl)-CO-SCH₃, -CH=C(Cl)-CO-SC₂H₅, -CH=C(Cl)-CO-S-n-C₃H₇, -CH=C(Cl)-CO-S-i-C₃H₇, -CH=C(Cl)-CO-S-n-C₄H₉, -CH=C(Cl)-CO-S-tert.-C₄H₉, -CH=C(Br)-CO-SCH₃, -CH=C(Br)-CO-SC₂H₅, -CH=C(Br)-CO-S-n-C₃H₇, -CH=C(Br)-CO-S-i-C₃H₇, -CH=C(Br)-CO-S-n-C₄H₉, -CH=C(Br)-CO-S-tert.-C₄H₉, -CH=C(CN)-CO-SCH₃, -CH=C(CN)-CO-SC₂H₅, -CH=C(CN)-CO-S-n-C₃H₇, -CH=C(CN)-CO-S-i-C₃H₇, -CH=C(CN)-CO-S-n-C₄H₉, -CH=C(CN)-CO-S-tert.-C₄H₉, -CH=C(COCH₃)-CO-OCH₃, -CH=C(COC₂H₅)-CO-OCH₃, -CH=C(CO-n-C₃H₇)-CO-OCH₃, -CH=C(COCH₃)-CO-OC₂H₅, -CH=C(COC₂H₅)-CO-OC₂H₅, -CH=C(CO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COCH₃)-CO-O-n-C₃H₇, -CH=C(COC₂H₅)-CO-O-n-C₃H₇, -CH=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-OCH₃, -CH=C(CF₃)-CO-OC₂H₅, -CH=C(CF₃)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-O-i-C₃H₇, -CH=C(CF₃)-CO-O-n-C₄H₉, -CH=C(CF₃)-CO-O-tert.-C₄H₉, -CH=C(COOCH₃)₂, -CH=C(COOC₂H₅)₂, -CH=C(COOCH₃)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)-CO-OCH₃, -CH=C(COO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)₂, -CH=CH-CH=CH-COOH, -CH=CH-CH=CH-CO-OCH₃, -CH=CH-CH=CH-CO-OC₂H₅, -CH=CH-CH=C(COOCH₃)₂, -CH=CH-CH=C(CN)-CO-OCH₃, -CH=CH-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-OCH₃, -CH=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CH=C(Cl)-CO-OCH₃, -CH=C(CH₃)-CH=C(Br)-CO-OCH₃, -CH=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-NH₂, -CH=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -CH=CH-(CH₂)₂-COOH, -CH=CH-(CH₂)₂-CO-OCH₃, -CH=CH-(CH₂)₂-CO-OC₂H₅, -CH=CH-CH₂-CH(COOCH₃)₂, -CH=CH-CH₂-CH(COOC₂H₅)₂, -CH=CH-CH₂-CH(CN)-CO-OCH₃, -CH=CH-CH₂-CH(CN)-CO-OC₂H₅, -CH=CH-CH₂-CH(CH₃)-CO-OCH₃, -CH=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -CH=CH-(CH₂)₂-CO-NH₂, -CH=CH-(CH₂)₂-CO-NH-CH₃, -CH=CH-CH₂-COOH, -CH=CH-CH₂-CO-OCH₃, -CH=CH-CH₂-CO-OC₂H₅, -CH=C(COOCH₃)-CH₂-CO-OCH₃, -CH=C(COOCH₃)-CH₂-CO-OC₂H₅, -CH=CH-CH₂-CO-NH₂, -CH=CH-CH₂-CO-NH-CH₃, -CH=CH-CH₂-CO-N(CH₃)₂, -CH(OCH₃)₂, -CH(SCH₃)₂, -CH(OC₂H₅)₂, -CH(SC₂H₅)₂, -CH(O-n-C₃H₇)₂, -CH(O-i-C₃H₇)₂, -CH(S-n-C₃H₇)₂, -CH(S-i-C₃H₇)₂, -CH(O-n-C₄H₉)₂, -CH(O-i-C₄H₉)₂, -CH(O-s-C₄H₉)₂, -CH(O-tert.-C₄H₉)₂, -CH(S-n-C₄H₉)₂, -CH(S-i-C₄H₉)₂, -CH(S-s-C₄H₉)₂, -CH(S-tert.-C₄H₉)₂, -CH(OC₅H₁₁)₂, 1,3-Dioxolan-2-yl, 1,3-Dithio­ lan-2-yl, 1,3-Oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 5-Methyl-1,3-oxathiolan-2-yl, 4-Ethyl-1,3-dioxolan-2-yl, 4-Ethyl- 1,4-dithiolan-2-yl, 4-Ethyl-1,3-oxathiolan-2-yl, 5-Ethyl-1,3-oxa­ thiolan-2-yl, 4,5-Dimethyl-1,3-dioxolan-2-yl, 4,4-Dimethyl-1,3- dioxolan-2-yl, 4,5-Dimethyl-1,3-dithiolan-2-yl, 5,5-Dimethyl-1,3- dithiolan-2-yl, 4,5-Dimethyl-1,3-oxathiolan-2-yl, 5,5-Dimethyl- 1,3-oxathiolan-2-yl, 4,4-Dimethyl-1,3-oxathiolan-2-yl, 4-Vinyl- 1,3-dioxolan-2-yl, 4-Vinyl-1,3-dithiolan-2-yl, 4-Vinyl-1,3-oxa­ thiolan-2-yl, 5-Vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3- dioxolan-2-yl, 4-Chlormethyl-1,3-dithiolan-2-yl, 4-Chlormethyl- 1,3-oxathiolan-2-yl, 5-Chlormethyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-1,3-dithio­ lan-2-yl, 4-Hydroxymethyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl- 1,3-oxathiolan-2-yl, 4-Methoxymethyl-1,3-dioxolan-2-yl, 4-Allyl­ oxymethyl-1,3-dioxolan-2-yl, 4-Propargyloxymethyl-1,3-dioxolan- 2-yl, 4-Acetoxymethyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-1,3-dithiolan-2-yl, 4-Propargyl- oxymethyl-1,3-dithiolan-2-yl, 4-Acetoxymethyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl-1,3-oxathiolan-2-yl, 5-Allyloxy­ methyl-1,3-oxathiolan-2-yl, 4-Propargyloxymethyl-1,3-oxathiolan-2-yl, 5-Propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxymethyl- 1,3-oxathiolan-2-yl, 5-Acetoxymethyl-1,3-oxathiolan-2-yl, 4-Methylthiomethyl-1,3-dioxolan-2-yl, 4-Methylthiomethyl-1,3- dithiolan-2-yl, 4-Carboxy-1,3-dioxolan-2-yl, 4-Carboxy-1,3- dithiolan-2-yl, 4-Methoxycarbonyl-1,3-dioxolan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-1,3-dithiolan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-4-methyl- 1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-di­ thiolan-2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-1,3- dithiolan-2-yl, 1,3-Dioxan-2-yl, 1,3-Dithian-2-yl, 1,3-Oxathian- 2-yl, 5-Methyl-1,3-dioxan-2-yl, 5-Methyl-1,3-dithian-2-yl, 5-Methyl-1,3-oxathian-2-yl, 5,5-Dimethyl-1,3-dioxan-2-yl, 4,6-Dimethyl- 1,3-dioxan-2-yl, 4,4-Dimethyl-1,3-dioxan-2-yl, 5,5-Dimethyl- 1,3-dithian-2-yl, 4,6-Dimethyl-1,3-dithian-2-yl, 4,4-Dimethyl- 1,3-dithian-2-yl, 5,5-Dimethyl-1,3-oxathian-2-yl, 4,4-Dimethyl- 1,3-oxathian-2-yl, 6,6-Dimethyl-1,3-oxathian-2-yl, 4-Hydroxymethyl-1,3-dioxan-2-yl, 4-Methoxymethyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-1,3-dithian-2-yl, 4-Methoxymethyl-1,3-dithian-2-yl, 4-Allyloxymethyl-1,3-dithian-2-yl, 4-Acetoxymethyl- 1,3-dithian-2-yl, 4-Chlormethyl-1,3-dioxan-2-yl, 4-Chlormethyl- 1,3-dithian-2-yl, 1,3-Dioxepan-2-yl, 1,3-Dithiepan-2-yl, 1,3-Dioxep-5-en-2-yl, 4-Methoxycarbonyl-1,3-dioxan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-1,3-dithian-2-yl, 4-n-Butoxycarbonyl-1,3-dithian-2-yl, 4-Methoxycarbonyl-4- methyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-Methoxy- carbonyl-4-methyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-4-methyl- 1,3-dithian-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithian-2-yl, -C(CH₃)(OCH₃)₂, -C(CH₃)(SCH₃)₂, -C(CH₃)(OC₂H₅)₂, -C(CH₃)(SC₂H₅)₂, -C(CH₃)(O-n-C₃H₇)₂, -C(CH₃)(O-i-C₃H₇)₂, -C(CH₃)(S-n-C₃H₇)₂, -C(CH₃)(S-i-C₃H₇)₂, -C(CH₃)(O-n-C₄H₉)₂, -C(CH₃)(O-i-C₄H₉)₂, -C(CH₃)(O-s-C₄H₉)₂, -C(CH₃)(O-tert.-C₄H₉)₂, -C(CH₃)(S-n-C₄H₉)₂, -C(CH₃)(S-i-C₄H₉)₂, -C(CH₃)(S-s-C₄H₉)₂, -C(CH₃)(S-tert.-C₄H₉)₂, -C(CH₃)(O-n-C₅H₁₁)′′, 2-Methyl-1,3-dioxolan-2-yl, 2-Methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-oxathiolan-2-yl, 2,4-Dimethyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-1,3- oxathiolan-2-yl, 2,5-Dimethyl-1,3-oxathiolan-2-yl, 4-Ethyl-2- methyl-1,3-dioxolan-2-yl, 4-Ethyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Ethyl-2-methyl-1,3- oxathiolan-2-yl, 2,4,5-Trimethyl-1,3-dioxolan-2-yl, 2,4,4-Trimethyl- 1,3-dioxolan-2-yl, 2,4,5-Trimethyl-1,3-dithiolan-2-yl, 2,4,4-Trimethyl-1,3-dithiolan-2-yl, 2,4,5-Trimethyl-1,3-oxathiolan-2-yl, 2,4,4-Trimethyl-1,3-oxathiolan-2-yl, 2-Methyl-4-vinyl- 1,3-dioxolan-2-yl, 2-Methyl-4-vinyl-1,3-dithiolan-2-yl, 2-Methyl- 4-vinyl-1,3-oxathiolan-2-yl, 2-Methyl-5-vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-dioxolan-2-yl, 4-Chlormethyl-2- methyl-1,3-dithiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl- 2-methyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-2- methyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dioxolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxy- 2-methyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dithiolan-2-yl, 4-Acetoxy-2- methyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl- 2-methyl-1,3-oxathiolan-2-yl, 5-Allyloxymetyl-2- methyl-1,3-oxathiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3- oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxy-2-methyl-1,3-oxathiolan-2-yl, 5-Acetoxy-2-methyl- 1,3-oxathiolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dioxolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-2- methyl-1,3-dioxolan-2-yl, 4-Carboxy-2-methyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-2- methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl- 2-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-2- methyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-ethoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4- ethoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-n-butoxy- carbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl-1,3- dithiolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-dioxan-2-yl, 2-Methyl-1,3-dithian-2-yl, 2-Methyl-1,3-oxathian-2-yl, 2,5- Dimethyl-1,3-dioxan-2-yl, 2,5-Dimethyl-1,3-dithian-2-yl, 2,5-Dimethyl- 1,3-oxathian-2-yl, 2,5,5-Trimethyl-1,3-dioxan-2-yl, 2,4,6- Trimethyl-1,3-dioxan-2-yl, 2,4,4-Trimethyl-1,3-dioxan-2-yl, 2,5,5-Trimethyl-1,3-dithian-2-yl, 2,4,6-Trimethyl-1,3-dithian-2-yl, 2,4,4-Trimethyl-1,3-dithian-2-yl, 2,5,5-Trimethyl-1,3-oxathian-2-yl, 2,4,4-Trimethyl-1,3-oxathian-2-yl, 2,6,6-Trimethyl- 1,3-oxathian-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-2- methyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dithian-2-yl, 4-Methoxymethyl-2- methyl-1,3-dithian-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithian-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dithian-2-yl, 4-Chlormethyl-2- methyl-1,3-dioxan-2-yl, 4-Chlormethyl-2-methyl-1,3-dithian-2-yl, -C(CH₃)=NH, -C(CH₃)=N-CH₃, -C(CH₃)=N-C₂H₅, -C(CH₃)=N-n-C₃H₇, -C(CH₃)=N-i-C₃H₇, -C(CH₃)=N-n-C₄H₉, -C(CH₃)=N-CH₂CH=CH₂, -C(CH₃)=N-CH₂CH=CH₂-CH₃, -C(CH₃)=N-CH₂C≡CH, -C(CH₃)=N-CH₂C≡C-CH₃, -C(CH₃)=N-cyclopropyl, -C(CH₃)=N-cyclobutyl, -C(CH₃)=N-cyclopentyl, -C(CH₃)=N-cyclohexyl, -C(CH₃)=N-cycloheptyl, -C(CH₃)=N-CH₂-CH₂Cl, -C(CH₃)=N-CH₂Cl, -C(CH₃)=N-C₆H₅, -C(CH₃)=N-(2-F-C₆H₄), -C(CH₃)=N-(3-F-C₆H₄), -C(CH₃)=N-(4-F-C₆H₄), -C(CH₃)=N-(2-Cl-C₆H₄), -C(CH₃)=N-(3-Cl-C₆H₄), -C(CH₃)=N-(4-Cl-C₆H₄), -C(CH₃)=N-(2-CH₃-C₆H₄), -C(CH₃)=N-(3-CH₃-C₆H₄), -C(CH₃)=N-(4-CH₃-C₆H₄), -C(CH₃)=N-(2-CF₃-C₆H₄), -C(CH₃)=N-(3-CF₃-C₆H₄), -C(CH₃)=N-(4-CF₃-C₆H₄), -C(CH₃)=N-(2-OCH₃-C₆H₄), -C(CH₃)=N-(3-OCH₃-C₆H₄), -C(CH₃)=N-(4-OCH₃-C₆H₄), -C(CH₃)=N-(4-NO₂-C₆H₄), -C(CH₃)=N-(4-CN-C₆H₄), -C(CH₃)=N-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-(2,4-(CH₃)₂-C₆H₃), -C(CH₃)=N-CH₂-OCH₃, -C(CH₃)=N-CH₂-OC₂H₅, -C(CH₃)=N-CH₂CH₂-OCH₃, -C(CH₃)=N-CH₂CH-OC₂H₅, -C(CH₃)=N-OH, -C(CH₃)=N-OCH₃, -C(CH₃)=N-OC₂H₅, -C(CH₃)=N-O-n-C₃H₇, -C(CH₃)=N-O-i-C₃H₇, -C(CH₃)=N-O-n-C₄H₉, -C(CH₃)=N-O-i-C₄H₉, -C(CH₃)=N-O-s-C₄H₉, -C(CH₃)=N-O-tert.-C₄H₉, -C(CH₃)=N-OCH₂-CH=CH₂, -C(CH₃)=N-OCH(CH₃)-CH=CH₂, -C(CH₃)=N-OCH₂-C≡CH, -C(CH₃)=N-CH(CH₃)-C≡CH, -C(CH₃)=N-OCH₂-CH=C-CH₃, -C(CH₃)=N-OCH₂CH₂-Cl, -C(CH₃)=N-OCH₂CH₂-F, -C(CH₃)=N-OCH₂-CF₃, -C(CH₃)=N-OCH₂-CH=CHCl, -C(CH₃)=N-OCH₂-C(Cl)=CH₂, -C(CH₃)=N-OCH₂-C(Br)=CH₂, -C(CH₃)=N-OCH₂-CH=C(Cl)-CH₃, -C(CH₃)=N-O-CO-CH₃, -C(CH₃)=N-O-CO-C₂H₅, -C(CH₃)=N-OCH₂-CN, -C(CH₃)=N-OCH₂-CH=CH-CH₂-OCH₃, -C(CH₃)=N-OCH₂-CH=CH-CH₂-O-tert.-C₄H₉, -C(CH₃)=N-O-(CH₂)₃-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-(4-Cl-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-C₆H₅, -C(CH₃)=N-OCH₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(3-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-CH₂-(4-CH₃O-C₆H₄), -C(CH₃)=N-OCH₂-CH=C(CH₃)-C₆H₅, -C(CH₃)=N-O-(CH₂)₂-CH=CH-(3,4-Cl₂-C₆H₃), -C(CH₃)=N-O-(CH₂)₃-C≡-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-OCH₃, -C(CH₃)=N-OCH₂CH₂-OCH₃, -C(CH₃)=N-OCH₂-OC₂H₅, -C(CH₃)=N-OCH(CH₃)-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=N-NH₂, -C(CH₃)=N-NH-CH₃, -C(CH₃)=N-NH-C₂H₅, -C(CH₃)=N-NH-n-C₃H₇, -C(CH₃)=N-NH-i-C₃H₇, -C(CH₃)=N-NH-n-C₄H₉, -C(CH₃)=N-NH-i-C₄H₉, -C(CH₃)=N-NH-s-C₄H₉, -C(CH₃)=N-NH-tert.-C₄H₉, -C(CH₃)=N-NH-cyclopropyl, -C(CH₃)=N-NH-cyclobutyl, -C(CH₃)=N-NH-cyclopentyl, -C(CH₃)=N-NH-cyclohexyl, -C(CH₃)=N-NH-cycloheptyl, -C(CH₃)=N-N(CH₃)₂, -C(CH₃)=N-N(C₂H₅)₂, -C(CH₃)=N-N(n-C₃H₇)₂, -C(CH₃)=N-N(i-C₃H₇)₂, -C(CH₃)=N-NH-CH₂-C=CH, -C(CH₃)=N-NH-CH₂-C≡CH, -C(CH₃)=N-N(CH₃)-CH₂-C≡CH, -C(CH₃)=N-NH-CH₂CF₃, -C(CH₃)=N-NH-CO-CH₃, -C(CH₃)=N-NH-CO-C₂H₅, -C(CH₃)=N-NH-CO-OCH₃, -C(CH₃)=N-NH-CO-OC₂H₅, -C(CH₃)=N-NH-CO-O-tert.-C₄H₉, -C(CH₃)=N-pyrrolidin-1-yl, -C(CH₃)=N-piperidin-1-yl, -C(CH₃)=N-morpholin-4-yl, -C(CH₃)=N-NH-C₆H₅, -C(CH₃)=N-NH-(4-Cl-C₆H₄), -C(CH₃)=N-NH-(4-NO₂-C₆H₄), -C(CH₃)=N-NH-(4-F-C₆H₄), -C(CH₃)=N-NH-(4-CH₃O-C₆H₄), -C(CH₃)=N-NH-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-NH-(2,4-(NO₂)₂-C₆H₃), -C(CH₃)=N-NH-CO-NH₂, -C(CH₃)=N-NH-CO-NHCH₃, -C(CH₃)=N-NH-CO-NHC₂H₅, -C(CH₃)=N-NH-CO-N(CH₃)₂, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=CH-CO-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -(CH₃)=CH-CO-O-n-C₄H₉, -C(CH₃)=CH-CO-O-tert.-C₄H₉, -C(CH₃)=CH-CO-O-cyclopropyl, -C(CH₃)=CH-CO-O-cyclobutyl, -C(CH₃)=CH-CO-O-cyclopentyl, -C(CH₃)=CH-CO-O-cyclohexyl, -C(CH₃)=CH-CO-O-cycloheptyl, -C(CH₃)=C(CH₃)-COOH, -C(CH₃)=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-cyclopropyl, -C(CH₃)=C(CH₃)-CO-O-cyclobutyl, -C(CH₃)=C(CH₃)-CO-O-cyclopentyl, -C(CH₃)=C(CH₃)-CO-O-cyclohexyl, -C(CH₃)=C(CH₃)-CO-O-cycloheptyl, -C(CH₃)=C(C₂H₅)-COOH, -C(CH₃)=C(C₂H₅)-CO-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-cyclo­ propyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-O- cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-O-cycloheptyl, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-O-n-C₄H₉, -C(CH₃)=C(Cl)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-O-cyclopropyl, -C(CH₃)=C(Cl)-CO-O-cyclobutyl, -C(CH₃)=C(Cl)-CO-O-cyclopentyl, -C(CH₃)=C(Cl)-CO-O-cyclohexyl, -C(CH₃)=C(Cl)-CO-O-cycloheptyl, -C(CH₃)=C(Br)-COOH, -C(CH₃)=C(Br)-CO-OCH₃, -C(CH₃)=C(Br)-CO-OC₂H₅, -C(CH₃)=C(Br)-CO-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-O-n-C₄H₉, -C(CH₃)=C(Br)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-O-cyclopropyl, -C(CH₃)=C(Br)-CO-O-cyclobutyl, -C(CH₃)=C(Br)-CO-O-cyclopentyl, -C(CH₃)=C(Br)-CO-O-cyclohexyl, -C(CH₃)=C(Br)-CO-O-cycloheptyl, -C(CH₃)=C(CN)-COOH, -C(CH₃)=C(CN)-CO-OCH₃, -C(CH₃)=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CN)-CO-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-O-n-C₄H₉, -C(CH₃)=C(CN)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-O-cyclopropyl, -C(CH₃)=C(CN)-CO-O-cyclobutyl, -C(CH₃)=C(CN)-CO-O-cyclopentyl, -C(CH₃)=C(CN)-CO-O-cyclohexyl, -C(CH₃)=C(CN)-CO-O-cycloheptyl, -C(CH₃)=CH-CO-OCH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-OCH(CH₃)-OCH₃, -C(CH₃)=CH-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=CH-CO-OCH₂CH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=(C₂H₅)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-O-i-C₃H₇, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -(CH₃)=C(Cl)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-O-i-C₃H₇, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-O-i-C₃H₇, -C(CH₃)=C(CN)-CO-OCH(CH₃)OCH₃, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-CF₃, -C(CH₃)=CH-CO-OCH₂-CCl₃, -C(CH₃)=CH-CO-OCH₂-oxiranyl, -C(CH₃)=CH-CO-(CH₂)₃-Br,-C(CH₃)=CH-CO-OCH₂-CH=CH₂, -C(CH₃)=CH-CO-OCH₂-C≡CH, -C(CH₃)=CH-CO-OCH₂-CN, -C(CH₃)=CH-CO-OCH₂CH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CF₃, -C(CH₃)=C(CH₃)-CO-OCH₂-CCl₃, -C(CH₃)=C(CH₃)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CH₃)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CH₃)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CH₃)-CO-OCH₂-C≡CH, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CF₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CCl₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-oxiranyl, -C(CH₃)=C(C₂H₅)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(C₂H₅)-CO-OCH₂-C≡CH, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂-CF₃, -C(CH₃)=C(Cl)-CO-OCH₂-CCl₃, -C(CH₃)=C(Cl)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Cl)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Cl)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Cl)-CO-OCH₂-C≡CH, -C(CH₃)=C(Cl)-CO-OCH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂-CF₃, -C(CH₃)=C(Br)-CO-OCH₂-CCl₃, -C(CH₃)=C(Br)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Br)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Br)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Br)-CO-OCH₂-C≡CH, -C(CH₃)=C(Br)-CO-OCH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂CH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂-CF₃, -C(CH₃)=C(CN)-CO-OCH₂-CCl₃, -C(CH₃)=C(CN)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CN)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CN)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CN)-CO-OCH₂-C≡CH, -C(CH₃)=C(CN)-CO-OCH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂CH₂-CN, -C(CH₃)=CH-CO-CH₃, -C(CH₃)=CH-CO-C₂H₅, -C(CH₃)=CH-CO-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-n-C₄H₉, -C(CH₃)=CH-CO-tert.-C₄H₉, -C(CH₃)=CH-CO-CH₂Cl, -C(CH₃)=CH-CO-CH₂Br, -C(CH₃)=CH-CO-CHCl₂, -C(CH₃)=CH-CO-CH₂-OCH₃, -C(CH₃)=CH-CO-CH(OCH₃)₂, -C(CH₃)=CH-CO-CH₂-SCH₃, -C(CH₃)=C(CH₃)-CO-CH₃, -C(CH₃)=C(CH₃)-CO-C₂H₅, -C(CH₃)=C(CH₃)-CO-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-CH₂Cl, -C(CH₃)=C(CH₃)-CO-CH₂Br, -C(CH₃)=C(CH₃)-CO-CHCl₂, -C(CH₃)=C(CH₃)-CO-CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-CH(OCH₃)₂, -C(CH₃)=C(CH₃)-CO-CH₂-SCH₃, -C(CH₃)=C(C₂H₅)-CO-CH₃, -C(CH₃)=C(C₂H₅)-CO-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-CH₂Cl, -C(CH₃)=C(C₂H₅)-CO-CH₂Br, -C(CH₃)=C(C₂H₅)-CO-CHCl₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-CH(OCH₃)₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-SCH₃, -C(CH₃)=C(Cl)-CO-CH₃, -C(CH₃)=C(Cl)-CO-C₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-n-C₄H₉, -C(CH₃)=C(Cl)-CO-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-CH₂Cl, -C(CH₃)=C(Cl)-CO-CHCl₂, -C(CH₃)=C(Cl)-CO-CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-CH(OCH₃)₂, -C(CH₃)=C(Cl)-CO-CH₂-SCH₃, -C(CH₃)=C(Br)-CO-CH₃, -C(CH₃)=C(Br)-CO-C₂H₅, -C(CH₃)=C(Br)-CO-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-n-C₄H₉, -C(CH₃)=C(Br)-CO-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-CH₂Cl, -C(CH₃)=C(Br)-CO-CH₂Br, -C(CH₃)=C(Br)-CO-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-CH(OCH₃)₂, -C(CH₃)=C(Br)-CO-CH₂-SCH₃, -C(CH₃)=C(CN)-CO-CH₃, -C(CH₃)=C(CN)-CO-C₂H₅, -C(CH₃)=C(CN)-CO-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-n-C₄H₉, -C(CH₃)=C(CN)-CO-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-CH₂Cl, -C(CH₃)=C(CN)-CO-CH₂Br, -C(CH₃)=C(CN)-CO-CHCl₂, -C(CH₃)=C(CN)-CO-CH₂-OCH₃, -C(CH₃)=C(CN)-CO-CH(OCH₃)₂, -C(CH₃)=C(CN)-CO-CH₂-SCH₃, -C(CH₃)=CH-CO-C₆H₅, -C(CH₃)=CH-CO-(4-Cl-C₆H₄), -C(CH₃)=C(CH₃)-CO-C₆H₅, -C(CH₃)=C(CH₃)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(C₂H₅)-CO-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(Cl)-CO-C₆H₅, -C(CH₃)=C(Br)-CO-C₆H₅, -C(CH₃)=C(CN)-CO-C₆H₅, -C(CH₃)=CH-CO-NH₂, -C(CH₃)=CH-CO-NHCH₃, -C(CH₃)=CH-CO-N(CH₃)₂, -C(CH₃)=CH-CO-NH-C₂H₅, -C(CH₃)=CH-CO-N(C₂H₅)₂, -C(CH₃)=CH-CO-NH-n-C₃H₇, -C(CH₃)=CH-CO-NH-i-C₃H₇, -C(CH₃)=CH-CO-NH-tert.-C₄H₉, -C(CH₃)=CH-CO-NH-cyclopropyl, -C(CH₃)=CH-CO-NH-cyclobutyl, -C(CH₃)=CH-CO-NH-cyclopentyl, -C(CH₃)=CH-CO-NH-cyclohexyl, -C(CH₃)=CH-CO-NH-cycloheptyl, -C(CH₃)=CH-CO-NH-cyclooctyl, -C(CH₃)=CH-CO-pyrrolidin-1-yl, -C(CH₃)=CH-CO-piperidin-1-yl, -C(CH₃)=CH-CO-morpholin-4-yl, -C(CH₃)=CH-CO-NH-CH₂CH=CH₂, -C(CH₃)=CH-CO-NH-CH₂C≡CH, -C(CH₃)=CH-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=CCH-CO-NH-(CH₂)₂Cl, -C(CH₃)=CH-CO-NH-C₆H₅, -C(CH₃)=C(CH₃)-CO-NH₂, -C(CH₃)=C(CH₃)-CO-NHCH₃, -C(CH₃)=C(CH₃)-CO-N(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-C₂H₅, -C(CH₃)=C(CH₃)-CO-N(C₂H₅)₂, -C(CH₃)=C(CH₃)-CO-NH-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-NH- cyclopropyl, -C(CH₃)=C(CH₃)-CO-NH-cyclobutyl, -C(CH₃)=C(CH₃)-CO-NH-cyclopentyl, -C(CH₃)=C(CH₃)-CO-NH- cyclohexyl, -C(CH₃)=C(CH₃)-CO-NH-cycloheptyl, -C(CH₃)=C(CH₃)-CO-NH-cyclooctyl, -C(CH₃)=C(CH₃)-CO- pyrrolidin-1-yl, -C(CH₃)=C(CH₃)-CO-piperidin-1-yl, -C(CH₃)=C(CH₃)-CO-morpholin-4-yl, -C(CH₃)=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-NH(CH₂)₂Cl, -C(CH₃)=C(CH₃)-CO-NH-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-NH₂, -C(CH₃)=C(C₂H₅)-CO-NHCH₃, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)₂, -C(CH₃)=C(C₂H₅)-CO-NH-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-N(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-NH- cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclo­ hexyl, -C(CH₃)=C(C₂H₅)-CO-NH-cycloheptyl, -C(CH₃)=C(C₂H₅)-CO-NH- cyclooctyl, -C(CH₃)=C(C₂H₅)-CO-pyrrolidin-1-yl, -C(CH₃)=C(C₂H₅)-CO-piperidin-1-yl, -C(CH₃)=C(C₂H₅)-CO- morpholin-4-yl, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(C₂H₅)-CO-NH-C₆H₅, -C(CH₃)=C(Cl)-CO-NH₂, -C(CH₃)=C(Cl)-CO-NHCH₃, -C(CH₃)=C(Cl)-CO-N(CH₃)₂, -C(CH₃)=C(Cl)-CO-NH-C₂H₅, -C(CH₃)=C(Cl)-CO-N(C₂H₅)₂, -C(CH₃)=C(Cl)-CO-NH-n-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-i-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-NH-cyclopropyl, -C(CH₃)=C(Cl)-CO-NH-cyclobutyl, -C(CH₃)=C(Cl)-CO-NH-cyclopentyl, -C(CH₃)=C(Cl)-CO-NH-cyclohexyl, -C(CH₃)=C(Cl)-CO-NH-cycloheptyl, -C(CH₃)=C(Cl)-CO-NH-cyclooctyl, -C(CH₃)=C(Cl)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Cl)-CO-piperidin-1- yl, -C(CH₃)=C(Cl)-CO-morpholin-4-yl, -C(CH₃)=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -C(Cl)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-N(CH₃)-CH₂≡CH, -C(CH₃)=C(Cl)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Cl)-NO-NH-C₆H₅, -C(CH₃)=C(Br)-CO-NH₂, -C(CH₃)=C(Br)-CO-NHCH₃, -C(CH₃)=C(Br)-CO-N(CH₃)₂, -C(CH₃)=C(Br)-CO-NH-C₂H₅, -C(CH₃)=C(Br)-CO-N(C₂H₅)₂, -C(CH₃)=C(Br)-CO-NH-n-C₃H₇, -C(CH₃)=C(Br)-CO-NH-i-C₃H₇, -C(CH₃)=C(Br)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-NH-cyclopropyl, -C(CH₃)=C(Br)-CO-NH-cyclobutyl, -C(CH₃)=C(Br)-CO-NH-cyclopentyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cycloheptyl, -C(CH₃)=C(Br)-CO-NH-cyclooctyl, -C(CH₃)=C(Br)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Br)-CO-piperidin-1-yl, -C(CH₃)=C(Br)-CO-morpholin-4-yl, -C(CH₃)=C(Br)-CO-NH-CH₂CH=C(Br)₂, -C(CH₃)=C(Br)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Br)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Br)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Br)-CO-NH-C₆H₅, -C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CN)-CO-NHCH₃, -C(CH₃)=C(CN)-CO-N(CH₃)₂, -C(CH₃)=C(CN)-CO-NH-C₂H₅, -C(CH₃)=C(CN)-CO-N(C₂H₅)₂, -C(CH₃)=C(CN)-CO-NH-n-C₃H₇, -C(CH₃)=C(CN)-CO-NH-i-C₃H₇, -C(CH₃)=C(CN)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-NH-cyclopropyl, -C(CH₃)=C(CN)-CO-NH-cyclobutyl, -C(CH₃)=C(CN)-CO-NH-cyclopentyl, -C(CH₃)=C(CN)-CO-NH-cyclohexyl, -C(CH₃)=C(CN)-CO-NH-cycloheptyl, -C(CH₃)=C(CN)-CO-NH-cyclooctyl, -C(CH₃)=C(CN)-CO-pyrrolidin-1-yl, -C(CH₃)=C(CN)-CO-piperidin-1-yl, -C(CH₃)=C(CN)-CO-morpholin-4-yl, -C(CH₃)=C(CN)-CO-NH-CH₂CH=C(CN)₂, -C(CH₃)=C(CN)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CN)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)=C(CN)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CN)-CO-NH-C₆H₅, -C(CH₃)=CH-SO-SCH₃, -C(CH₃)=CH-CO-SC₂H₅, -C(CH₃)=CH-CO-S-n-C₃H₇, -C(CH₃)=CH-CO-S-i-C₃H₇, -C(CH₃)=CH-CO-S-n-C₄H₉, -C(CH₃)=CH-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-SCH₃, -C(CH₃)=C(CH₃)-CO-SC₂H₅, -C(CH₃)=C(CH₃)CO-S-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-S-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-SCH₃, -C(CH₃)=C(C₂H₅)-CO-SC₂H₅, -C(CH₃)=C(C₂H₅)-CO-S-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-SCH₃, -C(CH₃)=C(Cl)-CO-SC₂H₅, -C(CH₃)=C(Cl)-CO-S-n-C₃H₇, -C(CH₃)=C(Cl)-CO-S-i-C₃H₇, -C(CH₃)=C(Cl)-CO-S-n-C₄H₉, -C(CH₃)=C(Cl)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-SCH₃, -C(CH₃)=C(Br)-CO-SC₂H₅, -C(CH₃)=C(Br)-CO-S-n-C₃H₇, -C(CH₃)=C(Br)-CO-S-i-C₃H₇, -C(CH₃)=C(Br)-CO-S-n-C₄H₉, -C(CH₃)=C(Br)-CO-S-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-SCH₃, -C(CH₃)=C(CN)-CO-SC₂H₅, -C(CH₃)=C(CN)-CO-S-n-C₃H₇, -C(CH₃)=C(CN)-CO-S-i-C₃H₇, -C(CH₃)=C(CN)-CO-S-N-C₄H₉, -C(CH₃)=C(CN)-CO-S-tert.-C₄H₉, -C(CH₃)=C(COCH₃)-CO-OCH₃, -C(CH₃)=C(COC₂H₅)-CO-OCH₃, -C(CH₃)=C(CO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COCH₃)-CO-OC₂H₅, -C(CH₃)=C(COC₂H₅)-CO-OC₂H₅, -C(CH₃)=C(CO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COCH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(COC₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-OCH₃, -C(CH₃)=C(CF₃)-CO-OC₂H₅, -C(CH₃)=C(CF₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CF₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(COOCH₃)₂, -C(CH₃)=C(COOC₂H₅)₂, -C(CH₃)=C(COOCH₃)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)₂, -C(CH₃)=CH-CH=CH-COOH, -C(CH₃)=CH-CH=CH-CO-OCH₃, -C(CH₃)=CH-CH=CH-CO-OC₂H₅, -C(CH₃)=CH-CH=C(COOCH₃)₂, -C(CH₃)=CH-CH=C(CN)-CO-OCH₃, -C(CH₃)=CH-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH₂, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -C(CH₃)=CH-(CH₂)₂-COOH, -C(CH₃)=CH-(CH₂)₂-CO-OCH₃, -C(CH₃)=CH-(CH₂)₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(COOCH₃)₂, -C(CH₃)=CH-CH₂-CH(COOC₂H₅)₂, -C(CH₃)=CH-CH₂-CH(CN)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CN)-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -C(CH₃)=CH-(CH₂)₂-CO-NH₂, -C(CH₃)=CH-(CH₂)₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-COOH, -C(CH₃)=CH-CH₂-CO-OCH₃, -C(CH₃)=CH-CH₂-CO-OC₂H₅, -C(CH₃)=C(COOCH₃)-CH₂-CO-OCH₃, -C(CH₃)=C(COOCH₃)-CH₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CO-NH₂, -C(CH₃)=CH-CH₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-CO-N(CH₃)₂.
wobei W für eine der folgenden Bedeutungen steht:
-CHO, -COCH₃, -COC₂H₅, -CO-n-C₃H₇, -CO-i-C₃H₇, -CO-n-C₄H₉, -CO-i-C₄H₉, -CO-s-C₄H₉, -CO-tert.-C₄H₉, -CO-CH₂CH=CH₂, -CO-CF₃, -COCCl₃, -COCH₂C≡CH, -CO-cyclopropyl, -CO-cyclobutyl, -CO-cyclopentyl, -CO-cyclohexyl, -CO-CN, -CO-COOCH₃, -CO-COOC₂H₅, -CH=NH, -CH=NCH₃, -CH=NC₂H₅, -CH=N-n-C₃H₅, -CH=N-i-C₃H₅, -CH=N-n-C₄H₉, -CH=NCH₂CH=CH₂, -CH=NCH₂CH=CH₂-CH₃, -CH=NCH₂≡CH, -CH=NCH₂C≡C-CH₃, -CH=N-cyclopropyl, -CH=N-cyclobutyl, -CH=N-cyclopentyl, -CH=N-cyclohexyl, -CH=N-cycloheptyl, -CH=N-CH₂-CH₂Cl, -CH=N-CH₂Cl, -CH=N-C₆H₅, -CH=N-(4-Br-C₆H₄), -CH=N-3-F-C₆H₄, -CH=N-4-F-C₆H₄, -CH=N-2-Cl-C₆H₄, -CH=N-3-Cl-C₆H₄, -CH=N-4-Cl-C₆H₄, -CH=N-2-Br-C₆H₄, -CH=N-2-F-C₆H₄, -CH=N-2-CH₃-C₆H₄, -CH=N-3-CH₃-C₆H₄, -CH=N-4-CH₃-C₆H₄, -CH=N-2-CF₃-C₆H₄, -CH=N-3-CF₃-C₆H₄, -CH=N-4-CF₃-C₆H₄, -CH=N-2-OCH₃-C₆H₄, -CH=N-3-OCH₃-C₆H₄, -CH=N-4-OCH₃-C₆H₄, -CH=N-4-NO₂-C₆H₄, -CH=N-4-CN-C₆H₄, -CH=N-2,4-(Cl,Cl)-C₆H₄, -CH=N-2,4-(CH₃,CH₃)-C₆H₄, -CH=N-CH₂OCH₃ -CH=N-CH₂OC₂H₅, -CH=N-CH₂CH₂OCH₃, -CH=N-CH₂CH₂OC₂H₅, -CH=N-OH, -CH=N-OCH₃, -CH=N-OC₂H₅, -CH=N-O-n-C₃H₇, -CH=N-O-i-C₃H₇, -CH=N-O-n-C₄H₉, -CH=N-O-i-C₄H₉, -CH=N-O-s-C₄H₉, -CH=N-O-tert.-C₄H₉, -CH=N-O-CH₂CH=CH₂, -CH=N-O-CH(CH₃)CH=CH₂, -CH=N-O-CH₂C≡CH, -CH=N-O-CH(CH₃)-C≡CH, -CH=N-O-CH₂-CH=CH-CH₃, -CH=N-O-CH₂-CH₂-Cl, -CH=N-O-CH₂-CH₂-F, -CH=N-O-CH₂-CF₃, -CH=N-O-CH₂-CH=CHCl, -CH=N-O-CH₂-CCl=CH₂, -CH=N-O-CH₂-CBr=CH₂, -CH=N-O-CH₂-CH=CCl-CH₃, -CH=N-OC(O)CH₃, -CH=N-OC(O)C₂H₅, -CH=N-O-CH₂-CN, -CH=N-O-CH₂-CH=CH-CH₂-O-CH₃, -CH=N-O-CH₂-CH=CH-CH₂-O-tert.-C₄H₉, -CH=N-O-(CH₂)₃-C₆H₅, -CH=N-O-(CH₂)₄-C₆H₅, -CH=N-O-(CH₂)₄-4-Cl-C₆H₄, -CH=N-O-(CH₂)₄-4-OCH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-CH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-C₆H₅, -CH=N-O-CH₂CH=CH-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CH-3-OCH₃-C₆H₄, -CH=N-O-(CH₂)₂CH=CH-4-F-C₆H₄, -CH=N-O-(CH₂)CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CHCH₂-4-OCH₃-C₆H₄, -CH=N-O-CH₂-CH=C(CH₃)-C₆H₄ -CH=N-O-(CH₂)₂CH=CH-3,4(Cl,Cl)-C₆H₃, -CH=N-O-(CH₂)₃C≡C-4-F-C₆H₄, -CH₂=N-OCHOCH₃, -CH=N-OC₂H₄OCH₃, -CH=N-OCH₂OC₂H₅, -CH=N-OCH(CH₃)OCH₃, -CH=N-OCH(CH₃)COOCH₃, -CH=N-OCH(CH₃)COO-n-C₄H₉, -CH=N-NH₂, -CH=N-NHCH₃, -CH=N-NHC₂H₅, -CH=N-NH-n-C₃H₇, -CH=N-NH-i-C₃H₇, -CH=N-NH-n-C₄H₉, -CH=N-NH-i-C₄H₉, -CH=N-NH-s-C₄H₉, -CH=N-NH-tert.-C₄H₉, -CH=N-NH-cyclopropyl, -CH=N-NH-cyclobutyl, -CH=N-NH-cyclopentyl, -CH=N-NH-cyclohexyl, -CH=N-NH-cycloheptyl, -CH=N-N(CH₃)₂, -CH=N-N(C₂H₅)₂, -CH=N-N(C₃H₇)₂, -CH=N-N(i-C₃H₇)(CH₃), -CH=N-NHCH₂-C=CH, -CH=N-NHCH₂-C≡CH, -CH=N-N(CH₃)-CH₂-C≡CH, -CH=N-NHCH₂CF₃, -CH=N-NH-CO-CH₃, -CH=N-NH-CO-CH₂H₅, -CH=N-NH-COOCH₃, -CH=N-NH-COOC₂H₅, -CH=N-NH-COO-tert.-C₄H₉, -CH=N-pyrrolidin-1-yl, -CH=N-piperidin-1-yl, -CH=N-morpholin-4-yl, -CH=N-NH-C₆H₅, -CH=N-NH-(4-Cl-C₆H₄), -CH=N-NH-(4-NO₂-C₆H₄), -CH=N-NH-(4-F-C₆H₄), -CH=N-NH-(4-CH₃O-C₆H₄), -CH=N-NH-(2,4-Cl₂-C₆H₃), -CH=N-NH-(2,4-(NO₂)₂-C₆H₃), -CH=N-NH-CO-NH₂, -CH=N-NH-CO-NHCH₃, -CH=N-NH-CO-NHC₂H₅, -CH=N-NH-CO-N(CH₃)₂, -CH=CH-COOH, -CH=CH-CO-OCH₃, -CH=CH-CO-OC₂H₅, -CH=CH-CO-O-n-C₃H₇, -CH=CH-CO-O-i-C₃H₇, -CH=CH-CO-O-n-C₄H₉, -CH=CH-CO-O-tert.-C₄H₉, -CH=CH-CO-O-cyclopropyl, -CH=CH-CO-O-cyclobutyl, -CH=CH-CO-O-cyclopentyl, -CH=CO-O-cyclohexyl, -CH=CH-CO-O-cycloheptyl, -CH=C(CH₃)-COOH, -CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CO-O-n-C₃H₇, -CH=C(CH₃)-CO-O-i-C₃H₇, -CH=C(CH₃)-CO-O-n-C₄H₉, -CH=C(CH₃)-CO-O-tert.-C₄H₉, -CH=C(CH₃)-CO-O-cyclopropyl, -CH=C(CH₃)-CO-O-cyclobutyl, -CH=C(CH₃)-CO-O-cyclopentyl, -CH=C(CH₃)-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cycloheptyl, -CH=C(C₂H₅)-COOH, -CH=C(C₂H₅)-CO-OCH₃, -CH=C(C₂H₅)-CO-OC₂H₅, -CH=C(C₂H₅)-CO-O-n-C₃H₇, -CH=C(C₂H₅)-CO-O-i-C₃H₇, -CH=C(C₂H₅)-CO-O-n-C₄H₉, -CH=C(C₂H₅)-CO-O-tert.-C₄H₉, -CH=C(C₂H₅)-CO-O-cyclopropyl, -CH=C(C₂H₅)-CO-O-cyclobutyl, -CH=C(C₂H₅)-CO-O-cyclopentyl, -CH=C(C₂H₅)-CO-O-cyclohexyl, -CH=C(C₂H₅)-CO-O-cycloheptyl, -CH=C(Cl)-COOH, -CH=C(Cl)-CO-OCH₃, -CH=C(Cl)-CO-OC₂H₅, -CH=C(Cl)-CO-O-n-C₃H₇, -CH=C(Cl)-CO-O-i-C₃H₇, -CH=C(Cl)-CO-O-n-C₄H₉, -CH=C(Cl)-CO-O-tert.-C₄H₉, -CH=C(Cl)-CO-O-cyclopropyl, -CH=C(Cl)-CO-O-cyclobutyl, -CH=C(Cl)-CO-O-cyclopentyl, -CH=C(Cl)-CO-O-cyclohexyl, -CH=C(Cl)-CO-O-cycloheptyl, -CH=C(Br)-COOH, -CH=C(Br)-CO-OCH₃, -CH=C(Br)-CO-OC₂H₅, -CH=C(Br)-CO-O-n-C₃H₇, -CH=C(Br)-CO-O-i-C₃H₇, -CH=C(Br)-CO-O-n-C₄H₉, -CH=C(Br)-CO-O-tert.-C₄H₉, -CH=C(Br)-CO-O-cyclopropyl, -CH=C(Br)-CO-O-cyclobutyl, -CH=C(Br)-CO-O-cyclopentyl, -CH=C(Br)-CO-O-cyclohexyl, -CH=C(Br)-CO-O-cycloheptyl, -CH=C(CN)-COOH, -CH=C(CN)-CO-OCH₃, -CH=C(CN)-CO-OC₂H₅, -CH=C(CN)-CO-O-n-C₃H₇, -CH=C(CN)-CO-O-i-C₃H₇, -CH=C(CN)-CO-O-n-C₄H₉, -CH=C(CN)-CO-O-tert.-C₄H₉, -CH=C(CN)-CO-O-cyclopropyl, -CH=C(CN)-CO-O-cyclobutyl, -CH=C(CN)-CO-O-cyclopentyl, -CH=C(CN)-CO-O-cyclohexyl, -CH=C(CN)-CO-O-cycloheptyl, -CH=CH-CO-OCH₂-OCH₃, -CH=CH-CO-OCH₂-OC₂H₅, -CH=CH-CO-OCH₂-O-n-C₃H₅, -CH=CH-CO-OCH₂-O-i-C₃H₅, -CH=CH-CO-OCH(CH₃)-OCH₃, -CH=CH-CO-OCH(CH₃)-OC₂H₅, -CH=CH-CO-O-CH₂CH₂-OCH₃, -CH=CH-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-OCH₃, -CH=C(CH₃)-CO-OCH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-O-n-C₃H₅, -CH=C(CH₃)-CO-OCH₂-O-i-C₃H₅, -CH=C(CH₃)-CO-OCH(CH₃)-OCH₃, -CH=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CH₃)-CO-O-CH₂CH₂-OCH₃, -CH=C(CH₃)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-OCH₃, -CH=C(C₂H₅)-CO-OCH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-O-n-C₃H₅, -CH=C(C₂H₅)-CO-OCH₂-O-i-C₃H₅, -CH=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -CH=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OCH₃, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-OCH₃, -CH=C(Cl)-CO-OCH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-O-n-C₃H₅, -CH=C(Cl)-CO-OCH₂-O-i-C₃H₅, -CH=C(Cl)-CO-OCH(CH₃)-OCH₃, -CH=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Cl)-CO-O-CH₂CH₂-OCH₃, -CH=C(Cl)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-OCH₃, -CH=C(Br)-CO-OCH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-O-n-C₃H₅, -CH=C(Br)-CO-OCH₂-O-i-C₃H₅, -CH=C(Br)-CO-OCH(CH₃)-OCH₃, -CH=C(Br)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Br)-CO-O-CH₂CH₂-OCH₃, -CH=C(Br)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-OCH₃, -CH=C(CN)-CO-OCH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-O-n-C₃H₅, -CH=C(CN)-CO-OCH₂-O-i-C₃H₅, -CH=C(CN)-CO-OCH(CH₃)-OCH₃, -CH=C(CN)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CN)-CO-O-CH₂CH₂-OCH₃, -CH=C(CN)-CO-O-CH₂CH₂-OC₂H₅, -CH=CH-CO-OCH₂-CF₃, -CH=CH-CO-OCH₂-CCl₃, -CH=CH-CO-OCH₂-oxiranyl, -CH=CH-CO-O(CH₂)₃-Br, -CH=CH-CO-OCH₂-CH=CH₂, -CH=CH-CO-OCH₂-C≡CH, -CH=CH-CO-OCH₂-CN, -CH=CH-CO-O(CH₂)₂-CN, -CH=C(CH₃)-CO-OCH₂-CF₃, -CH=C(CH₃)-CO-OCH₂-CCl₃, -CH=C(CH₃)-CO-OCH₂-oxiranyl, -CH=C(CH₃)-CO-O(CH₂)₃-Br, -CH=C(CH₃)-CO-OCH₂-CH=CH₂, -CH=C(CH₃)-CO-OCH₂-C≡CH, -CH=C(CH₃)-CO-OCH₂-CN, -CH=C(CH₃)-CO-O(CH₂)₂-CN, -CH=C(C₂H₅)-CO-OCH₂-CF₃, -CH=C(C₂H₅)-CO-OCH₂-CCl₃, -CH=C(C₂H₅)-CO-OCH₂-oxiranyl, -CH=C(C₂H₅)-CO-O(CH₂)₃-Br, -CH=C(C₂H₅)-CO-OCH₂-CH=CH₂, -CH=C(C₂H₅)-CO-OCH₂-C≡CH, -CH=C(C₂H₅)-CO-OCH₂-CN, -CH=C(C₂H₅)-CO-O(CH₂)₂-CN, -CH=C(Cl)-CO-OCH₂-CF₃, -CH=C(Cl)-CO-OCH₂-CCl₃, -CH=C(Cl)-CO-OCH₂-oxiranyl, -CH=C(Cl)-CO-O(CH₂)₃-Br, -CH=C(Cl)-CO-OCH₂-CH=CH₂, -CH=C(Cl)-CO-OCH₂-C≡CH, -CH=C(Cl)-CO-OCH₂-CN, -CH=C(Cl)-CO-O(CH₂)₂-CN, -CH=C(Br)-CO-OCH₂-CF₃, -CH=C(Br)-CO-OCH₂-CCl₃, -CH=C(Br)-CO-OCH₂-oxiranyl, -CH=C(Br)-CO-O(CH₂)₃-Br, -CH=C(Br)-CO-OCH₂-CH=CH₂, -CH=C(Br)-CO-OCH₂-C≡CH, -CH=C(Br)-CO-OCH₂-CN, -CH=C(Br)-CO-O(CH₂)₂-CN, -CH=C(CN)-CO-OCH₂-CF₃, -CH=C(CN)-CO-OCH₂-CCl₃, -CH=C(CN)-CO-OCH₂-oxiranyl -CH=C(CN)-CO-O(CH₂)₃-Br, -CH=C(CN)-CO-OCH₂-CH=CH₂, -CH=C(CN)-CO-OCH₂-C≡CH, -CH=C(CN)-CO-OCH₂-CN, -CH=C(CN)-CO-O(CH₂)₂-CN, -CH=CH-CO-CH₃, -CH=CH-CO-C₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-i-C₃H₇, -CH=CH-CO-n-C₄H₉, -CH=CH-CO-tert.-C₄H₉, -CH=CH-CO-CH₂Cl, -CH=CH-CO-CH₂Br, -CH=CH-CO-CHCl₂, -CH=CH-CO-CH₂-OCH₃, -CH=CH-CO-CH(OCH₃)₂, -CH=CH-CO-CH₂-SCH₃, -CH=C(CH₃)-CO-CH₃, -CH=C(CH₃)-CO-C₂H₅, -CH=C(CH₃)-CO-n-C₃H₇, -CH=C(CH₃)-CO-i-C₃H₇, -CH=C(CH₃)-CO-n-C₄H₉, -CH=C(CH₃)-CO-tert.-C₄H₉, -CH=C(CH₃)-CO-CH₂Cl, -CH=C(CH₃)-CO-CH₂Br, -CH=C(CH₃)-CO-CHCl₂, -CH=C(CH₃)-CO-CH₂-OCH₃, -CH=C(CH₃)-CO-CH(OCH₃)₂, -CH=C(CH₃)-CO-CH₂-SCH₃, -CH=C(C₂H₅)-CO-CH₃, -CH=C(C₂H₅)-CO-C₂H₅, -CH=C(C₂H₅)-CO-n-C₃H₇, -CH=C(C₂H₅)-CO-i-C₃H₇, -CH=C(C₂H₅)-CO-n-C₄H₉, -CH=C(C₂H₅)-CO-tert.-C₄H₉, -CH=C(C₂H₅)-CO-CH₂Cl, -CH=C(C₂H₅)-CO-CH₂Br, -CH=C(C₂H₅)-CO-CHCl₂, -CH=C(C₂H₅)-CO-CH₂-OCH₃, -CH=C(C₂H₅)-CO-CH(OCH₃)₂, -CH=C(C₂H₅)-CO-CH₂-SCH₃, -CH=C(Cl)-CO-CH₃, -CH=C(Cl)-CO-C₂H₅, -CH=C(Cl)-CO-n-C₃H₇, -CH=C(Cl)-CO-i-C₃H₇, -CH=C(Cl)-CO-n-C₄H₉, -CH=C(Cl)-CO-tert.-C₄H₉, -CH=C(Cl)-CO-CH₂Cl, -CH=C(Cl)-CO-CH₂Br, -CH=C(Cl)-CO-CHCl₂, -CH=C(Cl)-CO-CH₂-OCH₃, -CH=C(Cl)-CO-CH(OCH₃)₂, -CH=C(Cl)-CO-CH₂-SCH₃, -CH=C(Br)-CO-CH₃, -CH=C(Br)-CO-C₂H₅, -CH=C(Br)-CO-n-C₃H₇, -CH=C(Br)-CO-i-C₃H₇, -CH=C(Br)-CO-n-C₄H₉, -CH=C(Br)-CO-tert.-C₄H₉, -CH=C(Br)-CO-CH₂Cl, -CH=C(Br)-CO-CH₂Br, -CH=C(Br)-CO-CHCl₂, -CH=C(Br)-CO-CH₂-OCH₃, -CH=C(Br)-CO-CH(OCH₃)₂, -CH=C(Br)-CO-CH₂-SCH₃, -CH=C(CN)-CO-CH₃, -CH=C(CN)-CO-C₂H₅, -CH=C(CN)-CO-n-C₃H₇, -CH=C(CN)-CO-i-C₃H₇, -CH=C(CN)-CO-n-C₄H₉, -CH=C(CN)-CO-tert.-C₄H₉, -CH=C(CN)-CO-CH₂Cl, -CH=C(CN)-CO-CH₂Br, -CH=C(CN)-CO-CHCl₂, -CH=C(CN)-CO-CH₂-OCH₃, -CH=C(CN)-CO-CH(OCH₃)₂, -CH=C(CN)-CO-CH₂-SCH₃, -CH=CH-CO-C₆H₅, -CH=CH-CO-(4-Cl-C₆H₄), -CH=C(CH₃)-CO-C₆H₅, -CH=C(CH₃)-CO-(4-Cl-C₆H₄), -CH=C(C₂H₅)-CO-C₆H₅, -CH=C(C₂H₅)-CO-(4-Cl-C₆H₄), -CH=C(Cl)-CO-C₆H₅, -CH=C(Br)-CO-C₆H₅, -CH=C(CN)-CO-C₆H₅, -CH=CH-CO-NH₂, -CH=CH-CO-NHCH₃, -CH=CH-CO-N(CH₃)₂, -CH=CH-CO-NH-C₂H₅, -CH=CH-CO-N(C₂H₅)₂, -CH=CH-CO-NH-n-C₃H₇, -CH=CH-CO-NH-i-C₃H₇, -CH=CH-CO-NH-tert.-C₄H₉, -CH=CH-CO-NH-cyclopropyl, -CH=CH-CO-NH-cyclobutyl, -CH=CH-CO-NH-cyclopentyl, -CH=CH-CO-NH-cyclohexyl, -CH=CH-CO-NH-cycloheptyl, -CH=CH-CO-NH-cyclooctyl, -CH=CH-CO-pyrrolidin-1-yl, -CH=CH-CO-piperidin-1-yl, -CH=CH-CO-morpholin-4-yl, -CH=CH-CO-NH-CH₂CH=CH₂, -CH=CH-CO-NH-CH₂C≡CH, -CH=CH-CO-N(CH₃)-CH₂C≡CH, -CH=CH-CO-NH-(CH₂)₂Cl, -CH=CH-CO-NH-C₆H₅, -CH=C(CH₃)-CO-NH₂, -CH=C(CH₃)-CO-NHCH₃, -CH=C(CH₃)-CO-N(CH₃)₂, -CH=C(CH₃)-CO-NH-C₂H₅, -CH=C(CH₃)-CO-N(C₂H₅)₂, -CH=C(CH₃)-CO-NH-n-C₃H₇, -CH=C(CH₃)-CO-NH-i-C₃H₇, -CH=C(CH₃)-CO-NH-tert.-C₄H₉, -CH=C(CH₃)-CO-NH-cyclopropyl, -CH=C(CH₃)-CO-NH-cyclobutyl, -CH=C(CH₃)-CO-NH-cyclopentyl, -CH=C(CH₃)-CO-NH-cyclohexyl, -CH=C(CH₃)-CO-NH-cycloheptyl, -CH=C(CH₃)-CO-NH-cyclooctyl, -CH=C(CH₃)-CO-pyrrolidin-1-yl, -CH=C(CH₃)-CO-piperidin-1-yl, -CH=C(CH₃)-CO-morpholin-4-yl, -CH=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -CH=C(CH₃)-CO-NH-CH₂C≡CH, -CH=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CH₃)-CO-NH-(CH₂)₂Cl, -CH=C(CH₃)-CO-NH-C₆H₅, -CH=C(C₂H₅)-CO-NH₂, -CH=C(C₂H₅)-CO-NHCH₃, -CH=C(C₂H₅)-CO-N(CH₃)₂, -CH=C(C₂H₅)-CO-NH-C₂H₅, -CH=C(C₂H₅)-CO-N(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-n-C₃H₇, -CH=C(C₂H₅)-CO-NH-i-C₃H₇, -CH=C(C₂H₅)-CO-NH-tert.-C₄H₉, -CH=C(C₂H₅)-CO-NH-cyclopropyl, -CH=C(C₂H₅)-CO-NH-cyclobutyl, -CH=C(C₂H₅)-CO-NH-cyclopentyl, -CH=C(C₂H₅)-CO-NH-cyclohexyl, -CH=C(C₂H₅)-CO-NH-cycloheptyl, -CH=C(C₂H₅)-CO-NH-cyclooctyl, -CH=C(C₂H₅)-CO-pyrrolidin-1-yl, -CH=C(C₂H₅)-CO-piperidin-1-yl, -CH=C(C₂H₅)-CO-morpholin-4-yl, -CH=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-CH₂C≡CH, -CH=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -CH=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -CH=C(C₂H₅)-CO-NH-C₆H₅, -CH=C(Cl)-CO-NH₂, -CH=C(Cl)-CO-NHCH₃, -CH=C(Cl)-CO-N(CH₃)₂, -CH=C(Cl)-CO-NH-C₂H₅, -CH=C(Cl)-CO-N(C₂H₅)₂, -CH=C(Cl)-CO-NH-n-C₃H₇, -CH=C(Cl)-CO-NH-i-C₃H₇, -CH=C(Cl)-CO-NH-tert.-C₄H₉, -CH=C(Cl)-CO-NH-cyclopropyl, -CH=C(Cl)-CO-NH-cyclobutyl, -CH=C(Cl)-CO-NH-cyclopentyl, -CH=C(Cl)-CO-NH-cyclohexyl, -CH=C(Cl)-CO-NH-cycloheptyl, -CH=C(Cl)-CO-NH-cyclooctyl, -CH=C(Cl)-CO-pyrrolidin-1-yl, -CH=C(Cl)-CO-piperidin-1-yl, -CH=C(Cl)-CO-morpholin-4-yl, -CH=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -CH=C(Cl)-CO-NH-CH₂C≡CH, -CH=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Cl)-CO-NH-(CH₂)₂Cl, -CH=C(Cl)-CO-NH-C₆H₅, -CH=C(Br)-CO-NH₂, -CH=C(Br)-CO-NHCH₃, -CH=C(Br)-CO-N(CH₃)₂, -CH=C(Br)-CO-NH-C₂H₅, -CH=C(Br)-CO-N(C₂H₅)₂, -CH=C(Br)-CO-NH-n-C₃H₇, -CH=C(Br)-CO-NH-i-C₃H₇, -CH=C(Br)-CO-NH-tert.-C₄H₉, -CH=C(Br)-CO-NH-cyclopropyl, -CH=C(Br)-CO-NH-cyclobutyl, -CH=C(Br)-CO-NH-cyclopentyl, -CH=C(Br)-CO-NH-cyclohexyl, -CH=C(Br)-CO-NH-cycloheptyl, -CH=C(Br)-CO-NH-cyclooctyl, -CH=C(Br)-CO-pyrrolidin-1-yl, -CH=C(Br)-CO-piperidin-1-yl, -CH=C(Br)-CO-morpholin-4-yl, -CH=C(Br)-CO-NH-CH₂CH=C(Br)₂, -CH=C(Br)-CO-NH-CH₂C≡CH, -CH=C(Br)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Br)-CO-NH-(CH₂)₂Cl, -CH=C(Br)-CO-NH-C₆H₅, -CH=C(CN)-CO-NH₂, -CH=C(CN)-CO-NHCH₃, -CH=C(CN)-CO-N(CH₃)₂, -CH=C(CN)-CO-NH-C₂H₅, -CH=C(CN)-CO-N(C₂H₅)₂, -CH=C(CN)-CO-NH-n-C₃H₇, -CH=C(CN)-CO-NH-i-C₃H₇, -CH=C(CN)-CO-NH-tert.-C₄H₉, -CH=C(CN)-CO-NH-cyclopropyl, -CH=C(CN)-CO-NH-cyclobutyl, -CH=C(CN)-CO-NH-cyclopentyl, -CH=C(CN)-CO-NH-cyclohexyl, -CH=C(CN)-CO-NH-cycloheptyl, -CH=C(CN)-CO-NH-cyclooctyl, -CH=C(CN)-CO-pyrrolidin-1-yl, -CH=C(CN)-CO-piperidin-1-yl, -CH=C(CN)-CO-morpholin-4-yl, -CH=C(CN)-CO-NH-CH₂CH=C(CN)₂, -CH=C(CN)-CO-NH-CH₂C≡CH, -CH=C(CN)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CN)-CO-NH-(CH₂)₂Cl, -CH=C(CN)-CO-NH-C₆H₅, -CH=CH-CO-SCH₃, -CH=CH-CO-SC₂H₅, -CH=CH-CO-S-n-C₃H₇, -CH=CH-CO-S-i-C₃H₇, -CH=CH-CO-S-n-C₄H₉, -CH=CH-CO-S-tert.-C₄H₉, -CH=C(CH₃)-CO-SCH₃, -CH=C(CH₃)-CO-SC₂H₅, -CH=C(CH₃)-CO-S-n-C₃H₇, -CH=C(CH₃)-CO-S-i-C₃H₇, -CH=C(CH₃)-CO-S-n-C₄H₉, -CH=C(CH₃)-CO-S-tert.-C₄H₉, -CH=C(C₂H₅)-CO-SCH₃, -CH=C(C₂H₅)-CO-SC₂H₅, -CH=C(C₂H₅)-CO-S-n-C₃H₇, -CH=C(C₂H₅)-CO-S-i-C₃H₇, -CH=C(C₂H₅)-CO-S-n-C₄H₉, -CH=C(C₂H₅)-CO-S-tert.-C₄H₉, -CH=C(Cl)-CO-SCH₃, -CH=C(Cl)-CO-SC₂H₅, -CH=C(Cl)-CO-S-n-C₃H₇, -CH=C(Cl)-CO-S-i-C₃H₇, -CH=C(Cl)-CO-S-n-C₄H₉, -CH=C(Cl)-CO-S-tert.-C₄H₉, -CH=C(Br)-CO-SCH₃, -CH=C(Br)-CO-SC₂H₅, -CH=C(Br)-CO-S-n-C₃H₇, -CH=C(Br)-CO-S-i-C₃H₇, -CH=C(Br)-CO-S-n-C₄H₉, -CH=C(Br)-CO-S-tert.-C₄H₉, -CH=C(CN)-CO-SCH₃, -CH=C(CN)-CO-SC₂H₅, -CH=C(CN)-CO-S-n-C₃H₇, -CH=C(CN)-CO-S-i-C₃H₇, -CH=C(CN)-CO-S-n-C₄H₉, -CH=C(CN)-CO-S-tert.-C₄H₉, -CH=C(COCH₃)-CO-OCH₃, -CH=C(COC₂H₅)-CO-OCH₃, -CH=C(CO-n-C₃H₇)-CO-OCH₃, -CH=C(COCH₃)-CO-OC₂H₅, -CH=C(COC₂H₅)-CO-OC₂H₅, -CH=C(CO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COCH₃)-CO-O-n-C₃H₇, -CH=C(COC₂H₅)-CO-O-n-C₃H₇, -CH=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-OCH₃, -CH=C(CF₃)-CO-OC₂H₅, -CH=C(CF₃)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-O-i-C₃H₇, -CH=C(CF₃)-CO-O-n-C₄H₉, -CH=C(CF₃)-CO-O-tert.-C₄H₉, -CH=C(COOCH₃)₂, -CH=C(COOC₂H₅)₂, -CH=C(COOCH₃)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)-CO-OCH₃, -CH=C(COO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)₂, -CH=CH-CH=CH-COOH, -CH=CH-CH=CH-CO-OCH₃, -CH=CH-CH=CH-CO-OC₂H₅, -CH=CH-CH=C(COOCH₃)₂, -CH=CH-CH=C(CN)-CO-OCH₃, -CH=CH-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-OCH₃, -CH=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CH=C(Cl)-CO-OCH₃, -CH=C(CH₃)-CH=C(Br)-CO-OCH₃, -CH=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-NH₂, -CH=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -CH=CH-(CH₂)₂-COOH, -CH=CH-(CH₂)₂-CO-OCH₃, -CH=CH-(CH₂)₂-CO-OC₂H₅, -CH=CH-CH₂-CH(COOCH₃)₂, -CH=CH-CH₂-CH(COOC₂H₅)₂, -CH=CH-CH₂-CH(CN)-CO-OCH₃, -CH=CH-CH₂-CH(CN)-CO-OC₂H₅, -CH=CH-CH₂-CH(CH₃)-CO-OCH₃, -CH=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -CH=CH-(CH₂)₂-CO-NH₂, -CH=CH-(CH₂)₂-CO-NH-CH₃, -CH=CH-CH₂-COOH, -CH=CH-CH₂-CO-OCH₃, -CH=CH-CH₂-CO-OC₂H₅, -CH=C(COOCH₃)-CH₂-CO-OCH₃, -CH=C(COOCH₃)-CH₂-CO-OC₂H₅, -CH=CH-CH₂-CO-NH₂, -CH=CH-CH₂-CO-NH-CH₃, -CH=CH-CH₂-CO-N(CH₃)₂, -CH(OCH₃)₂, -CH(SCH₃)₂, -CH(OC₂H₅)₂, -CH(SC₂H₅)₂, -CH(O-n-C₃H₇)₂, -CH(O-i-C₃H₇)₂, -CH(S-n-C₃H₇)₂, -CH(S-i-C₃H₇)₂, -CH(O-n-C₄H₉)₂, -CH(O-i-C₄H₉)₂, -CH(O-s-C₄H₉)₂, -CH(O-tert.-C₄H₉)₂, -CH(S-n-C₄H₉)₂, -CH(S-i-C₄H₉)₂, -CH(S-s-C₄H₉)₂, -CH(S-tert.-C₄H₉)₂, -CH(OC₅H₁₁)₂, 1,3-Dioxolan-2-yl, 1,3-Dithio­ lan-2-yl, 1,3-Oxathiolan-2-yl, 4-Methyl-1,3-dioxolan-2-yl, 4-Methyl-1,3-dithiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 5-Methyl-1,3-oxathiolan-2-yl, 4-Ethyl-1,3-dioxolan-2-yl, 4-Ethyl- 1,4-dithiolan-2-yl, 4-Ethyl-1,3-oxathiolan-2-yl, 5-Ethyl-1,3-oxa­ thiolan-2-yl, 4,5-Dimethyl-1,3-dioxolan-2-yl, 4,4-Dimethyl-1,3- dioxolan-2-yl, 4,5-Dimethyl-1,3-dithiolan-2-yl, 5,5-Dimethyl-1,3- dithiolan-2-yl, 4,5-Dimethyl-1,3-oxathiolan-2-yl, 5,5-Dimethyl- 1,3-oxathiolan-2-yl, 4,4-Dimethyl-1,3-oxathiolan-2-yl, 4-Vinyl- 1,3-dioxolan-2-yl, 4-Vinyl-1,3-dithiolan-2-yl, 4-Vinyl-1,3-oxa­ thiolan-2-yl, 5-Vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3- dioxolan-2-yl, 4-Chlormethyl-1,3-dithiolan-2-yl, 4-Chlormethyl- 1,3-oxathiolan-2-yl, 5-Chlormethyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-1,3-dithio­ lan-2-yl, 4-Hydroxymethyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl- 1,3-oxathiolan-2-yl, 4-Methoxymethyl-1,3-dioxolan-2-yl, 4-Allyl­ oxymethyl-1,3-dioxolan-2-yl, 4-Propargyloxymethyl-1,3-dioxolan- 2-yl, 4-Acetoxymethyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-1,3-dithiolan-2-yl, 4-Propargyl- oxymethyl-1,3-dithiolan-2-yl, 4-Acetoxymethyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl-1,3-oxathiolan-2-yl, 5-Allyloxy- methyl-1,3-oxathiolan-2-yl, 4-Propargyloxymethyl-1,3-oxathiolan-2-yl, 5-Propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxymethyl- 1,3-oxathiolan-2-yl, 5-Acetoxymethyl-1,3-oxathiolan-2-yl, 4-Methylthiomethyl-1,3-dioxolan-2-yl, 4-Methylthiomethyl-1,3- dithiolan-2-yl, 4-Carboxy-1,3-dioxolan-2-yl, 4-Carboxy-1,3- dithiolan-2-yl, 4-Methoxycarbonyl-1,3-dioxolan-2-yl, 4-Ethoxy- carbonyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-1,3-dithiolan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-4-methyl- 1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-di­ thiolan-2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-1,3- dithiolan-2-yl, 1,3-Dioxan-2-yl, 1,3-Dithian-2-yl, 1,3-Oxathian- 2-yl, 5-Methyl-1,3-dioxan-2-yl, 5-Methyl-1,3-dithian-2-yl, 5-Methyl-1,3-oxathian-2-yl, 5,5-Dimethyl-1,3-dioxan-2-yl, 4,6-Dimethyl- 1,3-dioxan-2-yl, 4,4-Dimethyl-1,3-dioxan-2-yl, 5,5-Dimethyl- 1,3-dithian-2-yl, 4,6-Dimethyl-1,3-dithian-2-yl, 4,4-Dimethyl- 1,3-dithian-2-yl, 5,5-Dimethyl-1,3-oxathian-2-yl, 4,4-Dimethyl- 1,3-oxathian-2-yl, 6,6-Dimethyl-1,3-oxathian-2-yl, 4-Hydroxymethyl-1,3-dioxan-2-yl, 4-Methoxymethyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-1,3-dithian-2-yl, 4-Methoxymethyl-1,3-dithian-2-yl, 4-Allyloxymethyl-1,3-dithian-2-yl, 4-Acetoxymethyl- 1,3-dithian-2-yl, 4-Chlormethyl-1,3-dioxan-2-yl, 4-Chlormethyl- 1,3-dithian-2-yl, 1,3-Dioxepan-2-yl, 1,3-Dithiepan-2-yl, 1,3-Dioxep-5-en-2-yl, 4-Methoxycarbonyl-1,3-dioxan-2-yl, 4-Ethoxy- carbonyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-1,3-dithian-2-yl, 4-n-Butoxycarbonyl-1,3-dithian-2-yl, 4-Methoxycarbonyl-4- methyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-Methoxy- carbonyl-4-methyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-4-methyl- 1,3-dithian-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithian-2-yl, -C(CH₃)(OCH₃)₂, -C(CH₃)(SCH₃)₂, -C(CH₃)(OC₂H₅)₂, -C(CH₃)(SC₂H₅)₂, -C(CH₃)(O-n-C₃H₇)₂, -C(CH₃)(O-i-C₃H₇)₂, -C(CH₃)(S-n-C₃H₇)₂, -C(CH₃)(S-i-C₃H₇)₂, -C(CH₃)(O-n-C₄H₉)₂, -C(CH₃)(O-i-C₄H₉)₂, -C(CH₃)(O-s-C₄H₉)₂, -C(CH₃)(O-tert.-C₄H₉)₂, -C(CH₃)(S-n-C₄H₉)₂, -C(CH₃)(S-i-C₄H₉)₂, -C(CH₃)(S-s-C₄H₉)₂, -C(CH₃)(S-tert.-C₄H₉)₂, -C(CH₃)(O-n-C₅H₁₁)′′, 2-Methyl-1,3-dioxolan-2-yl, 2-Methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-oxathiolan-2-yl, 2,4-Dimethyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-1,3- oxathiolan-2-yl, 2,5-Dimethyl-1,3-oxathiolan-2-yl, 4-Ethyl-2- methyl-1,3-dioxolan-2-yl, 4-Ethyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Ethyl-2-methyl-1,3- oxathiolan-2-yl, 2,4,5-Trimethyl-1,3-dioxolan-2-yl, 2,4,4-Trimethyl- 1,3-dioxolan-2-yl, 2,4,5-Trimethyl-1,3-dithiolan-2-yl, 2,4,4-Trimethyl-1,3-dithiolan-2-yl, 2,4,5-Trimethyl-1,3-oxathiolan-2-yl, 2,4,4-Trimethyl-1,3-oxathiolan-2-yl, 2-Methyl-4-vinyl- 1,3-dioxolan-2-yl, 2-Methyl-4-vinyl-1,3-dithiolan-2-yl, 2-Methyl- 4-vinyl-1,3-oxathiolan-2-yl, 2-Methyl-5-vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-dioxolan-2-yl, 4-Chlormethyl-2- methyl-1,3-dithiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl- 2-methyl-1,3-dioxolan-2-yl, 5-Allyloxymethyl-2-methyl- 1,3-oxathiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-2- methyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dioxolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxy- 2-methyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dithiolan-2-yl, 4-Acetoxy-2- methyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl- 2-methyl-1,3-oxathiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3- oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxy-2-methyl-1,3-oxathiolan-2-yl, 5-Acetoxy-2-methyl- 1,3-oxathiolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dioxolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-2- methyl-1,3-dioxolan-2-yl, 4-Carboxy-2-methyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-2- methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl- 2-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-2- methyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-ethoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4- ethoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-n-butoxy- carbony-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl-1,3- dithiolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-dioxan-2-yl, 2-Methyl-1,3-dithian-2-yl, 2-Methyl-1,3-oxathian-2-yl, 2,5- Dimethyl-1,3-dioxan-2-yl, 2,5-Dimethyl-1,3-dithian-2-yl, 2,5-Dimethyl- 1,3-oxathian-2-yl, 2,5,5-Trimethyl-1,3-dioxan-2-yl, 2,4,6- Trimethyl-1,3-dioxan-2-yl, 2,2,4-Trimethyl-1,3-dioxan-2-yl, 2,5,5-Trimethyl-1,3-dithian-2-yl, 2,4,6-Trimethyl-1,3-dithian-2-yl, 2,4,4-Trimethyl-1,3-dithian-2-yl, 2,5,5-Trimethyl-1,3-oxathian-2-yl, 2,4,4-Trimethyl-1,3-oxathian-2-yl, 2,6,6-Trimethyl- 1,3-oxathian-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-2- methyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dithian-2-yl, 4-Methoxymethyl-2- methyl-1,3-dithian-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithian-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dithian-2-yl, 4-Chlormethyl-2- methyl-1,3-dioxan-2-yl, 4-Chlormethyl-2-methyl-1,3-dithian-2-yl, -C(CH₃)=NH, -C(CH₃)=N-CH₃, -C(CH₃)=N-C₂H₅, -C(CH₃)=N-n-C₃H₇, -(CH₃)=N-i-C₃H₇, -C(CH₃)=N-n-C₄H₉, -C(CH₃)=N-CH₂CH=CH₂, -C(CH₃)=N-CH₂CH=CH₂-CH₃, -C(CH₃)=N-CH₂C≡CH, -C(CH₃)=N-CH₂C≡C-CH₃, -C(CH₃)=N-cyclopropyl, -C(CH₃)=N-cyclobutyl, -C(CH₃)=N-cyclopentyl, -C(CH₃)=N-cyclohexyl, -C(CH₃)=N-cycloheptyl, -C(CH₃)=N-CH₂-CH₂Cl, -C(CH₃)=N-CH₂Cl, -C(CH₃)=N-C₆H₅, -C(CH₃)=N-(2-F-C₆H₄), -C(CH₃)=N-(3-F-C₆H₄), -C(CH₃)=N-(4-F-C₆H₄), -C(CH₃)=N-(2-Cl-C₆H₄), -C(CH₃)=N-(3-Cl-C₆H₄), -C(CH₃)=N-(4-Cl-C₆H₄), -C(CH₃)=N-(2-CH₃-C₆H₄), -C(CH₃)=N-(3-CH₃-C₆H₄), -C(CH₃)=N-(4-CH₃-C₆H₄), -C(CH₃)=N-(2-CF₃-C₆H₄), -C(CH₃)=N-(3-CF₃-C₆H₄), -C(CH₃)=N-(4-CF₃-C₆H₄), -C(CH₃)=N-(2-OCH₃-C₆H₄), -C(CH₃)=N-(3-OCH₃-C₆H₄), -C(CH₃)=N-(4-OCH₃-C₆H₄), -C(CH₃)=N-(4-NO₂-C₆H₄), -C(CH₃)=N-(4-CN-C₆H₄), -C(CH₃)=N-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-(2,4-(CH₃)₂-C₆H₃), -C(CH₃)=N-CH₂-OCH₃, -C(CH₃)=N-CH₂-OC₂H₅, -C(CH₃)=N-CH₂CH₂-OCH₃, -C(CH₃)=N-CH₂CH-OC₂H₅, -C(CH₃)=N-OH, -C(CH₃)=N-OCH₃, -C(CH₃)=N-OC₂H₅, -C(CH₃)=N-O-n-C₃H₇, -C(CH₃)=N-O-i-C₃H₇, -C(CH₃)=N-O-n-C₄H₉, -C(CH₃)=N-O-i-C₄H₉, -C(CH₃)=N-O-s-C₄H₉, -C(CH₃)=N-O-tert.-C₄H₉, -C(CH₃)=N-OCH₂-CH=CH₂, -C(CH₃)=N-OCH(CH₃)-CH=CH₂, -C(CH₃)=N-OCH₂-C≡CH, -C(CH₃)=N-CH(CH₃)-C≡CH, -C(CH₃)=N-OCH₂-CH=C-CH₃, -C(CH₃)=N-OCH₂CH₂-Cl, -C(CH₃)=N-OCH₂CH₂-F, -C(CH₃)=N-OCH₂-CF₃, -C(CH₃)=N-OCH₂-CH=CHCl, -C(CH₃)=N-OCH₂-C(Cl)=CH₂, -C(CH₃)=N-OCH₂-C(Br)=CH₂, -C(CH₃)=N-OCH₂-CH=C(Cl)-CH₃, -C(CH₃)=N-O-CO-CH₃, -C(CH₃)=N-O-CO-C₂H₅, -C(CH₃)=N-OCH₂-CN, -C(CH₃)=N-OCH₂-CH=CH-CH₂-OCH₃, -C(CH₃)=N-OCH₂-CH=CH-CH₂-O-tert.-C₄H₉, -C(CH₃)=N-O-(CH₂)₃-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-(4-Cl-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-C₆H₅, -C(CH₃)=N-OCH₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(3-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-CH₂-(4-CH₃O-C₆H₄), -C(CH₃)=N-OCH₂-CH=C(CH₃)-C₆H₅, -C(CH₃)=N-O-(CH₂)₂-CH=CH-(3,4-Cl₂-C₆H₃), -C(CH₃)=N-O-(CH₂)₃-C≡-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-OCH₃, -C(CH₃)=N-OCH₂CH₂-OCH₃, -C(CH₃)=N-OCH₂-OC₂H₅, -C(CH₃)=N-OCH(CH₃)-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=N-NH₂, -C(CH₃)=N-NH-CH₃, -C(CH₃)=N-NH-C₂H₅, -C(CH₃)=N-NH-n-C₃H₇, -C(CH₃)=N-NH-i-C₃H₇, -C(CH₃)=N-NH-n-C₄H₉, -C(CH₃)=N-NH-i-C₄H₉, -C(CH₃)=N-NH-s-C₄H₉, -C(CH₃)=N-NH-tert.-C₄H₉, -C(CH₃)=N-NH-cyclopropyl, -C(CH₃)=N-NH-cyclobutyl, -C(CH₃)=N-NH-cyclopentyl, -C(CH₃)=N-NH-cyclohexyl, -C(CH₃)=N-NH-cycloheptyl, -C(CH₃)=N-N(CH₃)₂, -C(CH₃)=N-N(C₂H₅)₂, -C(CH₃)=N-N(n-C₃H₇)₂, -C(CH₃)=N-N(i-C₃H₇)₂, -C(CH₃)=N-NH-CH₂-C=CH, -C(CH₃)=N-NH-CH₂-C≡CH, -C(CH₃)=N-N(CH₃)-CH₂-C≡CH, -C(CH₃)=N-NH-CH₂CF₃, -C(CH₃)=N-NH-CO-CH₃, -C(CH₃)=N-NH-CO-C₂H₅, -C(CH₃)=N-NH-CO-OCH₃, -C(CH₃)=N-NH-CO-OC₂H₅, -C(CH₃)=N-NH-CO-O-tert.-C₄H₉, -C(CH₃)=N-pyrrolidin-1-yl, -C(CH₃)=N-piperidin-1-yl, -C(CH₃)=N-morpholin-4 99999 00070 552 001000280000000200012000285919988800040 0002004131038 00004 99880-yl, -C(CH₃)=N-NH-C₆H₅, -C(CH₃)=N-NH-(4-Cl-C₆H₄), -C(CH₃)=N-NH-(4-NO₂-C₆H₄), -C(CH₃)=N-NH-(4-F-C₆H₄), -C(CH₃)=N-NH-(4-CH₃O-C₆H₄), -C(CH₃)=N-NH-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-NH-(2,4-(NO₂)₂-C₆H₃), -C(CH₃)=N-NH-CO-NH₂, -C(CH₃)=N-NH-CO-NHCH₃, -C(CH₃)=N-NH-CO-NHC₂H₅, -C(CH₃)=N-NH-CO-N(CH₃)₂, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=CH-CO-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -(CH₃)=CH-CO-O-n-C₄H₉, -C(CH₃)=CH-CO-O-tert.-C₄H₉, -C(CH₃)=CH-CO-O-cyclopropyl, -C(CH₃)=CH-CO-O-cyclobutyl, -C(CH₃)=CH-CO-O-cyclopentyl, -C(CH₃)=CH-CO-O-cyclohexyl, -C(CH₃)=CH-CO-O-cycloheptyl, -C(CH₃)=C(CH₃)-COOH, -C(CH₃)=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-cyclopropyl, -C(CH₃)=C(CH₃)-CO-O-cyclobutyl, -C(CH₃)=C(CH₃)-CO-O-cyclopentyl, -C(CH₃)=C(CH₃)-CO-O-cyclohexyl, -C(CH₃)=C(CH₃)-CO-O-cycloheptyl, -C(CH₃)=C(C₂H₅)-COOH, -C(CH₃)=C(C₂H₅)-CO-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-cyclo­ propyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-O- cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-O-cycloheptyl, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-O-n-C₄H₉, -C(CH₃)=C(Cl)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-O-cyclopropyl, -C(CH₃)=C(Cl)-CO-O-cyclobutyl, -C(CH₃)=C(Cl)-CO-O-cyclopentyl, -C(CH₃)=C(Cl)-CO-O-cyclohexyl, -C(CH₃)=C(Cl)-CO-O-cycloheptyl, -C(CH₃)=C(Br)-COOH, -C(CH₃)=C(Br)-CO-OCH₃, -C(CH₃)=C(Br)-CO-OC₂H₅, -C(CH₃)=C(Br)-CO-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-O-n-C₄H₉, -C(CH₃)=C(Br)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-O-cyclopropyl, -C(CH₃)=C(Br)-CO-O-cyclobutyl, -C(CH₃)=C(Br)-CO-O-cyclopentyl, -C(CH₃)=C(Br)-CO-O-cyclohexyl, -C(CH₃)=C(Br)-CO-O-cycloheptyl, -C(CH₃)=C(CN)-COOH, -C(CH₃)=C(CN)-CO-OCH₃, -C(CH₃)=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CN)-CO-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-O-n-C₄H₉, -C(CH₃)=C(CN)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-O-cyclopropyl, -C(CH₃)=C(CN)-CO-O-cyclobutyl, -C(CH₃)=C(CN)-CO-O-cyclopentyl, -C(CH₃)=C(CN)-CO-O-cyclohexyl, -C(CH₃)=C(CN)-CO-O-cycloheptyl, -C(CH₃)=CH-CO-OCH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-OCH(CH₃)-OCH₃, -C(CH₃)=CH-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=CH-CO-OCH₂CH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=(C₂H₅)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-O-i-C₃H₇, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -(CH₃)=C(Cl)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-O-i-C₃H₇, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-O-i-C₃H₇, -C(CH₃)=C(CN)-CO-OCH(CH₃)OCH₃, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-CF₃, -C(CH₃)=CH-CO-OCH₂-CCl₃, -C(CH₃)=CH-CO-OCH₂-oxiranyl, -C(CH₃)=CH-CO-(CH₂)₃-Br, -C(CH₃)=CH-CO-OCH₂-CH=CH₂, -C(CH₃)=CH-CO-OCH₂-C≡CH, -C(CH₃)=CH-CO-OCH₂-CN, -C(CH₃)=CH-CO-OCH₂CH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CF₃, -C(CH₃)=C(CH₃)-CO-OCH₂-CCl₃, -C(CH₃)=C(CH₃)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CH₃)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CH₃)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CH₃)-CO-OCH₂-C≡CH, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CF₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CCl₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-oxiranyl, -C(CH₃)=C(C₂H₅)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(C₂H₅)CO-OCH₂-C≡CH, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂-CF₃, -C(CH₃)=C(Cl)-CO-OCH₂-CCl₃, -C(CH₃)=C(Cl)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Cl)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Cl)-CO-OCH₂-CH≡CH₂, -C(CH₃)=C(Cl)-CO-OCH₂-C≡CH, -C(CH₃)=C(Cl)-CO-OCH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂-CF₃, -C(CH₃)=C(Br)-CO-OCH₂-CCl₃, -C(CH₃)=C(Br)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Br)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Br)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Br)-CO-OCH₂-C≡CH, -C(CH₃)=C(Br)-CO-OCH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂CH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂-CF₃, -C(CH₃)=C(CN)-CO-OCH₂-CCl₃, -C(CH₃)=C(CN)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CN)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CN)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CN)-CO-OCH₂-C≡CH, -C(CH₃)=C(CN)-CO-OCH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂CH₂-CN, -C(CH₃)=CH-CO-CH₃, -C(CH₃)=CH-CO-C₂H₅, -C(CH₃)=CH-CO-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-n-C₄H₉, -C(CH₃)=CH-CO-tert.-C₄H₉, -C(CH₃)=CH-CO-CH₂Cl, -C(CH₃)=CH-CO-CH₂Br, -C(CH₃)=CH-CO-CHCl₂, -C(CH₃)=CH-CO-CH₂-OCH₃, -C(CH₃)=CH-CO-CH(OCH₃)₂, -C(CH₃)=CH-CO-CH₂-SCH₃, -C(CH₃)=C(CH₃)-CO-CH₃, -C(CH₃)=C(CH₃)-CO-C₂H₅, -C(CH₃)=C(CH₃)-CO-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-CH₂Cl, -C(CH₃)=C(CH₃)-CO-CH₂Br, -C(CH₃)=C(CH₃)-CO-CHCl₂, -C(CH₃)=C(CH₃)-CO-CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-CH(OCH₃)₂, -C(CH₃)=C(CH₃)-CO-CH₂-SCH₃, -C(CH₃)=C(C₂H₅)-CO-CH₃, -C(CH₃)=C(C₂H₅)-CO-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-CH₂Cl, -C(CH₃)=C(C₂H₅)-CO-CH₂Br, -C(CH₃)=C(C₂H₅)-CO-CHCl₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-CH(OCH₃)₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-SCH₃, -C(CH₃)=C(Cl)-CO-CH₃, -C(CH₃)=C(Cl)-CO-C₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-n-C₄H₉, -C(CH₃)=C(Cl)-CO-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-CH₂Cl, -C(CH₃)=C(Cl)-CO-CHCl₂, -C(CH₃)=C(Cl)-CO-CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-CH(OCH₃)₂, -C(CH₃)=C(Cl)-CO-CH₂-SCH₃, -C(CH₃)=C(Br)-CO-CH₃, -C(CH₃)=C(Br)-CO-C₂H₅, -C(CH₃)=C(Br)-CO-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-n-C₄H₉, -C(CH₃)=C(Br)-CO-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-CH₂Cl, -C(CH₃)=C(Br)-CO-CH₂Br, -C(CH₃)=C(Br)-CO-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-CH(OCH₃)₂, -C(CH₃)=C(Br)-CO-CH₂-SCH₃, -C(CH₃)=C(CN)-CO-CH₃, -C(CH₃)=C(CN)-CO-C₂H₅, -C(CH₃)=C(CN)-CO-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-n-C₄H₉, -C(CH₃)=C(CN)-CO-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-CH₂Cl, -C(CH₃)=C(CN)-CO-CH₂Br, -C(CH₃)=C(CN)-CO-CHCl₂, -C(CH₃)=C(CN)-CO-CH₂-OCH₃, -C(CH₃)=C(CN)-CO-CH(OCH₃)₂, -C(CH₃)=C(CN)-CO-CH₂-SCH₃, -C(CH₃)=CH-CO-C₆H₅, -C(CH₃)=CH-CO-(4-Cl-C₆H₄), -C(CH₃)=C(CH₃)-CO-C₆H₅, -C(CH₃)=C(CH₃)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(C₂H₅)-CO-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(Cl)-CO-C₆H₅, -C(CH₃)=C(Br)-CO-C₆H₅, -C(CH₃)=C(CN)-CO-C₆H₅, -C(CH₃)=CH-CO-NH₂, -C(CH₃)=CH-CO-NHCH₃, -C(CH₃)=CH-CO-N(CH₃)₂, -C(CH₃)=CH-CO-NH-C₂H₅, -C(CH₃)=CH-CO-N(C₂H₅)₂, -C(CH₃)=CH-CO-NH-n-C₃H₇, -C(CH₃)=CH-CO-NH-i-C₃H₇, -C(CH₃)=CH-CO-NH-tert.-C₄H₉, -C(CH₃)=CH-CO-NH-cyclopropyl, -C(CH₃)=CH-CO-NH-cyclobutyl, -C(CH₃)=CH-CO-NH-cyclopentyl, -C(CH₃)=CH-CO-NH-cyclohexyl, -C(CH₃)=CH-CO-NH-cycloheptyl, -C(CH₃)=CH-CO-NH-cyclooctyl, -C(CH₃)=CH-CO-pyrrolidin-1-yl, -C(CH₃)=CH-CO-piperidin-1-yl, -C(CH₃)=CH-CO-morpholin-4-yl, -C(CH₃)=CH-CO-NH-CH₂CH=CH₂, -C(CH₃)=CH-CO-NH-CH₂C≡CH, -C(CH₃)=CH-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=CH-CO-NH-(CH₂)₂Cl, -C(CH₃)=CH-CO-NH-C₆H₅, -C(CH₃)=C(CH₃)-CO-NH₂, -C(CH₃)=C(CH₃)-CO-NHCH₃, -C(CH₃)=C(CH₃)-CO-N(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-C₂H₅, -C(CH₃)=C(CH₃)-CO-N(C₂H₅)₂, -C(CH₃)=C(CH₃)-CO-NH-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-NH- cyclopropyl, -C(CH₃)=C(CH₃)-CO-NH-cyclobutyl, -C(CH₃)=C(CH₃)-CO-NH-cyclopentyl, -C(CH₃)=C(CH₃)-CO-NH- cyclohexyl, -C(CH₃)=C(CH₃)-CO-NH-cycloheptyl, -C(CH₃)=C(CH₃)-CO-NH-cyclooctyl, -C(CH₃)=C(CH₃)-CO- pyrrolidin-1-yl, -C(CH₃)=C(CH₃)-CO-piperidin-1-yl, -C(CH₃)=C(CH₃)-CO-morpholin-4-yl, -C(CH₃)=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-NH(CH₂)₂Cl, -C(CH₃)=C(CH₃)-CO-NH-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-NH₂, -C(CH₃)=C(C₂H₅)-CO-NHCH₃, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)₂, -C(CH₃)=C(C₂H₅)-CO-NH-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-N(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-NH- cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-NH-cycloheptyl, -C(CH₃)=C(C₂H₅)-CO-NH- cyclooctyl, -C(CH₃)=C(C₂H₅)-CO-pyrrolidin-1-yl, -C(CH₃)=C(C₂H₅)-CO-piperidin-1-yl, -C(CH₃)=C(C₂H₅)-CO- morpholin-4-yl, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(C₂H₅)-CO-NH-C₆H₅, -C(CH₃)=C(Cl)-CO-NH₂, -C(CH₃)=C(CH₃)=C(Cl)-CO-NHCH₃, -C(CH₃)=C(Cl)-CO-N(CH₃)₂, -C(CH₃)=C(Cl)-CO-NH-C₂H₅, -C(CH₃)=C(Cl)-CO-N(C₂H₅)₂, -C(CH₃)=C(Cl)-CO-NH-n-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-i-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-NH-cyclopropyl, -C(CH₃)=C(Cl)-CO-NH-cyclobutyl, -C(CH₃)=C(Cl)-CO-NH-cyclopentyl, -C(CH₃)=C(Cl)-CO-NH-cyclohexyl, -C(CH₃)=C(Cl)-CO-NH-cycloheptyl, -C(CH₃)=C(Cl)-CO-NH-cyclooctyl, -C(CH₃)=C(Cl)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Cl)-CO-piperidin-1- yl, -C(CH₃)=C(Cl)-CO-morpholin-4-yl, -C(CH₃)=C(Cl)-CO-NH-CH₂CH=C(Cl)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-N(CH₃)-CH₂≡CH, -C(CH₃)=C(Cl)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Cl)-NO-NH-C₆H₅, -C(CH₃)=C(Br)-CO-NH₂, -C(CH₃)=C(Br)-CO-NHCH₃, -C(CH₃)=C(Br)-CO-N(CH₃)₂, -C(CH₃)=C(Br)-CO-NH-C₂H₅, -C(CH₃)=C(Br)-CO-N(C₂H₅)₂, -C(CH₃)=C(Br)-CO-NH-n-C₃H₇, -C(CH₃)=C(Br)-CO-NH-i-C₃H₇, -C(CH₃)=C(Br)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-NH-cyclopropyl, -C(CH₃)=C(Br)-CO-NH-cyclobutyl, -C(CH₃)=C(Br)-CO-NH-cyclopentyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cycloheptyl, -C(CH₃)=C(Br)-CO-NH-cyclooctyl, -C(CH₃)=C(Br)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Br)-CO-piperidin-1-yl, -C(CH₃)=C(Br)-CO-morpholin-4-yl, -C(CH₃)=C(Br)-CO-NH-CH₂CH=C(CH₃)=C(Br)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Br)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Br)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Br)-CO-NH-C₆H₅, -C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CN)-CO-NHCH₃, -C(CH₃)=C(CN)-CO-N(CH₃)₂, -C(CH₃)=C(CN)-CO-NH-C₂H₅, -C(CH₃)=C(CN)-CO-N(C₂H₅)₂, -C(CH₃)=C(CN)-CO-NH-n-C₃H₇, -C(CH₃)=C(CN)-CO-NH-i-C₃H₇, -C(CH₃)=C(CN)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-NH-cyclopropyl, -C(CH₃)=C(CN)-CO-NH-cyclobutyl, -C(CH₃)=C(CN)-CO-NH-cyclopentyl, -C(CH₃)=C(CN)-CO-NH-cyclohexyl, -C(CH₃)=C(CN)-CO-NH-cycloheptyl, -C(CH₃)=C(CN)-CO-NH-cyclooctyl, -C(CH₃)=C(CN)-CO-pyrrolidin-1-yl, -C(CH₃)=C(CN)-CO-piperidin-1-yl, -C(CH₃)=C(CN)-CO-morpholin-4-yl, -C(CH₃)=C(CN)-CO-NH-CH₂CH=C(CN)₂, -C(CH₃)=C(CN)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CN)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)=(CN)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CN)-CO-NH-C₆H₅, -C(CH₃)=CH-SO-SCH₃, -C(CH₃)=CH-CO-SC₂H₅, -C(CH₃)=CH-CO-S-n-C₃H₇, -C(CH₃)=CH-CO-S-i-C₃H₇, -C(CH₃)=CH-CO-S-n-C₄H₉, -C(CH₃)=CH-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-SCH₃, -C(CH₃)=C(CH₃)-CO-SC₂H₅, -C(CH₃)=C(CH₃)CO-S-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-S-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-SCH₃, -C(CH₃)=C(C₂H₅)-CO-SC₂H₅, -C(CH₃)=C(C₂H₅)-CO-S-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-SCH₃, -C(CH₃)=C(Cl)-CO-SC₂H₅, -C(CH₃)=C(Cl)-CO-S-n-C₃H₇, -C(CH₃)=C(Cl)-CO-S-i-C₃H₇, -C(CH₃)=C(Cl)-CO-S-n-C₄H₉, -C(CH₃)=C(Cl)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-SCH₃, -C(CH₃)=C(Br)-CO-SC₂H₅, -C(CH₃)=C(Br)-CO-S-n-C₃H₇, -C(CH₃)=C(Br)-CO-S-i-C₃H₇, -C(CH₃)=C(Br)-CO-S-n-C₄H₉, -C(CH₃)=C(Br)-CO-S-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-SCH₃, -C(CH₃)=C(CN)-CO-SC₂H₅, -C(CH₃)=C(CN)-CO-S-n-C₃H₇, -C(CH₃)=C(CN)-CO-S-i-C₃H₇, -C(CH₃)=C(CN)-CO-S-N-C₄H₉, -C(CH₃)=C(CN)-CO-S-tert.-C₄H₉, -C(CH₃)=C(COCH₃)-CO-OCH₃, -C(CH₃)=C(COC₂H₅)-CO-OCH₃, -C(CH₃)=C(CO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COCH₃)-CO-OC₂H₅, -C(CH₃)=C(COC₂H₅)-CO-OC₂H₅, -C(CH₃)=C(CO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COCH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(COC₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-OCH₃, -C(CH₃)=C(CF₃)-CO-OC₂H₅, -C(CH₃)=C(CF₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CF₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(COOCH₃)₂, -C(CH₃)=C(COOC₂H₅)₂, -C(CH₃)=C(COOCH₃)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)₂, -C(CH₃)=CH-CH=CH-COOH, -C(CH₃)=CH-CH=CH-CO-OCH₃, -C(CH₃)=CH-CH=CH-CO-OC₂H₅, -C(CH₃)=CH-CH=C(COOCH₃)₂, -C(CH₃)=CH-CH=C(CN)-CO-OCH₃, -C(CH₃)=CH-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH₂, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -C(CH₃)=CH-(CH₂)₂-COOH, -C(CH₃)=CH-(CH₂)₂-CO-OCH₃, -C(CH₃)=CH-(CH₂)₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(COOCH₃)₂, -C(CH₃)=CH-CH₂-CH(COOC₂H₅)₂, -C(CH₃)=CH-CH₂-CH(CN)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CN)-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -C(CH₃)=CH-(CH₂)₂-CO-NH₂, -C(CH₃)=CH-(CH₂)₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-COOH, -C(CH₃)=CH-CH₂-CO-OCH₃, -C(CH₃)=CH-CH₂-CO-OC₂H₅, -C(CH₃)=C(COOCH₃)-CH₂-CO-OCH₃, -C(CH₃)=C(COOCH₃)-CH₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CO-NH₂, -C(CH₃)=CH-CH₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-CO-N(CH₃)₂.
wobei W für eine der folgenden Bedeutungen steht:
-CHO, -COCH₃, -COC₂H₅, -CO-n-C₃H₇, -CO-i-C₃H₇, -CO-n-C₄H₉, -CO-i-C₄H₉, -CO-s-C₄H₉, -CO-tert.-C₄H₉, -CO-CH₂CH=CH₂, -CO-CF₃, -COCCl₃, -COCH₂C≡CH, -CO-cyclopropyl, -CO-cyclobutyl, -CO-cyclopentyl, -CO-cyclohexyl, -CO-CN, -CO-COOCH₃, -CO-COOC₂H₅, -CH=NH, -CH=NCH₃, -CH=NC₂H₅, -CH=N-n-C₃H₅, -CH=N-i-C₃H₅, -CH=N-n-C₄H₉, -CH=NCH₂CH=CH₂, -CH=NCH₂CH=CH₂-CH₃, -CH=NCH₂C≡CH, -CH=NCH₂C≡C-CH₃, -CH=N-cyclopropyl, -CH=N-cyclobutyl, -CH=N-cyclopentyl, -CH=N-cyclohexyl, -CH=N-cycloheptyl, -CH=N-CH₂-CH₂Cl, -CH=N-CH₂Cl, -CH=N-C₆H₅, -CH=N-4-Br-C₆H₄, -CH=N-3-F-C₆H₄, -CH=N-4-F-C₆H₄, -CH=N-2-Cl-C₆H₄, -CH=N-3-Cl-C₆H₄, -CH=N-4-Cl-C₆H₄, -CH=N-2-Br-C₆H₄, -CH=N-2-F-C₆H₄, -CH=N-2-CH₃-C₆H₄, -CH=N-3-CH₃-C₆H₄, -CH=N-4-CH₃-C₆H₄, -CH=N-2-CF₃-C₆H₄, -CH=N-3-CF₃-C₆H₄, -CH=N-4-CF₃-C₆H₄, -CH=N-2-OCH₃-C₆H₄, -CH=N-3-OCH₃-C₆H₄, -CH=N-4-OCH₃-C₆H₄, -CH=N-4-NO₂-C₆H₄, -CH=N-4-CN-C₆H₄, -CH=N-2,4-(Cl,Cl)-C₆H₄, -CH=N-2,4-(CH₃,CH₃)-C₆H₄, -CH=N-CH₂OCH₃ -CH=N-CH₂OC₂H₅, -CH=N-CH₂CH₂OCH₃, -CH=N-CH₂CH₂OC₂H₅, -CH=N-OH, -CH=N-OCH₃, -CH=N-OC₂H₅, -CH=N-O-n-C₃H₇, -CH=N-O-i-C₃H₇, -CH=N-O-n-C₄H₉, -CH=N-O-i-C₄H₉, -CH=N-O-s-C₄H₉, -CH=N-O-tert.-C₄H₉, -CH=N-O-CH₂CH=CH₂, -CH=N-O-CH(CH₃)CH=CH₂, -CH=N-O-CH₂C≡CH, -CH=N-O-CH(CH₃)-C≡CH, -CH=N-O-CH₂-CH=CH-CH₃, -CH=N-O-CH₂-CH₂-Cl, -CH=N-O-CH₂-CH₂-F, -CH=N-O-CH₂-CF₃, -CH=N-O-CH₂-CH=CHCl, -CH=N-O-CH₂-CCl=CH₂, -CH=N-O-CH₂-CBr=CH₂, -CH=N-O-CH₂-CH=CCl-CH₃, -CH=N-OC(O)CH₃, -CH=N-OC(O)C₂H₅, -CH=N-O-CH₂-CN, -CH=N-O-CH₂-CH=CH-CH₂-O-CH₃, -CH=N-O-CH₂-CH=CH-CH₂-O-tert.-C₄H₉, -CH=N-O-(CH₂)₃-C₆H₅, -CH=N-O-(CH₂)₄-C₆H₅, -CH=N-O-(CH₂)₄-4-Cl-C₆H₄, -CH=N-O-(CH₂)₄-4-OCH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-CH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-C₆H₅, -CH=N-O-CH₂CH=CH-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CH-3-OCH₃-C₆H₄, -CH=N-O-(CH₂)₂CH=CH-4-F-C₆H₄, -CH=N-O-(CH₂)CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CHCH₂-4-OCH₃-C₆H₄, -CH=N-O-CH₂-CH=C(CH₃)-C₆H₅, -CH=N-O-(CH₂)₂CH=CH-3,4(Cl,Cl)-C₆H₃, -CH=N-O-(CH₂)₃C≡C-4-F-C₆H₄, -CH₂=N-OCHOCH₃, -CH=N-OC₂H₄OCH₃, -CH=N-OCH₂OC₂H₅, -CH=N-OCH(CH₃)OCH₃, -CH=N-OCH(CH₃)COOCH₃, -CH=N-OCH(CH₃)COO-n-C₄H₉, -CH=N-NH₂, -CH=N-NHCH₃, -CH=N-NHC₂H₅, -CH=N-NH-n-C₃H₇, -CH=N-NH-i-C₃H₇, -CH=N-NH-n-C₄H₉, -CH=N-NH-i-C₄H₉, -CH=N-NH-s-C₄H₉, -CH=N-NH-tert.-C₄H₉, -CH=N-NH-cyclopropyl, -CH=N-NH-cyclobutyl, -CH=N-NH-cyclopentyl, -CH=N-NH-cyclohexyl, -CH=N-NH-cycloheptyl, -CH=N-N(CH₃)₂, -CH=N-N(C₂H₅)₂, -CH=N-N(C₃H₇)₂, -CH=N-N(i-C₃H₇)(CH₃), -CH=N-NHCH₂-C=CH, -CH=N-NHCH₂-C≡CH, -CH=N-N(CH₃)-CH₂-C≡CH, -CH=N-NHCH₂CF₃, -CH=N-NH-CO-CH₃, -CH=N-NH-CO-CH₂H₅, -CH=N-NH-COOCH₃, -CH=N-NH-COOC₂H₅, -CH=N-NH-COO-tert.-C₄H₉, -CH=N-pyrrolidin-1-yl, -CH=N-piperidin-1-yl, -CH=N-morpholin-4-yl, -CH=N-NH-C₆H₅, -CH=N-NH-(4-Cl-C₆H₄), -CH=N-NH-(4-NO₂-C₆H₄), -CH=N-NH-(4-F-C₆H₄), -CH=N-NH-(4-CH₃O-C₆H₄), -CH=N-NH-(2,4-Cl₂-C₆H₃), -CH=N-NH-(2,4-(NO₂)₂-C₆H₃), -CH=N-NH-CO-NH₂, -CH=N-NH-CO-NHCH₃, -CH=N-NH-CO-NHC₂H₅, -CH=N-NH-CO-N(CH₃)₂, -CH=CH-COOH, -CH=CH-CO-OCH₃, -CH=C-CO-OC₂H₅, -CH=CH-CO-O-n-C₃H₇, -CH=CH-CO-O-i-C₃H₇, -CH=CH-CO-O-n-C₄H₉, -CH=CH-CO-O-tert.-C₄H₉, -CH=CH-CO-O-cyclopropyl, -CH=CH-CO-O-cyclobutyl, -CH=CH-CO-O-cyclopentyl, -CH=CH-CO-O-cyclohexyl, -CH=CH-CO-O-cycloheptyl, -CH=C(CH₃)-COOH, -CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CO-O-n-C₃H₇, -CH=C(CH₃)-CO-O-i-C₃H₇, -CH=C(CH₃)-CO-O-n-C₄H₉, -CH=C(CH₃)-CO-O-tert.-C₄H₉, -CH=C(CH₃)-CO-O-cyclopropyl, -CH=C(CH₃)-CO-O-cyclobutyl, -CH=C(CH₃)-CO-O-cyclopentyl, -CH=CH-CO-O-cyclopentyl, -CH=CH-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cycloheptyl, -CH=C(C₂H₅)-COOH, -CH=C(C₂H₅)-CO-OCH₃, -CH=C(C₂H₅)-CO-OC₂H₅, -CH=C(C₂H₅)-CO-O-n-C₃H₇, -CH=C(C₂H₅)-CO-O-i-C₃H₇, -CH=C(C₂H₅)-CO-O-n-C₄H₉, -CH=C(C₂H₅)-CO-O-tert.-C₄H₉, -CH=C(C₂H₅)-CO-O-cyclopropyl, -CH=C(C₂H₅)-CO-O-cyclobutyl, -CH=C(C₂H₅)-CO-O-cyclopentyl, -CH=C(C₂H₅)-CO-O-cyclohexyl, -CH=C(C₂H₅)-CO-O-cycloheptyl, -CH=C(Cl)-COOH, -CH=C(Cl)-CO-OCH₃, -CH=C(Cl)-CO-OC₂H₅, -CH=C(Cl)-CO-O-n-C₃H₇, -CH=C(Cl)-CO-O-i-C₃H₇, -CH=C(Cl)-CO-O-n-C₄H₉, -CH=C(Cl)-CO-O-tert.-C₄H₉, -CH=C(Cl)-CO-O-cyclopropyl, -CH=C(Cl)-CO-O-cyclobutyl, -CH=C(Cl)-CO-O-cyclopentyl, -CH=C(Cl)-CO-O-cyclohexyl, -CH=C(Cl)-CO-O-cycloheptyl, -CH=C(Br)-COOH, -CH=C(Br)-CO-OCH₃, -CH=C(Br)-CO-OC₂H₅, -CH=C(Br)-CO-O-n-C₃H₇, -CH=C(Br)-CO-O-i-C₃H₇, -CH=C(Br)-CO-O-n-C₄H₉, -CH=C(Br)-CO-O-tert.-C₄H₉, -CH=C(Br)-CO-O-cyclopropyl, -CH=C(Br)-CO-O-cyclobutyl, -CH=C(Br)-CO-O-cyclopentyl, -CH=C(Br)-CO-O-cyclohexyl, -CH=C(Br)-CO-O-cycloheptyl, -CH=C(CN)-COOH, -CH=C(CN)-CO-OCH₃, -CH=C(CN)-CO-OC₂H₅, -CH=C(CN)-CO-O-n-C₃H₇, -CH=C(CN)-CO-O-i-C₃H₇, -CH=C(CN)-CO-O-n-C₄H₉, -CH=C(CN)-CO-O-tert.-C₄H₉, -CH=C(CN)-CO-O-cyclopropyl, -CH=C(CN)-CO-O-cyclobutyl, -CH=C(CN)-CO-O-cyclopentyl, -CH=C(CN)-CO-O-cyclohexyl, -CH=C(CN)-CO-O-cycloheptyl, -CH=CH-CO-OCH₂-OCH₃, -CH=CH-CO-OCH₂-OC₂H₅, -CH=CH-CO-OCH₂-O-n-C₃H₅, -CH=CH-CO-OCH₂-O-i-C₃H₅, -CH=CH-CO-OCH(CH₃)-OCH₃, -CH=CH-CO-OCH(CH₃)-OC₂H₅, -CH=CH-CO-O-CH₂CH₂-OCH₃, -CH=CH-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-OCH₃, -CH=C(CH₃)-CO-OCH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-O-n-C₃H₅, -CH=C(CH₃)-CO-OCH₂-O-i-C₃H₅, -CH=C(CH₃)-CO-OCH(CH₃)-OCH₃, -CH=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CH₃)-CO-O-CH₂CH₂-OCH₃, -CH=C(CH₃)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-OCH₃, -CH=C(C₂H₅)-CO-OCH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-O-n-C₃H₅, -CH=C(C₂H₅)-CO-OCH₂-O-i-C₃H₅, -CH=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -CH=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OCH₃, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-OCH₃, -CH=C(Cl)-CO-OCH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-O-n-C₃H₅, -CH=C(Cl)-CO-OCH₂-O-i-C₃H₅, -CH=C(Cl)-CO-OCH(CH₃)-OCH₃, -CH=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Cl)-CO-O-CH₂CH₂-OCH₃, -CH=C(Cl)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-OCH₃, -CH=C(Br)-CO-OCH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-O-n-C₃H₅, -CH=C(Br)-CO-OCH₂-O-i-C₃H₅, -CH=C(Br)-CO-OCH(CH₃)-OCH₃, -CH=C(Br)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Br)-CO-O-CH₂CH₂-OCH₃, -CH=C(Br)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-OCH₃, -CH=C(CN)-CO-OCH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-O-n-C₃H₅, -CH=C(CN)-CO-OCH₂-O-i-C₃H₅, -CH=C(CN)-CO-OCH(CH₃)-OCH₃, -CH=C(CN)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CN)-CO-O-CH₂CH₂-OCH₃, -CH=C(CN)-CO-O-CH₂CH₂-OC₂H₅, -CH=CH-CO-OCH₂-CF₃, -CH=CH-CO-OCH₂-CCl₃, -CH=CH-CO-OCH₂-oxiranyl, -CH=CH-CO-O(CH₂)₃-Br, -CH=CH-CO-OCH₂-CH=CH₂, -CH=CH-CO-OCH₂-C≡CH, -CH=CH-CO-OCH₂-CN, -CH=CH-CO-O(CH₂)₂-CN, -CH=C(CH₃)-CO-OCH₂-CF₃, -CH=C(CH₃)-CO-OCH₂-CCl₃, -CH=C(CH₃)-CO-OCH₂-oxiranyl, -CH=C(CH₃)-CO-O(CH₂)₃-Br, -CH=C(CH₃)-CO-OCH₂-CH=CH₂, -CH=C(CH₃)-CO-OCH₂-C≡CH, -CH=C(CH₃)-CO-OCH₂-CN, -CH=C(CH₃)-CO-O(CH₂)₂-CN, -CH=C(C₂H₅)-CO-OCH₂-CF₃, -CH=C(C₂H₅)-CO-OCH₂-CCl₃, -CH=C(C₂H₅)-CO-OCH₂-oxiranyl, -CH=C(C₂H₅)-CO-O(CH₂)₃-Br, -CH=C(C₂H₅)-CO-OCH₂-CH=CH₂, -CH=C(C₂H₅)-CO-OCH₂-C≡CH, -CH=C(C₂H₅)-CO-OCH₂-CN, -CH=C(C₂H₅)-CO-O(CH₂)₂-CN, -CH=C(Cl)-CO-OCH₂-CF₃, -CH=C(Cl)-CO-OCH₂-CCl₃, -CH=C(Cl)-CO-OCH₂-oxiranyl, -CH=C(Cl)-CO-O(CH₂)₃-Br, -CH=C(Cl)-CO-OCH₂-CH=CH₂, -CH=C(Cl)-CO-OCH₂-C≡CH, -CH=C(Cl)-CO-OCH₂-CN, -CH=C(Cl)-CO-O(CH₂)₂-CN, -CH=C(Br)-CO-OCH₂-CF₃, -CH=C(Br)-CO-OCH₂-CCl₃, -CH=C(Br)-CO-OCH₂-oxiranyl, -CH=C(Br)-CO-O(CH₂)₃-Br, -CH=C(Br)-CO-OCH₂-CH=CH₂, -CH=C(Br)-CO-OCH₂-C≡CH, -CH=C(Br)-CO-OCH₂-CN, -CH=C(Br)-CO-O(CH₂)₂-CN, -CH=C(CN)-CO-OCH₂-CF₃, -CH=C(CN)-CO-OCH₂-CCl₃, -CH=C(CN)-CO-OCH₂-oxiranyl -CH=C(CN)-CO-O(CH₂)₃-Br, -CH=C(CN)-CO-OCH₂-CH=CH₂, -CH=C(CN)-CO-OCH₂-C≡CH, -CH=C(CN)-CO-OCH₂-CN, -CH=C(CN)-CO-O(CH₂)₂-CN, -CH=CH-CO-CH₃, -CH=CH-CO-C₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-i-C₃H₇, -CH=CH-CO-n-C₄H₉, -CH=CH-CO-tert.-C₄H₉, -CH=CH-CO-CH₂Cl, -CH=CH-CO-CH₂Br, -CH=CH-CO-CHCl₂, -CH=CH-CO-CH₂-OCH₃, -CH=CH-CO-CH(OCH₃)₂, -CH=CH-CO-CH₂-SCH₃, -CH=C(CH₃)-CO-CH₃, -CH=C(CH₃)-CO-C₂H₅, -CH=C(CH₃)-CO-n-C₃H₇, -CH=C(CH₃)-CO-i-C₃H₇, -CH=C(CH₃)-CO-n-C₄H₉, -CH=C(CH₃)-CO-tert.-C₄H₉, -CH=C(CH₃)-CO-CH₂Cl, -CH=C(CH₃)-CO-CH₂Br, -CH=C(CH₃)-CO-CHCl₂, -CH=C(CH₃)-CO-CH₂-OCH₃, -CH=C(CH₃)-CO-CH(OCH₃)₂, -CH=C(CH₃)-CO-CH₂-SCH₃, -CH=C(C₂H₅)-CO-CH₃, -CH=C(C₂H₅)-CO-C₂H₅, -CH=C(C₂H₅)-CO-n-C₃H₇, -CH=C(C₂H₅)-CO-i-C₃H₇, -CH=C(C₂H₅)-CO-n-C₄H₉, -CH=C(C₂H₅)-CO-tert.-C₄H₉, -CH=C(C₂H₅)-CO-CH₂Cl, -CH=C(C₂H₅)-CO-CH₂Br, -CH=C(C₂H₅)-CO-CHCl₂, -CH=C(C₂H₅)-CO-CH₂-OCH₃, -CH=C(C₂H₅)-CO-CH(OCH₃)₂, -CH=C(C₂H₅)-CO-CH₂-SCH₃, -CH=C(Cl)-CO-CH₃, -CH=C(Cl)-CO-C₂H₅, -CH=C(Cl)-CO-n-C₃H₇, -CH=C(Cl)-CO-i-C₃H₇, -CH=C(Cl)-CO-n-C₄H₉, -CH=C(Cl)-CO-tert.-C₄H₉, -CH=C(Cl)-CO-CH₂Cl, -CH=C(Cl)-CO-CH₂Br, -CH=C(Cl)-CO-CHCl₂, -CH=C(Cl)-CO-CH₂-OCH₃, -CH=C(Cl)-CO-CH(OCH₃)₂, -CH=C(Cl)-CO-CH₂-SCH₃, -CH=C(Br)-CO-CH₃, -CH=C(Br)-CO-C₂H₅, -CH=C(Br)-CO-n-C₃H₇, -CH=C(Br)-CO-i-C₃H₇, -CH=C(Br)-CO-n-C₄H₉, -CH=C(Br)-CO-tert.-C₄H₉, -CH=C(Br)-CO-CH₂Cl, -CH=C(Br)-CO-CH₂Br, -CH=C(Br)-CO-CHCl₂, -CH=C(Br)-CO-CH₂-OCH₃, -CH=C(Br)-CO-CH(OCH₃)₂, -CH=C(Br)-CO-CH₂-SCH₃, -CH=C(CN)-CO-CH₃, -CH=C(CN)-CO-C₂H₅, -CH=C(CN)-CO-n-C₃H₇, -CH=C(CN)-CO-i-C₃H₇, -CH=C(CN)-CO-n-C₄H₉, -CH=C(CN)-CO-tert.-C₄H₉, -CH=C(CN)-CO-CH₂Cl, -CH=C(CN)-CO-CH₂Br, -CH=C(CN)-CO-CHCl₂, -CH=C(CN)-CO-CH₂-OCH₃, -CH=C(CN)-CO-CH(OCH₃)₂, -CH=C(CN)-CO-CH₂-SCH₃, -CH=CH-CO-C₆H₅, -CH=CH-CO-(4-Cl-C₆H₄), -CH=C(CH₃)-CO-C₆H₅, -CH=C(CH₃)-CO-(4-Cl-C₆H₄), -CH=C(C₂H₅)-CO-C₆H₅, -CH=C(C₂H₅)-CO-(4-Cl-C₆H₄), -CH=C(Cl)-CO-C₆H₅, -CH=C(Br)-CO-C₆H₅, -CH=C(CN)-CO-C₆H₅, -CH=CH-CO-NH₂, -CH=CH-CO-NHCH₃, -CH=CH-CO-N(CH₃)₂, -CH=CH-CO-NH-C₂H₅, -CH=CH-CO-N(C₂H₅)₂, -CH=CH-CO-NH-n-C₃H₇, -CH=CH-CO-NH-i-C₃H₇, -CH=CH-CO-NH-tert.-C₄H₉, -CH=CH-CO-NH-cyclopropyl, -CH=CH-CO-NH-cyclobutyl, -CH=CH-CO-NH-cyclopentyl, -CH=CH-CO-NH-cyclohexyl, -CH=CH-CO-NH-cycloheptyl, -CH=CH-CO-NH-cyclooctyl, -CH=CH-CO-pyrrolidin-1-yl, -CH=CH-CO-piperidin-1-yl, -CH=CH-CO-morpholin-4-yl, -CH=CH-CO-NH-CH₂CH=CH₂, -CH=CH-CO-NH-CH₂C≡CH, -CH=CH-CO-N(CH₃)-CH₂C≡CH, -CH=CH-CO-NH-(CH₂)₂Cl, -CH=CH-CO-NH-C₆H₅, -CH=C(CH₃)-CO-NH₂, -CH=C(CH₃)-CO-NHCH₃, -CH=C(CH₃)-CO-N(CH₃)₂, -CH=C(CH₃)-CO-NH-C₂H₅, -CH=C(CH₃)-CO-N(C₂H₅)₂, -CH=C(CH₃)-CO-NH-n-C₃H₇, -CH=C(CH₃)-CO-NH-i-C₃H₇, -CH=C(CH₃)-CO-NH-tert.-C₄H₉, -CH=C(CH₃)-CO-NH-cyclopropyl, -CH=C(CH₃)-CO-NH-cyclobutyl, -CH=C(CH₃)-CO-NH-cyclopentyl, -CH=C(CH₃)-CO-NH-cyclohexyl, -CH=C(CH₃)-CO-NH-cycloheptyl, -CH=C(CH₃)-CO-NH-cyclooctyl, -CH=C(CH₃)-CO-pyrrolidin-1-yl, -CH=C(CH₃)-CO-piperidin-1-yl, -CH=C(CH₃)-CO-morpholin-4-yl, -CH=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -CH=C(CH₃)-CO-NH-CH₂C≡CH, -CH=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CH₃)-CO-NH-(CH₂)₂Cl, -CH=C(CH₃)-CO-NH-C₆H₅, -CH=C(C₂H₅)-CO-NH₂, -CH=C(C₂H₅)-CO-NHCH₃, -CH=C(C₂H₅)-CO-N(CH₃)₂, -CH=C(C₂H₅)-CO-NH-C₂H₅, -CH=C(C₂H₅)-CO-N(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-n-C₃H₇, -CH=C(C₂H₅)-CO-NH-i-C₃H₇, -CH=C(C₂H₅)-CO-NH-tert.-C₄H₉, -CH=C(C₂H₅)-CO-NH-cyclopropyl, -CH=C(C₂H₅)-CO-NH-cyclobutyl, -CH=C(C₂H₅)-CO-NH-cyclopentyl, -CH=C(C₂H₅)-CO-NH-cyclohexyl, -CH=C(C₂H₅)-CO-NH-cycloheptyl, -CH=C(C₂H₅)-CO-NH-cyclooctyl, -CH=C(C₂H₅)-CO-pyrrolidin-1-yl, -CH=C(C₂H₅)-CO-piperidin-1-yl, -CH=C(C₂H₅)-CO-morpholin-4-yl, -CH=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-CH₂C≡CH, -CH=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -CH=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -CH=C(C₂H₅)-CO-NH-C₆H₅, -CH=C(Cl)-CO-NH₂, -CH=C(Cl)-CO-NHCH₃, -CH=C(Cl)-CO-N(CH₃)₂, -CH=C(Cl)-CO-NH-C₂H₅, -CH=C(Cl)-CO-N(C₂H₅)₂, -CH=C(Cl)-CO-NH-n-C₃H₇, -CH=C(Cl)-CO-NH-i-C₃H₇, -CH=C(Cl)-CO-NH-tert.-C₄H₉, -CH=C(Cl)-CO-NH-cyclopropyl, -CH=C(Cl)-CO-NH-cyclobutyl, -CH=C(Cl)-CO-NH-cyclopentyl, -CH=C(Cl)-CO-NH-cyclohexyl, -CH=C(Cl)-CO-NH-cycloheptyl, -CH=C(Cl)-CO-NH-cyclooctyl, -CH=C(Cl)-CO-pyrrolidin-1-yl, -CH=C(Cl)-CO-piperidin-1-yl, -CH=C(Cl)-CO-morpholin-4-yl, -CH=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -CH=C(Cl)-CO-NH-CH₂C≡CH, -CH=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Cl)-CO-NH-(CH₂)₂Cl, -CH=C(Cl)-CO-NH-C₆H₅, -CH=C(Br)-CO-NH₂, -CH=C(Br)-CO-NHCH₃, -CH=C(Br)-CO-N(CH₃)₂, -CH=C(Br)-CO-NH-C₂H₅, -CH=C(Br)-CO-N(C₂H₅)₂, -CH=C(Br)-CO-NH-n-C₃H₇, -CH=C(Br)-CO-NH-i-C₃H₇, -CH=C(Br)-CO-NH-tert.-C₄H₉, -CH=C(Br)-CO-NH-cyclopropyl, -CH=C(Br)-CO-NH-cyclobutyl, -CH=C(Br)-CO-NH-cyclopentyl, -CH=C(Br)-CO-NH-cyclohexyl, -CH=C(Br)-CO-NH-cycloheptyl, -CH=C(Br)-CO-NH-cyclooctyl, -CH=C(Br)-CO-pyrrolidin-1-yl, -CH=C(Br)-CO-piperidin-1-yl, -CH=C(Br)-CO-morpholin-4-yl, -CH=C(Br)-CO-NH-CH₂CH=C(Br)₂, -CH=C(Br)-CO-NH-CH₂C≡CH, -CH=C(Br)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Br)-CO-NH-(CH₂)₂Cl, -CH=C(Br)-CO-NH-C₆H₅, -CH=C(CN)-CO-NH₂, -CH=C(CN)-CO-NHCH₃, -CH=C(CN)-CO-N(CH₃)₂, -CH=C(CN)-CO-NH-C₂H₅, -CH=C(CN)-CO-N(C₂H₅)₂, -CH=C(CN)-CO-NH-n-C₃H₇, -CH=C(CN)-CO-NH-i-C₃H₇, -CH=C(CN)-CO-NH-tert.-C₄H₉, -CH=C(CN)-CO-NH-cyclopropyl, -CH=C(CN)-CO-NH-cyclobutyl, -CH=C(CN)-CO-NH-cyclopentyl, -CH=C(CN)-CO-NH-cyclohexyl, -CH=C(CN)-CO-NH-cycloheptyl, -CH=C(CN)-CO-NH-cyclooctyl, -CH=C(CN)-CO-pyrrolidin-1-yl, -CH=C(CN)-CO-piperidin-1-yl, -CH=C(CN)-CO-morpholin-4-yl, -CH=C(CN)-CO-NH-CH₂CH=C(CN)₂, -CH=C(CN)-CO-NH-CH₂C≡CH, -CH=C(CN)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CN)-CO-NH-(CH₂)₂Cl, -CH=C(CN)-CO-NH-C₆H₅, -CH=CH-CO-SCH₃, -CH=CH-CO-SC₂H₅, -CH=CH-CO-S-n-C₃H₇, -CH=CH-CO-S-i-C₃H₇, -CH=CH-CO-S-n-C₄H₉, -CH=CH-CO-S-tert.-C₄H₉, -CH=C(CH₃)-CO-SCH₃, -CH=C(CH₃)-CO-SC₂H₅, -CH=C(CH₃)-CO-S-n-C₃H₇, -CH=C(CH₃)-CO-S-i-C₃H₇, -CH=C(CH₃)-CO-S-n-C₄H₉, -CH=C(CH₃)-CO-S-tert.-C₄H₉, -CH=C(C₂H₅)-CO-SCH₃, -CH=C(C₂H₅)-CO-SC₂H₅, -CH=C(C₂H₅)-CO-S-n-C₃H₇, -CH=C(C₂H₅)-CO-S-i-C₃H₇, -CH=C(C₂H₅)-CO-S-n-C₄H₉, -CH=C(C₂H₅)-CO-S-tert.-C₄H₉, -CH=C(Cl)-CO-SCH₃, -CH=C(Cl)-CO-SC₂H₅, -CH=C(Cl)-CO-S-n-C₃H₇, -CH=C(Cl)-CO-S-i-C₃H₇, -CH=C(Cl)-CO-S-n-C₄H₉, -CH=C(Cl)-CO-S-tert.-C₄H₉, -CH=C(Br)-CO-SCH₃, -CH=C(Br)-CO-SC₂H₅, -CH=C(Br)-CO-S-n-C₃H₇, -CH=C(Br)-CO-S-i-C₃H₇, -CH=C(Br)-CO-S-n-C₄H₉, -CH=C(Br)-CO-S-tert.-C₄H₉, -CH=C(CN)-CO-SCH₃, -CH=C(CN)-CO-SC₂H₅, -CH=C(CN)-CO-S-n-C₃H₇, -CH=C(CN)-CO-S-i-C₃H₇, -CH=C(CN)-CO-S-n-C₄H₉, -CH=C(CN)-CO-S-tert.-C₄H₉, -CH=C(COCH₃)-CO-OCH₃, -CH=C(COC₂H₅)-CO-OCH₃, -CH=C(CO-n-C₃H₇)-CO-OCH₃, -CH=C(COCH₃)-CO-OC₂H₅, -CH=C(COC₂H₅)-CO-OC₂H₅, -CH=C(CO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COCH₃)-CO-O-n-C₃H₇, -CH=C(COC₂H₅)-CO-O-n-C₃H₇, -CH=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-OCH₃, -CH=C(CF₃)-CO-OC₂H₅, -CH=C(CF₃)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-O-i-C₃H₇, -CH=C(CF₃)-CO-O-n-C₄H₉, -CH=C(CF₃)-CO-O-tert.-C₄H₉, -CH=C(COOCH₃)₂, -CH=C(COOC₂H₅)₂, -CH=C(COOCH₃)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)-CO-OCH₃, -CH=C(COO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)₂, -CH=CH-CH=CH-COOH, -CH=CH-CH=CH-CO-OCH₃, -CH=CH-CH=CH-CO-OC₂H₅, -CH=CH-CH=C(COOCH₃)₂, -CH=CH-CH=C(CN)-CO-OCH₃, -CH=CH-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-OCH₃, -CH=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CH=C(Cl)-CO-OCH₃, -CH=C(CH₃)-CH=C(Br)-CO-OCH₃, -CH=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-NH₂, -CH=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -CH=CH-(CH₂)₂-COOH, -CH=CH-(CH₂)₂-CO-OCH₃, -CH=CH-(CH₂)₂-CO-OC₂H₅, -CH=CH-CH₂-CH(COOCH₃)₂, -CH=CH-CH₂-CH(COOC₂H₅)₂, -CH=CH-CH₂-CH(CN)-CO-OCH₃, -CH=CH-CH₂-CH(CN)-CO-OC₂H₅, -CH=CH-CH₂-CH(CH₃)-CO-OCH₃, -CH=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -CH=CH-(CH₂)₂-CO-NH₂, -CH=CH-(CH₂)₂-CO-NH-CH₃, -CH=CH-CH₂-COOH, -CH=CH-CH₂-CO-OCH₃, -CH=CH-CH₂-CO-OC₂H₅, -CH=C(COOCH₃)-CH₂-CO-OCH₃, -CH=C(COOCH₃)-CH₂-CO-OC₂H₅, -CH=CH-CH₂-CO-NH₂, -CH=CH-CH₂-CO-NH-CH₃, -CH=CH-CH₂-CO-N(CH₃)₂, -CH(OCH₃)₂, -CH(SCH₃)₂, -CH(OC₂H₅)₂, -CH(SC₂H₅)₂, -CH(O-n-C₃H₇)₂, -CH(O-i-C₃H₇)₂, -CH(S-n-C₃H₇)₂, -CH(S-i-C₃H₇)₂, -CH(O-n-C₄H₉)₂, -CH(O-i-C₄H₉)₂, -CH(O-s-C₄H₉)₂, -CH(O-tert.-C₄H₉)₂, -CH(S-n-C₄H₉)₂, -CH(S-i-C₄H₉)₂, -CH(S-s-C₄H₉)₂, -CH(S-tert.-C₄H₉)₂, -CH(OC₅H₁₁)₂, 1,3-Dioxolan-2-yl, 1,3-Dithiolan- 2-yl, 1,3-Oxathiolan-2-yl, 4-Methyl-1,3-dioxolan-2-yl, 4-Methyl-1,3-dithiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 5-Methyl-1,3-oxathiolan-2-yl, 4-Ethyl-1,3-dioxolan-2-yl, 4-Ethyl- 1,4-dithiolan-2-yl, 4-Ethyl-1,3-oxathiolan-2-yl, 5-Ethyl-1,3-oxathiolan- 2-yl, 4,5-Dimethyl-1,3-dioxolan-2-yl, 4,4-Dimethyl-1,3- dioxolan-2-yl, 4,5-Dimethyl-1,3-dithiolan-2-yl, 5,5-Dimethyl-1,3- dithiolan-2-yl, 4,5-Dimethyl-1,3-oxathiolan-2-yl, 5,5-Dimethyl- 1,3-oxathiolan-2-yl, 4,4-Dimethyl-1,3-oxathiolan-2-yl, 4-Vinyl- 1,3-dioxolan-2-yl, 4-Vinyl-1,3-dithiolan-2-yl, 4-Vinyl-1,3-oxathiolan- 2-yl, 5-Vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3- dioxolan-2-yl, 4-Chlormethyl-1,3-dithiolan-2-yl, 4-Chlormethyl- 1,3-oxathiolan-2-yl, 5-Chlormethyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-1,3-dithiolan- 2-yl, 4-Hydroxymethyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl- 1,3-oxathiolan-2-yl, 4-Methoxymethyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl- oxymethyl-1,3-dioxolan-2-yl, 4-Propargyloxymethyl-1,3-dioxolan- 2-yl, 4-Acetoxymethyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-1,3-dithiolan-2-yl, 4-Propargyl- oxymethyl-1,3-dithiolan-2-yl, 4-Acetoxymethyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-1,3-oxathiolan- 2-yl, 4-Allyloxymethyl-1,3-oxathiolan-2-yl, 5-Allyloxy- methyl-1,3-oxathiolan-2-yl, 4-Propargyloxymethyl-1,3-oxathiolan- 2-yl, 5-Propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxymethyl- 1,3-oxathiolan-2-yl, 5-Acetoxymethyl-1,3-oxathiolan-2-yl, 4-Methylthiomethyl-1,3-dioxolan-2-yl, 4-Methylthiomethyl-1,3- dithiolan-2-yl, 4-Carboxy-1,3-dioxolan-2-yl, 4-Carboxy-1,3- dithiolan-2-yl, 4-Methoxycarbonyl-1,3-dioxolan-2-yl, 4-Ethoxy- carbonyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-1,3-dithiolan- 2-yl, 4-n-Butoxycarbonyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-4-methyl- 1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithiolan- 2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-1,3- dithiolan-2-yl, 1,3-Dioxan-2-yl, 1,3-Dithian-2-yl, 1,3-Oxathian- 2-yl, 5-Methyl-1,3-dioxan-2-yl, 5-Methyl-1,3-dithian-2-yl, 5-Methyl-1,3-oxathian-2-yl, 5,5-Dimethyl-1,3-dioxan-2-yl, 4,6-Dimethyl- 1,3-dioxan-2-yl, 4,4-Dimethyl-1,3-dioxan-2-yl, 5,5-Dimethyl- 1,3-dithian-2-yl, 4,6-Dimethyl-1,3-dithian-2-yl, 4,4-Dimethyl- 1,3-dithian-2-yl, 5,5-Dimethyl-1,3-oxathian-2-yl, 4,4-Dimethyl- 1,3-oxathian-2-yl, 6,6-Dimethyl-1,3-oxathian-2-yl, 4-Hydroxymethyl-1,3-dioxan-2-yl, 4-Methoxymethyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-1,3-dioxan-2- yl, 4-Hydroxymethyl-1,3-dithian-2-yl, 4-Methoxymethyl-1,3-dithian- 2-yl, 4-Allyloxymethyl-1,3-dithian-2-yl, 4-Acetoxymethyl- 1,3-dithian-2-yl, 4-Chlormethyl-1,3-dioxan-2-yl, 4-Chlormethyl- 1,3-dithian-2-yl, 1,3-Dioxepan-2-yl, 1,3-Dithiepan-2-yl, 1,3-Dioxep- 5-en-2-yl, 4-Methoxycarbonyl-1,3-dioxan-2-yl, 4-Ethoxy- carbonyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-1,3-dithian- 2-yl, 4-n-Butoxycarbonyl-1,3-dithian-2-yl, 4-Methoxycarbonyl-4- methyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxan-2- yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-Methoxy- carbonyl-4-methyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-4-methyl- 1,3-dithian-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithian-2-yl, -C(CH₃)(OCH₃)₂, -C(CH₃)(SCH₃)₂, -C(CH₃)(OC₂H₅)₂, -C(CH₃)(SC₂H₅)₂, -C(CH₃)(O-n-C₃H₇)₂, -C(CH₃)(O-i-C₃H₇)₂, -C(CH₃)(S-n-C₃H₇)₂, -C(CH₃)(S-i-C₃H₇)₂, -C(CH₃)(O-n-C₄H₉)₂, -C(CH₃)(O-i-C₄H₉)₂, -C(CH₃)(O-s-C₄H₉)₂, -C(CH₃)(O-tert.-C₄H₉)₂, -C(CH₃)(S-n-C₄H₉)₂, -C(CH₃)(S-i-C₄H₉)₂, -C(CH₃)(S-s-C₄H₉)₂, -C(CH₃)(S-tert.-C₄H₉)₂, -C(CH₃)(O-n-C₅H₁₁)′′, 2-Methyl-1,3-dioxolan-2-yl, 2-Methyl-1,3-dithiolan- 2-yl, 2-Methyl-1,3-oxathiolan-2-yl, 2,4-Dimethyl-1,3- dioxolan-2-yl, 2,4-Dimethyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-1,3- oxathiolan-2-yl, 2,5-Dimethyl-1,3-oxathiolan-2-yl, 4-Ethyl-2- methyl-1,3-dioxolan-2-yl, 4-Ethyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Ethyl-2-methyl-1,3- oxathiolan-2-yl, 2,4,5-Trimethyl-1,3-dioxolan-2-yl, 2,4,4-Trimethyl- 1,3-dioxolan-2-yl, 2,4,5-Trimethyl-1,3-dithiolan-2-yl, 2,4,4-Trimethyl-1,3-dithiolan-2-yl, 2,4,5-Trimethyl-1,3-oxathiolan- 2-yl, 2,4,4-Trimethyl-1,3-oxathiolan-2-yl, 2-Methyl-4-vinyl- 1,3-dioxolan-2-yl, 2-Methyl-4-vinyl-1,3-dithiolan-2-yl, 2-Methyl- 4-vinyl-1,3-oxathiolan-2-yl, 2-Methyl-5-vinyl-1,3-oxathiolan-2- yl, 4-Chlormethyl-2-methyl-1,3-dioxolan-2-yl, 4-Chlormethyl-2- methyl-1,3-dithiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-oxathiolan- 2-yl, 5-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl- 2-methyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-2- methyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dioxolan- 2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxy- 2-methyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dithiolan-2-yl, 4-Acetoxy-2- methyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-oxathiolan- 2-yl, 5-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl- 2-methyl-1,3-oxathiolan-2-yl, 5- Allyoxymethyl-2- methyl-1,3-oxathiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3- oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3-oxathiolan-2- yl, 4-Acetoxy-2-methyl-1,3-oxathiolan-2-yl, 5-Acetoxy-2-methyl- 1,3-oxathiolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dioxolan-2- yl, 2-Methyl-4-methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-2- methyl-1,3-dioxolan-2-yl, 4-Carboxy-2-methyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-2- methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-2-methyl-1,3-dioxolan- 2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl- 2-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-2- methyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dioxolan- 2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-ethoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4- ethoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-n-butoxy- carbony-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl-1,3- dithiolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-dioxan-2-yl, 2-Methyl-1,3-dithian-2-yl, 2-Methyl-1,3-oxathian-2-yl, 2,5- Dimethyl-1,3-dioxan-2-yl, 2,5-Dimethyl-1,3-dithian-2-yl, 2,5-Dimethyl- 1,3-oxathian-2-yl, 2,5,5-Trimethyl-1,3-dioxan-2-yl, 2,4,6- Trimethyl-1,3-dioxan-2-yl, 2,2,4-Trimethyl-1,3-dioxan-2-yl, 2,5,5-Trimethyl-1,3-dithian-2-yl, 2,4,6-Trimethyl-1,3-dithian-2-yl, 2,4,4-Trimethyl-1,3-dithian-2-yl, 2,5,5-Trimethyl-1,3-oxathian- 2-yl, 2,4,4-Trimethyl-1,3-oxathian-2-yl, 2,6,6-Trimethyl- 1,3-oxathian-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-2- methyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dithian-2-yl, 4-Methoxymethyl-2- methyl-1,3-dithian-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithian-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dithian-2-yl, 4-Chlormethyl-2- methyl-1,3-dioxan-2-yl, 4-Chlormethyl-2-methyl-1,3-dithian-2-yl, -C(CH₃)=NH, -C(CH₃)=N-CH₃, -C(CH₃)=N-C₂H₅, -C(CH₃)=N-n-C₃H₇, -C(CH₃)=N-i-C₃H₇, -C(CH₃)=N-n-C₄H₉, -C(CH₃)=N-CH₂CH=CH₂, -C(CH₃)=N-CH₂CH=CH₂-CH₃, -C(CH₃)=N-CH₂C≡CH, -C(CH₃)=N-CH₂C≡C-CH₃, -C(CH₃)=N-cyclopropyl, -C(CH₃)=N-cyclobutyl, -C(CH₃)=N-cyclopentyl, -C(CH₃)=N-cyclohexyl, -C(CH₃)=N-cycloheptyl, -C(CH₃)=N-CH₂-CH₂Cl, -C(CH₃)=N-CH₂Cl, -C(CH₃)=N-C₆H₅, -C(CH₃)=N-(2-F-C₆H₄), -C(CH₃)=N-(3-F-C₆H₄), -C(CH₃)=N-(4-F-C₆H₄), -C(CH₃)=N-(2-Cl-C₆H₄), -C(CH₃)=N-(3-Cl-C₆H₄), -C(CH₃)=N-(4-Cl-C₆H₄), -C(CH₃)=N-(2-CH₃-C₆H₄), -C(CH₃)=N-(3-CH₃-C₆H₄), -C(CH₃)=N-(4-CH₃-C₆H₄), -C(CH₃)=N-(2-CF₃-C₆H₄), -C(CH₃)=N-(3-CF₃-C₆H₄), -C(CH₃)=N-(4-CF₃-C₆H₄), -C(CH₃)=N-(2-OCH₃-C₆H₄), -C(CH₃)=N-(3-OCH₃-C₆H₄), -C(CH₃)=N-(4-OCH₃-C₆H₄), -C(CH₃)=N-(4-NO₂-C₆H₄), -C(CH₃)=N-(4-CN-C₆H₄), -C(CH₃)=N-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-(2,4-(CH₃)₂-C₆H₃), -C(CH₃)=N-CH₂-OCH₃, -C(CH₃)=N-CH₂-OC₂H₅, -C(CH₃)=N-CH₂CH₂-OCH₃, -C(CH₃)=N-CH₂CH-OC₂H₅, -C(CH₃)=N-OH, -C(CH₃)=N-OCH₃, -C(CH₃)=N-OC₂H₅, -C(CH₃)=N-O-n-C₃H₇, -C(CH₃)=N-O-i-C₃H₇, -C(CH₃)=N-O-n-C₄H₉, -C(CH₃)=N-O-i-C₄H₉, -C(CH₃)=N-O-s-C₄H₉, -C(CH₃)=N-O-tert.-C₄H₉, -C(CH₃)=N-OCH₂-CH=CH₂, -C(CH₃)=N-OCH(CH₃)-CH=CH₂, -C(CH₃)=N-OCH₂-C≡CH, -C(CH₃)=N-CH(CH₃)-C≡CH, -C(CH₃)=N-OCH₂-CH=C-CH₃, -C(CH₃)=N-OCH₂CH₂-Cl, -C(CH₃)=N-OCH₂CH₂-F, -C(CH₃)=N-OCH₂-CF₃, -C(CH₃)=N-OCH₂-CH=CHCl, -C(CH₃)=N-OCH₂-C(Cl)=CH₂, -C(CH₃)=N-OCH₂-C(Br)=CH₂, -C(CH₃)=N-OCH₂-CH=C(Cl)-CH₃, -C(CH₃)=N-O-CO-CH₃, -C(CH₃)=N-O-CO-C₂H₅, -C(CH₃)=N-OCH₂-CN, -C(CH₃)=N-OCH₂-CH=CH-CH₂-OCH₃, -C(CH₃)=N-OCH₂-CH=CH-CH₂-O-tert.-C₄H₉, -C(CH₃)=N-O-(CH₂)₃-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-(4-Cl-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-C₆H₅, -C(CH₃)=N-OCH₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(3-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-CH₂-(4-CH₃O-C₆H₄), -C(CH₃)=N-OCH₂-CH=C(CH₃)-C₆H₅, -C(CH₃)=N-O-(CH₂)₂-CH=CH-(3,4-Cl₂-C₆H₃), -C(CH₃)=N-O-(CH₂)₃-C≡-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-OCH₃, -C(CH₃)=N-OCH₂CH₂-OCH₃, -C(CH₃)=N-OCH₂-OC₂H₅, -C(CH₃)=N-OCH(CH₃)-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=N-NH₂, -C(CH₃)=N-NH-CH₃, -C(CH₃)=N-NH-C₂H₅, -C(CH₃)=N-NH-n-C₃H₇, -C(CH₃)=N-NH-i-C₃H₇, -C(CH₃)=N-NH-n-C₄H₉, -C(CH₃)=N-NH-i-C₄H₉, -C(CH₃)=N-NH-s-C₄H₉, -C(CH₃)=N-NH-tert.-C₄H₉, -C(CH₃)=N-NH-cyclopropyl, -C(CH₃)=N-NH- cyclobutyl, -C(CH₃)=N-NH-cyclopentyl, -C(CH₃)=N-NH-cyclohexyl, -C(CH₃)=N-NH-cycloheptyl, -C(CH₃)=N-N(CH₃)₂, -C(CH₃)=N-N(C₂H₅)₂, -C(CH₃)=N-N(n-C₃H₇)₂, -C(CH₃)=N-N(i-C₃H₇)₂, -C(CH₃)=N-NH-CH₂-C=CH, -C(CH₃)=N-NH-CH₂-C≡CH, -C(CH₃)=N-N(CH₃)-CH₂-C≡CH, -C(CH₃)=N-NH-CH₂CF₃, -C(CH₃)=N-NH-CO-CH₃, -C(CH₃)=N-NH-CO-C₂H₅, -C(CH₃)=N-NH-CO-OCH₃, -C(CH₃)=N-NH-CO-OC₂H₅, -C(CH₃)=N-NH-CO-O-tert.-C₄H₉, -C(CH₃)=N- pyrrolidin-1-yl, -C(CH₃)=N-piperidin-1-yl, -C(CH₃)=N-morpholin- 4-yl, -C(CH₃)=N-NH-C₆H₅, -C(CH₃)=N-NH-(4-Cl-C₆H₄), -C(CH₃)=N-NH-(4-NO₂-C₆H₄), -C(CH₃)=N-NH-(4-F-C₆H₄), -C(CH₃)=N-NH-(4-CH₃O-C₆H₄), -C(CH₃)=N-NH-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-NH-(2,4-(NO₂)₂-C₆H₃), -C(CH₃)=N-NH-CO-NH₂, -C(CH₃)=N-NH-CO-NHCH₃, -C(CH₃)=N-NH-CO-NHC₂H₅, -C(CH₃)=N-NH-CO-N(CH₃)₂, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=CH-CO-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -(CH₃)=CH-CO-O-n-C₄H₉, -C(CH₃)=CH-CO-O-tert.-C₄H₉, -C(CH₃)=CH-CO-O-cyclopropyl, -C(CH₃)=CH-CO-O-cyclobutyl, -C(CH₃)=CH-CO-O-cyclopentyl, -C(CH₃)=CH-CO-O-cyclohexyl, -C(CH₃)=CH-CO-O-cycloheptyl, -C(CH₃)=C(CH₃)-COOH, -C(CH₃)=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-cyclopropyl, -C(CH₃)=C(CH₃)-CO-O-cyclobutyl, -C(CH₃)=C(CH₃)-CO-O-cyclopentyl, -C(CH₃)=C(CH₃)-CO-O-cyclohexyl, -C(CH₃)=C(CH₃)-CO-O-cycloheptyl, -C(CH₃)=C(C₂H₅)-COOH, -C(CH₃)=C(C₂H₅)-CO-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-O- cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-O-cycloheptyl, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-O-n-C₄H₉, -C(CH₃)=C(Cl)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-O-cyclopropyl, -C(CH₃)=C(Cl)-CO-O-cyclobutyl, -C(CH₃)=C(Cl)-CO-O-cyclopentyl, -C(CH₃)=C(Cl)-CO-O-cyclohexyl, -C(CH₃)=C(Cl)-CO-O-cycloheptyl, -C(CH₃)=C(Br)-COOH, -C(CH₃)=C(Br)-CO-OCH₃, -C(CH₃)=C(Br)-CO-OC₂H₅, -C(CH₃)=C(Br)-CO-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-O-n-C₄H₉, -C(CH₃)=C(Br)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-O-cyclopropyl, -C(CH₃)=C(Br)-CO-O-cyclobutyl, -C(CH₃)=C(Br)-CO-O-cyclopentyl, -C(CH₃)=C(Br)-CO-O-cyclohexyl, -C(CH₃)=C(Br)-CO-O-cycloheptyl, -C(CH₃)=C(CN)-COOH, -C(CH₃)=C(CN)-CO-OCH₃, -C(CH₃)=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CN)-CO-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-O-n-C₄H₉, -C(CH₃)=C(CN)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-O-cyclopropyl, -C(CH₃)=C(CN)-CO-O-cyclobutyl, -C(CH₃)=C(CN)-CO-O-cyclopentyl, -C(CH₃)=C(CN)-CO-O-cyclohexyl, -C(CH₃)=C(CN)-CO-O-cycloheptyl, -C(CH₃)=CH-CO-OCH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-OCH(CH₃)-OCH₃, -C(CH₃)=CH-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=CH-CO-OCH₂CH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-O-i-C₃H₇, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -(CH₃)=C(Cl)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-O-i-C₃H₇, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-O-i-C₃H₇, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-CF₃, -C(CH₃)=CH-CO-OCH₂-CCl₃, -C(CH₃)=CH-CO-OCH₂-oxiranyl, -C(CH₃)=CH-CO-(CH₂)₃-Br, -C(CH₃)=CH-CO-OCH₂-CH=CH₂, -C(CH₃)=CH-CO-OCH₂-C≡CH, -C(CH₃)=CH-CO-OCH₂-CN, -C(CH₃)=CH-CO-OCH₂CH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CF₃, -C(CH₃)=C(CH₃)-CO-OCH₂-CCl₃, -C(CH₃)=C(CH₃)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CH₃)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(CH₃)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CH₃)-CO-OCH₂-C≡CH, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CF₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CCl₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-oxiranyl, -C(CH₃)=C(C₂H₅)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(C₂H₅)CO-OCH₂-C≡CH, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-C₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂-CF₃, -C(CH₃)=C(Cl)-CO-OCH₂-CCl₃, -C(CH₃)=C(Cl)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Cl)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Cl)-CO-OCH₂-CH≡CH₂, -C(CH₃)=C(Cl)-CO-OCH₂-C≡CH, -C(CH₃)=C(Cl)-CO-OCH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂-CF₃, -C(CH₃)=C(Br)-CO-OCH₂-CCl₃, -C(CH₃)=C(Br)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Br)-CO-O(CH₂)₃-Br, -C(CH₃)=C(Br)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Br)-CO-OCH₂-C≡CH, -C(CH₃)=C(Br)-CO-OCH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂CH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂-CF₃, -C(CH₃)=C(CN)-CO-OCH₂-CCl₃, -C(CH₃)=C(CN)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CN)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CN)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CN)-CO-OCH₂-C≡CH, -C(CH₃)=C(CN)-CO-OCH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂CH₂-CN, -C(CH₃)=CH-CO-CH₃, -C(CH₃)=CH-CO-C₂H₅, -C(CH₃)=CH-CO-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-n-C₄H₉, -C(CH₃)=CH-CO-tert.-C₄H₉, -C(CH₃)=CH-CO-CH₂Cl, -C(CH₃)=CH-CO-CH₂Br, -C(CH₃)=CH-CO-CHCl₂, -C(CH₃)=CH-CO-CH₂-OCH₃, -C(CH₃)=CH-CO-CH(OCH₃)₂, -C(CH₃)=CH-CO-CH₂-SCH₃, -C(CH₃)=C(CH₃)-CO-CH₃, -C(CH₃)=C(CH₃)-CO-C₂H₅, -C(CH₃)=C(CH₃)-CO-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-CH₂Cl, -C(CH₃)=C(CH₃)-CO-CH₂Br, -C(CH₃)=C(CH₃)-CO-CHCl₂, -C(CH₃)=C(CH₃)-CO-CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-CH(OCH₃)₂, -C(CH₃)=C(CH₃)-CO-CH₂-SCH₃, -C(CH₃)=C(C₂H₅)-CO-CH₃, -C(CH₃)=C(C₂H₅)-CO-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-CH₂Cl, -C(CH₃)=C(C₂H₅)-CO-CH₂Br, -C(CH₃)=C(C₂H₅)-CO-CHCl₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-CH(OCH₃)₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-SCH₃, -C(CH₃)=C(Cl)-CO-CH₃, -C(CH₃)=C(Cl)-CO-C₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-n-C₄H₉, -C(CH₃)=C(Cl)-CO-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-CH₂Cl, -C(CH₃)=C(Cl)-CO-CHCl₂, -C(CH₃)=C(Cl)-CO-CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-CH(OCH₃)₂, -C(CH₃)=C(Cl)-CO-CH₂-SCH₃, -C(CH₃)=C(Br)-CO-CH₃, -C(CH₃)=C(Br)-CO-C₂H₅, -C(CH₃)=C(Br)-CO-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-n-C₄H₉, -C(CH₃)=C(Br)-CO-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-CH₂Cl, -C(CH₃)=C(Br)-CO-CH₂Br, -C(CH₃)=C(Br)-CO-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-CH(OCH₃)₂, -C(CH₃)=C(Br)-CO-CH₂-SCH₃, -C(CH₃)=C(CN)-CO-CH₃, -C(CH₃)=C(CN)-CO-C₂H₅, -C(CH₃)=C(CN)-CO-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-n-C₄H₉, -C(CH₃)=C(CN)-CO-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-CH₂Cl, -C(CH₃)=C(CN)-CO-CH₂Br, -C(CH₃)=C(CN)-CO-CHCl₂, -C(CH₃)=C(CN)-CO-CH₂-OCH₃, -C(CH₃)=C(CN)-CO-CH(OCH₃)₂, -C(CH₃)=C(CN)-CO-CH₂-SCH₃, -C(CH₃)=CH-CO-C₆H₅, -C(CH₃)=CH-CO-(4-Cl-C₆H₄), -C(CH₃)=C(CH₃)-CO-C₆H₅, -C(CH₃)=C(CH₃)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(C₂H₅)-CO-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(Cl)-CO-C₆H₅, -C(CH₃)=C(Br)-CO-C₆H₅, -C(CH₃)=C(CN)-CO-C₆H₅, -C(CH₃)=CH-CO-NH₂, -C(CH₃)=CH-CO-NHCH₃, -C(CH₃)=CH-CO-N(CH₃)₂, -C(CH₃)=CH-CO-NH-C₂H₅, -C(CH₃)=CH-CO-N(C₂H₅)₂, -C(CH₃)=CH-CO-NH-n-C₃H₇, -C(CH₃)=CH-CO-NH-i-C₃H₇, -C(CH₃)=CH-CO-NH-tert.-C₄H₉, -C(CH₃)=CH-CO-NH-cyclopropyl, -C(CH₃)=CH-CO-NH-cyclobutyl, -C(CH₃)=CH-CO-NH-cyclopentyl, -C(CH₃)=CH-CO-NH-cyclohexyl, -C(CH₃)=CH-CO-NH-cycloheptyl, -C(CH₃)=CH-CO-NH-cyclooctyl, -C(CH₃)=CH-CO-pyrrolidin-1-yl, -C(CH₃)=CH-CO-piperidin-1-yl, -C(CH₃)=CH-CO-morpholin-4-yl, -C(CH₃)=CH-CO-NH-CH₂CH=CH₂, -C(CH₃)=CH-CO-NH-CH₂C≡CH, -C(CH₃)=CH-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=CH-CO-NH-(CH₂)₂Cl, -C(CH₃)=CH-CO-NH-C₆H₅, -C(CH₃)=C(CH₃)-CO-NH₂, -C(CH₃)=C(CH₃)-CO-NHCH₃, -C(CH₃)=C(CH₃)-CO-N(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-C₂H₅, -C(CH₃)=C(CH₃)-CO-N(C₂H₅)₂, -C(CH₃)=C(CH₃)-CO-NH-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-NH- cyclopropyl, -C(CH₃)=C(CH₃)-CO-NH-cyclobutyl, -C(CH₃)=C(CH₃)-CO-NH-cyclopentyl, -C(CH₃)=C(CH₃)-CO-NH- cyclohexyl, -C(CH₃)=C(CH₃)-CO-NH-cycloheptyl, -C(CH₃)=C(CH₃)-CO-NH-cyclooctyl, -C(CH₃)=C(CH₃)-CO- pyrrolidin-1-yl, -C(CH₃)=C(CH₃)-CO-piperidin-1-yl, -C(CH₃)=C(CH₃)-CO-morpholin-4-yl, -C(CH₃)=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CH₃)-CO-NH-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-NH₂, -C(CH₃)=C(C₂H₅)-CO-NHCH₃, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)₂, -C(CH₃)=C(C₂H₅)-CO-NH-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-N(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-NH- cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-NH-cycloheptyl, -C(CH₃)=C(C₂H₅)-CO-NH- cyclooctyl, -C(CH₃)=C(C₂H₅)-CO-pyrrolidin-1-yl, -C(CH₃)=C(C₂H₅)-CO-piperidin-1-yl, -C(CH₃)=C(C₂H₅)-CO- morpholin-4-yl, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(C₂H₅)-CO-NH-C₆H₅, -C(CH₃)=C(Cl)-CO-NH₂, -C(CH₃)=C(Cl)-CO-NHCH₃, -C(CH₃)=C(Cl)-CO-N(CH₃)₂, -C(CH₃)=C(Cl)-CO-NH-C₂H₅, -C(CH₃)=C(Cl)-CO-N(C₂H₅)₂, -C(CH₃)=C(Cl)-CO-NH-n-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-i-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-NH-cyclopropyl, -C(CH₃)=C(Cl)-CO-NH-cyclobutyl, -C(CH₃)=C(Cl)-CO-NH-cyclopentyl, -C(CH₃)=C(Cl)-CO-NH-cyclohexyl, -C(CH₃)=C(Cl)-CO-NH-cycloheptyl, -C(CH₃)=C(Cl)-CO-NH-cyclooctyl, -C(CH₃)=C(Cl)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Cl)-CO-piperidin-1- yl, -C(CH₃)=C(Cl)-CO-morpholin-4-yl, -C(CH₃)=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -C(CH₃)=C(Cl)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-N(CH₃)-CH₂≡CH, -C(CH₃)=C(Cl)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Cl)-NO-NH-C₆H₅, -C(CH₃)=C(Br)-CO-NH₂, -C(CH₃)=C(Br)-CO-NHCH₃, -C(CH₃)=C(Br)-CO-N(CH₃)₂, -C(CH₃)=C(Br)-CO-NH-C₂H₅, -C(CH₃)=C(Br)-CO-N(C₂H₅)₂, -C(CH₃)=C(Br)-CO-NH-n-C₃H₇, -C(CH₃)=C(Br)-CO-NH-i-C₃H₇, -C(CH₃)=C(Br)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-NH-cyclopropyl, -C(CH₃)=C(Br)-CO-NH-cyclobutyl, -C(CH₃)=C(Br)-CO-NH-cyclopentyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cycloheptyl, -C(CH₃)=C(Br)-CO-NH-cyclooctyl, -C(CH₃)=C(Br)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Br)-CO-piperidin-1-yl, -C(CH₃)=C(Br)-CO-morpholin-4-yl, -C(CH₃)=C(Br)-CO-NH-CH₂CH=C(Br)₂, -C(CH₃)=C(Br)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Br)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Br)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Br)-CO-NH-C₆H₅, -C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CN)-CO-NHCH₃, -C(CH₃)=C(CN)-CO-N(CH₃)₂, -C(CH₃)=C(CN)-CO-NH-C₂H₅, -C(CH₃)=C(CN)-CO-N(C₂H₅)₂, -C(CH₃)=C(CN)-CO-NH-n-C₃H₇, -C(CH₃)=C(CN)-CO-NH-i-C₃H₇, -C(CH₃)=C(CN)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-NH-cyclopropyl, -C(CH₃)=C(CN)-CO-NH-cyclobutyl, -C(CH₃)=C(CN)-CO-NH-cyclopentyl, -C(CH₃)=C(CN)-CO-NH-cyclohexyl, -C(CH₃)=C(CN)-CO-NH-cycloheptyl, -C(CH₃)=C(CN)-CO-NH-cyclooctyl, -C(CH₃)=C(CN)-CO-pyrrolidin-1-yl, -C(CH₃)=C(CN)-CO-piperidin-1-yl, -C(CH₃)=C(CN)-CO-morpholin-4-yl, -C(CH₃)=C(CN)-CO-NH-CH₂CH=C(CN)₂, -C(CH₃)=C(CN)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CN)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CN)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CN)-CO-NH-C₆H₅, -C(CH₃)=CH-CO-SCH₃, -C(CH₃)=CH-CO-SC₂H₅, -C(CH₃)=CH-CO-S-n-C₃H₇, -C(CH₃)=CH-CO-S-i-C₃H₇, -C(CH₃)=CH-CO-S-n-C₄H₉, -C(CH₃)=CH-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-SCH₃, -C(CH₃)=C(CH₃)-CO-SC₂H₅, -C(CH₃)=C(CH₃)CO-S-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-S-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-SCH₃, -C(CH₃)=C(C₂H₅)-CO-SC₂H₅, -C(CH₃)=C(C₂H₅)-CO-S-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-SCH₃, -C(CH₃)=C(Cl)-CO-SC₂H₅, -C(CH₃)=C(Cl)-CO-S-n-C₃H₇, -C(CH₃)=C(Cl)-CO-S-i-C₃H₇, -C(CH₃)=C(Cl)-CO-S-n-C₄H₉, -C(CH₃)=C(Cl)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-SCH₃, -C(CH₃)=C(Br)-CO-SC₂H₅, -C(CH₃)=C(Br)-CO-S-n-C₃H₇, -C(CH₃)=C(Br)-CO-S-i-C₃H₇, -C(CH₃)=C(Br)-CO-S-n-C₄H₉, -C(CH₃)=C(Br)-CO-S-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-SCH₃, -C(CH₃)=C(CN)-CO-SC₂H₅, -C(CH₃)=C(CN)-CO-S-n-C₃H₇, -C(CH₃)=C(CN)-CO-S-i-C₃H₇, -C(CH₃)=C(CN)-CO-S-n-C₄H₉, -C(CH₃)=C(CN)-CO-S-tert.-C₄H₉, -C(CH₃)=C(COCH₃)-CO-OCH₃, -C(CH₃)=C(COC₂H₅)-CO-OCH₃, -C(CH₃)=C(CO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COCH₃)-CO-OC₂H₅, -C(CH₃)=C(COC₂H₅)-CO-OC₂H₅, -C(CH₃)=C(CO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COCH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(COC₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-OCH₃, -C(CH₃)=C(CF₃)-CO-OC₂H₅, -C(CH₃)=C(CF₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CF₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(COOCH₃)₂, -C(CH₃)=C(COOC₂H₅)₂, -C(CH₃)=C(COOCH₃)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)₂, -C(CH₃)=CH-CH=CH-COOH, -C(CH₃)=CH-CH=CH-CO-OCH₃, -C(CH₃)=CH-CH=CH-CO-OC₂H₅, -C(CH₃)=CH-CH=C(COOCH₃)₂, -C(CH₃)=CH-CH=C(CN)-CO-OCH₃, -C(CH₃)=CH-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH₂, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -C(CH₃)=CH-(CH₂)₂-COOH, -C(CH₃)=CH-(CH₂)₂-CO-OCH₃, -C(CH₃)=CH-(CH₂)₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(COOCH₃)₂, -C(CH₃)=CH-CH₂-CH(COOC₂H₅)₂, -C(CH₃)=CH-CH₂-CH(CN)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CN)-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -C(CH₃)=CH-(CH₂)₂-CO-NH₂, -C(CH₃)=CH-(CH₂)₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-COOH, -C(CH₃)=CH-CH₂-CO-OCH₃, -C(CH₃)=CH-CH₂-CO-OC₂H₅, -C(CH₃)=C(COOCH₃)-CH₂-CO-OCH₃, -C(CH₃)=C(COOCH₃)-CH₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CO-NH₂, -C(CH₃)=CH-CH₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-CO-N(CH₃)₂.
wobei W für eine der folgenden Bedeutungen steht:
-CHO, -COCH₃, -COC₂H₅, -CO-n-C₃H₇, -CO-i-C₃H₇, -CO-n-C₄H₉, -CO-i-C₄H₉, -CO-s-C₄H₉, -CO-tert.-C₄H₉, -CO-CH₂CH=CH₂, -CO-CF₃, -COCCl₃, -COCH₂≡CH, -CO-cyclopropyl, -CO-cyclobutyl, -CO-cyclo­ pentyl, -CO-cyclohexyl, -CO-CN, -CO-COOCH₃, -CO-COOC₂H₅, -CH=NH, -CH=NCH₃, -CH=NC₂H₅, -CH=N-n-C₃H₅, -CH=N-i-C₃H₅, -CH=N-n-C₄H₉, -CH=NCH₂CH=CH₂, -CH=NCH₂CH=CH₂-CH₃, -CH=NCH₂C≡CH, -CH=NCH₂C≡C-CH₃, -CH=N-cyclopropyl, -CH=N-cyclobutyl, -CH=N-cyclopentyl, -CH=N-cyclohexyl, -CH=N-cycloheptyl, -CH=N-CH₂-CH₂Cl, -CH=N-CH₂Cl, -CH=N-C₆H₅, -CH=N-4-Br-C₆H₄, -CH=N-3-F-C₆H₄, -CH=N-4-F-C₆H₄, -CH=N-2-Cl-C₆H₄, -CH=N-3-Cl-C₆H₄, -CH=N-4-Cl-C₆H₄, -CH=N-2-Br-B₆H₄, -CH=N-2-F-C₆H₄, -CH=N-2-CH₃-C₆H₄, -CH=N-3-CH₃-C₆H₄, -CH=N-4-CH₃-C₆H₄, -CH=N-2-CF₃-C₆H₄, -CH-N-3-CF₃-C₆H₄, -CH=N-4-CF₃-C₆H₄, -CH=N-2-OCH₃-C₆H₄, -CH=N-3-OCH₃-C₆H₄, -CH=N-4-OCH₃-C₆H₄, -CH=N-4-NO₂-C₆H₄, -CH=N-4-CN-C₆H₄, -CH=N-2,4-(Cl, Cl)-C₆H₄, -CH=N-2,4-(CH₃, CH₃)-C₆H₄, -CH=N-CH₂OCH₃, -CH=N-CH₂OC₂H₅, -CH=N-CH₂CH₂OCH₃, -CH=N-CH₂CH₂OC₂H₅, -CH=N-OH, -CH=N-OCH₃, -CH=N-OC₂H₅, -CH=N-O-n-C₃H₇, -CH=N-O-i-C₃H₇, -CH=N-O-n-C₄H₉, -CH=N-O-i-C₄H₉, -CH=N-O-s-C₄H₉, -CH=N-O-tert.-C₄H₉, -CH=N-O-CH₂CH=CH₂, -CH=N-O-CH(CH₃)CH=CH₂, -CH=N-O-CH₂C≡CH, -CH=N-O-CH(CH₃)-C≡CH, -CH=N-O-CH₂-CH=CH-CH₃, -CH=N-O-CH₂-CH₂-Cl, -CH=N-O-CH₂-CH₂-F, -CH=N-O-CH₂CF₃, -CH=N-O-CH₂-CH=CHCl, -CH=N-O-CH₂-CCl=CH₂, -CH=N-O-CH₂-CBr=CH₂, -CH=N-O-CH₂-CH=CCl-CH₃, -CH=N-OC(O)CH₃, -CH=N-OC(O)C₂H₅, -CH=N-O-CH₂-CN, -CH=N-O-CH₂-CH=CH-CH₂-O-CH₃, -CH=N-O-CH₂-CH=CH-CH₂-O-tert.-C₄H₉, -CH=N-O-(CH₂)₃-C₆H₅, -CH=N-O-(CH₂)₄-C₆H₅, -CH=N-O-(CH₂)₄-4-Cl-C₆H₄, -CH=N-O-(CH₂)₄-4-OCH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-CH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-C₆H₅, -CH=N-O-CH₂CH=CH-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CH-3-OCH₃-C₆H₄, -CH=N-O-(CH₂)₂CH=CH-4-F-C₆H₄, -CH=N-O-(CH₂)CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CHCH₂-4-OCH₃-C₆H₄, -CH=N-O-CH₂-CH=C(CH₃)-C₆H₅, -CH=N-O-(CH₂)₂CH=CH-3,4(Cl,Cl)-C₆H₃, -CH=N-O-(CH₂)₃C≡C-4-F-C₆H₄, -CH₂=N-OCHOCH₃, -CH=N-OC₂H₄OCH₃, -CH=N-OCH₂OC₂H₅, -CH=N-OCH(CH₃)OCH₃, -CH=N-OCH(CH₃)COOCH₃, -CH=N-OCH(CH₃)COO-n-C₄H₉, -CH=N-NH₂, -CH=N-NHCH₃, -CH=N-NHC₂H₅, -CH=N-NH-n-C₃H₇, -CH=N-NH-i-C₃H₇, -CH=N-NH-n-C₄H₉, -CH=N-NH-i-C₄H₉, -CH=N-NH-s-C₄H₉, -CH=N-NH-tert.-C₄H₉, -CH=N-NH-cyclopropyl, -CH=N-NH-cyclobutyl, -CH=N-NH-cyclopentyl, -CH=N-NH-cyclohexyl, -CH=N-NH-cycloheptyl, -CH=N-N(CH₃)₂, -CH=N-N(C₂H₅)₂, -CH=N-N(C₃H₇)₂, -CH=N-N(i-C₃H₇)(CH₃), -CH=N-NHCH₂-C=CH, -CH=N-NHCH₂-C≡CH, -CH=N-N(CH₃)-CH₂-C≡CH, -CH=N-NHCH₂CF₃, - 99999 00070 552 001000280000000200012000285919988800040 0002004131038 00004 99880CH=N-NH-CO-CH₃, -CH=N-NH-CO-CH₂H₅, -CH=N-NH-COOCH₃, -CH=N-NH-COOC₂H₅, -CH=N-NH-COO-tert.-C₄H₉, -CH=N-pyrrolidin-1-yl, -CH=N-piperidin-1-yl, -CH=N-morpholin-4-yl, -CH=N-NH-C₆H₅, -CH=N-NH-(4-Cl-C₆H₄), -CH=N-NH-(4-NO₂-C₆H₄), -CH=N-NH-(4-F-C₆H₄), -CH=N-NH-(4-CH₃O-C₆H₄), -CH=N-NH-(2,4-Cl₂-C₆H₃), -CH=N-NH-(2,4-(NO₂)₂-C₆H₃), -CH=N-NH-CO-NH₂, -CH=N-NH-CO-NHCH₃, -CH=N-NH-CO-NHC₂H₅, -CH=N-NH-CO-N(CH₃)₂, -CH=CH-COOH, -CH=CH-CO-OCH₃, -CH=CH-CO-OC₂H₅, -CH=CH-CO-O-n-C₃H₇, -CH=CH-CO-O-i-C₃H₇, -CH=CH-CO-O-n-C₄H₉, -CH=CH-CO-O-tert.-C₄H₉, -CH=CH-CO-O-cyclopropyl, -CH=CH-CO-O-cyclobutyl, -CH=CH-CO-O-cyclopentyl, -CH=CH-CO-O-cyclohexyl, -CH=CH-CO-O-cycloheptyl, -CH=C(CH₃)-COOH, -CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CO-O-n-C₃H₇, -CH=C(CH₃)-CO-O-i-C₃H₇, -CH=C(CH₃)-CO-O-n-C₄H₉, -CH=C(CH₃)-CO-O-tert.-C₄H₉, -CH=C(CH₃)-CO-O-cyclopropyl, -CH=C(CH₃)-CO-O-cyclobutyl, -CH=C(CH₃)-CO-O-cyclopentyl, -CH=C(CH₃)-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cycloheptyl, -CH=C(C₂H₅)-COOH, -CH=C(C₂H₅)-CO-OCH₃, -CH=C(C₂H₅)-CO-OC₂H₅, -CH=C(C₂H₅)-CO-O-n-C₃H₇, -CH=C(C₂H₅)-CO-O-i-C₃H₇, -CH=C(C₂H₅)-CO-O-n-C₄H₉, -CH=C(C₂H₅)-CO-O-tert.-C₄H₉, -CH=C(C₂H₅)-CO-O-cyclopropyl, -CH=C(₂H₅)-CO-O-cyclobutyl, -CH=C(C₂H₅)-CO-O-cyclopentyl, -CH=C(C₂H₅)-CO-O-cyclohexyl, -CH=C(C₂H₅)-CO-O-cycloheptyl, -CH=C(Cl)-COOH, -CH=C(Cl)-CO-OCH₃, -CH=C(Cl)-CO-OC₂H₅, -CH=C(Cl)-CO-O-n-C₃H₇, -CH=C(Cl)-CO-O-i-C₃H₇, -CH=C(Cl)-CO-O-n-C₄H₉, -CH=C(Cl)-CO-O-tert.-C₄H₉, -CH=C(Cl)-CO-O-cyclopropyl, -CH=C(Cl)-CO-O-cyclobutyl, -CH=C(Cl)-CO-O-cyclopentyl, -CH=C(Cl)-CO-O-cyclohexyl, -CH=C(Cl)-CO-O-cycloheptyl, -CH=C(Br)-COOH, -CH=C(Br)-CO-OCH₃, -CH=C(Br)-CO-OC₂H₅, -CH=C(Br)-CO-O-n-C₃H₇, -CH=C(Br)-CO-O-i-C₃H₇, -CH=C(Br)-CO-O-n-C₄H₉, -CH=C(Br)-CO-O-tert.-C₄H₉, -CH=C(Br)-CO-O-cyclopropyl, -CH=C(Br)-CO-O-cyclobutyl, -CH=C(Br)-CO-O-cyclopentyl, -CH=C(Br)-CO-O-cyclohexyl, -CH=C(Br)-CO-O-cycloheptyl, -CH=C(CN)-COOH, -CH=C(CN)-CO-OCH₃, -CH=C(CN)-CO-OC₂H₅, -CH=C(CN)-CO-O-n-C₃H₇, -CH=C(CN)-CO-O-i-C₃H₇, -CH=C(CN)-CO-O-n-C₄H₉, -CH=C(CN)-CO-O-tert.-C₄H₉, -CH=C(CN)-CO-O-cyclopropyl, -CH=C(CN)-CO-O-cyclobutyl, -CH=C(CN)-CO-O-cyclopentyl, -CH=C(CN)-CO-O-cyclohexyl, -CH=C(CN)-CO-O-cycloheptyl, -CH=CH-CO-OCH₂-OCH₃, -CH=CH-CO-OCH₂-OC₂H₅, -CH=CH-CO-OCH₂-O-n-C₃H₅, -CH=CH-CO-OCH₂-O-i-C₃H₅, -CH=CH-CO-OCH(CH₃)-OCH₃, -CH=CH-CO-OCH(CH₃)-OC₂H₅, -CH=CH-CO-O-CH₂CH₂-OCH₃, -CH=CH-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-OCH₃, -CH=C(CH₃)-CO-OCH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-O-n-C₃H₅, -CH=C(CH₃)-CO-OCH₂-O-i-C₃H₅, -CH=C(CH₃)-CO-OCH(CH₃)-OCH₃, -CH=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CH₃)-CO-O-CH₂CH₂-OCH₃, -CH=C(CH₃)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-OCH₃, -CH=C(C₂H₅)-CO-OCH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-O-n-C₃H₅, -CH=C(C₂H₅)-CO-OCH₂-O-i-C₃H₅, -CH=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -CH=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OCH₃, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-OCH₃, -CH=C(Cl)-CO-OCH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-O-n-C₃H₅, -CH=C(Cl)-CO-OCH₂-O-i-C₃H₅, -CH=C(Cl)-CO-OCH(CH₃)-OCH₃, -CH=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Cl)-CO-O-CH₂CH₂-OCH₃, -CH=C(Cl)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-OCH₃, -CH=C(Br)-CO-OCH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-O-n-C₃H₅, -CH=C(Br)-CO-OCH₂-O-i-C₃H₅, -CH=C(Br)-CO-OCH(CH₃)-OCH₃, -CH=C(Br)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Br)-CO-O-CH₂CH₂-OCH₃, -CH=C(Br)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-OCH₃, -CH=C(CN)-CO-OCH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-O-n-C₃H₅, -CH=C(CN)-CO-OCH₂-O-i-C₃H₅, -CH=C(CN)-CO-OCH(CH₃)-OCH₃, -CH=C(CN)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CN)-CO-O-CH₂CH₂-OCH₃, -CH=C(CN)-CO-O-CH₂CH₂-OC₂H₅, -CH=CH-CO-OCH₂-CF₃, -CH=CH-CO-OCH₂-CCl₃, -CH=CH-CO-OCH₂-oxiranyl, -CH=CH-CO-O(CH₂)₃-Br, -CH=CH-CO-OCH₂-CH=CH₂, -CH=CH-CO-OCH₂-C≡CH, -CH=CH-CO-OCH₂-CN, -CH=CH-CO-O(CH₂)₂-CN, -CH=C(CH₃)-CO-OCH₂-CF₃, -CH=C(CH₃)-CO-OCH₂-CCl₃, -CH=C(CH₃)-CO-OCH₂-oxiranyl, -CH=C(CH₃)-CO-O(CH₂)₃-Br, -CH=C(CH₃)-CO-OCH₂-CH=CH₂, -CH=C(CH₃)-CO-OCH₂-C≡CH, -CH=C(CH₃)-CO-OCH₂-CN, -CH=C(CH₃)-CO-O(CH₂)₂-CN, -CH=C(C₂H₅)-CO-OCH₂-CF₃, -CH=C(C₂H₅)-CO-OCH₂-CCl₃, -CH=C(C₂H₅)-CO-OCH₂-oxiranyl, -CH=C(C₂H₅)-CO-O(CH₂)₃-Br, -CH=C(C₂H₅)-CO-OCH₂-CH=CH₂, -CH=C(C₂H₅)-CO-OCH₂-C≡CH, -CH=C(C₂H₅)-CO-OCH₂-CN, -CH=C(C₂H₅)-CO-O(CH₂)₂-CN, -CH=C(Cl)-CO-OCH₂-CF₃, -CH=C(Cl)-CO-OCH₂-CCl₃, -CH=C(Cl)-CO-OCH₂-oxiranyl, -CH=C(Cl)-CO-O(CH₂)₃-Br, -CH=C(Cl)-CO-OCH₂-CH=CH₂, -CH=C(Cl)-CO-OCH₂-C≡CH, -CH=C(Cl)-CO-OCH₂-CN, -CH=C(Cl)-CO-O(CH₂)₂-CN, -CH=C(Br)-CO-OCH₂-CF₃, -CH=C(Br)-CO-OCH₂-CCl₃, -CH=C(Br)-CO-OCH₂-oxiranyl, -CH=C(Br)-CO-O(CH₂)₃-Br, -CH=C(Br)-CO-OCH₂-CH=CH₂, -CH=C(Br)-CO-OCH₂-C≡CH, -CH=C(Br)-CO-OCH₂-CN, -CH=C(Br)-CO-O(CH₂)₂-CN, -CH=C(CN)-CO-OCH₂-CF₃, -CH=C(CN)-CO-OCH₂-CCl₃, -CH=C(CN)-CO-OCH₂-oxiranyl, -CH=C(CN)-CO-O(CH₂)₃-Br, -CH=C(CN)-CO-OCH₂-CH=CH₂, -CH=C(CN)-CO-OCH₂-C≡CH, -CH=C(CN)-CO-OCH₂-CN, -CH=C(CN)-CO-O(CH₂)₂-CN, -CH=CH-CO-CH₃, -CH=CH-CO-C₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-i-C₃H₇, -CH=CH-CO-n-C₄H₉, -CH=CH-CO-tert.-C₄H₉, -CH=CH-CO-CH₂Cl, -CH=CH-CO-CH₂Br, -CH=CH-CO-CHCl₂, -CH=CH-CO-CH₂-OCH₃, -CH=CH-CO-CH(OCH₃)₂, -CH=CH-CO-CH₂-SCH₃, -CH=C(CH₃)-CO-CH₃, -CH=C(CH₃)-CO-C₂H₅, -CH=C(CH₃)-CO-n-C₃H₇, -CH=C(CH₃)-CO-i-C₃H₇, -CH=C(CH₃)-CO-n-C₄H₉, -CH=C(CH₃)-CO-tert.-C₄H₉, -CH=C(CH₃)-CO-CH₂Cl, -CH=C(CH₃)-CO-CH₂Br, -CH=C(CH₃)-CO-CHCl₂, -CH=C(CH₃)-CO-CH₂-OCH₃, -CH=C(CH₃)-CO-CH(OCH₃)₂, -CH=C(CH₃)-CO-CH₂-SCH₃, -CH=C(C₂H₅)-CO-CH₃, -CH=C(C₂H₅)-CO-C₂H₅, -CH=C(C₂H₅)-CO-n-C₃H₇, -CH=C(C₂H₅)-CO-i-C₃H₇, -CH=C(C₂H₅)-CO-n-C₄H₉, -CH=C(C₂H₅)-CO-tert.-C₄H₉, -CH=C(C₂H₅)-CO-CH₂Cl, -CH=C(C₂H₅)-CO-CH₂Br, -CH=C(C₂H₅)-CO-CHCl₂, -CH=C(C₂H₅)-CO-CH₂-OCH₃, -CH=C(C₂H₅)-CO-CH(OCH₃)₂, -CH=C(C₂H₅)-CO-CH₂-SCH₃, -CH=C(Cl)-CO-CH₃, -CH=C(Cl)-CO-C₂H₅, -CH=C(Cl)-CO-n-C₃H₇, -CH=C(Cl)-CO-i-C₃H₇, -CH=C(Cl)-CO-n-C₄H₉, -CH=C(Cl)-CO-tert.-C₄H₉, -CH=C(Cl)-CO-CH₂Cl, -CH=C(Cl)-CO-CH₂Br, -CH=C(Cl)-CO-CHCl₂, -CH=C(Cl)-CO-CH₂-OCH₃, -CH=C(Cl)-CO-CH(OCH₃)₂, -CH=C(Cl)-CO-CH₂-SCH₃, -CH=C(Br)-CO-CH₃, -CH=C(Br)-CO-C₂H₅, -CH=C(Br)-CO-n-C₃H₇, -CH=C(Br)-CO-i-C₃H₇, -CH=C(Br)-CO-n-C₄H₉, -CH=C(Br)-CO-tert.-C₄H₉, -CH=C(Br)-CO-CH₂Cl, -CH=C(Br)-CO-CH₂Br, -CH=C(Br)-CO-CHCl₂, -CH=C(Br)-CO-CH₂-OCH₃, -CH=C(Br)-CO-CH(OCH₃)₂, -CH=C(Br)-CO-CH₂-SCH₃, -CH=C(CN)-CO-CH₃, -CH=C(CN)-CO-C₂H₅, -CH=C(CN)-CO-n-C₃H₇, -CH=C(CN)-CO-i-C₃H₇, -CH=C(CN)-CO-n-C₄H₉, -CH=C(CN)-CO-tert.-C₄H₉, -CH=C(CN)-CO-CH₂Cl, -CH=C(CN)-CO-CH₂Br, -CH=C(CN)-CO-CHCl₂, -CH=C(CN)-CO-CH₂-OCH₃, -CH=C(CN)-CO-CH(OCH₃)₂, -CH=C(CN)-CO-CH₂-SCH₃, -CH=CH-CO-C₆H₅, -CH=CH-CO-(4-Cl-C₆H₄), -CH=C(CH₃)-CO-C₆H₅, -CH=C(CH₃)-CO-(4-Cl-C₆H₄), -CH=C(C₂H₅)-CO-C₆H₅, -CH=C(C₂H₅)-CO-(4-Cl-C₆H₄), -CH=C(Cl)-CO-C₆H₅, -CH=C(Br)-CO-C₆H₅, -CH=C(CN)-CO-C₆H₅, -CH=CH-CO-NH₂, -CH=CH-CO-NHCH₃, -CH=CH-CO-N(CH₃)₂, -CH=CH-CO-NH-C₂H₅, -CH=CH-CO-N(C₂H₅)₂, -CH=CH-CO-NH-n-C₃H₇, -CH=CH-CO-NH-i-C₃H₇, -CH=CH-CO-NH-tert.-C₄H₉, -CH=CH-CO-NH-cyclopropyl, -CH=CH-CO-NH-cyclobutyl, -CH=CH-CO-NH-cyclopentyl, -CH=CH-CO-NH-cyclohexyl, -CH=CH-CO-NH-cycloheptyl, -CH=CH-CO-NH-cyclooctyl, -CH=CH-CO-pyrrolidin-1-yl, -CH=CH-CO-piperidin-1-yl, -CH=CH-CO-morpholin-4-yl, -CH=CH-CO-NH-CH₂CH=CH₂, -CH=CH-CO-NH-CH₂C≡CH, -CH=CH-CO-N(CH₃)-CH₂C≡CH, -CH=CH-CO-NH-(CH₂)₂Cl, -CH=CH-CO-NH-C₆H₅, -CH=C(CH₃)-CO-NH₂, -CH=C(CH₃)-CO-NHCH₃, -CH=C(CH₃)-CO-N(CH₃)₂, -CH=C(CH₃)-CO-NH-C₂H₅, -CH=C(CH₃)-CO-N(C₂H₅)₂, -CH=C(CH₃)-CO-NH-n-C₃H₇, -CH=C(CH₃)-CO-NH-i-C₃H₇, -CH=C(CH₃)-CO-NH-tert.-C₄H₉, -CH=C(CH₃)-CO-NH-cyclopropyl, -CH=C(CH₃)-CO-NH-cyclobutyl, -CH=C(CH₃)-CO-NH-cyclopentyl, -CH=C(CH₃)-CO-NH-cyclohexyl, -CH=C(CH₃)-CO-NH-cycloheptyl, -CH=C(CH₃)-CO-NH-cyclooctyl, -CH=C(CH₃)-CO-pyrrolidin-1-yl, -CH=C(CH₃)-CO-piperidin-1-yl, -CH=C(CH₃)-CO-morpholin-4-yl, -CH=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -CH=C(CH₃)-CO-NH-CH₂C≡CH, -CH=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CH₃)-CO-NH-(CH₂)₂Cl, -CH=C(CH₃)-CO-NH-C₆H₅, -CH=C(C₂H₅)-CO-NH₂, -CH=C(C₂H₅)-CO-NHCH₃, -CH=C(C₂H₅)-CO-N(CH₃)₂, -CH=C(C₂H₅)-CO-NH-C₂H₅, -CH=C(C₂H₅)-CO-N(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-n-C₃H₇, -CH=C(C₂H₅)-CO-NH-i-C₃H₇, -CH=C(C₂H₅)-CO-NH-tert.-C₄H₉, -CH=C(C₂H₅)-CO-NH-cyclopropyl, -CH=C(C₂H₅)-CO-NH-cyclobutyl, -CH=C(C₂H₅)-CO-NH-cyclopentyl, -CH=C(C₂H₅)-CO-NH-cyclohexyl, -CH=C(C₂H₅)-CO-NH-cycloheptyl, -CH=C(C₂H₅)-CO-NH-cyclooctyl, -CH=C(C₂H₅)-CO-pyrrolidin-1-yl, -CH=C(C₂H₅)-CO-piperidin-1-yl, -CH=C(C₂H₅)-CO-morpholin-4-yl, -CH=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-CH₂C≡CH, -CH=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -CH=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -CH=C(C₂H₅)-CO-NH-C₆H₅, -CH=C(Cl)-CO-NH₂, -CH=C(Cl)-CO-NHCH₃, -CH=C(Cl)-CO-N(CH₃)₂, -CH=C(Cl)-CO-NH-C₂H₅, -CH=C(Cl)-CO-N(C₂H₅)₂, -CH=C(Cl)-CO-NH-n-C₃H₇, -CH=C(Cl)-CO-NH-i-C₃H₇, -CH=C(Cl)-CO-NH-tert.-C₄H₉, -CH=C(Cl)-CO-NH-cyclopropyl, -CH=C(Cl)-CO-NH-cyclobutyl, -CH=C(Cl)-CO-NH-cyclopentyl, -CH=C(Cl)-CO-NH-cyclohexyl, -CH=C(Cl)-CO-NH-cycloheptyl, -CH=C(Cl)-CO-NH-cyclooctyl, -CH=C(Cl)-CO-pyrrolidin-1-yl, -CH=C(Cl)-CO-piperidin-1-yl, -CH=C(Cl)-CO-morpholin-4-yl, -CH=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -CH=C(Cl)-CO-NH-CH₂C≡CH, -CH=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Cl)-CO-NH-(CH₂)₂Cl, -CH=C(Cl)-CO-NH-C₆H₅, -CH=C(Br)-CO-NH₂, -CH=C(Br)-CO-NHCH₃, -CH=C(Br)-CO-N(CH₃)₂, -CH=C(Br)-CO-NH-C₂H₅, -CH=C(Br)-CO-N(C₂H₅)₂, -CH=C(Br)-CO-NH-n-C₃H₇, -CH=C(Br)-CO-NH-i-C₃H₇, -CH=C(Br)-CO-NH-tert.-C₄H₉, -CH=C(Br)-CO-NH-cyclopropyl, -CH=C(Br)-CO-NH-cyclobutyl, -CH=C(Br)-CO-NH-cyclopentyl, -CH=C(Br)-CO-NH-cyclohexyl, -CH=C(Br)-CO-NH-cycloheptyl, -CH=C(Br)-CO-NH-cyclooctyl, -CH=C(Br)-CO-pyrrolidin-1-yl, -CH=C(Br)-CO-piperidin-1-yl, -CH=C(Br)-CO-morpholin-4-yl, -CH=C(Br)-CO-NH-CH₂CH=C(Br)₂, -CH=C(Br)-CO-NH-CH₂C≡CH, -CH=C(Br)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Br)-CO-NH-(CH₂)₂Cl, -CH=C(Br)-CO-NH-C₆H₅, -CH=C(CN)-CO-NH₂, -CH=C(CN)-CO-NHCH₃, -CH=C(CN)-CO-N(CH₃)₂, -CH=C(CN)-CO-NH-C₂H₅, -CH=C(CN)-CO-N(C₂H₅)₂, -CH=C(CN)-CO-NH-n-C₃H₇, -CH=C(CN)-CO-NH-i-C₃H₇, -CH=C(CN)-CO-NH-tert.-C₄H₉, -CH=C(CN)-CO-NH-cyclopropyl, -CH=C(CN)-CO-NH-cyclobutyl, -CH=C(CN)-CO-NH-cyclopentyl, -CH=C(CN)-CO-NH-cyclohexyl, -CH=C(CN)-CO-NH-cycloheptyl, -CH=C(CN)-CO-NH-cyclooctyl, -CH=C(CN)-CO-pyrrolidin-1-yl, -CH=C(CN)-CO-piperidin-1-yl, -CH=C(CN)-CO-morpholin-4-yl, -CH=C(CN)-CO-NH-CH₂CH=C(CN)₂, -CH=C(CN)-CO-NH-CH₂C≡CH, -CH=C(CN)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CN)-CO-NH-(CH₂)₂Cl, -CH=C(CN)-CO-NH-C₆H₅, -CH=CH-CO-SCH₃, -CH=CH-CO-SC₂H₅, -CH=CH-CO-S-n-C₃H₇, -CH=CH-CO-S-i-C₃H₇, -CH=CH-CO-S-n-C₄H₉, -CH=CH-CO-S-tert.-C₄H₉, -CH=C(CH₃)-CO-SCH₃, -CH=C(CH₃)-CO-SC₂H₅, -CH=C(CH₃)-CO-S-n-C₃H₇, -CH=C(CH₃)-CO-S-i-C₃H₇, -CH=C(CH₃)-CO-S-n-C₄H₉, -CH=C(CH₃)-CO-S-tert.-C₄H₉, -CH=C(C₂H₅)-CO-SCH₃, -CH=C(C₂H₅)-CO-SC₂H₅, -CH=C(C₂H₅)-CO-S-n-C₃H₇, -CH=C(C₂H₅)-CO-S-i-C₃H₇, -CH=C(C₂H₅)-CO-S-n-C₄H₉, -CH=C(C₂H₅)-CO-S-tert.-C₄H₉, -CH=C(Cl)-CO-SCH₃, -CH=C(Cl)-CO-SC₂H₅, -CH=C(Cl)-CO-S-n-C₃H₇, -CH=C(Cl)-CO-S-i-C₃H₇, -CH=C(Cl)-CO-S-n-C₄H₉, -CH=C(Cl)-CO-S-tert.-C₄H₉, -CH=C(Br)-CO-SCH₃, -CH=C(Br)-CO-SC₂H₅, -CH=C(Br)-CO-S-n-C₃H₇, -CH=C(Br)-CO-S-i-C₃H₇, -CH=C(Br)-CO-S-n-C₄H₉, -CH=C(Br)-CO-S-tert.-C₄H₉, -CH=C(CN)-CO-SCH₃, -CH=C(CN)-CO-SC₂H₅, -CH=C(CN)-CO-S-n-C₃H₇, -CH=C(CN)-CO-S-i-C₃H₇, -CH=C(CN)-CO-S-n-C₄H₉, -CH=C(CN)-CO-S-tert.-C₄H₉, -CH=C(COCH₃)-CO-OCH₃, -CH=C(COC₂H₅)-CO-OCH₃, -CH=C(CO-n-C₃H₇)-CO-OCH₃, -CH=C(COCH₃)-CO-OC₂H₅, -CH=C(COC₂H₅)-CO-OC₂H₅, -CH=C(CO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COCH₃)-CO-O-n-C₃H₇, -CH=C(COC₂H₅)-CO-O-n-C₃H₇, -CH=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-OCH₃, -CH=C(CF₃)-CO-OC₂H₅, -CH=C(CF₃)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-O-i-C₃H₇, -CH=C(CF₃)-CO-O-n-C₄H₉, -CH=C(CF₃)-CO-O-tert.-C₄H₉, -CH=C(COOCH₃)₂, -CH=C(COOC₂H₅)₂, -CH=C(COOCH₃)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)-CO-OCH₃, -CH=C(COO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)₂, -CH=CH-CH=CH-COOH, -CH=CH-CH=CH-CO-OCH₃, -CH=CH-CH=CH-CO-OC₂H₅, -CH=CH-CH=C(COOCH₃)₂, -CH=CH-CH=C(CN)-CO-OCH₃, -CH=CH-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-OCH₃, -CH=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CH=C(Cl)-CO-OCH₃, -CH=C(CH₃)-CH=C(Br)-CO-OCH₃, -CH=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-NH₂, -CH=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -CH=CH-(CH₂)₂-COOH, -CH=CH-(CH₂)₂-CO-OCH₃, -CH=CH-(CH₂)₂-CO-OC₂H₅, -CH=CH-CH₂-CH(COOCH₃)₂, -CH=CH-CH₂-CH(COOC₂H₅)₂, -CH=CH-CH₂-CH(CN)-CO-OCH₃, -CH=CH-CH₂-CH(CN)-CO-OC₂H₅, -CH=CH-CH₂-CH(CH₃)-CO-OCH₃, -CH=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -CH=CH-(CH₂)₂-CO-NH₂, -CH=CH-(CH₂)₂-CO-NH-CH₃, -CH=CH-CH₂-COOH, -CH=CH-CH₂-CO-OCH₃, -CH=CH-CH₂-CO-OC₂H₅, -CH=C(COOCH₃)-CH₂-CO-OCH₃, -CH=C(COOCH₃)-CH₂-CO-OC₂H₅, -CH=CH-CH₂-CO-NH₂, -CH=CH-CH₂-CO-NH-CH₃, -CH=CH-CH₂-CO-N(CH₃)₂, -CH(OCH₃)₂, -CH(SCH₃)₂, -CH(OC₂H₅)₂, -CH(SC₂H₅)₂, -CH(O-n-C₃H₇)₂, -CH(O-i-C₃H₇)₂, -CH(S-n-C₃H₇)₂, -CH(S-i-C₃H₇)₂, -CH(O-n-C₄H₉)₂, -CH(O-i-C₄H₉)₂, -CH(O-s-C₄H₉)₂, -CH(O-tert.-C₄H₉)₂, -CH(S-n-C₄H₉)₂, -CH(S-i-C₄H₉)₂, -CH(S-s-C₄H₉)₂, -CH(S-tert.-C₄H₉)₂, -CH(OC₅H₁₁)₂, 1,3-Dioxolan-2-yl, 1,3-Dithio­ lan-2-yl, 1,3-Oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 4-Methyl-1,3-dithiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 5-Methyl-1,3-oxathiolan-2-yl, 4-Ethyl-1,3-dioxolan-2-yl, 4-Ethyl- 1,4-dithiolan-2-yl, 4-Ethyl-1,3-oxathiolan-2-yl, 5-Ethyl-1,3-oxa­ thiolan-2-yl, 4,5-Dimethyl-1,3-dioxolan-2-yl, 4,4-Dimethyl-1,3- dioxolan-2-yl, 4,5-Dimethyl-1,3-dithiolan-2-yl, 5,5-Dimethyl-1,3- dithiolan-2-yl, 4,5-Dimethyl-1,3-oxathiolan-2-yl, 5,5-Dimethyl- 1,3-oxathiolan-2-yl, 4,4-Dimethyl-1,3-oxathiolan-2-yl, 4-Vinyl- 1,3-dioxolan-2-yl, 4-Vinyl-1,3-dithiolan-2-yl, 4-Vinyl-1,3-oxa­ thiolan-2-yl, 5-Vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3- dioxolan-2-yl, 4-Chlormethyl-1,3-dithiolan-2-yl, 4-Chlormethyl- 1,3-oxathiolan-2-yl, 5-Chlormethyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-1,3-dithio­ lan-2-yl, 4-Hydroxymethyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl- 1,3-oxathiolan-2-yl, 4-Methoxymethyl-1,3-dioxolan-2-yl, 4-Allyl­ oxymethyl-1,3-dioxolan-2-yl, 4-Propargyloxymethyl-1,3-dioxolan- 2-yl, 4-Acetoxymethyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-1,3-dithiolan-2-yl, 4-Propargyl­ oxymethyl-1,3-dithiolan-2-yl, 4-Acetoxymethyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-1,3-oxa­ thiolan-2-yl, 4-Allyloxymethyl-1,3-oxathiolan-2-yl, 5-Allyloxy- methyl-1,3-oxathiolan-2-yl, 4-Propargyloxymethyl-1,3-oxathiolan- 2-yl, 5-Propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxymethyl- 1,3-oxathiolan-2-yl, 5-Acetoxymethyl-1,3-oxathiolan-2-yl, 4-Methylthiomethyl-1,3-dioxolan-2-yl, 4-Methylthiomethyl-1,3- dithiolan-2-yl, 4-Carboxy-1,3-dioxolan-2-yl, 4-Carboxy-1,3- dithiolan-2-yl, 4-Methoxycarbonyl-1,3-dioxolan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-1,3-di­ thiolan-2-yl, 4-n-Butoxycarbonyl-1,3-dithiolan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-4-methyl- 1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-di­ thiolan-2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-1,3- dithiolan-2-yl, 1,3-Dioxan-2-yl, 1,3-Dithian-2-yl, 1,3-Oxathian- 2-yl, 5-Methyl-1,3-dioxan-2-yl, 5-Methyl-1,3-dithian-2-yl, 5-Methyl-1,3-oxathian-2-yl, 5,5-Dimethyl-1,3-dioxan-2-yl, 4,6-Di­ methyl-1,3-dioxan-2-yl, 4,4-Dimethyl-1,3-dioxan-2-yl, 5,5-Di­ methyl-1,3-dithian-2-yl, 4,6-Dimethyl-1,3-dithian-2-yl, 4,4-Di­ methyl-1,3-dithian-2-yl, 5,5-Dimethyl-1,3-oxathian-2-yl, 4,4-Di­ methyl-1,3-oxathian-2-yl, 6,6-Dimethyl-1,3-oxathian-2-yl, 4-Hydroxymethyl-1,3-dioxan-2-yl, 4-Methoxymethyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-1,3-dioxan-2- yl, 4-Hydroxymethyl-1,3-dithian-2-yl, 4-Methoxymethyl-1,3-di­ thian-2-yl, 4-Allyloxymethyl-1,3-dithian-2-yl, 4-Acetoxymethyl- 1,3-dithian-2-yl, 4-Chlormethyl-1,3-dioxan-2-yl, 4-Chlormethyl- 1,3-dithian-2-yl, 1,3-Dioxepan-2-yl, 1,3-Dithiepan-2-yl, 1,3-Di­ oxep-5-en-2-yl, 4-Methoxycarbonyl-1,3-dioxan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-1,3-dithian- 4-yl, 4-n-Butoxycarbonyl-1,3-dithian-2-yl, 4-Methoxycarbonyl-4- methyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxan-2- yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-4-methyl- 1,3-dithian-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithian-2-yl, -C(CH₃)(OCH₃)₂, -C(CH₃)(SCH₃)₂, -C(CH₃)(OC₂H₅)₂, -C(CH₃)(SC₂H₅)₂, -C(CH₃)(O-n-C₃H₇)₂, -C(CH₃)(O-i-C₃H₇)₂, -C(CH₃)(S-n-C₃H₇)₂, -C(CH₃)(S-i-C₃H₇)₂, -C(CH₃)(O-n-C₄H₉)₂, -C(CH₃)(O-i-C₄H₉)₂, -C(CH₃)(O-s-C₄H₉)₂, -C(CH₃)(O-tert.-C₄H₉)₂, -C(CH₃)(S-n-C₄H₉)₂, -C(CH₃)(S-i-C₄H₉)₂, -C(CH₃)(S-s-C₄H₉)₂, -C(CH₃)(S-tert.-C₄H₉)₂, -C(CH₃)(O-n-C₅H₁₁)′′, 2-Methyl-1,3-dioxolan-2-yl, 2-Methyl-1,3-di­ thiolan-2-yl, 2-Methyl-1,3-oxathiolan-2-yl, 2,4-Dimethyl-1,3- dioxolan-2-yl, 2,4-Dimethyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-1,3- oxathiolan-2-yl, 2,5-Dimethyl-1,3-oxathiolan-2-yl, 4-Ethyl-2- methyl-1,3-dioxolan-2-yl, 4-Ethyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Ethyl-2-methyl-1,3- oxathiolan-2-yl, 2,4,5-Trimethyl-1,3-dioxolan-2-yl, 2,4,4-Tri­ methyl-1,3-dioxolan-2-yl, 2,4,5-Trimethyl-1,3-dithiolan-2-yl, 2,4,4-Trimethyl-1,3-dithiolan-2-yl, 2,4,5-Trimethyl-1,3-oxathio­ lan-2-yl, 2,4,4-Trimethyl-1,3-oxathiolan-2-yl, 2-Methyl-4-vinyl- 1,3-dioxolan-2-yl, 2-Methyl-4-vinyl-1,3-dithiolan-2-yl, 2-Methyl- 4-vinyl-1,3-oxathiolan-2-yl, 2-Methyl-5-vinyl-1,3-oxathiolan-2- yl, 4-Chlormethyl-2-methyl-1,3-dioxolan-2-yl, 4-Chlormethyl-2- methyl-1,3-dithiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-oxathio­ lan-2-yl, 5-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Hydroxy­ methyl-2-methyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-2- methyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dioxolan- 2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxy- 2-methyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dithiolan-2-yl, 4-Acetoxy-2- methyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-oxathio­ lan-2-yl, 5-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Allyl­ oxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Allyloxymethyl-2- methyl-1,3-oxathiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3- oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3-oxathiolan-2- yl, 4-Acetoxy-2-methyl-1,3-oxathiolan-2-yl, 5-Acetoxy-2-methyl- 1,3-oxathiolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dioxolan-2- yl, 2-Methyl-4-methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-2- methyl-1,3-dioxolan-2-yl, 4-Carboxy-2-methyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-2- methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-2-methyl-1,3-dioxo­ lan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-Eth­ oxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-2- methyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-di­ oxolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-ethoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4- ethoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-n-butoxy­ carbony-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl-1,3- dithiolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-dioxan-2- yl, 2-Methyl-1,3-dithian-2-yl, 2-Methyl-1,3-oxathian-2-yl, 2,5- Dimethyl-1,3-dioxan-2-yl, 2,5-Dimethyl-1,3-dithian-2-yl, 2,5-Di­ methyl-1,3-oxathian-2-yl, 2,5,5-Trimethyl-1,3-dioxan-2-yl, 2,4,6- Trimethyl-1,3-dioxan-2-yl, 2,4,4-Trimethyl-1,3-dioxan-2-yl, 2,5,5-Trimethyl-1,3-dithian-2-yl, 2,4,6-Trimethyl-1,3-dithian-2- yl, 2,4,4-Trimethyl-1,3-dithian-2-yl, 2,5,5-Trimethyl-1,3-oxa­ thian-2-yl, 2,4,4-Trimethyl-1,3-oxathian-2-yl, 2,6,6-Trimethyl- 1,3-oxathian-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-2- methyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dithian-2-yl, 4-Methoxymethyl-2- methyl-1,3-dithian-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithian-2- yl, 4-Acetoxymethyl-2-methyl-1,3-dithian-2-yl, 4-Chlormethyl-2- methyl-1,3-dioxan-2-yl, 4-Chlormethyl-2-methyl-1,3-dithian-2-yl, -C(CH₃)=NH, -C(CH₃)=N-CH₃, -C(CH₃)=N-C₂H₅, -C(CH₃)=N-n-C₃H₇, -(CH₃)=N-i-C₃H₇, -C(CH₃)=N-n-C₄H₉, -C(CH₃)=N-CH₂CH=CH₂, -C(CH₃)=N-CH₂CH=CH₂-CH₃, -C(CH₃)=N-CH₂C≡CH, -C(CH₃)=N-CH₂C≡C-CH₃, -C(CH₃)=N-cyclopropyl, -C(CH₃)=N-cyclobutyl, -C(CH₃)=N-cyclo­ pentyl, -C(CH₃)=N-cyclohexyl, -C(CH₃)=N-cycloheptyl, -C(CH₃)=N-CH₂-CH₂Cl, -C(CH₃)=N-CH₂Cl, -C(CH₃)=N-C₆H₅, -C(CH₃)=N-(2-F-C₆H₄), -C(CH₃)=N-(3-F-C₆H₄), -C(CH₃)=N-(4-F-C₆H₄), -C(CH₃)=N-(2-Cl-C₆H₄), -C(CH₃)=N-(3-Cl-C₆H₄), -C(CH₃)=N-(4-Cl-C₆H₄), -C(CH₃)=N-(2-CH₃-C₆H₄), -C(CH₃)=N-(3-CH₃-C₆H₄), -C(CH₃)=N-(4-CH₃-C₆H₄), -C(CH₃)=N-(2-CF₃-C₆H₄), -C(CH₃)=N-(3-CF₃-C₆H₄), -C(CH₃)=N-(4-CF₃-C₆H₄), -C(CH₃)=N-(2-OCH₃-C₆H₄), -C(CH₃)=N-(3-OCH₃-C₆H₄), -C(CH₃)=N-(4-OCH₃-C₆H₄), -C(CH₃)=N-(4-NO₂-C₆H₄), -C(CH₃)=N-(4-CN-C₆H₄), -C(CH₃)=N-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-(2,4-(CH₃)₂-C₆H₃), -C(CH₃)=N-CH₂-OCH₃, -C(CH₃)=N-CH₂-OC₂H₅, -C(CH₃)=N-CH₂CH₂-OCH₃, -C(CH₃)=N-CH₂CH₂-OC₂H₅, -C(CH₃)=N-OH, -C(CH₃)=N-OCH₃, -C(CH₃)=N-OC₂H₅, -C(CH₃)=N-O-n-C₃H₇, -C(CH₃)=N-O-i-C₃H₇, -C(CH₃)=N-O-n-C₄H₉, -C(CH₃)=N-O-i-C₄H₉, -C(CH₃)=N-O-s-C₄H₉, -C(CH₃)=N-O-tert.-C₄H₉, -C(CH₃)=N-OCH₂-CH=CH₂, -C(CH₃)=N-OCH(CH₃)-CH=CH₂, -C(CH₃)=N-OCH₂-C≡CH, -C(CH₃)=N-CH(CH₃)-C≡CH, -C(CH₃)=N-OCH₂-CH=C-CH₃, -C(CH₃)=N-OCH₂CH₂-Cl, -C(CH₃)=N-OCH₂CH₂-F, -C(CH₃)=N-OCH₂-CF₃, -C(CH₃)=N-OCH₂-CH=CHCl, -C(CH₃)=N-OCH₂-C(Cl)=CH₂, -C(CH₃)=N-OCH₂-C(Br)=CH₂, -C(CH₃)=N-OCH₂-CH=C(Cl)-CH₃, -C(CH₃)=N-O-CO-CH₃, -C(CH₃)=N-O-CO-C₂H₅, -C(CH₃)=N-OCH₂-CN, -C(CH₃)=N-OCH₂-CH=CH-CH₂-OCH₃, -C(CH₃)=N-OCH₂-CH=CH-CH₂-O-tert.-C₄H₉, -C(CH₃)=N-O-(CH₂)₃-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-(4-Cl-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-C₆H₅, -C(CH₃)=N-OCH₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(3-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-CH₂-(4-CH₃O-C₆H₄), -C(CH₃)=N-OCH₂-CH=C(CH₃)-C₆H₅, -C(CH₃)=N-O-(CH₂)₂-CH=CH-(3,4-Cl₂-C₆H₃), -C(CH₃)=N-O-(CH₂)₃-C≡-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-OCH₃, -C(CH₃)=N-OCH₂CH₂-OCH₃, -C(CH₃)=N-OCH₂-OC₂H₅, -C(CH₃)=N-OCH(CH₃)-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=N-NH₂, -C(CH₃)=N-NH-CH₃, -C(CH₃)=N-NH-C₂H₅, -C(CH₃)=N-NH-n-C₃H₇, -C(CH₃)=N-NH-i-C₃H₇, -C(CH₃)=N-NH-n-C₄H₉, -C(CH₃)=N-NH-i-C₄H₉, -C(CH₃)=N-NH-s-C₄H₉, -C(CH₃)=N-NH-tert.-C₄H₉, -C(CH₃)=N-NH-cyclopropyl, -C(CH₃)=N-NH- cyclobutyl, -C(CH₃)=N-NH-cyclopentyl, -C(CH₃)=N-NH-cyclohexyl, -C(CH₃)=N-NH-cycloheptyl, -C(CH₃)=N-N(CH₃)₂, -C(CH₃)=N-N(C₂H₅)₂, -C(CH₃)=N-N(n-C₃H₇)₂, -C(CH₃)=N-N(i-C₃H₇)₂, -C(CH₃)=N-NH-CH₂-C=CH, -C(CH₃)=N-NH-CH₂-C≡CH, -C(CH₃)=N-N(CH₃)-CH₂-C≡CH, -C(CH₃)=N-NH-CH₂CF₃, -C(CH₃)=N-NH-CO-CH₃, -C(CH₃)=N-NH-CO-C₂H₅, -C(CH₃)=N-NH-CO-OCH₃, -C(CH₃)=N-NH-CO-OC₂H₅, -C(CH₃)=N-NH-CO-O-tert.-C₄H₉, -C(CH₃)=N- pyrrolidin-1-yl, -C(CH₃)=N-piperidin-1-yl, -C(CH₃)=N-morpholin- 4-yl, -C(CH₃)=N-NH-C₆H₅, -C(CH₃)=N-NH-(4-Cl-C₆H₄), -C(CH₃)=N-NH-(4-NO₂-C₆H₄), -C(CH₃)=N-NH-(4-F-C₆H₄), -C(CH₃)=N-NH-(4-CH₃O-C₆H₄), -C(CH₃)=N-NH-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-NH-(2,4-(NO₂)₂-C₆H₃), -C(CH₃)=N-NH-CO-NH₂, -C(CH₃)=N-NH-CO-NHCH₃, -C(CH₃)=N-NH-CO-NHC₂H₅, -C(CH₃)=N-NH-CO-N(CH₃)₂, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=CH-CO-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -(CH₃)=CH-CO-O-n-C₄H₉, -C(CH₃)=CH-CO-O-tert.-C₄H₉, -C(CH₃)=CH-CO-O-cyclopropyl, -C(CH₃)=CH-CO-O-cyclobutyl, -C(CH₃)=CH-CO-O-cyclopentyl, -C(CH₃)=CH-CO-O-cyclohexyl, -C(CH₃)=CH-CO-O-cycloheptyl, -C(CH₃)=C(CH₃)-COOH, -C(CH₃)=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-cyclopropyl, -C(CH₃)=C(CH₃)-CO-O-cyclobutyl, -C(CH₃)=C(CH₃)-CO-O-cyclopentyl, -C(CH₃)=C(CH₃)-CO-O-cyclohexyl, -C(CH₃)=C(CH₃)-CO-O-cycloheptyl, -C(CH₃)=C(C₂H₅)-COOH, -C(CH₃)=C(C₂H₅)-CO-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-cyclo­ propyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-O- cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-O-cycloheptyl, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=C(Cl)-CO-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-O-n-C₄H₉, -C(CH₃)=C(Cl)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-O-cyclopropyl, -C(CH₃)=C(Cl)-CO-O-cyclobutyl, -C(CH₃)=C(Cl)-CO-O-cyclopentyl, -C(CH₃)=C(Cl)-CO-O-cyclohexyl, -C(CH₃)=C(Cl)-CO-O-cycloheptyl, -C(CH₃)=C(Br)-COOH, -C(CH₃)=C(Br)-CO-OCH₃, -C(CH₃)=C(Br)-CO-OC₂H₅, -C(CH₃)=C(Br)-CO-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-O-n-C₄H₉, -C(CH₃)=C(Br)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-O-cyclopropyl, -C(CH₃)=C(Br)-CO-O-cyclobutyl, -C(CH₃)=C(Br)-CO-O-cyclopentyl, -C(CH₃)=C(Br)-CO-O-cyclohexyl, -C(CH₃)=C(Br)-CO-O-cycloheptyl, -C(CH₃)=C(CN)-COOH, -C(CH₃)=C(CN)-CO-OCH₃, -C(CH₃)=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CN)-CO-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-O-n-C₄H₉, -C(CH₃)=C(CN)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-O-cyclopropyl, -C(CH₃)=C(CN)-CO-O-cyclobutyl, -C(CH₃)=C(CN)-CO-O-cyclopentyl, -C(CH₃)=C(CN)-CO-O-cyclohexyl, -C(CH₃)=C(CN)-CO-O-cycloheptyl, -C(CH₃)=CH-CO-OCH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=CH-CO-O-i-C₃H₇, -C(CH₃)=CH-CO-OCH(CH₃)-OCH₃, -C(CH₃)=CH-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=CH-CO-OCH₂CH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=(C₂H₅)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-O-i-C₃H₇, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -(CH₃)=C(Cl)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-O-i-C₃H₇, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-O-i-C₃H₇, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-CF₃, -C(CH₃)=CH-CO-OCH₂-CCl₃, -C(CH₃)=CH-CO-OCH₂-oxiranyl, -C(CH₃)=CH-CO-(CH₂)₃-Br,-C(CH₃)=CH-CO-OCH₂-CH=CH₂, -C(CH₃)=CH-CO-OCH₂-C≡CH, -C(CH₃)=CH-CO-OCH₂-CN, -C(CH₃)=CH-CO-OCH₂CH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CF₃, -C(CH₃)=C(CH₃)-CO-OCH₂-CCl₃, -C(CH₃)=C(CH₃)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CH₃)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(CH₃)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CH₃)-CO-OCH₂-C≡CH, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CF₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CCl₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-oxiranyl, -C(CH₃)=C(C₂H₅)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(C₂H₅)-CO-OCH₂-C≡CH, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-C₂, -C(CH₃)=C(Cl)-CO-OCH₂-CF₃, -C(CH₃)=C(Cl)-CO-OCH₂-CCl₃, -C(CH₃)=C(Cl)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Cl)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Cl)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Cl)-CO-OCH₂-C≡CH, -C(CH₃)=C(Cl)-CO-OCH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂-CF₃, -C(CH₃)=C(Br)-CO-OCH₂-CCl₃, -C(CH₃)=C(Br)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Br)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Br)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Br)-CO-OCH₂-C≡CH, -C(CH₃)=C(Br)-CO-OCH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂CH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂-CF₃, -C(CH₃)=C(CN)-CO-OCH₂-CCl₃, -C(CH₃)=C(CN)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CN)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(CN)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CN)-CO-OCH₂-C≡CH, -C(CH₃)=C(CN)-CO-OCH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂CH₂-CN, -C(CH₃)=CH-CO-CH₃, -C(CH₃)=CH-CO-C₂H₅, -C(CH₃)=CH-CO-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-n-C₄H₉, -C(CH₃)=CH-CO-tert.-C₄H₉, -C(CH₃)=CH-CO-CH₂Cl, -C(CH₃)=CH-CO-CH₂Br, -C(CH₃)=CH-CO-CHCl₂, -C(CH₃)=CH-CO-CH₂-OCH₃, -C(CH₃)=CH-CO-CH(OCH₃)₂, -C(CH₃)=CH-CO-CH₂-SCH₃, -C(CH₃)=C(CH₃)-CO-CH₃, -C(CH₃)=C(CH₃)-CO-C₂H₅, -C(CH₃)=C(CH₃)-CO-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-CH₂Cl, -C(CH₃)=C(CH₃)-CO-CH₂Br, -C(CH₃)=C(CH₃)-CO-CHCl₂, -C(CH₃)=C(CH₃)-CO-CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-CH(OCH₃)₂, -C(CH₃)=C(CH₃)-CO-CH₂-SCH₃, -C(CH₃)=C(C₂H₅)-CO-CH₃, -C(CH₃)=C(C₂H₅)-CO-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-CH₂Cl, -C(CH₃)=C(C₂H₅)-CO-CH₂Br, -C(CH₃)=C(C₂H₅)-CO-CHCl₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-CH(OCH₃)₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-SCH₃, -C(CH₃)=C(Cl)-CO-CH₃, -C(CH₃)=C(Cl)-CO-C₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-n-C₄H₉, -C(CH₃)=C(Cl)-CO-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-CH₂Cl, -C(CH₃)=C(Cl)-CO-CHCl₂, -C(CH₃)=C(Cl)-CO-CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-CH(OCH₃)₂, -C(CH₃)=C(Cl)-CO-CH₂-SCH₃, -C(CH₃)=C(Br)-CO-CH₃, -C(CH₃)=C(Br)-CO-C₂H₅, -C(CH₃)=C(Br)-CO-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-n-C₄H₉, -C(CH₃)=C(Br)-CO-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-CH₂Cl, -C(CH₃)=C(Br)-CO-CH₂Br, -C(CH₃)=C(Br)-CO-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-CH(OCH₃)₂, -C(CH₃)=C(Br)-CO-CH₂-SCH₃, -C(CH₃)=C(CN)-CO-CH₃, -C(CH₃)=C(CN)-CO-C₂H₅, -C(CH₃)=C(CN)-CO-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-n-C₄H₉, -C(CH₃)=C(CN)-CO-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-CH₂Cl, -C(CH₃)=C(CN)-CO-CH₂Br, -C(CH₃)=C(CN)-CO-CHCl₂, -C(CH₃)=C(CN)-CO-CH₂-OCH₃, -C(CH₃)=C(CN)-CO-CH(OCH₃)₂, -C(CH₃)=C(CN)-CO-CH₂-SCH₃, -C(CH₃)=CH-CO-C₆H₅, -C(CH₃)=CH-CO-(4-Cl-C₆H₄), -C(CH₃)=C(CH₃)-CO-C₆H₅, -C(CH₃)=C(CH₃)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(C₂H₅)-CO-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(Cl)-CO-C₆H₅, -C(CH₃)=C(Br)-CO-C₆H₅, -C(CH₃)=C(CN)-CO-C₆H₅, -C(CH₃)=CH-CO-NH₂, -C(CH₃)=CH-CO-NHCH₃, -C(CH₃)=CH-CO-N(CH₃)₂, -C(CH₃)=CH-CO-NH-C₂H₅, -C(CH₃)=CH-CO-N(C₂H₅)₂, -C(CH₃)=CH-CO-NH-n-C₃H₇, -C(CH₃)=CH-CO-NH-i-C₃H₇, -C(CH₃)=CH-CO-NH-tert.-C₄H₉, -C(CH₃)=CH-CO-NH-cyclopropyl, -C(CH₃)=CH-CO-NH-cyclobutyl, -C(CH₃)=CH-CO-NH-cyclopentyl, -C(CH₃)=CH-CO-NH-cyclohexyl, -C(CH₃)=CH-CO-NH-cycloheptyl, -C(CH₃)=CH-CO-NH-cyclooctyl, -C(CH₃)=CH-CO-pyrrolidin-1-yl, -C(CH₃)=CH-CO-piperidin-1-yl, -C(CH₃)=CH-CO-morpholin-4-yl, -C(CH₃)=CH-CO-NH-CH₂CH=CH₂, -C(CH₃)=CH-CO-NH-CH₂C≡CH, -C(CH₃)=CH-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=CH-CO-NH-(CH₂)₂Cl, -C(CH₃)=CH-CO-NH-C₆H₅, -C(CH₃)=C(CH₃)-CO-NH₂, -C(CH₃)=C(CH₃)-CO-NHCH₃, -C(CH₃)=C(CH₃)-CO-N(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-C₂H₅, -C(CH₃)=C(CH₃)-CO-N(C₂H₅)₂, -C(CH₃)=C(CH₃)-CO-NH-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-NH- cyclopropyl, -C(CH₃)=C(CH₃)-CO-NH-cyclobutyl, -C(CH₃)=C(CH₃)-CO-NH-cyclopentyl, -C(CH₃)=C(CH₃)-CO-NH- cyclohexyl, -C(CH₃)=C(CH₃)-CO-NH-cycloheptyl, -C(CH₃)=C(CH₃)-CO-NH-cyclooctyl, -C(CH₃)=C(CH₃)-CO- pyrrolidin-1-yl, -C(CH₃)=C(CH₃)-CO-piperidin-1-yl, -C(CH₃)=C(CH₃)-CO-morpholin-4-yl, -C(CH₃)=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-NH(CH₂)₂Cl, -C(CH₃)=C(CH₃)-CO-NH-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-NH₂, -C(CH₃)=C(C₂H₅)-CO-NHCH₃, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)₂, -C(CH₃)=C(C₂H₅)-CO-NH-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-N(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-NH- cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclo­ hexyl, -C(CH₃)=C(C₂H₅)-CO-NH-cycloheptyl, -C(CH₃)=C(C₂H₅)-CO-NH- cyclooctyl, -C(CH₃)=C(C₂H₅)-CO-pyrrolidin-1-yl, -C(CH₃)=C(C₂H₅)-CO-piperidin-1-yl, -C(CH₃)=C(C₂H₅)-CO- morpholin-4-yl, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(C₂H₅)-CO-NH-C₆H₅, -C(CH₃)=C(Cl)-CO-NH₂, -C(CH₃)=C(CH₃)=C(Cl)-CO-NHCH₃, -C(CH₃)=C(Cl)-CO-N(CH₃)₂, -C(CH₃)=C(Cl)-CO-NH-C₂H₅, -C(CH₃)=C(Cl)-CO-N(C₂H₅)₂, -C(CH₃)=C(Cl)-CO-NH-n-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-i-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-NH-cyclopropyl, -C(CH₃)=C(Cl)-CO-NH-cyclobutyl, -C(CH₃)=C(Cl)-CO-NH-cyclopentyl, -C(CH₃)=C(Cl)-CO-NH-cyclohexyl, -C(CH₃)=C(Cl)-CO-NH-cycloheptyl, -C(CH₃)=C(Cl)-CO-NH-cyclooctyl, -C(CH₃)=C(Cl)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Cl)-CO-piperidin-1- yl, -C(CH₃)=C(Cl)-CO-morpholin-4-yl, -C(CH₃)=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -(CH₃)=C(Cl)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-N(CH₃)-CH₂≡CH, -C(CH₃)=C(Cl)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Cl)-NO-NH-C₆H₅, -C(CH₃)=C(Br)-CO-NH₂, -C(CH₃)=C(Br)-CO-NHCH₃, -C(CH₃)=C(Br)-CO-N(CH₃)₂, -C(CH₃)=C(Br)-CO-NH-C₂H₅, -C(CH₃)=C(Br)-CO-N(C₂H₅)₂, -C(CH₃)=C(Br)-CO-NH-n-C₃H₇, -C(CH₃)=C(Br)-CO-NH-i-C₃H₇, -C(CH₃)=C(Br)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-NH-cyclopropyl, -C(CH₃)=C(Br)-CO-NH-cyclobutyl, -C(CH₃)=C(Br)-CO-NH-cyclopentyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cycloheptyl, -C(CH₃)=C(Br)-CO-NH-cyclooctyl, -C(CH₃)=C(Br)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Br)-CO-piperidin-1-yl, -C(CH₃)=C(Br)-CO-morpholin-4-yl, -C(CH₃)=C(Br)-CO-NH-CH₂CH=C(Br)₂, -C(CH₃)=C(Br)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Br)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Br)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Br)-CO-NH-C₆H₅, -C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CN)-CO-NHCH₃, -C(CH₃)=C(CN)-CO-N(CH₃)₂, -C(CH₃)=C(CN)-CO-NH-C₂H₅, -C(CH₃)=C(CN)-CO-N(C₂H₅)₂, -C(CH₃)=C(CN)-CO-NH-n-C₃H₇, -C(CH₃)=C(CN)-CO-NH-i-C₃H₇, -C(CH₃)=C(CN)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-NH-cyclopropyl, -C(CH₃)=C(CN)-CO-NH-cyclobutyl, -C(CH₃)=C(CN)-CO-NH-cyclopentyl, -C(CH₃)=C(CN)-CO-NH-cyclohexyl, -C(CH₃)=C(CN)-CO-NH-cycloheptyl, -C(CH₃)=C(CN)-CO-NH-cyclooctyl, -C(CH₃)=C(CN)-CO-pyrrolidin-1-yl, -C(CH₃)=C(CN)-CO-piperidin-1-yl, -C(CH₃)=C(CN)-CO-morpholin-4-yl, -C(CH₃)=C(CN)-CO-NH-CH₂CH=C(CN)₂, -C(CH₃)=C(CN)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CN)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)=(CN)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CN)-CO-NH-C₆H₅, -C(CH₃)=CH-CO-SCH₃, -C(CH₃)=CH-CO-SC₂H₅, -C(CH₃)=CH-CO-S-n-C₃H₇, -C(CH₃)=CH-CO-S-i-C₃H₇, -C(CH₃)=CH-CO-S-n-C₄H₉, -C(CH₃)=CH-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-SCH₃, -C(CH₃)=C(CH₃)-CO-SC₂H₅, -C(CH₃)=C(CH₃)-CO-S-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-S-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-SCH₃, -C(CH₃)=C(C₂H₅)-CO-SC₂H₅, -C(CH₃)=C(C₂H₅)-CO-S-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-SCH₃, -C(CH₃)=C(Cl)-CO-SC₂H₅, -C(CH₃)=C(Cl)-CO-S-n-C₃H₇, -C(CH₃)=C(Cl)-CO-S-i-C₃H₇, -C(CH₃)=C(Cl)-CO-S-n-C₄H₉, -C(CH₃)=C(Cl)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-SCH₃, -C(CH₃)=C(Br)-CO-SC₂H₅, -C(CH₃)=C(Br)-CO-S-n-C₃H₇, -C(CH₃)=C(Br)-CO-S-i-C₃H₇, -C(CH₃)=C(Br)-CO-S-n-C₄H₉, -C(CH₃)=C(Br)-CO-S-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-SCH₃, -C(CH₃)=C(CN)-CO-SC₂H₅, -C(CH₃)=C(CN)-CO-S-n-C₃H₇, -C(CH₃)=C(CN)-CO-S-i-C₃H₇, -C(CH₃)=C(CN)-CO-S-N-C₄H₉, -C(CH₃)=C(CN)-CO-S-tert.-C₄H₉, -C(CH₃)=C(COCH₃)-CO-OCH₃, -C(CH₃)=C(COC₂H₅)-CO-OCH₃, -C(CH₃)=C(CO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COCH₃)-CO-OC₂H₅, -C(CH₃)=C(COC₂H₅)-CO-OC₂H₅, -C(CH₃)=C(CO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COCH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(COC₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-OCH₃, -C(CH₃)=C(CF₃)-CO-OC₂H₅, -C(CH₃)=C(CF₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CF₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(COOCH₃)₂, -C(CH₃)=C(COOC₂H₅)₂, -C(CH₃)=C(COOCH₃)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)₂, -C(CH₃)=CH-CH=CH-COOH, -C(CH₃)=CH-CH=CH-CO-OCH₃, -C(CH₃)=CH-CH=CH-CO-OC₂H₅, -C(CH₃)=CH-CH=C(COOCH₃)₂, -C(CH₃)=CH-CH=C(CN)-CO-OCH₃, -C(CH₃)=CH-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH₂, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -C(CH₃)=CH-(CH₂)₂-COOH, -C(CH₃)=CH-(CH₂)₂-CO-OCH₃, -C(CH₃)=CH-(CH₂)₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(COOCH₃)₂, -C(CH₃)=CH-CH₂-CH(COOC₂H₅)₂, -C(CH₃)=CH-CH₂-CH(CN)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CN)-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -C(CH₃)=CH-(CH₂)₂-CO-NH₂, -C(CH₃)=CH-(CH₂)₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-COOH, -C(CH₃)=CH-CH₂-CO-OCH₃, -C(CH₃)=CH-CH₂-CO-OC₂H₅, -C(CH₃)=C(COOCH₃)-CH₂-CO-OCH₃, -C(CH₃)=C(COOCH₃)-CH₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CO-NH₂, -C(CH₃)=CH-CH₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-CO-N(CH₃)₂.
wobei W für eine der folgenden Bedeutungen steht:
-CHO, -COCH₃, -COC₂H₅, -CO-n-C₃H₇, -CO-i-C₃H₇, -CO-n-C₄H₉, -CO-i-C₄H₉, -CO-s-C₄H₉, -CO-tert.-C₄H₉, -CO-CH₂CH=CH₂, -CO-CF₃, -COCCl₃, -COCH₂C≡CH, -CO-cyclopropyl, -CO-cyclobutyl, -CH-cyclo­ pentyl, -CO-cyclhexyl, -CO-CN, -CO-COOCH₃, -CO-COOC₂H₅, -CH=NH, -CH=NCH₃, -CH=NC₂H₅, -CH=N-n-C₃H₅, -CH=N-i-C₃H₅, -CH=N-n-C₄H₉, -CH=NCH₂CH=CH₂, -CH=NCH₂CH=CH₂-CH₃, -CH=NCH₂C≡CH, -CH=NCH₂C≡C-CH₃, -CH=N-cyclopropyl, -CH=N-cyclobutyl, -CH=N-cyclopentyl, -CH=N-cyclohexyl, -CH=N-cycloheptyl, -CH=N-CH₂-CH₂Cl, -CH=N-CH₂Cl, -CH=N-C₆H₅, -CH=N-4-Br-C₆H₄, -CH=N-3-F-C₆H₄, -CH=N-4-F-C₆H₄, -CH=N-2-Cl-C₆H₄, -CH=N-3-Cl-C₆H₄, -CH=N-4-Cl-C₆H₄, -CH=N-2-Br-C₆H₄, -CH=N-2-F-C₆H₄, -CH=N-2-CH₃-C₆H₄, -CH=N-3-CH₃-C₆H₄, -CH=N-4-CH₃-C₆H₄, -CH=N-2-CF₃-C₆H₄, -CH=N-3-CF₃-C₆H₄, -CH=N-4-CF₃-C₆H₄, -CH=N-2-OCH₃-C₆H₄, -CH=N-3-OCH₃-C₆H₄, -CH=N-4-OCH₃-C₆H₄, -CH=N-4-NO₂-C₆H₄, -CH=N-4-CN-C₆H₄, -CH=N-2,4-(Cl,Cl)-C₆H₄, -CH=N-2,4-(CH₃,CH₃)-C₆H₄, -CH=N-CH₂OCH₃ -CH=N-CH₂OC₂H₅, -CH=N-CH₂CH₂OCH₃, -CH=N-CH₂CH₂OC₂H₅, -CH=N-OH, -CH=N-OCH₃, -CH=N-OC₂H₅, -CH=N-O-n-C₃H₇, -CH=N-O-i-C₃H₇, -CH=N-O-n-C₄H₉, -CH=N-O-i-C₄H₉, -CH=N-O-s-C₄H₉, -CH=N-O-tert.-C₄H₉, -CH=N-O-CH₂CH=CH₂, -CH=N-O-CH(CH₃)CH=CH₂, -CH=N-O-CH₂C≡CH, -CH=N-O-CH(CH₃)-C≡CH, -CH=N-O-CH₂-CH=CH-CH₃, -CH=N-O-CH₂-CH₂-Cl, -CH=N-O-CH₂-CH₂-F, -CH=N-O-CH₂-CF₃, -CH=N-O-CH₂-CH=CHCl, -CH=N-O-CH₂-CCl=CH₂, -CH=N-O-CH₂-CBr=CH₂, -CH=N-O-CH₂-CH=CCl-CH₃, -CH=N-OC(O)CH₃, -CH=N-OC(O)C₂H₅, -CH=N-O-CH₂-CN, -CH=N-O-CH₂-CH=CH-CH₂-O-CH₃, -CH=N-O-CH₂-CH=CH-CH₂-O-tert.-C₄H₉, -CH=N-O-(CH₂)₃-C₆H₅, -CH=N-O-(CH₂)₄-C₆H₅, -CH=N-O-(CH₂)₄-4-Cl-C₆H₄, -CH=N-O-(CH₂)₄-4-OCH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-CH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-C₆H₅, -CH=N-O-CH₂CH=CH-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CH-3-OCH₃-C₆H₄, -CH=N-O-(CH₂)₂CH=CH-4-F-C₆H₄, -CH=N-O-(CH₂)CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CHCH₂-4-OCH₃-C₆H₄, -CH=N-O-CH₂-CH=C(CH₃)-C₆H₄ -CH=N-O-(CH₂)₂CH=CH-3,4(Cl,Cl)-C₆H₃, -CH=N-O-(CH₂)₃C≡C-4-F-C₆H₄, -CH₂=N-OCHOCH₃, -CH=N-OC₂H₄OCH₃, -CH=N-OCH₂OC₂H₅, -CH=N-OCH(CH₃)OCH₃, -CH=N-OCH(CH₃)COOCH₃, -CH=N-OCH(CH₃)COO-n-C₄H₉, -CH=N-NH₂, -CH=N-NHCH₃, -CH=N-NHC₂H₅, -CH=N-NH-n-C₃H₇, -CH=N-NH-i-C₃H₇, -CH=N-NH-n-C₄H₉, -CH=N-NH-i-C₄H₉, -CH=N-NH-s-C₄H₉, -CH=N-NH-tert.-C₄H₉, -CH=N-NH-cyclopropyl, -CH=N-NH-cyclobutyl, -CH=N-NH-cyclopentyl, -CH=N-NH-cyclohexyl, -CH=N-NH-cycloheptyl, -CH=N-N(CH₃)₂, -CH=N-N(C₂H₅)₂, -CH=N-N(C₃H₇)₂, -CH=N-N(i-C₃H₇)(CH₃), -CH=N-NHCH₂-C=CH, -CH=N-NHCH₂-C≡CH, -CH=N-N(CH₃)-CH₂-C≡CH, -CH=N-NHCH₂CF₃, -CH=N-NH-CO-CH₃, -CH=N-NH-CO-CH₂H₅, -CH=N-NH-COOCH₃, -CH=N-NH-COOC₂H₅, -CH=N-NH-COO-tert.-C₄H₉, -CH=N-pyrrolidin-1-yl, -CH=N-piperidin-1-yl, -CH=N-morpholin-4-yl, -CH=N-NH-C₆H₅, -CH=N-NH-(4-Cl-C₆H₄), -CH=N-NH-(4-NO₂-C₆H₄), -CH=N-NH-(4-F-C₆H₄), -CH=N-NH-(4-CH₃O-C₆H₄), -CH=N-NH-(2,4-Cl₂-C₆H₃), -CH=N-NH-(2,4-(NO₂)₂-C₆H₃), -CH=N-NH-CO-NH₂, -CH=N-NH-CO-NHCH₃, -CH=N-NH-CO-NHC₂H₅, -CH=N-NH-CO-N(CH₃)₂, -CH=CH-COOH, -CH=CH-CO-OCH₃, -CH=CH-CO-OC₂H₅, -CH=CH-CO-O-n-C₃H₇, -CH=CH-CO-O-i-C₃H₇, -CH=CH-CO-O-n-C₄H₉, -CH=CH-CO-O-tert.-C₄H₉, -CH=CH-CO-O-cyclopropyl, -CH=CH-CO-O-cyclobutyl, -CH=CH-CO-O-cyclopentyl, -CH=CH-CO-O-cyclohexyl, -CH=CH-CO-O-cycloheptyl, -CH=C(CH₃)-COOH, -CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CO-O-n-C₃H₇, -CH=C(CH₃)-CO-O-i-C₃H₇, -CH=C(CH₃)-CO-O-n-C₄H₉, -CH=C(CH₃)-CO-O-tert.-C₄H₉, -CH=C(CH₃)-CO-O-cyclopropyl, -CH=C(CH₃)-CO-O-cyclobutyl, -CH=C(CH₃)-CO-O-cyclopentyl, -CH=C(CH₃)-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cycloheptyl, -CH=C(C₂H₅)-COOH, -CH=C(C₂H₅)-CO-OCH₃, -CH=C(C₂H₅)-CO-OC₂H₅, -CH=C(C₂H₅)-CO-O-n-C₃H₇, -CH=C(C₂H₅)-CO-O-i-C₃H₇, -CH=C(C₂H₅)-CO-O-n-C₄H₉, -CH=C(C₂H₅)-CO-O-tert.-C₄H₉, -CH=C(C₂H₅)-CO-O-cyclopropyl, -CH=C(C₂H₅)-CO-O-cyclobutyl, -CH=C(C₂H₅)-CO-O-cyclopentyl, -CH=C(C₂H₅)-CO-O-cyclohexyl, -CH=C(C₂H₅)-CO-O-cycloheptyl, -CH=C(Cl)-COOH, -CH=C(Cl)-CO-OCH₃, -CH=C(Cl)-CO-OC₂H₅, -CH=C(Cl)-CO-O-n-C₃H₇, -CH=C(Cl)-CO-O-i-C₃H₇, -CH=C(Cl)-CO-O-n-C₄H₉, -CH=C(Cl)-CO-O-tert.-C₄H₉, -CH=C(Cl)-CO-O-cyclopropyl, -CH=C(Cl)-CO-O-cyclobutyl, -CH=C(Cl)-CO-O-cyclopentyl, -CH=C(Cl)-CO-O-cyclohexyl, -CH=C(Cl)-CO-O-cycloheptyl, -CH=C(Br)-COOH, -CH=C(Br)-CO-OCH₃, -CH=C(Br)-CO-OC₂H₅, -CH=C(Br)-CO-O-n-C₃H₇, -CH=C(Br)-CO-O-i-C₃H₇, -CH=C(Br)-CO-O-n-C₄H₉, -CH=C(Br)-CO-O-tert.-C₄H₉, -CH=C(Br)-CO-O-cyclopropyl, -CH=C(Br)-CO-O-cyclobutyl, -CH=C(Br)-CO-O-cyclopentyl, -CH=C(Br)-CO-O-cyclohexyl, -CH=C(Br)-CO-O-cycloheptyl, -CH=C(CN)-COOH, -CH=C(CN)-CO-OCH₃, -CH=C(CN)-CO-OC₂H₅, -CH=C(CN)-CO-O-n-C₃H₇, -CH=C(CN)-CO-O-i-C₃H₇, -CH=C(CN)-CO-O-n-C₄H₉, -CH=C(CN)-CO-O-tert.-C₄H₉, -CH=C(CN)-CO-O-cyclopropyl, -CH=C(CN)-CO-O-cyclobutyl, -CH=C(CN)-CO-O-cyclopentyl, -CH=C(CN)-CO-O-cyclohexyl, -CH=C(CN)-CO-O-cycloheptyl, -CH=CH-CO-OCH₂-OCH₃, -CH=CH-CO-OCH₂-OC₂H₅, -CH=CH-CO-OCH₂-O-n-C₃H₅, -CH=CH-CO-OCH₂-O-i-C₃H₅, -CH=CH-CO-OCH(CH₃)-OCH₃, -CH=CH-CO-OCH(CH₃)-OC₂H₅, -CH=CH-CO-O-CH₂CH₂-OCH₃, -CH=CH-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-OCH₃, -CH=C(CH₃)-CO-OCH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-O-n-C₃H₅, -CH=C(CH₃)-CO-OCH₂-O-i-C₃H₅, -CH=C(CH₃)-CO-OCH(CH₃)-OCH₃, -CH=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CH₃)-CO-O-CH₂CH₂-OCH₃, -CH=C(CH₃)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-OCH₃, -CH=C(C₂H₅)-CO-OCH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-O-n-C₃H₅, -CH=C(C₂H₅)-CO-OCH₂-O-i-C₃H₅, -CH=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -CH=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OCH₃, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-OCH₃, -CH=C(Cl)-CO-OCH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-O-n-C₃H₅, -CH=C(Cl)-CO-OCH₂-O-i-C₃H₅, -CH=C(Cl)-CO-OCH(CH₃)-OCH₃, -CH=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Cl)-CO-O-CH₂CH₂-OCH₃, -CH=C(Cl)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-OCH₃, -CH=C(Br)-CO-OCH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-O-n-C₃H₅, -CH=C(Br)-CO-OCH₂-O-i-C₃H₅, -CH=C(Br)-CO-OCH(CH₃)-OCH₃, -CH=C(Br)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Br)-CO-O-CH₂CH₂-OCH₃, -CH=C(Br)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-OCH₃, -CH=C(CN)-CO-OCH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-O-n-C₃H₅, -CH=C(CN)-CO-OCH₂-O-i-C₃H₅, -CH=C(CN)-CO-OCH(CH₃)-OCH₃, -CH=C(CN)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CN)-CO-O-CH₂CH₂-OCH₃, -CH=C(CN)-CO-O-CH₂CH₂-OC₂H₅, -CH=CH-CO-OCH₂-CF₃, -CH=CH-CO-OCH₂-CCl₃, -CH=CH-CO-OCH₂-oxiranyl, -CH=CH-CO-O(CH₂)₃-Br, -CH=CH-CO-OCH₂-CH=CH₂, -CH=CH-CO-OCH₂-C≡CH, -CH=CH-CO-OCH₂-CN, -CH=CH-CO-O(CH₂)₂-CN, -CH=C(CH₃)-CO-OCH₂-CF₃, -CH=C(CH₃)-CO-OCH₂-CCl₃, -CH=C(CH₃)-CO-OCH₂-oxiranyl, -CH=C(CH₃)-CO-O(CH₂)₃-Br, -CH=C(CH₃)-CO-OCH₂-CH=CH₂, -CH=C(CH₃)-CO-OCH₂-C≡CH, -CH=C(CH₃)-CO-OCH₂-CN, -CH=C(CH₃)-CO-O(CH₂)₂-CN, -CH=C(C₂H₅)-CO-OCH₂-CF₃, -CH=C(C₂H₅)-CO-OCH₂-CCl₃, -CH=C(C₂H₅)-CO-OCH₂-oxiranyl, -CH=C(C₂H₅)-CO-O(CH₂)₃-Br, -CH=C(C₂H₅)-CO-OCH₂-CH=CH₂, -CH=C(C₂H₅)-CO-OCH₂-C≡CH, -CH=C(C₂H₅)-CO-OCH₂-CN, -CH=C(C₂H₅)-CO-O(CH₂)₂-CN, -CH=C(Cl)-CO-OCH₂-CF₃, -CH=C(Cl)-CO-OCH₂-CCl₃, -CH=C(Cl)-CO-OCH₂-oxiranyl, -CH=C(Cl)-CO-O(CH₂)₃-Br, -CH=C(Cl)-CO-OCH₂-CH=CH₂, -CH=C(Cl)-CO-OCH₂-C≡CH, -CH=C(Cl)-CO-OCH₂-CN, -CH=C(Cl)-CO-O(CH₂)₂-CN, -CH=C(Br)-CO-OCH₂-CF₃, -CH=C(Br)-CO-OCH₂-CCl₃, -CH=C(Br)-CO-OCH₂-oxiranyl, -CH=C(Br)-CO-O(CH₂)₃-Br, -CH=C(Br)-CO-OCH₂-CH=CH₂, -CH=C(Br)-CO-OCH₂-C≡CH, -CH=C(Br)-CO-OCH₂-CN, -CH=C(Br)-CO-O(CH₂)₂-CN, -CH=C(CN)-CO-OCH₂-CF₃, -CH=C(CN)-CO-OCH₂-CCl₃, -CH=C(CN)-CO-OCH₂-oxiranyl -CH=C(CN)-CO-O(CH₂)₃-Br, -CH=C(CN)-CO-OCH₂-CH=CH₂, -CH=C(CN)-CO-OCH₂-C≡CH, -CH=C(CN)-CO-OCH₂-CN, -CH=C(CN)-CO-O(CH₂)₂-CN, -CH=CH-CO-CH₃, -CH=CH-CO-C₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-i-C₃H₇, -CH=CH-CO-n-C₄H₉, -CH=CH-CO-tert.-C₄H₉, -CH=CH-CO-CH₂Cl, -CH=CH-CO-CH₂Br, -CH=CH-CO-CHCl₂, -CH=CH-CO-CH₂-OCH₃, -CH=CH-CO-CH(OCH₃)₂, -CH=CH-CO-CH₂-SCH₃, -CH=C(CH₃)-CO-CH₃, -CH=C(CH₃)-CO-C₂H₅, -CH=C(CH₃)-CO-n-C₃H₇, -CH=C(CH₃)-CO-i-C₃H₇, -CH=C(CH₃)-CO-n-C₄H₉, -CH=C(CH₃)-CO-tert.-C₄H₉, -CH=C(CH₃)-CO-CH₂Cl, -CH=C(CH₃)-CO-CH₂Br, -CH=C(CH₃)-CO-CHCl₂, -CH=C(CH₃)-CO-CH₂-OCH₃, -CH=C(CH₃)-CO-CH(OCH₃)₂, -CH=C(CH₃)-CO-CH₂-SCH₃, -CH=C(C₂H₅)-CO-CH₃, -CH=C(C₂H₅)-CO-C₂H₅, -CH=C(C₂H₅)-CO-n-C₃H₇, -CH=C(C₂H₅)-CO-i-C₃H₇, -CH=C(C₂H₅)-CO-n-C₄H₉, -CH=C(C₂H₅)-CO-tert.-C₄H₉, -CH=C(C₂H₅)-CO-CH₂Cl, -CH=C(C₂H₅)-CO-CH₂Br, -CH=C(C₂H₅)-CO-CHCl₂, -CH=C(C₂H₅)-CO-CH₂-OCH₃, -CH=C(C₂H₅)-CO-CH(OCH₃)₂, -CH=C(C₂H₅)-CO-CH₂-SCH₃, -CH=C(Cl)-CO-CH₃, -CH=C(Cl)-CO-C₂H₅, -CH=C(Cl)-CO-n-C₃H₇, -CH=C(Cl)-CO-i-C₃H₇, -CH=C(Cl)-CO-n-C₄H₉, -CH=C(Cl)-CO-tert.-C₄H₉, -CH=C(Cl)-CO-CH₂Cl, -CH=C(Cl)-CO-CH₂Br, -CH=C(Cl)-CO-CHCl₂, -CH=C(Cl)-CO-CH₂-OCH₃, -CH=C(Cl)-CO-CH(OCH₃)₂, -CH=C(Cl)-CO-CH₂-SCH₃, -CH=C(Br)-CO-CH₃, -CH=C(Br)-CO-C₂H₅, -CH=C(Br)-CO-n-C₃H₇, -CH=C(Br)-CO-i-C₃H₇, -CH=C(Br)-CO-n-C₄H₉, -CH=C(Br)-CO-tert.-C₄H₉, -CH=C(Br)-CO-CH₂Cl, -CH=C(Br)-CO-CH₂Br, -CH=C(Br)-CO-CHCl₂, -CH=C(Br)-CO-CH₂-OCH₃, -CH=C(Br)-CO-CH(OCH₃)₂, -CH=C(Br)-CO-CH₂-SCH₃, -CH=C(CN)-CO-CH₃, -CH=C(CN)-CO-C₂H₅, -CH=C(CN)-CO-n-C₃H₇, -CH=C(CN)-CO-i-C₃H₇, -CH=C(CN)-CO-n-C₄H₉, -CH=C(CN)-CO-tert.-C₄H₉, -CH=C(CN)-CO-CH₂Cl, -CH=C(CN)-CO-CH₂Br, -CH=C(CN)-CO-CHCl₂, -CH=C(CN)-CO-CH₂-OCH₃, -CH=C(CN)-CO-CH(OCH₃)₂, -CH=C(CN)-CO-CH₂-SCH₃, -CH=CH-CO-C₆H₅, -CH=CH-CO-(4-Cl-C₆H₄), -CH=C(CH₃)-CO-C₆H₅, -CH=C(CH₃)-CO-(4-Cl-C₆H₄), -CH=C(C₂H₅)-CO-C₆H₅, -CH=C(C₂H₅)-CO-(4-Cl-C₆H₄), -CH=C(Cl)-CO-C₆H₅, -CH=C(Br)-CO-C₆H₅, -CH=C(CN)-CO-C₆H₅, -CH=CH-CO-NH₂, -CH=CH-CO-NHCH₃, -CH=CH-CO-N(CH₃)₂, -CH=CH-CO-NH-C₂H₅, -CH=CH-CO-N(C₂H₅)₂, -CH=CH-CO-NH-n-C₃H₇, -CH=CH-CO-NH-i-C₃H₇, -CH=CH-CO-NH-tert.-C₄H₉, -CH=CH-CO-NH-cyclopropyl, -CH=CH-CO-NH-cyclobutyl, -CH=CH-CO-NH-cyclopentyl, -CH=CH-CO-NH-cyclohexyl, -CH=CH-CO-NH-cycloheptyl, -CH=CH-CO-NH-cyclooctyl, -CH=CH-CO-pyrrolidin-1-yl, -CH=CH-CO-piperidin-1-yl, -CH=CH-CO-morpholin-4-yl, -CH=CH-CO-NH-CH₂CH=CH₂, -CH=CH-CO-NH-CH₂C≡CH, -CH=CH-CO-N(CH₃)-CH₂C≡CH, -CH=CH-CO-NH-(CH₂)₂Cl, -CH=CH-CO-NH-C₆H₅, -CH=C(CH₃)-CO-NH₂, -CH=C(CH₃)-CO-NHCH₃, -CH=C(CH₃)-CO-N(CH₃)₂, -CH=C(CH₃)-CO-NH-C₂H₅, -CH=C(CH₃)-CO-N(C₂H₅)₂, -CH=C(CH₃)-CO-NH-n-C₃H₇, -CH=C(CH₃)-CO-NH-i-C₃H₇, -CH=C(CH₃)-CO-NH-tert.-C₄H₉, -CH=C(CH₃)-CO-NH-cyclopropyl, -CH=C(CH₃)-CO-NH-cyclobutyl, -CH=C(CH₃)-CO-NH-cyclopentyl, -CH=C(CH₃)-CO-NH-cyclohexyl, -CH=C(CH₃)-CO-NH-cycloheptyl, -CH=C(CH₃)-CO-NH-cyclooctyl, -CH=C(CH₃)-CO-pyyrolidin-1-yl, -CH=C(CH₃)-CO-piperidin-1-yl, -CH=C(CH₃)-CO-morpholin-4-yl, -CH=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -CH=C(CH₃)-CO-NH-CH₂C≡CH, -CH=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CH₃)-CO-NH-(CH₂)₂Cl, -CH=C(CH₃)-CO-NH-C₆H₅, -CH=C(C₂H₅)-CO-NH₂, -CH=C(C₂H₅)-CO-NHCH₃, -CH=C(C₂H₅)-CO-N(CH₃)₂, -CH=C(C₂H₅)-CO-NH-C₂H₅, -CH=C(C₂H₅)-CO-N(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-n-C₃H₇, -CH=C(C₂H₅)-CO-NH-i-C₃H₇, -CH=C(C₂H₅)-CO-NH-tert.-C₄H₉, -CH=C(C₂H₅)-CO-NH-cyclopropyl, -CH=C(C₂H₅)-CO-NH-cyclobutyl, -CH=C(C₂H₅)-CO-NH-cyclopentyl, -CH=C(C₂H₅)-CO-NH-cyclohexyl, -CH=C(C₂H₅)-CO-NH-cycloheptyl, -CH=C(C₂H₅)-CO-NH-cyclooctyl, -CH=C(C₂H₅)-CO-pyrrolidin-1-yl, -CH=C(C₂H₅)-CO-piperidin-1-yl, -CH=C(C₂H₅)-CO-morpholin-4-yl, -CH=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-CH₂C≡CH, -CH=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -CH=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -CH=C(C₂H₅)-CO-NH-C₆H₅, -CH=C(Cl)-CO-NH₂, -CH=C(Cl)-CO-NHCH₃, -CH=C(Cl)-CO-N(CH₃)₂, -CH=C(Cl)-CO-NH-C₂H₅, -CH=C(Cl)-CO-N(C₂H₅)₂, -CH=C(Cl)-CO-NH-n-C₃H₇, -CH=C(Cl)-CO-NH-i-C₃H₇, -CH=C(Cl)-CO-NH-tert.-C₄H₉, -CH=C(Cl)-CO-NH-cyclopropyl, -CH=C(Cl)-CO-NH-cyclobutyl, -CH=C(Cl)-CO-NH-cyclopentyl, -CH=C(Cl)-CO-NH-cyclohexyl, -CH=C(Cl)-CO-NH-cycloheptyl, -CH=C(Cl)-CO-NH-cyclooctyl, -CH=C(Cl)-CO-pyrrolidin-1-yl, -CH=C(Cl)-CO-piperidin-1-yl, -CH=C(Cl)-CO-morpholin-4-yl, -CH=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -CH=C(Cl)-CO-NH-CH₂C≡CH, -CH=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Cl)-CO-NH-(CH₂)₂Cl, -CH=C(Cl)-CO-NH-C₆H₅, -CH=C(Br)-CO-NH₂, -CH=C(Br)-CO-NHCH₃, -CH=C(Br)-CO-N(CH₃)₂, -CH=C(Br)-CO-NH-C₂H₅, -CH=C(Br)-CO-N(C₂H₅)₂, -CH=C(Br)-CO-NH-n-C₃H₇, -CH=C(Br)-CO-NH-i-C₃H₇, -CH=C(Br)-CO-NH-tert.-C₄H₉, -CH=C(Br)-CO-NH-cyclopropyl, -CH=C(Br)-CO-NH-cyclobutyl, -CH=C(Br)-CO-NH-cyclopentyl, -CH=C(Br)-CO-NH-cyclohexyl, -CH=C(Br)-CO-NH-cycloheptyl, -CH=C(Br)-CO-NH-cyclooctyl, -CH=C(Br)-CO-pyrrolidin-1-yl, -CH=C(Br)-CO-piperidin-1-yl, -CH=C(Br)-CO-morpholin-4-yl, -CH=C(Br)-CO-NH-CH₂CH=C(Br)₂, -CH=C(Br)-CO-NH-CH₂C≡CH, -CH=C(Br)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Br)-CO-NH-(CH₂)₂Cl, -CH=C(Br)-CO-NH-C₆H₅, -CH=C(CN)-CO-NH₂, -CH=C(CN)-CO-NHCH₃, -CH=C(CN)-CO-N(CH₃)₂, -CH=C(CN)-CO-NH-C₂H₅, -CH=C(CN)-CO-N(C₂H₅)₂, -CH=C(CN)-CO-NH-n-C₃H₇, -CH=C(CN)-CO-NH-i-C₃H₇, -CH=C(CN)-CO-NH-tert.-C₄H₉, -CH=C(CN)-CO-NH-cyclopropyl, -CH=C(CN)-CO-NH-cyclobutyl, -CH=C(CN)-CO-NH-cyclopentyl, -CH=C(CN)-CO-NH-cyclohexyl, -CH=C(CN)-CO-NH-cycloheptyl, -CH=C(CN)-CO-NH-cyclooctyl, -CH=C(CN)-CO-pyrrolidin-1-yl, -CH=C(CN)-CO-piperidin-1-yl, -CH=C(CN)-CO-morpholin-4-yl, -CH=C(CN)-CO-NH-CH₂CH=C(CN)₂, -CH=C(CN)-CO-NH-CH₂C≡CH, -CH=C(CN)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CN)-CO-NH-(CH₂)₂Cl, -CH=C(CN)-CO-NH-C₆H₅, -CH=CH-CO-SCH₃, -CH=CH-CO-SC₂H₅, -CH=CH-CO-S-n-C₃H₇, -CH=CH-CO-S-i-C₃H₇, -CH=CH-CO-S-n-C₄H₉, -CH=CH-CO-S-tert.-C₄H₉, -CH=C(CH₃)-CO-SCH₃, -CH=C(CH₃)-CO-SC₂H₅, -CH=C(CH₃)-CO-S-n-C₃H₇, -CH=C(CH₃)-CO-S-i-C₃H₇, -CH=C(CH₃)-CO-S-n-C₄H₉, -CH=C(CH₃)-CO-S-tert.-C₄H₉, -CH=C(C₂H₅)-CO-SCH₃, -CH=C(C₂H₅)-CO-SC₂H₅, -CH=C(C₂H₅)-CO-S-n-C₃H₇, -CH=C(C₂H₅)-CO-S-i-C₃H₇, -CH=C(C₂H₅)-CO-S-n-C₄H₉, -CH=C(C₂H₅)-CO-S-tert.-C₄H₉, -CH=C(Cl)-CO-SCH₃, -CH=C(Cl)-CO-SC₂H₅, -CH=C(Cl)-CO-S-n-C₃H₇, -CH=C(Cl)-CO-S-i-C₃H₇, -CH=C(Cl)-CO-S-n-C₄H₉, -CH=C(Cl)-CO-S-tert.-C₄H₉, -CH=C(Br)-CO-SCH₃, -CH=C(Br)-CO-SC₂H₅, -CH=C(Br)-CO-S-n-C₃H₇, -CH=C(Br)-CO-S-i-C₃H₇, -CH=C(Br)-CO-S-n-C₄H₉, -CH=C(Br)-CO-S-tert.-C₄H₉, -CH=C(CN)-CO-SCH₃, -CH=C(CN)-CO-SC₂H₅, -CH=C(CN)-CO-S-n-C₃H₇, -CH=C(CN)-CO-S-i-C₃H₇, -CH=C(CN)-CO-S-n-C₄H₉, -CH=C(CN)-CO-S-tert.-C₄H₉, -CH=C(COCH₃)-CO-OCH₃, -CH=C(COC₂H₅)-CO-OCH₃, -CH=C(CO-n-C₃H₇)-CO-OCH₃, -CH=C(COCH₃)-CO-OC₂H₅, -CH=C(COC₂H₅)-CO-OC₂H₅, -CH=C(CO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COCH₃)-CO-O-n-C₃H₇, -CH=C(COC₂H₅)-CO-O-n-C₃H₇, -CH=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-OCH₃, -CH=C(CF₃)-CO-OC₂H₅, -CH=C(CF₃)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-O-i-C₃H₇, -CH=C(CF₃)-CO-O-n-C₄H₉, -CH=C(CF₃)-CO-O-tert.-C₄H₉, -CH=C(COOCH₃)₂, -CH=C(COOC₂H₅)₂, -CH=C(COOCH₃)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)-CO-OCH₃, -CH=C(COO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)₂, -CH=CH-CH=CH-COOH, -CH=CH-CH=CH-CO-OCH₃, -CH=CH-CH=CH-CO-OC₂H₅, -CH=CH-CH=C(COOCH₃)₂, -CH=CH-CH=C(CN)-CO-OCH₃, -CH=CH-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-OCH₃, -CH=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CH=C(Cl)-CO-OCH₃, -CH=C(CH₃)-CH=C(Br)-CO-OCH₃, -CH=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-NH₂, -CH=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -CH=CH-(CH₂)₂-COOH, -CH=CH-(CH₂)₂-CO-OCH₃, -CH=CH-(CH₂)₂-CO-OC₂H₅, -CH=CH-CH₂-CH(COOCH₃)₂, -CH=CH-CH₂-CH(COOC₂H₅)₂, -CH=CH-CH₂-CH(CN)-CO-OCH₃, -CH=CH-CH₂-CH(CN)-CO-OC₂H₅, -CH=CH-CH₂-CH(CH₃)-CO-OCH₃, -CH=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -CH=CH-(CH₂)₂-CO-NH₂, -CH=CH-(CH₂)₂-CO-NH-CH₃, -CH=CH-CH₂-COOH, -CH=CH-CH₂-CO-OCH₃, -CH=CH-CH₂-CO-OC₂H₅, -CH=C(COOCH₃)-CH₂-CO-OCH₃, -CH=C(COOCH₃)-CH₂-CO-OC₂H₅, -CH=CH-CH₂-CO-NH₂, -CH=CH-CH₂-CO-NH-CH₃, -CH=CH-CH₂-CO-N(CH₃)₂, -CH(OCH₃)₂, -CH(SCH₃)₂, -CH(OC₂H₅)₂, -CH(SC₂H₅)₂, -CH(O-n-C₃H₇)₂, -CH(O-i-C₃H₇)₂, -CH(S-n-C₃H₇)₂, -CH(S-i-C₃H₇)₂, -CH(O-n-C₄H₉)₂, -CH(O-i-C₄H₉)₂, -CH(O-s-C₄H₉)₂, -CH(O-tert.-C₄H₉)₂, -CH(S-n-C₄H₉)₂, -CH(S-i-C₄H₉)₂, -CH(S-s-C₄H₉)₂, -CH(S-tert.-C₄H₉)₂, -CH(OC₅H₁₁)₂, 1,3-Dioxolan-2-yl, 1,3-Dithio­ lan-2-yl, 1,3-Oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 5-Methyl-1,3-oxathiolan-2-yl, 4-Ethyl-1,3-dioxolan-2-yl, 4-Ethyl- 1,4-dithiolan-2-yl, 4-Ethyl-1,3-oxathiolan-2-yl, 5-Ethyl-1,3-oxa­ thiolan-2-yl, 4,5-Dimethyl-1,3-dioxolan-2-yl, 4,4-Dimethyl-1,3- dioxolan-2-yl, 4,5-Dimethyl-1,3-dithiolan-2-yl, 5,5-Dimethyl-1,3- dithiolan-2-yl, 4,5-Dimethyl-1,3-oxathiolan-2-yl, 5,5-Dimethyl- 1,3-oxathiolan-2-yl, 4,4-Dimethyl-1,3-oxathiolan-2-yl, 4-Vinyl- 1,3-dioxolan-2-yl, 4-Vinyl-1,3-dithiolan-2-yl, 4-Vinyl-1,3-oxa­ thiolan-2-yl, 5-Vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3- dioxolan-2-yl, 4-Chlormethyl-1,3-dithiolan-2-yl, 4-Chlormethyl- 1,3-oxathiolan-2-yl, 5-Chlormethyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-1,3-dithio­ lan-2-yl, 4-Hydroxymethyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl- 1,3-oxathiolan-2-yl, 4-Methoxymethyl-1,3-dioxolan-2-yl, 4-Allyl­ oxymethyl-1,3-dioxolan-2-yl, 4-Propargyloxymethyl-1,3-dioxolan- 2-yl, 4-Acetoxymethyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-1,3-dithiolan-2-yl, 4-Propargyl- oxymethyl-1,3-dithiolan-2-yl, 4-Acetoxymethyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl-1,3-oxathiolan-2-yl, 5-Allyloxy- methyl-1,3-oxathiolan-2-yl, 4-Propargyloxymethyl-1,3-oxathiolan-2-yl, 5-Propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxymethyl- 1,3-oxathiolan-2-yl, 5-Acetoxymethyl-1,3-oxathiolan-2-yl, 4-Methylthiomethyl-1,3-dioxolan-2-yl, 4-Methylthiomethyl-1,3- dithiolan-2-yl, 4-Carboxy-1,3-dioxolan-2-yl, 4-Carboxy-1,3- dithiolan-2-yl, 4-Methoxycarbonyl-1,3-dioxolan-2-yl, 4-Ethoxy- carbonyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-1,3-dithiolan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-4-methyl- 1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-di­ thiolan-2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-1,3- dithiolan-2-yl, 1,3-Dioxan-2-yl, 1,3-Dithian-2-yl, 1,3-Oxathian- 2-yl, 5-Methyl-1,3-dioxan-2-yl, 5-Methyl-1,3-dithian-2-yl, 5-Methyl-1,3-oxathian-2-yl, 5,5-Dimethyl-1,3-dioxan-2-yl, 4,6-Dimethyl- 1,3-dioxan-2-yl, 4,4-Dimethyl-1,3-dioxan-2-yl, 5,5-Dimethyl- 1,3-dithian-2-yl, 4,6-Dimethyl-1,3-dithian-2-yl, 4,4-Dimethyl- 1,3-dithian-2-yl, 5,5-Dimethyl-1,3-oxathian-2-yl, 4,4-Dimethyl- 1,3-oxathian-2-yl, 6,6-Dimethyl-1,3-oxathian-2-yl, 4-Hydroxymethyl-1,3-dioxan-2-yl, 4-Methoxymethyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-1,3-dithian-2-yl, 4-Methoxymethyl-1,3-dithian-2-yl, 4-Allyloxymethyl-1,3-dithian-2-yl, 4-Acetoxymethyl- 1,3-dithian-2-yl, 4-Chlormethyl-1,3-dioxan-2-yl, 4-Chlormethyl- 1,3-dithian-2-yl, 1,3-Dioxepan-2-yl, 1,3-Dithiepan-2-yl, 1,3-Dioxep-5-en-2-yl, 4-Methoxycarbonyl-1,3-dioxan-2-yl, 4-Ethoxy- carbonyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-1,3-dithian-2-yl, 4-n-Butoxycarbonyl-1,3-dithian-2-yl, 4-Methoxycarbonyl-4- methyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-Methoxy- carbonyl-4-methyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-4-methyl- 1,3-dithian-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithian-2-yl, -C(CH₃)(OCH₃)₂, -C(CH₃)(SCH₃)₂, -C(CH₃)(OC₂H₅)₂, -C(CH₃)(SC₂H₅)₂, -C(CH₃)(O-n-C₃H₇)₂, -C(CH₃)(O-i-C₃H₇)₂, -C(CH₃)(S-n-C₃H₇)₂, -C(CH₃)(S-i-C₃H₇)₂, -C(CH₃)(O-n-C₄H₉)₂, -C(CH₃)(O-i-C₄H₉)₂, -C(CH₃)(O-s-C₄H₉)₂, -C(CH₃)(O-tert.-C₄H₉)₂, -C(CH₃)(S-n-C₄H₉)₂, -C(CH₃)(S-i-C₄H₉)₂, -C(CH₃)(S-s-C₄H₉)₂, -C(CH₃)(S-tert.-C₄H₉)₂, -C(CH₃)(O-n-C₅H₁₁)′′, 2-Methyl-1,3-dioxolan-2-yl, 2-Methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-oxathiolan-2-yl, 2,4-Dimethyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-1,3- oxathiolan-2-yl, 2,5-Dimethyl-1,3-oxathiolan-2-yl, 4-Ethyl-2- methyl-1,3-dioxolan-2-yl, 4-Ethyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Ethyl-2-methyl-1,3- oxathiolan-2-yl, 2,4,5-Trimethyl-1,3-dioxolan-2-yl, 2,4,4-Trimethyl- 1,3-dioxolan-2-yl, 2,4,5-Trimethyl-1,3-dithiolan-2-yl, 2,4,4-Trimethyl-1,3-dithiolan-2-yl, 2,4,5-Trimethyl-1,3-oxathiolan-2-yl, 2,4,4-Trimethyl-1,3-oxathiolan-2-yl, 2-Methyl-4-vinyl- 1,3-dioxolan-2-yl, 2-Methyl-4-vinyl-1,3-dithiolan-2-yl, 2-Methyl- 4-vinyl-1,3-oxathiolan-2-yl, 2-Methyl-5-vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-dioxolan-2-yl, 4-Chlormethyl-2- methyl-1,3-dithiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl- 2-methyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-2- methyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dioxolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxy- 2-methyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dithiolan-2-yl, 4-Acetoxy-2- methyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Allyloxymethyl- 2-methyl-1,3-oxathiolan-2-yl, 5-Allyloxymethyl-2- methyl-1,3-oxathiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3- oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxy-2-methyl-1,3-oxathiolan-2-yl, 5-Acetoxy-2-methyl- 1,3-oxathiolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dioxolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-2- methyl-1,3-dioxolan-2-yl, 4-Carboxy-2-methyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-2- methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl- 2-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-2- methyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-ethoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4- ethoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-n-butoxy- carbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl-1,3- dithiolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-dioxan-2-yl, 2-Methyl-1,3-dithian-2-yl, 2-Methyl-1,3-oxathian-2-yl, 2,5- Dimethyl-1,3-dioxan-2-yl, 2,5-Dimethyl-1,3-dithian-2-yl, 2,5-Dimethyl- 1,3-oxathian-2-yl, 2,5,5-Trimethyl-1,3-dioxan-2-yl, 2,4,6- Trimethyl-1,3-dioxan-2-yl, 2,2,4-Trimethyl-1,3-dioxan-2-yl, 2,5,5-Trimethyl-1,3-dithian-2-yl, 2,4,6-Trimethyl-1,3-dithian-2-yl, 2,4,4-Trimethyl-1,3-dithian-2-yl, 2,5,5-Trimethyl-1,3-oxathian-2-yl, 2,4,4-Trimethyl-1,3-oxathian-2-yl, 2,6,6-Trimethyl- 1,3-oxathian-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-2- methyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dithian-2-yl, 4-Methoxymethyl-2- methyl-1,3-dithian-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithian-2-yl, 99999 00070 552 001000280000000200012000285919988800040 0002004131038 00004 998804-Acetoxymethyl-2-methyl-1,3-dithian-2-yl, 4-Chlormethyl-2- methyl-1,3-dioxan-2-yl, 4-Chlormethyl-2-methyl-1,3-dithian-2-yl, -C(CH₃)=NH, -C(CH₃)=N-CH₃, -C(CH₃)=N-C₂H₅, -C(CH₃)=N-n-C₃H₇, -(CH₃)=N-i-C₃H₇, -C(CH₃)=N-n-C₄H₉, -C(CH₃)=N-CH₂CH=CH₂, -C(CH₃)=N-CH₂CH=CH₂-CH₃, -C(CH₃)=N-CH₂C≡CH, -C(CH₃)=N-CH₂C≡C-CH₃, -C(CH₃)=N-cyclopropyl, -C(CH₃)=N-cyclobutyl, -C(CH₃)=N-cyclopentyl, -C(CH₃)=N-cyclohexyl, -C(CH₃)=N-cycloheptyl, -C(CH₃)=N-CH₂-CH₂Cl, -C(CH₃)=N-CH₂Cl, -C(CH₃)=N-C₆H₅, -C(CH₃)=N-(2-F-C₆H₄), -C(CH₃)=N-(3-F-C₆H₄), -C(CH₃)=N-(4-F-C₆H₄), -C(CH₃)=N-(2-Cl-C₆H₄), -C(CH₃)=N-(3-Cl-C₆H₄), -C(CH₃)=N-(4-Cl-C₆H₄), -C(CH₃)=N-(2-CH₃-C₆H₄), -C(CH₃)=N-(3-CH₃-C₆H₄), -C(CH₃)=N-(4-CH₃-C₆H₄), -C(CH₃)=N-(2-CF₃-C₆H₄), -C(CH₃)=N-(3-CF₃-C₆H₄), -C(CH₃)=N-(4-CF₃-C₆H₄), -C(CH₃)=N-(2-OCH₃-C₆H₄), -C(CH₃)=N-(3-OCH₃-C₆H₄), -C(CH₃)=N-(4-OCH₃-C₆H₄), -C(CH₃)=N-(4-NO₂-C₆H₄), -C(CH₃)=N-(4-CN-C₆H₄), -C(CH₃)=N-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-(2,4-(CH₃)₂-C₆H₃), -C(CH₃)=N-CH₂-OCH₃, -C(CH₃)=N-CH₂-OC₂H₅, -C(CH₃)=N-CH₂CH₂-OCH₃, -C(CH₃)=N-CH₂CH-OC₂H₅, -C(CH₃)=N-OH, -C(CH₃)=N-OCH₃, -C(CH₃)=N-OC₂H₅, -C(CH₃)=N-O-n-C₃H₇, -C(CH₃)=N-O-i-C₃H₇, -C(CH₃)=N-O-n-C₄H₉, -C(CH₃)=N-O-i-C₄H₉, -C(CH₃)=N-O-s-C₄H₉, -C(CH₃)=N-O-tert.-C₄H₉, -C(CH₃)=N-OCH₂-CH=CH₂, -C(CH₃)=N-OCH(CH₃)-CH=CH₂, -C(CH₃)=N-OCH₂-C≡CH, -C(CH₃)=N-CH(CH₃)-C≡CH, -C(CH₃)=N-OCH₂-CH=C-CH₃, -C(CH₃)=N-OCH₂CH₂-Cl, -C(CH₃)=N-OCH₂CH₂-F, -C(CH₃)=N-OCH₂-CF₃, -C(CH₃)=N-OCH₂-CH=CHCl, -C(CH₃)=N-OCH₂-C(Cl)=CH₂, -C(CH₃)=N-OCH₂-C(Br)=CH₂, -C(CH₃)=N-OCH₂-CH=C(Cl)-CH₃, -C(CH₃)=N-O-CO-CH₃, -C(CH₃)=N-O-CO-C₂H₅, -C(CH₃)=N-OCH₂-CN, -C(CH₃)=N-OCH₂-CH=CH-CH₂-OCH₃, -C(CH₃)=N-OCH₂-CH=CH-CH₂-O-tert.-C₄H₉, -C(CH₃)=N-O-(CH₂)₃-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-(4-Cl-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-C₆H₅, -C(CH₃)=N-OCH₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(3-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-CH₂-(4-CH₃O-C₆H₄), -C(CH₃)=N-OCH₂-CH=C(CH₃)-C₆H₅, -C(CH₃)=N-O-(CH₂)₂-CH=CH-(3,4-Cl₂-C₆H₃), -C(CH₃)=N-O-(CH₂)₃-C≡C-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-OCH₃, -C(CH₃)=N-OCH₂CH₂-OCH₃, -C(CH₃)=N-OCH₂-OC₂H₅, -C(CH₃)=N-OCH(CH₃)-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=N-NH₂, -C(CH₃)=N-NH-CH₃, -C(CH₃)=N-NH-C₂H₅, -C(CH₃)=N-NH-n-C₃H₇, -C(CH₃)=N-NH-i-C₃H₇, -C(CH₃)=N-NH-n-C₄H₉, -C(CH₃)=N-NH-i-C₄H₉, -C(CH₃)=N-NH-s-C₄H₉, -C(CH₃)=N-NH-tert.-C₄H₉, -C(CH₃)=N-NH-cyclopropyl, -C(CH₃)=N-NH-cyclobutyl, -C(CH₃)=N-NH-cyclopentyl, -C(CH₃)=N-NH-cyclohexyl, -C(CH₃)=N-NH-cycloheptyl, -C(CH₃)=N-N(CH₃)₂, -C(CH₃)=N-N(C₂H₅)₂, -C(CH₃)=N-N(n-C₃H₇)₂, -C(CH₃)=N-N(i-C₃H₇)₂, -C(CH₃)=N-NH-CH₂-C=CH, -C(CH₃)=N-NH-CH₂-C≡CH, -C(CH₃)=N-N(CH₃)-CH₂-C≡CH, -C(CH₃)=N-NH-CH₂CF₃, -C(CH₃)=N-NH-CO-CH₃, -C(CH₃)=N-NH-CO-C₂H₅, -C(CH₃)=N-NH-CO-OCH₃, -C(CH₃)=N-NH-CO-OC₂H₅, -C(CH₃)=N-NH-CO-O-tert.-C₄H₉, -C(CH₃)=N-pyrrolidin-1-yl, -C(CH₃)=N-piperidin-1-yl, -C(CH₃)=N-morpholin-4-yl, -C(CH₃)=N-NH-C₆H₅, -C(CH₃)=N-NH-(4-Cl-C₆H₄), -C(CH₃)=N-NH-(4-NO₂-C₆H₄), -C(CH₃)=N-NH-(4-F-C₆H₄), -C(CH₃)=N-NH-(4-CH₃O-C₆H₄), -C(CH₃)=N-NH-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-NH-(2,4-(NO₂)₂-C₆H₃), -C(CH₃)=N-NH-CO-NH₂, -C(CH₃)=N-NH-CO-NHCH₃, -C(CH₃)=N-NH-CO-NHC₂H₅, -C(CH₃)=N-NH-CO-N(CH₃)₂, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=CH-CO-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -(CH₃)=CH-CO-O-n-C₄H₉, -C(CH₃)=CH-CO-O-tert.-C₄H₉, -C(CH₃)=CH-CO-O-cyclopropyl, -C(CH₃)=CH-CO-O-cyclobutyl, -C(CH₃)=CH-CO-O-cyclopentyl, -C(CH₃)=CH-CO-O-cyclohexyl, -C(CH₃)=CH-CO-O-cycloheptyl, -C(CH₃)=C(CH₃)-COOH, -C(CH₃)=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-cyclopropyl, -C(CH₃)=C(CH₃)-CO-O-cyclobutyl, -C(CH₃)=C(CH₃)-CO-O-cyclopentyl, -C(CH₃)=C(CH₃)-CO-O-cyclohexyl, -C(CH₃)=C(CH₃)-CO-O-cycloheptyl, -C(CH₃)=C(C₂H₅)-COOH, -C(CH₃)=C(C₂H₅)-CO-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-cyclo­ propyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-O- cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-O-cycloheptyl, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-O-n-C₄H₉, -C(CH₃)=C(Cl)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-O-cyclopropyl, -C(CH₃)=C(Cl)-CO-O-cyclobutyl, -C(CH₃)=C(Cl)-CO-O-cyclopentyl, -C(CH₃)=C(Cl)-CO-O-cyclohexyl, -C(CH₃)=C(Cl)-CO-O-cycloheptyl, -C(CH₃)=C(Br)-COOH, -C(CH₃)=C(Br)-CO-OCH₃, -C(CH₃)=C(Br)-CO-OC₂H₅, -C(CH₃)=C(Br)-CO-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-O-n-C₄H₉, -C(CH₃)=C(Br)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-O-cyclopropyl, -C(CH₃)=C(Br)-CO-O-cyclobutyl, -C(CH₃)=C(Br)-CO-O-cyclopentyl, -C(CH₃)=C(Br)-CO-O-cyclohexyl, -C(CH₃)=C(Br)-CO-O-cycloheptyl, -C(CH₃)=C(CN)-COOH, -C(CH₃)=C(CN)-CO-OCH₃, -C(CH₃)=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CN)-CO-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-O-n-C₄H₉, -C(CH₃)=C(CN)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-O-cyclopropyl, -C(CH₃)=C(CN)-CO-O-cyclobutyl, -C(CH₃)=C(CN)-CO-O-cyclopentyl, -C(CH₃)=C(CN)-CO-O-cyclohexyl, -C(CH₃)=C(CN)-CO-O-cycloheptyl, -C(CH₃)=CH-CO-OCH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-OCH(CH₃)-OCH₃, -C(CH₃)=CH-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=CH-CO-OCH₂CH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=(C₂H₅)-CO-OCH₂CH₂-OCH₃, -(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-O-i-C₃H₇, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-O-i-C₃H₇, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-O-i-C₃H₇, -C(CH₃)=C(CN)-CO-OCH(CH₃)OCH₃, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-CF₃, -C(CH₃)=CH-CO-OCH₂-CCl₃, -C(CH₃)=CH-CO-OCH₂-oxiranyl, -C(CH₃)=CH-CO-(CH₂)₃-Br,-C(CH₃)=CH-CO-OCH₂-CH=CH₂, -C(CH₃)=CH-CO-OCH₂-C≡CH, -C(CH₃)=CH-CO-OCH₂-CN, -C(CH₃)=CH-CO-OCH₂CH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CF₃, -C(CH₃)=C(CH₃)-CO-OCH₂-CCl₃, -C(CH₃)=C(CH₃)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CH₃)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CH₃)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CH₃)-CO-OCH₂-C≡CH, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CF₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CCl₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-oxiranyl, -C(CH₃)=C(C₂H₅)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(C₂H₅)CO-OCH₂-C≡CH, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂-CF₃, -C(CH₃)=C(Cl)-CO-OCH₂-CCl₃, -C(CH₃)=C(Cl)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Cl)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Cl)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Cl)-CO-OCH₂-C≡CH, -C(CH₃)=C(Cl)-CO-OCH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂-CF₃, -C(CH₃)=C(Br)-CO-OCH₂-CCl₃, -C(CH₃)=C(Br)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Br)-CO-O(CH₂)₃-Br, -C(CH₃)=C(Br)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Br)-CO-OCH₂-C≡CH, -C(CH₃)=C(Br)-CO-OCH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂CH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂-CF₃, -C(CH₃)=C(CN)-CO-OCH₂-CCl₃, -C(CH₃)=C(CN)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CN)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(CN)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CN)-CO-OCH₂-C≡CH, -C(CH₃)=C(CN)-CO-OCH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂CH₂-CN, -C(CH₃)=CH-CO-CH₃, -C(CH₃)=CH-CO-C₂H₅, -C(CH₃)=CH-CO-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-n-C₄H₉, -C(CH₃)=CH-CO-tert.-C₄H₉, -C(CH₃)=CH-CO-CH₂Cl, -C(CH₃)=CH-CO-CH₂Br, -C(CH₃)=CH-CO-CHCl₂, -C(CH₃)=CH-CO-CH₂-OCH₃, -C(CH₃)=CH-CO-CH(OCH₃)₂, -C(CH₃)=CH-CO-CH₂-SCH₃, -C(CH₃)=C(CH₃)-CO-CH₃, -C(CH₃)=C(CH₃)-CO-C₂H₅, -C(CH₃)=C(CH₃)-CO-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-CH₂Cl, -C(CH₃)=C(CH₃)-CO-CH₂Br, -C(CH₃)=C(CH₃)-CO-CHCl₂, -C(CH₃)=C(CH₃)-CO-CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-CH(OCH₃)₂, -C(CH₃)=C(CH₃)-CO-CH₂-SCH₃, -C(CH₃)=C(C₂H₅)-CO-CH₃, -C(CH₃)=C(C₂H₅)-CO-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-CH₂Cl, -C(CH₃)=C(C₂H₅)-CO-CH₂Br, -C(CH₃)=C(C₂H₅)-CO-CHCl₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-CH(OCH₃)₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-SCH₃, -C(CH₃)=C(Cl)-CO-CH₃, -C(CH₃)=C(Cl)-CO-C₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-n-C₄H₉, -C(CH₃)=C(Cl)-CO-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-CH₂Cl, -C(CH₃)=C(Cl)-CO-CHCl₂, -C(CH₃)=C(Cl)-CO-CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-CH(OCH₃)₂, -C(CH₃)=C(Cl)-CO-CH₂-SCH₃, -C(CH₃)=C(Br)-CO-CH₃, -C(CH₃)=C(Br)-CO-C₂H₅, -C(CH₃)=C(Br)-CO-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-n-C₄H₉, -C(CH₃)=C(Br)-CO-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-CH₂Cl, -C(CH₃)=C(Br)-CO-CH₂Br, -C(CH₃)=C(Br)-CO-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-CH(OCH₃)₂, -C(CH₃)=C(Br)-CO-CH₂-SCH₃, -C(CH₃)=C(CN)-CO-CH₃, -C(CH₃)=C(CN)-CO-C₂H₅, -C(CH₃)=C(CN)-CO-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-n-C₄H₉, -C(CH₃)=C(CN)-CO-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-CH₂Cl, -C(CH₃)=C(CN)-CO-CH₂Br, -C(CH₃)=C(CN)-CO-CHCl₂, -C(CH₃)=C(CN)-CO-CH₂-OCH₃, -C(CH₃)=C(CN)-CO-CH(OCH₃)₂, -C(CH₃)=C(CN)-CO-CH₂-SCH₃, -C(CH₃)=CH-CO-C₆H₅, -C(CH₃)=CH-CO-(4-Cl-C₆H₄), -C(CH₃)=C(CH₃)-CO-C₆H₅, -C(CH₃)=C(CH₃)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(C₂H₅)-CO-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(Cl)-CO-C₆H₅, -C(CH₃)=C(Br)-CO-C₆H₅, -C(CH₃)=C(CN)-CO-C₆H₅, -C(CH₃)=CH-CO-NH₂, -C(CH₃)=CH-CO-NHCH₃, -C(CH₃)=CH-CO-N(CH₃)₂, -C(CH₃)=CH-CO-NH-C₂H₅, -C(CH₃)=CH-CO-N(C₂H₅)₂, -C(CH₃)=CH-CO-NH-n-C₃H₇, -C(CH₃)=CH-CO-NH-i-C₃H₇, -C(CH₃)=CH-CO-NH-tert.-C₄H₉, -C(CH₃)=CH-CO-NH-cyclopropyl, -C(CH₃)=CH-CO-NH-cyclobutyl, -C(CH₃)=CH-CO-NH-cyclopentyl, -C(CH₃)=CH-CO-NH-cyclohexyl, -C(CH₃)=CH-CO-NH-cycloheptyl, -C(CH₃)=CH-CO-NH-cyclooctyl, -C(CH₃)=CH-CO-pyrrolidin-1-yl, -C(CH₃)=CH-CO-piperidin-1-yl, -C(CH₃)=CH-CO-morpholin-4-yl, -C(CH₃)=CH-CO-NH-CH₂CH=CH₂, -C(CH₃)=CH-CO-NH-CH₂C≡CH, -C(CH₃)=CH-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=CH-CO-NH-(CH₂)₂Cl, -C(CH₃)=CH-CO-NH-C₆H₅, -C(CH₃)=C(CH₃)-CO-NH₂, -C(CH₃)=C(CH₃)-CO-NHCH₃, -C(CH₃)=C(CH₃)-CO-N(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-C₂H₅, -C(CH₃)=C(CH₃)-CO-N(C₂H₅)₂, -C(CH₃)=C(CH₃)-CO-NH-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-NH- cyclopropyl, -C(CH₃)=C(CH₃)-CO-NH-cyclobutyl, -C(CH₃)=C(CH₃)-CO-NH-cyclopentyl, -C(CH₃)=C(CH₃)-CO-NH- cyclohexyl, -C(CH₃)=C(CH₃)-CO-NH-cycloheptyl, -C(CH₃)=C(CH₃)-CO-NH-cyclooctyl, -C(CH₃)=C(CH₃)-CO- pyrrolidin-1-yl, -C(CH₃)=C(CH₃)-CO-piperidin-1-yl, -C(CH₃)=C(CH₃)-CO-morpholin-4-yl, -C(CH₃)=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-NH(CH₂)₂Cl, -C(CH₃)=C(CH₃)-CO-NH-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-NH₂, -C(CH₃)=C(C₂H₅)-CO-NHCH₃, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)₂, -C(CH₃)=C(C₂H₅)-CO-NH-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-N(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-NH- cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclo­ hexyl, -C(CH₃)=C(C₂H₅)-CO-NH-cycloheptyl, -C(CH₃)=C(C₂H₅)-CO-NH- cyclooctyl, -C(CH₃)=C(C₂H₅)-CO-pyrrolidin-1-yl, -C(CH₃)=C(C₂H₅)-CO-piperidin-1-yl, -C(CH₃)=C(C₂H₅)-CO- morpholin-4-yl, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(C₂H₅)-CO-NH-C₆H₅, -C(CH₃)=C(Cl)-CO-NH₂, -C(CH₃)=C(Cl)-CO-NHCH₃, -C(CH₃)=C(Cl)-CO-N(CH₃)₂, -C(CH₃)=C(Cl)-CO-NH-C₂H₅, -C(CH₃)=C(Cl)-CO-N(C₂H₅)₂, -C(CH₃)=C(Cl)-CO-NH-n-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-i-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-NH-cyclopropyl, -C(CH₃)=C(Cl)-CO-NH-cyclobutyl, -C(CH₃)=C(Cl)-CO-NH-cyclopentyl, -C(CH₃)=C(Cl)-CO-NH-cyclohexyl, -C(CH₃)=C(Cl)-CO-NH-cycloheptyl, -C(CH₃)=C(Cl)-CO-NH-cyclooctyl, -C(CH₃)=C(Cl)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Cl)-CO-piperidin-1- yl, -C(CH₃)=C(Cl)-CO-morpholin-4-yl, -C(CH₃)=C(Cl)-CO-NH-CH₂CH=C(Cl)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Cl)-CO-NH-C₆H₅, -C(CH₃)=C(Br)-CO-NH₂, -C(CH₃)=C(Br)-CO-NHCH₃, -C(CH₃)=C(Br)-CO-N(CH₃)₂, -C(CH₃)=C(Br)-CO-NH-C₂H₅, -C(CH₃)=C(Br)-CO-N(C₂H₅)₂, -C(CH₃)=C(Br)-CO-NH-n-C₃H₇, -C(CH₃)=C(Br)-CO-NH-i-C₃H₇, -C(CH₃)=C(Br)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-NH-cyclopropyl, -C(CH₃)=C(Br)-CO-NH-cyclobutyl, -C(CH₃)=C(Br)-CO-NH-cyclopentyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cycloheptyl, -C(CH₃)=C(Br)-CO-NH-cyclooctyl, -C(CH₃)=C(Br)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Br)-CO-piperidin-1-yl, -C(CH₃)=C(Br)-CO-morpholin-4-yl, -C(CH₃)=C(Br)-CO-NH-CH₂CH=C(Br)₂, -C(CH₃)=C(Br)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Br)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Br)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Br)-CO-NH-C₆H₅, -C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CN)-CO-NHCH₃, -C(CH₃)=C(CN)-CO-N(CH₃)₂, -C(CH₃)=C(CN)-CO-NH-C₂H₅, -C(CH₃)=C(CN)-CO-N(C₂H₅)₂, -C(CH₃)=C(CN)-CO-NH-n-C₃H₇, -C(CH₃)=C(CN)-CO-NH-i-C₃H₇, -C(CH₃)=C(CN)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-NH-cyclopropyl, -C(CH₃)=C(CN)-CO-NH-cyclobutyl, -C(CH₃)=C(CN)-CO-NH-cyclopentyl, -C(CH₃)=C(CN)-CO-NH-cyclohexyl, -C(CH₃)=C(CN)-CO-NH-cycloheptyl, -C(CH₃)=C(CN)-CO-NH-cyclooctyl, -C(CH₃)=C(CN)-CO-pyrrolidin-1-yl, -C(CH₃)=C(CN)-CO-piperidin-1-yl, -C(CH₃)=C(CN)-CO-morpholin-4-yl, -C(CH₃)=C(CN)-CO-NH-CH₂CH=C(CN)₂, -C(CH₃)=C(CN)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CN)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)=C(CN)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CN)-CO-NH-C₆H₅, -C(CH₃)=CH-CO-SCH₃, -C(CH₃)=CH-CO-SC₂H₅, -C(CH₃)=CH-CO-S-n-C₃H₇, -C(CH₃)=CH-CO-S-i-C₃H₇, -C(CH₃)=CH-CO-S-n-C₄H₉, -C(CH₃)=CH-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-SCH₃, -C(CH₃)=C(CH₃)-CO-SC₂H₅, -C(CH₃)=C(CH₃)CO-S-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-S-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-SCH₃, -C(CH₃)=C(C₂H₅)-CO-SC₂H₅, -C(CH₃)=C(C₂H₅)-CO-S-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-SCH₃, -C(CH₃)=C(Cl)-CO-SC₂H₅, -C(CH₃)=C(Cl)-CO-S-n-C₃H₇, -C(CH₃)=C(Cl)-CO-S-i-C₃H₇, -C(CH₃)=C(Cl)-CO-S-n-C₄H₉, -C(CH₃)=C(Cl)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-SCH₃, -C(CH₃)=C(Br)-CO-SC₂H₅, -C(CH₃)=C(Br)-CO-S-n-C₃H₇, -C(CH₃)=C(Br)-CO-S-i-C₃H₇, -C(CH₃)=C(Br)-CO-S-n-C₄H₉, -C(CH₃)=C(Br)-CO-S-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-SCH₃, -C(CH₃)=C(CN)-CO-SC₂H₅, -C(CH₃)=C(CN)-CO-S-n-C₃H₇, -C(CH₃)=C(CN)-CO-S-i-C₃H₇, -C(CH₃)=C(CN)-CO-S-N-C₄H₉, -C(CH₃)=C(CN)-CO-S-tert.-C₄H₉, -C(CH₃)=C(COCH₃)-CO-OCH₃, -C(CH₃)=C(COC₂H₅)-CO-OCH₃, -C(CH₃)=C(CO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COCH₃)-CO-OC₂H₅, -C(CH₃)=C(COC₂H₅)-CO-OC₂H₅, -C(CH₃)=C(CO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COCH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(COC₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-OCH₃, -C(CH₃)=C(CF₃)-CO-OC₂H₅, -C(CH₃)=C(CF₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CF₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(COOCH₃)₂, -C(CH₃)=C(COOC₂H₅)₂, -C(CH₃)=C(COOCH₃)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)₂, -C(CH₃)=CH-CH=CH-COOH, -C(CH₃)=CH-CH=CH-CO-OCH₃, -C(CH₃)=CH-CH=CH-CO-OC₂H₅, -C(CH₃)=CH-CH=C(COOCH₃)₂, -C(CH₃)=CH-CH=C(CN)-CO-OCH₃, -C(CH₃)=CH-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH₂, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -C(CH₃)=CH-(CH₂)₂-COOH, -C(CH₃)=CH-(CH₂)₂-CO-OCH₃, -C(CH₃)=CH-(CH₂)₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(COOCH₃)₂, -C(CH₃)=CH-CH₂-CH(COOC₂H₅)₂, -C(CH₃)=CH-CH₂-CH(CN)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CN)-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -C(CH₃)=CH-(CH₂)₂-CO-NH₂, -C(CH₃)=CH-(CH₂)₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-COOH, -C(CH₃)=CH-CH₂-CO-OCH₃, -C(CH₃)=CH-CH₂-CO-OC₂H₅, -C(CH₃)=C(COOCH₃)-CH₂-CO-OCH₃, -C(CH₃)=C(COOCH₃)-CH₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CO-NH₂, -C(CH₃)=CH-CH₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-CO-N(CH₃)₂.
wobei W für eine der folgenden Bedeutungen steht:
-CHO, -COCH₃, -COC₂H₅, -COn-C₃H₇, -CO-i-C₃H₇, -CO-n-C₄H₉, -CO-i-C₄H₉, -CO-s-C₄H₉, -CO-tert.-C₄H₉, -CO-CH₂CH=CH₂, -CO-CF₃, -COCCl₃, -COCH₂C≡CH, -CO-cyclopropyl, -CO-cyclobutyl, -CO-cyclopentyl, -CO-cyclohexyl, -CO-CN, -CO-COOCH₃, -CO-COOC₂H₅, -CH=NH, -CH=NCH₃, -CH=NC₂H₅, -CH=N-n-C₃H₅, -CH=N-i-C₃H₅, -CH=N-n-C₄H₉, -CH=NCH₂CH=CH₂, -CH=NCH₂CH=CH₂-CH₃, -CH=NCH₂≡CH, -CH=NCH₂C≡C-CH₃, -CH=N-cyclopropyl, -CH=N-cyclobutyl, -CH=N-cyclopentyl, -CH=N-cyclohexyl, -CH=N-cycloheptyl, -CH=N-CH₂-CH₂Cl, -CH=N-CH₂Cl, -CH=N-₆H₅, -CH=N-(4-Br-C₆H₄), -CH=N-3-F-C₆H₄, -CH=N-4-F-C₆H₄, -CH=N-2-Cl-C₆H₄, -CH=N-3-Cl-C₆H₄, -CH=N-4-Cl-C₆H₄, -CH=N-2-Br-C₆H₄, -CH=N-2-F-C₆H₄, -CH=N-2-CH₃-C₆H₄, -CH=N-3-CH₃-C₆H₄, -CH=N-4-CH₃-C₆H₄, -CH=N-2-CF₃-C₆H₄, -CH=N-3-CF₃-C₆H₄, -CH=N-4-CF₃-C₆H₄, -CH=N-2-OCH₃-C₆H₄, -CH=N-3-OCH₃-C₆H₄, -CH=N-4-OCH₃-C₆H₄, -CH=N-4-NO₂-C₆H₄, -CH=N-4-CN-C₆H₄, -CH=N-2,4-(Cl,Cl)-C₆H₄, -CH=N-2,4-(CH₃,CH₃)-C₆H₄, -CH=N-CH₂OCH₃ -CH=N-CH₂OC₂H₅, -CH=N-CH₂CH₂OCH₃, -CH=N-CH₂CH₂OC₂H₅, -CH=N-OH, -CH=N-OCH₃, -CH=N-OC₂H₅, -CH=N-O-n-C₃H₇, -CH=N-O-i-C₃H₇, -CH=N-O-n-C₄H₉, -CH=N-O-i-C₄H₉, -CH=N-O-s-C₄H₉, -CH=N-O-tert.-C₄H₉, -CH=N-O-CH₂CH=CH₂, -CH=N-O-CH(CH₃)CH=CH₂, -CH=N-O-CH₂C≡CH, -CH=N-O-CH(CH₃)-C≡CH, -CH=N-O-CH₂-CH=CH-CH₃, -CH=N-O-CH₂-CH₂-Cl, -CH=N-O-CH₂-CH₂-F, -CH=N-O-CH₂-CF₃, -CH=N-O-CH₂-CH=CHCl, -CH=N-O-CH₂-CCl=CH₂, -CH=N-O-CH₂-CBr=CH₂, -CH=N-O-CH₂-CH=CCl-CH₃, -CH=N-OC(O)CH₃, -CH=N-OC(O)C₂H₅, -CH=N-O-CH₂-CN, -CH=N-O-CH₂-CH=CH-CH₂-O-CH₃, -CH=N-O-CH₂-CH=CH-CH₂-O-tert.-C₄H₉, -CH=N-O-(CH₂)₃-C₆H₅, -CH=N-O-(CH₂)₄-C₆H₅, -CH=N-O-(CH₂)₄-4-Cl-C₆H₄, -CH=N-O-(CH₂)₄-4-OCH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-CH₃-C₆H₄, -CH=N-O-(CH₂)₄-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-C₆H₅, -CH=N-O-CH₂CH=CH-4-F-C₆H₄, -CH=N-O-CH₂CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CH-3-OCH₃-C₆H₄, -CH=N-O-(CH₂)₂CH=CH-4-F-C₆H₄, -CH=N-O-(CH₂)CH=CH-4-Cl-C₆H₄, -CH=N-O-CH₂CH=CHCH₂-4-OCH₃-C₆H₄, -CH=N-O-CH₂-CH=C(CH₃)-C₆H₄ -CH=N-O-(CH₂)₂CH=CH-3,4(Cl,Cl)-C₆H₃, -CH=N-O-(CH₂)₃C≡C-4-F-C₆H₄, -CH₂=N-OCHOCH₃, -CH=N-OC₂H₄OCH₃, -CH=N-OCH₂OC₂H₅, -CH=N-OCH(CH₃)OCH₃, -CH=N-OCH(CH₃)COOCH₃, -CH=N-OCH(CH₃)COO-n-C₄H₉, -CH=N-NH₂, -CH=N-NHCH₃, -CH=N-NHC₂H₅, -CH=N-NH-n-C₃H₇, -CH=N-NH-i-C₃H₇, -CH=N-NH-n-C₄H₉, -CH=N-NH-cyclopropyl, -CH=N-NH-cyclobutyl, -CH=N-NH-cyclopentyl, -CH=N-NH-cyclohexyl, -CH=N-NH-cycloheptyl, -CH=N-N(CH₃)₂, -CH=N-N(C₂H₅)₂, -CH=N-N(C₃H₇)₂, -CH=N-N(i-C₃H₇)(CH₃), -CH=N-NHCH₂-C=CH, -CH=N-NHCH₂-C≡CH, -CH=N-N(CH₃)-CH₂-C≡CH, -CH=N-NHCH₂CF₃, -CH=N-NH-CO-CH₃, -CH=N-NH-CO-CH₂H₅, -CH=N-NH-COOCH₃, -CH=N-NH-COOC₂H₅, -CH=N-NH-COO-tert.-C₄H₉, -CH=N-pyrrolidin-1-yl, -CH=N-piperidin-1-yl, -CH=N-morpholin-4-yl, -CH=N-NH-C₆H₅, -CH=N-NH-(4-Cl-C₆H₄), -CH=N-NH-(4-NO₂-C₆H₄), -CH=N-NH-(4-F-C₆H₄), -CH=N-NH-(4-CH₃O-C₆H₄), -CH=N-NH-(2,4-Cl₂-C₆H₃), -CH=N-NH-(2,4-(NO₂)₂-C₆H₃), -CH=N-NH-CO-NH₂, -CH=N-NH-CO-NHCH₃, -CH=N-NH-CO-NHC₂H₅, -CH=N-NH-CO-N(CH₃)₂, -CH=CH-COOH, -CH=CH-CO-OCH₃, -CH=C-CO-OC₂H₅, -CH=CH-CO-O-n-C₃H₇, -CH=CH-CO-O-i-C₃H₇, -CH=CH-CO-O-n-C₄H₉, -CH=CH-CO-O-tert.-C₄H₉, -CH=CH-CO-O-cyclopropyl, -CH=CH-CO-O-cyclobutyl, -CH=CH-CO-O-cyclopentyl, -CH=CH-CO-O-cyclohexyl, -CH=CH-CO-O-cycloheptyl, -CH=C(CH₃)-COOH, -CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CO-O-n-C₃H₇, -CH=C(CH₃)-CO-O-i-C₃H₇, -CH=C(CH₃)-CO-O-n-C₄H₉, -CH=C(CH₃)-CO-O-tert.-C₄H₉, -CH=C(CH₃)-CO-O-cyclopropyl, -CH=C(CH₃)-CO-O-cyclobutyl, -CH=C(CH₃)-CO-O-cyclopentyl, -CH=C(CH₃)-CO-O-cyclohexyl, -CH=C(CH₃)-CO-O-cycloheptyl, -CH=C(C₂H₅)-COOH, -CH=C(C₂H₅)-CO-OCH₃, -CH=C(C₂H₅)-CO-OC₂H₅, -CH=C(C₂H₅)-CO-O-n-C₃H₇, -CH=C(C₂H₅)-CO-O-i-C₃H₇, -CH=C(C₂H₅)-CO-O-n-C₄H₉, -CH=C(C₂H₅)-CO-O-tert.-C₄H₉, -CH=C(C₂H₅)-CO-O-cyclopropyl, -CH=C(C₂H₅)-CO-O-cyclobutyl, -CH=C(C₂H₅)-CO-O-cyclopentyl, -CH=C(C₂H₅)-CO-O-cyclohexyl, -CH=C(C₂H₅)-CO-O-cycloheptyl, -CH=C(Cl)-COOH, -CH=C(Cl)-CO-OCH₃, -CH=C(Cl)-CO-OC₂H₅, -CH=C(Cl)-CO-O-n-C₃H₇, -CH=C(Cl)-CO-O-i-C₃H₇, -CH=C(Cl)-CO-O-n-C₄H₉, -CH=C(Cl)-CO-O-tert.-C₄H₉, -CH=C(Cl)-CO-O-cyclopropyl, -CH=C(Cl)-CO-O-cyclobutyl, -CH=C(Cl)-CO-O-cyclopentyl, -CH=C(Cl)-CO-O-cyclohexyl, -CH=C(Cl)-CO-O-cycloheptyl, -CH=C(Br)-COOH, -CH=C(Br)-CO-OCH₃, -CH=C(Br)-CO-OC₂H₅, -CH=C(Br)-CO-O-n-C₃H₇, -CH=C(Br)-CO-O-i-C₃H₇, -CH=C(Br)-CO-O-n-C₄H₉, -CH=C(Br)-CO-O-tert.-C₄H₉, -CH=C(Br)-CO-O-cyclopropyl, -CH=C(Br)-CO-O-cyclobutyl, -CH=C(Br)-CO-O-cyclopentyl, -CH=C(Br)-CO-O-cyclohexyl, -CH=C(Br)-CO-O-cycloheptyl, -CH=C(CN)-COOH, -CH=C(CN)-CO-OCH₃, -CH=C(CN)-CO-OC₂H₅, -CH=C(CN)-CO-O-n-C₃H₇, -CH=C(CN)-CO-O-i-C₃H₇, -CH=C(CN)-CO-O-n-C₄H₉, -CH=C(CN)-CO-O-tert.-C₄H₉, -CH=C(CN)-CO-O-cyclopropyl, -CH=C(CN)-CO-O-cyclobutyl, -CH=C(CN)-CO-O-cyclopentyl, -CH=C(CN)-CO-O-cyclohexyl, -CH=C(CN)-CO-O-cycloheptyl, -CH=CH-CO-OCH₂-OCH₃, -CH=CH-CO-OCH₂-OC₂H₅, -CH=CH-CO-OCH₂-O-n-C₃H₅, -CH=CH-CO-OCH₂-O-i-C₃H₅, -CH=CH-CO-OCH(CH₃)-OCH₃, -CH=CH-CO-OCH(CH₃)-OC₂H₅, -CH=CH-CO-O-CH₂CH₂-OCH₃, -CH=CH-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-OCH₃, -CH=C(CH₃)-CO-OCH₂-OC₂H₅, -CH=C(CH₃)-CO-OCH₂-O-n-C₃H₅, -CH=C(CH₃)-CO-OCH₂-O-i-C₃H₅, -CH=C(CH₃)-CO-OCH(CH₃)-OCH₃, -CH=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CH₃)-CO-O-CH₂CH₂-OCH₃, -CH=C(CH₃)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-OCH₃, -CH=C(C₂H₅)-CO-OCH₂-OC₂H₅, -CH=C(C₂H₅)-CO-OCH₂-O-n-C₃H₅, -CH=C(C₂H₅)-CO-OCH₂-O-i-C₃H₅, -CH=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -CH=C(C₂H₅)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-OCH₃, -CH=C(Cl)-CO-OCH₂-OC₂H₅, -CH=C(Cl)-CO-OCH₂-O-n-C₃H₅, -CH=C(Cl)-CO-OCH₂-O-i-C₃H₅, -CH=C(Cl)-CO-OCH(CH₃)-OCH₃, -CH=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Cl)-CO-O-CH₂CH₂-OCH₃, -CH=C(Cl)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-OCH₃, -CH=C(Br)-CO-OCH₂-OC₂H₅, -CH=C(Br)-CO-OCH₂-O-n-C₃H₅, -CH=C(Br)-CO-OCH₂-O-i-C₃H₅, -CH=C(Br)-CO-OCH(CH₃)-OCH₃, -CH=C(Br)-CO-OCH(CH₃)-OC₂H₅, -CH=C(Br)-CO-O-CH₂CH₂-OCH₃, -CH=C(Br)-CO-O-CH₂CH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-OCH₃, -CH=C(CN)-CO-OCH₂-OC₂H₅, -CH=C(CN)-CO-OCH₂-O-n-C₃H₅, -CH=C(CN)-CO-OCH₂-O-i-C₃H₅, -CH=C(CN)-CO-OCH(CH₃)-OCH₃, -CH=C(CN)-CO-OCH(CH₃)-OC₂H₅, -CH=C(CN)-CO-O-CH₂CH₂-OCH₃, -CH=C(CN)-CO-O-CH₂CH₂-OC₂H₅, -CH=CH-CO-OCH₂-CF₃, -CH=CH-CO-OCH₂-CCl₃, -CH=CH-CO-OCH₂-oxiranyl, -CH=CH-CO-O(CH₂)₃-Br, -CH=CH-CO-OCH₂-CH=CH₂, -CH=CH-CO-OCH₂-C≡CH, -CH=CH-CO-OCH₂-CN, -CH=CH-CO-O(CH₂)₂-CN, -CH=C(CH₃)-CO-OCH₂-CF₃, -CH=C(CH₃)-CO-OCH₂-CCl₃, -CH=C(CH₃)-CO-OCH₂-oxiranyl, -CH=C(CH₃)-CO-O(CH₂)₃-Br, -CH=C(CH₃)-CO-OCH₂-CH=CH₂, -CH=C(CH₃)-CO-OCH₂-C≡CH, -CH=C(CH₃)-CO-OCH₂-CN, -CH=C(CH₃)-CO-O(CH₂)₂-CN, -CH=C(C₂H₅)-CO-OCH₂-CF₃, -CH=C(C₂H₅)-CO-OCH₂-CCl₃, -CH=C(C₂H₅)-CO-OCH₂-oxiranyl, -CH=C(C₂H₅)-CO-O(CH₂)₃-Br, -CH=C(C₂H₅)-CO-OCH₂-CH=CH₂, -CH=C(C₂H₅)-CO-OCH₂-C≡CH, -CH=C(C₂H₅)-CO-OCH₂-CN, -CH=C(C₂H₅)-CO-O(CH₂)₂-CN, -CH=C(Cl)-CO-OCH₂-CF₃, -CH=C(Cl)-CO-OCH₂-CCl₃, -CH=C(Cl)-CO-OCH₂-oxiranyl, -CH=C(Cl)-CO-O(CH₂)₃-Br, -CH=C(Cl)-CO-OCH₂-CH=CH₂, -CH=C(Cl)-CO-OCH₂-C≡CH, -CH=C(Cl)-CO-OCH₂-CN, -CH=C(Cl)-CO-O(CH₂)₂-CN, -CH=C(Br)-CO-OCH₂-CF₃, -CH=C(Br)-CO-OCH₂-CCl₃, -CH=C(Br)-CO-OCH₂-oxiranyl, -CH=C(Br)-CO-O(CH₂)₃-Br, -CH=C(Br)-CO-OCH₂-CH=CH₂, -CH=C(Br)-CO-OCH₂-C≡CH, -CH=C(Br)-CO-OCH₂-CN, -CH=C(Br)-CO-O(CH₂)₂-CN, -CH=C(CN)-CO-OCH₂-CF₃, -CH=C(CN)-CO-OCH₂-CCl₃, -CH=C(CN)-CO-OCH₂-oxiranyl -CH=C(CN)-CO-O(CH₂)₃-Br, -CH=C(CN)-CO-OCH₂-CH=CH₂, -CH=C(CN)-CO-OCH₂-C≡CH, -CH=C(CN)-CO-OCH₂-CN, -CH=C(CN)-CO-O(CH₂)₂-CN, -CH=CH-CO-CH₃, -CH=CH-CO-C₂H₅, -CH=CH-CO-n-C₃H₇, -CH=CH-CO-i-C₃H₇, -CH=CH-CO-n-C₄H₉, -CH=CH-CO-tert.-C₄H₉, -CH=CH-CO-CH₂Cl, -CH=CH-CO-CH₂Br, -CH=CH-CO-CHCl₂, -CH=CH-CO-CH₂-OCH₃, -CH=CH-CO-CH(OCH₃)₂, -CH=CH-CO-CH₂-SCH₃, -CH=C(CH₃)-CO-CH₃, -CH=C(CH₃)-CO-C₂H₅, -CH=C(CH₃)-CO-n-C₃H₇, -CH=C(CH₃)-CO-i-C₃H₇, -CH=C(CH₃)-CO-n-C₄H₉, -CH=C(CH₃)-CO-tert.-C₄H₉, -CH=C(CH₃)-CO-CH₂Cl, -CH=C(CH₃)-CO-CH₂Br, -CH=C(CH₃)-CO-CHCl₂, -CH=C(CH₃)-CO-CH₂-OCH₃, -CH=C(CH₃)-CO-CH(OCH₃)₂, -CH=C(CH₃)-CO-CH₂-SCH₃, -CH=C(C₂H₅)-CO-CH₃, -CH=C(C₂H₅)-CO-C₂H₅, -CH=C(C₂H₅)-CO-n-C₃H₇, -CH=C(C₂H₅)-CO-i-C₃H₇, -CH=C(C₂H₅)-CO-n-C₄H₉, -CH=C(C₂H₅)-CO-tert.-C₄H₉, -CH=C(C₂H₅)-CO-CH₂Cl, -CH=C(C₂H₅)-CO-CH₂Br, -CH=C(C₂H₅)-CO-CHCl₂, -CH=C(C₂H₅)-CO-CH₂-OCH₃, -CH=C(C₂H₅)-CO-CH(OCH₃)₂, -CH=C(C₂H₅)-CO-CH₂-SCH₃, -CH=C(Cl)-CO-CH₃, -CH=C(Cl)-CO-C₂H₅, -CH=C(Cl)-CO-n-C₃H₇, -CH=C(Cl)-CO-i-C₃H₇, -CH=C(Cl)-CO-n-C₄H₉, -CH=C(Cl)-CO-tert.-C₄H₉, -CH=C(Cl)-CO-CH₂Cl, -CH=C(Cl)-CO-CH₂Br, -CH=C(Cl)-CO-CHCl₂, -CH=C(Cl)-CO-CH₂-OCH₃, -CH=C(Cl)-CO-CH(OCH₃)₂, -CH=C(Cl)-CO-CH₂-SCH₃, -CH=C(Br)-CO-CH₃, -CH=C(Br)-CO-C₂H₅, -CH=C(Br)-CO-n-C₃H₇, -CH=C(Br)-CO-i-C₃H₇, -CH=C(Br)-CO-n-C₄H₉, -CH=C(Br)-CO-tert.-C₄H₉, -CH=C(Br)-CO-CH₂Cl, -CH=C(Br)-CO-CH₂Br, -CH=C(Br)-CO-CHCl₂, -CH=C(Br)-CO-CH₂-OCH₃, -CH=C(Br)-CO-CH(OCH₃)₂, -CH=C(Br)-CO-CH₂-SCH₃, -CH=C(CN)-CO-CH₃, -CH=C(CN)-CO-C₂H₅, -CH=C(CN)-CO-n-C₃H₇, -CH=C(CN)-CO-i-C₃H₇, -CH=C(CN)-CO-n-C₄H₉, -CH=C(CN)-CO-tert.-C₄H₉, -CH=C(CN)-CO-CH₂Cl, -CH=C(CN)-CO-CH₂Br, -CH=C(CN)-CO-CHCl₂, -CH=C(CN)-CO-CH₂-OCH₃, -CH=C(CN)-CO-CH(OCH₃)₂, -CH=C(CN)-CO-CH₂-SCH₃, -CH=CH-CO-C₆H₅, -CH=CH-CO-(4-Cl-C₆H₄), -CH=C(CH₃)-CO-C₆H₅, -CH=C(CH₃)-CO-(4-Cl-C₆H₄), -CH=C(C₂H₅)-CO-C₆H₅, -CH=C(C₂H₅)-CO-(4-Cl-C₆H₄), -CH=C(Cl)-CO-C₆H₅, -CH=C(Br)-CO-C₆H₅, -CH=C(CN)-CO-C₆H₅, -CH=CH-CO-NH₂, -CH=CH-CO-NHCH₃, -CH=CH-CO-N(CH₃)₂, -CH=CH-CO-NH-C₂H₅, -CH=CH-CO-N(C₂H₅)₂, -CH=CH-CO-NH-n-C₃H₇, -CH=CH-CO-NH-i-C₃H₇, -CH=CH-CO-NH-tert.-C₄H₉, -CH=CH-CO-NH-cyclopropyl, -CH=CH-CO-NH-cyclobutyl, -CH=CH-CO-NH-cyclopentyl, -CH=CH-CO-NH-cyclohexyl, -CH=CH-CO-cycloheptyl, -CH=CH-CO-NH-cyclooctyl, -CH=CH-CO-pyrrolidin-1-yl, -CH=CH-CO-piperidin-1-yl, -CH=CH-CO-morpholin-4-yl, -CH=CH-CO-NH-CH₂CH=CH₂, -CH=CH-CO-NH-CH₂C≡CH, -CH=CH-CO-N(CH₃)-CH₂C≡CH, -CH=CH-CO-NH-(CH₂)₂Cl, -CH=CH-CO-NH-C₆H₅, -CH=C(CH₃)-CO-NH₂, -CH=C(CH₃)-CO-NHCH₃, -CH=C(CH₃)-CO-N(CH₃)₂, -CH=C(CH₃)-CO-NH-C₂H₅, -CH=C(CH₃)-CO-N(C₂H₅)₂, -CH=C(CH₃)-CO-NH-n-C₃H₇, -CH=C(CH₃)-CO-NH-i-C₃H₇, -CH=C(CH₃)-CO-NH-tert.-C₄H₉, -CH=C(CH₃)-CO-NH-cyclopropyl, -CH=C(CH₃)-CO-NH-cyclobutyl, -CH=C(CH₃)-CO-NH-cyclopentyl, -CH=C(CH₃)-CO-NH-cyclohexyl, -CH=C(CH₃)-CO-NH-cycloheptyl, -CH=C(CH₃)-CO-NH-cyclooctyl, -CH=C(CH₃)-CO-pyyrolidin-1-yl, -CH=C(CH₃)-CO-piperidin-1-yl, -CH=C(CH₃)-CO-morpholin-4-yl, -CH=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -CH=C(CH₃)-CO-NH-CH₂C≡CH, -CH=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CH₃)-CO-NH-(CH₂)₂Cl, -CH=C(CH₃)-CO-NH-C₆H₅, -CH=C(C₂H₅)-CO-NH₂, -CH=C(C₂H₅)-CO-NHCH₃, -CH=C(C₂H₅)-CO-N(CH₃)₂, -CH=C(C₂H₅)-CO-NH-C₂H₅, -CH=C(C₂H₅)-CO-N(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-n-C₃H₇, -CH=C(C₂H₅)-CO-NH-i-C₃H₇, -CH=C(C₂H₅)-CO-NH-tert.-C₄H₉, -CH=C(C₂H₅)-CO-NH-cyclopropyl, -CH=C(C₂H₅)-CO-NH-cyclobutyl, -CH=C(C₂H₅)-CO-NH-cyclopentyl, -CH=C(C₂H₅)-CO-NH-cyclohexyl, -CH=C(C₂H₅)-CO-NH-cycloheptyl, -CH=C(C₂H₅)-CO-NH-cyclooctyl, -CH=C(C₂H₅)-CO-pyrrolidin-1-yl, -CH=C(C₂H₅)-CO-piperidin-1-yl, -CH=C(C₂H₅)-CO-morpholin-4-yl, -CH=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -CH=C(C₂H₅)-CO-NH-CH₂C≡CH, -CH=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -CH=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -CH=C(C₂H₅)-CO-NH-C₆H₅, -CH=C(Cl)-CO-NH₂, -CH=C(Cl)-CO-NHCH₃, -CH=C(Cl)-CO-N(CH₃)₂, -CH=C(Cl)-CO-NH-C₂H₅, -CH=C(Cl)-CO-N(C₂H₅)₂, -CH=C(Cl)-CO-NH-n-C₃H₇, -CH=C(Cl)-CO-NH-i-C₃H₇, -CH=C(Cl)-CO-NH-tert.-C₄H₉, -CH=C(Cl)-CO-NH-cyclopropyl, -CH=C(Cl)-CO-NH-cyclobutyl, -CH=C(Cl)-CO-NH-cyclopentyl, -CH=C(Cl)-CO-NH-cyclohexyl, -CH=C(Cl)-CO-NH-cycloheptyl, -CH=C(Cl)-CO-NH-cyclooctyl, -CH=C(Cl)-CO-pyrrolidin-1-yl, -CH=C(Cl)-CO-piperidin-1-yl, -CH=C(Cl)-CO-morpholin-4-yl, -CH=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -CH=C(Cl)-CO-NH-CH₂C≡CH, -CH=C(Cl)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Cl)-CO-NH-(CH₂)₂Cl, -CH=C(Cl)-CO-NH-C₆H₅, -CH=C(Br)-CO-NH₂, -CH=C(Br)-CO-NHCH₃, -CH=C(Br)-CO-N(CH₃)₂, -CH=C(Br)-CO-NH-C₂H₅, -CH=C(Br)-CO-N(C₂H₅)₂, -CH=C(Br)-CO-NH-n-C₃H₇, -CH=C(Br)-CO-NH-i-C₃H₇, -CH=C(Br)-CO-NH-tert.-C₄H₉, -CH=C(Br)-CO-NH-cyclopropyl, -CH=C(Br)-CO-NH-cyclobutyl, -CH=C(Br)-CO-NH-cyclopentyl, -CH=C(Br)-CO-NH-cyclohexyl, -CH=C(Br)-CO-NH-cycloheptyl, -CH=C(Br)-CO-NH-cyclooctyl, -CH=C(Br)-CO-pyrrolidin-1-yl, -CH=C(Br)-CO-piperidin-1-yl, -CH=C(Br)-CO-morpholin-4-yl, -CH=C(Br)-CO-NH-CH₂CH=C(Br)₂, -CH=C(Br)-CO-NH-CH₂C≡CH, -CH=C(Br)-CO-N(CH₃)-CH₂C≡CH, -CH=C(Br)-CO-NH-(CH₂)₂Cl, -CH=C(Br)-CO-NH-C₆H₅, -CH=C(CN)-CO-NH₂, -CH=C(CN)-CO-NHCH₃, -CH=C(CN)-CO-N(CH₃)₂, -CH=C(CN)-CO-NH-C₂H₅, -CH=C(CN)-CO-N(C₂H₅)₂, -CH=C(CN)-CO-NH-n-C₃H₇, -CH=C(CN)-CO-NH-i-C₃H₇, -CH=C(CN)-CO-NH-tert.-C₄H₉, -CH=C(CN)-CO-NH-cyclopropyl, -CH=C(CN)-CO-NH-cyclobutyl, -CH=C(CN)-CO-NH-cyclopentyl, -CH=C(CN)-CO-NH-cyclohexyl, -CH=C(CN)-CO-NH-cycloheptyl, -CH=C(CN)-CO-NH-cyclooctyl, -CH=C(CN)-CO-pyrrolidin-1-yl, -CH=C(CN)-CO-piperidin-1-yl, -CH=C(CN)-CO-morpholin-4-yl, -CH=C(CN)-CO-NH-CH₂CH=C(CN)₂, -CH=C(CN)-CO-NH-CH₂C≡CH, -CH=C(CN)-CO-N(CH₃)-CH₂C≡CH, -CH=C(CN)-CO-NH-(CH₂)₂Cl, -CH=C(CN)-CO-NH-C₆H₅, -CH=CH-CO-SCH₃, -CH=CH-CO-SC₂H₅, -CH=CH-CO-S-n-C₃H₇, -CH=CH-CO-S-i-C₃H₇, -CH=CH-CO-S-n-C₄H₉, -CH=CH-CO-S-tert.-C₄H₉, -CH=C(CH₃)-CO-SCH₃, -CH=C(CH₃)-CO-SC₂H₅, -CH=C(CH₃)-CO-S-n-C₃H₇, -CH=C(CH₃)-CO-S-i-C₃H₇, -CH=C(CH₃)-CO-S-n-C₄H₉, -CH=C(CH₃)-CO-S-tert.-C₄H₉, -CH=C(C₂H₅)-CO-SCH₃, -CH=C(C₂H₅)-CO-SC₂H₅, -CH=C(C₂H₅)-CO-S-n-C₃H₇, -CH=C(C₂H₅)-CO-S-i-C₃H₇, -CH=C(C₂H₅)-CO-S-n-C₄H₉, -CH=C(C₂H₅)-CO-S-tert.-C₄H₉, -CH=C(Cl)-CO-SCH₃, -CH=C(Cl)-CO-SC₂H₅, -CH=C(Cl)-CO-S-n-C₃H₇, -CH=C(Cl)-CO-S-i-C₃H₇, -CH=C(Cl)-CO-S-n-C₄H₉, -CH=C(Cl)-CO-S-tert.-C₄H₉, -CH=C(Br)-CO-SCH₃, -CH=C(Br)-CO-SC₂H₅, -CH=C(Br)-CO-S-n-C₃H₇, -CH=C(Br)-CO-S-i-C₃H₇, -CH=C(Br)-CO-S-n-C₄H₉, -CH=C(Br)-CO-S-tert.-C₄H₉, -CH=C(CN)-CO-SCH₃, -CH=C(CN)-CO-SC₂H₅, -CH=C(CN)-CO-S-n-C₃H₇, -CH=C(CN)-CO-S-i-C₃H₇, -CH=C(CN)-CO-S-n-C₄H₉, -CH=C(CN)-CO-S-tert.-C₄H₉, -CH=C(COCH₃)-CO-OCH₃, -CH=C(COC₂H₅)-CO-OCH₃, -CH=C(CO-n-C₃H₇)-CO-OCH₃, -CH=C(COCH₃)-CO-OC₂H₅, -CH=C(COC₂H₅)-CO-OC₂H₅, -CH=C(CO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COCH₃)-CO-O-n-C₃H₇, -CH=C(COC₂H₅)-CO-O-n-C₃H₇, -CH=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-OCH₃, -CH=C(CF₃)-CO-OC₂H₅, -CH=C(CF₃)-CO-O-n-C₃H₇, -CH=C(CF₃)-CO-O-i-C₃H₇, -CH=C(CF₃)-CO-O-n-C₄H₉, -CH=C(CF₃)-CO-O-tert.-C₄H₉, -CH=C(COOCH₃)₂, -CH=C(COOC₂H₅)₂, -CH=C(COOCH₃)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)-CO-OCH₃, -CH=C(COO-n-C₃H₇)-CO-OC₂H₅, -CH=C(COO-n-C₃H₇)₂, -CH=CH-CH=CH-COOH, -CH=CH-CH=CH-CO-OCH₃, -CH=CH-CH=CH-CO-OC₂H₅, -CH=CH-CH=C(COOCH₃)₂, -CH=CH-CH=C(CN)-CO-OCH₃, -CH=CH-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-OCH₃, -CH=C(CH₃)-CH=C(CN)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -CH=C(CH₃)-CH=C(Cl)-CO-OCH₃, -CH=C(CH₃)-CH=C(Br)-CO-OCH₃, -CH=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -CH=C(CH₃)-CH=C(CN)-CO-NH₂, -CH=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -CH=CH-(CH₂)₂-COOH, -CH=CH-(CH₂)₂-CO-OCH₃, -CH=CH-(CH₂)₂-CO-OC₂H₅, -CH=CH-CH₂-CH(COOCH₃)₂, -CH=CH-CH₂-CH(COOC₂H₅)₂, -CH=CH-CH₂-CH(CN)-CO-OCH₃, -CH=CH-CH₂-CH(CN)-CO-OC₂H₅, -CH=CH-CH₂-CH(CH₃)-CO-OCH₃, -CH=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -CH=CH-(CH₂)₂-CO-NH₂, -CH=CH-(CH₂)₂-CO-NH-CH₃, -CH=CH-CH₂-COOH, -CH=CH-CH₂-CO-OCH₃, -CH=CH-CH₂-CO-OC₂H₅, -CH=C(COOCH₃)-CH₂-CO-OCH₃, -CH=C(COOCH₃)-CH₂-CO-OC₂H₅, -CH=CH-CH₂-CO-NH₂, -CH=CH-CH₂-CO-NH-CH₃, -CH=CH-CH₂-CO-N(CH₃)₂, -CH(OCH₃)₂, -CH(SCH₃)₂, -CH(OC₂H₅)₂, -CH(SC₂H₅)₂, -CH(O-n-C₃H₇)₂, -CH(O-i-C₃H₇)₂, -CH(S-n-C₃H₇)₂, -CH(S-i-C₃H₇)₂, -CH(O-n-C₄H₉)₂, -CH(O-i-C₄H₉)₂, -CH(O-s-C₄H₉)₂, -CH(O-tert.-C₄H₉)₂, -CH(S-n-C₄H₉)₂, -CH(S-i-C₄H₉)₂, -CH(S-s-C₄H₉)₂, -CH(S-tert.-C₄H₉)₂, -CH(OC₅H₁₁)₂, 1,3-Dioxolan-2-yl, 1,3-Dithio­ lan-2-yl, 1,3-Oxathiolan-2-yl, 4-Methyl-1,3-dioxolan-2-yl, 4-Methyl-1,3-dithiolan-2-yl, 4-Methyl-1,3-oxathiolan-2-yl, 5-Methyl-1,3-oxathiolan-2-yl, 4-Ethyl-1,3-dioxolan-2-yl, 4-Ethyl- 1,4-dithiolan-2-yl, 4-Ethyl-1,3-oxathiolan-2-yl, 5-Ethyl-1,3-oxa­ thiolan-2-yl, 4,5-Dimethyl-1,3-dioxolan-2-yl, 4,4-Dimethyl-1,3- dioxolan-2-yl, 4,5-Dimethyl-1,3-dithiolan-2-yl, 5,5-Dimethyl-1,3- dithiolan-2-yl, 4,5-Dimethyl-1,3-oxathiolan-2-yl, 5,5-Dimethyl- 1,3-oxathiolan-2-yl, 4,4-Dimethyl-1,3-oxathiolan-2-yl, 4-Vinyl- 1,3-dioxolan-2-yl, 4-Vinyl-1,3-dithiolan-2-yl, 4-Vinyl-1,3-oxa­ thiolan-2-yl, 5-Vinyl-1,3-oxathiolan-2-yl, 4-Chlormethyl-1,3- dioxolan-2-yl, 4-Chlormethyl-1,3-dithiolan-2-yl, 4-Chlormethyl- 1,3-oxathiolan-2-yl, 5-Chlormethyl-1,3-oxathiolan-2-yl, 4-Hydroxymethyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-1,3-dithio­ lan-2-yl, 4-Hydroxymethyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl- 1,3-oxathiolan-2-yl, 4-Methoxymethyl-1,3-dioxolan-2-yl, 4-Allyl­ oxymethyl-1,3-dioxolan-2-yl, 4-Propargyloxymethyl-1,3-dioxolan- 2-yl, 4-Acetoxymethyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-1,3-dithiolan-2-yl, 4-Propargyl­ oxymethyl-1,3-dithiolan-2-yl, 4-Acetoxymethyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-1,3-oxathiolan-2-yl, 5-Methoxymethyl-1,3-oxathiolan- 2-yl, 4-Allyloxymethyl-1,3-oxathiolan-2-yl, 5-Allyloxy­ methyl-1,3-oxathiolan-2-yl, 4-Propargyloxymethyl-1,3-oxathiolan- 2-yl, 5-Propargyloxymethyl-1,3-oxathiolan-2-yl, 4-Acetoxymethyl- 1,3-oxathiolan-2-yl, 5-Acetoxymethyl-1,3-oxathiolan-2-yl, 4-Methylthiomethyl-1,3-dioxolan-2-yl, 4-Methylthiomethyl-1,3- dithiolan-2-yl, 4-Carboxy-1,3-dioxolan-2-yl, 4-Carboxy-1,3- dithiolan-2-yl, 4-Methoxycarbonyl-1,3-dioxolan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-1,3-di­ thiolan-2-yl, 4-n-Butoxycarbonyl-1,3-dithiolan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Methoxycarbonyl-4-methyl- 1,3-dithiolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl- 4-methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-di­ thiolan-2-yl, 4-Cyanomethyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-1,3- dithiolan-2-yl, 1,3-Dioxan-2-yl, 1,3-Dithian-2-yl, 1,3-Oxathian- 2-yl, 5-Methyl-1,3-dioxan-2-yl, 5-Methyl-1,3-dithian-2-yl, 5-Methyl-1,3-oxathian-2-yl, 5,5-Dimethyl-1,3-dioxan-2-yl, 4,6-Di­ methyl-1,3-dioxan-2-yl, 4,4-Dimethyl-1,3-dioxan-2-yl, 5,5-Di­ methyl-1,3-dithian-2-yl, 4,6-Dimethyl-1,3-dithian-2-yl, 4,4-Di­ methyl-1,3-dithian-2-yl, 5,5-Dimethyl-1,3-oxathian-2-yl, 4,4-Di­ methyl-1,3-oxathian-2-yl, 6,6-Dimethyl-1,3-oxathian-2-yl, 4-Hydroxymethyl-1,3-dioxan-2-yl, 4-Methoxymethyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-1,3-dioxan-2- yl, 4-Hydroxymethyl-1,3-dithian-2-yl, 4-Methoxymethyl-1,3-di­ thian-2-yl, 4-Allyloxymethyl-1,3-dithian-2-yl, 4-Acetoxymethyl- 1,3-dithian-2-yl, 4-Chlormethyl-1,3-dioxan-2-yl, 4-Chlormethyl- 1,3-dithian-2-yl, 1,3-Dioxepan-2-yl, 1,3-Dithiepan-2-yl, 1,3-Di­ oxep-5-en-2-yl, 4-Methoxycarbonyl-1,3-dioxan-2-yl, 4-Ethoxy­ carbonyl-1,3-dioxan-2-yl, 4-n-Butoxycarbonyl-1,3-dioxan-2-yl, 4-Methoxycarbonyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-1,3-dithian- 2-yl, 4-n-Butoxycarbonyl-1,3-dithian-2-yl, 4-Methoxycarbonyl-4- methyl-1,3-dioxan-2-yl, 4-Ethoxycarbonyl-4-methyl-1,3-dioxan-2- yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dioxan-2-yl, 4-Methoxy­ carbonyl-4-methyl-1,3-dithian-2-yl, 4-Ethoxycarbonyl-4-methyl- 1,3-dithian-2-yl, 4-n-Butoxycarbonyl-4-methyl-1,3-dithian-2-yl, -C(CH₃)(OCH₃)₂, -C(CH₃)(SCH₃)₂, -C(CH₃)(OC₂H₅)₂, -C(CH₃)(SC₂H₅)₂, -C(CH₃)(O-n-C₃H₇)₂, -C(CH₃)(O-i-C₃H₇)₂, -C(CH₃)(S-n-C₃H₇)₂, -C(CH₃)(S-i-C₃H₇)₂, -C(CH₃)(O-n-C₄H₉)₂, -C(CH₃)(O-i-C₄H₉)₂, -C(CH₃)(O-s-C₄H₉)₂, -C(CH₃)(O-tert.-C₄H₉)₂, -C(CH₃)(S-n-C₄H₉)₂, -C(CH₃)(S-i-C₄H₉)₂, -C(CH₃)(S-s-C₄H₉)₂, -C(CH₃)(S-tert.-C₄H₉)₂, -C(CH₃)(O-n-C₅H₁₁)′′, 2-Methyl-1,3-dioxolan-2-yl, 2-Methyl-1,3-di- thiolan-2-yl, 2-Methyl-1,3-oxathiolan-2-yl, 2,4-Dimethyl-1,3- dioxolan-2-yl, 2,4-Dimethyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-1,3- oxathiolan-2-yl, 2,5-Dimethyl-1,3-oxathiolan-2-yl, 4-Ethyl-2- methyl-1,3-dioxolan-2-yl, 4-Ethyl-2-methyl-1,3-dithiolan-2-yl, 4-Ethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Ethyl-2-methyl-1,3- oxathiolan-2-yl, 2,4,5-Trimethyl-1,3-dioxolan-2-yl, 2,4,4-Tri­ methyl-1,3-dioxolan-2-yl, 2,4,5-Trimethyl-1,3-dithiolan-2-yl, 2,4,4-Trimethyl-1,3-dithiolan-2-yl, 2,4,5-Trimethyl-1,3-oxathio­ lan-2-yl, 2,4,4-Trimethyl-1,3-oxathiolan-2-yl, 2-Methyl-4-vinyl- 1,3-dioxolan-2-yl, 2-Methyl-4-vinyl-1,3-dithiolan-2-yl, 2-Methyl- 4-vinyl-1,3-oxathiolan-2-yl, 2-Methyl-5-vinyl-1,3-oxathiolan-2- yl, 4-Chlormethyl-2-methyl-1,3-dioxolan-2-yl, 4-Chlormethyl-2- methyl-1,3-dithiolan-2-yl, 4-Chlormethyl-2-methyl-1,3-oxathio- lan-2-yl, 5-Chlormethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Hydroxy­ methyl-2-methyl-1,3-dioxolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Hydroxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Methoxymethyl-2- methyl-1,3-dioxolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dioxolan- 2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dioxolan-2-yl, 4-Acetoxy- 2-methyl-1,3-dioxolan-2-yl, 4-Methoxymethyl-2-methyl-1,3- dithiolan-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3-dithiolan-2-yl, 4-Acetoxy-2- methyl-1,3-dithiolan-2-yl, 4-Methoxymethyl-2-methyl-1,3-oxathio­ lan-2-yl, 5-Methoxymethyl-2-methyl-1,3-oxathiolan-2-yl, 4-Allyl­ oxymethyl-2-methyl-1,3-oxathiolan-2-yl, 5-Allyloxymethyl-2- methyl-1,3-oxathiolan-2-yl, 2-Methyl-4-propargyloxymethyl-1,3- oxathiolan-2-yl, 2-Methyl-5-propargyloxymethyl-1,3-oxathiolan-2- yl, 4-Acetoxy-2-methyl-1,3-oxathiolan-2-yl, 5-Acetoxy-2-methyl- 1,3-oxathiolan-2-yl, 2-Methyl-4-methylthiomethyl-1,3-dioxolan-2- yl, 2-Methyl-4-methylthiomethyl-1,3-dithiolan-2-yl, 4-Carboxy-2- methyl-1,3-dioxolan-2-yl, 4-Carboxy-2-methyl-1,3-dithiolan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dioxolan-2-yl, 4-Ethoxycarbonyl-2- methyl-1,3-dioxolan-2-yl, 4-n-Butoxycarbonyl-2-methyl-1,3-dioxo­ lan-2-yl, 4-Methoxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-Eth­ oxycarbonyl-2-methyl-1,3-dithiolan-2-yl, 4-n-Butoxycarbonyl-2- methyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-di­ oxolan-2-yl, 2,4-Dimethyl-4-methoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-ethoxycarbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4- ethoxycarbonyl-1,3-dithiolan-2-yl, 2,4-Dimethyl-4-n-butoxy­ carbonyl-1,3-dioxolan-2-yl, 2,4-Dimethyl-4-n-butoxycarbonyl-1,3- dithiolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dioxolan-2-yl, 4-Cyanomethyl-2-methyl-1,3-dithiolan-2-yl, 2-Methyl-1,3-dioxan-2- yl, 2-Methyl-1,3-dithian-2-yl, 2-Methyl-1,3-oxathian-2-yl, 2,5- Dimethyl-1,3-dioxan-2-yl, 2,5-Dimethyl-1,3-dithian-2-yl, 2,5-Di­ methyl-1,3-oxathian-2-yl, 2,5,5-Trimethyl-1,3-dioxan-2-yl, 2,4,6- Trimethyl-1,3-dioxan-2-yl, 2,2,4-Trimethyl-1,3-dioxan-2-yl, 2,5,5-Trimethyl-1,3-dithian-2-yl, 2,4,6-Trimethyl-1,3-dithian-2- yl, 2,4,4-Trimethyl-1,3-dithian-2-yl, 2,5,5-Trimethyl-1,3-oxa­ thian-2-yl, 2,4,4-Trimethyl-1,3-oxathian-2-yl, 2,6,6-Trimethyl- 1,3-oxathian-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Methoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Allyloxymethyl-2- methyl-1,3-dioxan-2-yl, 4-Acetoxymethyl-2-methyl-1,3-dioxan-2-yl, 4-Hydroxymethyl-2-methyl-1,3-dithian-2-yl, 4-Methoxymethyl-2- methyl-1,3-dithian-2-yl, 4-Allyloxymethyl-2-methyl-1,3-dithian-2- yl, 4-Acetoxymethyl-2-methyl-1,3-dithian-2-yl, 4-Chlormethyl-2- methyl-1,3-dioxan-2-yl, 4-Chlormethyl-2-methyl-1,3-dithian-2-yl, -C(CH₃)=NH, -C(CH₃)=N-CH₃, -C(CH₃)=N-C₂H₅, -C(CH₃)=N-n-C₃H₇, -C(CH₃)=N-i-C₃H₇, -C(CH₃)=N-n-C₄H₉, -C(CH₃)=N-CH₂CH=CH₂, -C(CH₃)=N-CH₂CH=CH₂-CH₃, -C(CH₃)=N-CH₂C≡CH, -C(CH₃)=N-CH₂C≡C-CH₃, -C(CH₃)=N-cyclopropyl, -C(CH₃)=N-cyclobutyl, -C(CH₃)=N-cyclo­ pentyl, -C(CH₃)=N-cyclohexyl, -C(CH₃)=N-cycloheptyl, -C(CH₃)=N-CH₂-CH₂Cl, -C(CH₃)=N-CH₂Cl, -C(CH₃)=N-C₆H₅, -C(CH₃)=N-(2-F-C₆H₄), -C(CH₃)=N-(3-F-C₆H₄), -C(CH₃)=N-(4-F-C₆H₄), -C(CH₃)=N-(2-Cl-C₆H₄), -C(CH₃)=N-(3-Cl-C₆H₄), -C(CH₃)=N-(4-Cl-C₆H₄), -C(CH₃)=N-(2-CH₃-C₆H₄), -C(CH₃)=N-(3-CH₃-C₆H₄), -C(CH₃)=N-(4-CH₃-C₆H₄), -C(CH₃)=N-(2-CF₃-C₆H₄), -C(CH₃)=N-(3-CF₃-C₆H₄), -C(CH₃)=N-(4-CF₃-C₆H₄), -C(CH₃)=N-(2-OCH₃-C₆H₄), -C(CH₃)=N-(3-OCH₃-C₆H₄), -C(CH₃)=N-(4-OCH₃-C₆H₄), -C(CH₃)=N-(4-NO₂-C₆H₄), -C(CH₃)=N-(4-CN-C₆H₄), -C(CH₃)=N-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-(2,4-(CH₃)₂-C₆H₃), -C(CH₃)=N-CH₂-OCH₃, -C(CH₃)=N-CH₂-OC₂H₅, -C(CH₃)=N-CH₂CH₂-OCH₃, -C(CH₃)=N-CH₂CH₂-OC₂H₅, -C(CH₃)=N-OH, -C(CH₃)=N-OCH₃, -C(CH₃)=N-OC₂H₅, -C(CH₃)=N-O-n-C₃H₇, -C(CH₃)=N-O-i-C₃H₇, -C(CH₃)=N-O-n-C₄H₉, -C(CH₃)=N-O-i-C₄H₉, -C(CH₃)=N-O-s-C₄H₉, -C(CH₃)=N-O-tert.-C₄H₉, -C(CH₃)=N-OCH₂-CH=CH₂, -C(CH₃)=N-OCH(CH₃)-CH=CH₂, -C(CH₃)=N-OCH₂-C≡CH, -C(CH₃)=N-CH(CH₃)-C≡CH, -C(CH₃)=N-OCH₂-CH=C-CH₃, -C(CH₃)=N-OCH₂CH₂-Cl, -C(CH₃)=N-OCH₂CH₂-F, -C(CH₃)=N-OCH₂-CF₃, -C(CH₃)=N-OCH₂-CH=CHCl, -C(CH₃)=N-OCH₂-C(Cl)=CH₂, -C(CH₃)=N-OCH₂-C(Br)=CH₂, -C(CH₃)=N-OCH₂-CH=C(Cl)-CH₃, -C(CH₃)=N-O-CO-CH₃, -C(CH₃)=N-O-CO-C₂H₅, -C(CH₃)=N-OCH₂-CN, -C(CH₃)=N-OCH₂-CH=CH-CH₂-OCH₃, -C(CH₃)=N-OCH₂-CH=CH-CH₂-O-tert.-C₄H₉, -C(CH₃)=N-O-(CH₂)₃-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-C₆H₅, -C(CH₃)=N-O-(CH₂)₄-(4-Cl-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-CH₃-C₆H₄), -C(CH₃)=N-O-(CH₂)₄-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-C₆H₅, -C(CH₃)=N-OCH₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-(3-CH₃O-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-F-C₆H₄), -C(CH₃)=N-O-(CH₂)₂-CH=CH-(4-Cl-C₆H₄), -C(CH₃)=N-OCH₂-CH=CH-CH₂-(4-CH₃O-C₆H₄), -C(CH₃)=N-OCH₂-CH=C(CH₃)-C₆H₅, -C(CH₃)=N-O-(CH₂)₂-CH=CH-(3,4-Cl₂-C₆H₃), -C(CH₃)=N-O-(CH₂)₃-C≡-(4-F-C₆H₄), -C(CH₃)=N-OCH₂-OCH₃, -C(CH₃)=N-OCH₂CH₂-OCH₃, -C(CH₃)=N-OCH₂-OC₂H₅, -C(CH₃)=N-OCH(CH₃)-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-OCH₃, -C(CH₃)=N-OCH(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=N-NH₂, -C(CH₃)=N-NH-CH₃, -C(CH₃)=N-NH-C₂H₅, -C(CH₃)=N-NH-n-C₃H₇, -C(CH₃)=N-NH-i-C₃H₇, -C(CH₃)=N-NH-n-C₄H₉, -C(CH₃)=N-NH-i-C₄H₉, -C(CH₃)=N-NH-s-C₄H₉, -C(CH₃)=N-NH-tert.-C₄H₉, -C(CH₃)=N-NH-cyclopropyl, -C(CH₃)=N-NH- cyclobutyl, -C(CH₃)=N-NH-cyclopentyl, -C(CH₃)=N-NH-cyclohexyl, -C(CH₃)=N-NH-cycloheptyl, -C(CH₃)=N-N(CH₃)₂, -C(CH₃)=N-N(C₂H₅)₂, -C(CH₃)=N-N(n-C₃H₇)₂, -C(CH₃)=N-N(i-C₃H₇)₂, -C(CH₃)=N-NH-CH₂-C=CH, -C(CH₃)=N-NH-CH₂-C≡CH, -C(CH₃)=N-N(CH₃)-CH₂-C≡CH, -C(CH₃)=N-NH-CH₂CF₃, -C(CH₃)=N-NH-CO-CH₃, -C(CH₃)=N-NH-CO-C₂H₅, -C(CH₃)=N-NH-CO-OCH₃, -C(CH₃)=N-NH-CO-OC₂H₅, -C(CH₃)=N-NH-CO-O-tert.-C₄H₉, -C(CH₃)=N- pyrrolidin-1-yl, -C(CH₃)=N-piperidin-1-yl, -C(CH₃)=N-morpholin- 4-yl, -C(CH₃)=N-NH-C₆H₅, -C(CH₃)=N-NH-(4-Cl-C₆H₄), -C(CH₃)=N-NH-(4-NO₂-C₆H₄), -C(CH₃)=N-NH-(4-F-C₆H₄), -C(CH₃)=N-NH-(4-CH₃O-C₆H₄), -C(CH₃)=N-NH-(2,4-Cl₂-C₆H₃), -C(CH₃)=N-NH-(2,4-(NO₂)₂-C₆H₃), -C(CH₃)=N-NH-CO-NH₂, -C(CH₃)=N-NH-CO-NHCH₃, -C(CH₃)=N-NH-CO-NHC₂H₅, -C(CH₃)=N-NH-CO-N(CH₃)₂, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=CH-CO-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -(CH₃)=CH-CO-O-n-C₄H₉, -C(CH₃)=CH-CO-O-tert.-C₄H₉, -C(CH₃)=CH-CO-O-cyclopropyl, -C(CH₃)=CH-CO-O-cyclobutyl, -C(CH₃)=CH-CO-O-cyclopentyl, -C(CH₃)=CH-CO-O-cyclohexyl, -C(CH₃)=CH-CO-O-cycloheptyl, -C(CH₃)=C(CH₃)-COOH, -C(CH₃)=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-O-cyclopropyl, -C(CH₃)=C(CH₃)-CO-O-cyclobutyl, -C(CH₃)=C(CH₃)-CO-O-cyclopentyl, -C(CH₃)=C(CH₃)-CO-O-cyclohexyl, -C(CH₃)=C(CH₃)-CO-O-cycloheptyl, -C(CH₃)=C(C₂H₅)-COOH, -C(CH₃)=C(C₂H₅)-CO-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-O-cyclo­ propyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-O- cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-O-cyclohexyl, -C(CH₃)=C(C₂H₅)-CO-O-cycloheptyl, -C(CH₃)=CH-COOH, -C(CH₃)=CH-CO-OCH₃, -C(CH₃)=CH-CO-OC₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-O-n-C₄H₉, -C(CH₃)=C(Cl)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-O-cyclopropyl, -C(CH₃)=C(Cl)-CO-O-cyclobutyl, -C(CH₃)=C(Cl)-CO-O-cyclopentyl, -C(CH₃)=C(Cl)-CO-O-cyclohexyl, -C(CH₃)=C(Cl)-CO-O-cycloheptyl, -C(CH₃)=C(Br)-COOH, -C(CH₃)=C(Br)-CO-OCH₃, -C(CH₃)=C(Br)-CO-OC₂H₅, -C(CH₃)=C(Br)-CO-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-O-n-C₄H₉, -C(CH₃)=C(Br)-CO-O-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-O-cyclopropyl, -C(CH₃)=C(Br)-CO-O-cyclobutyl, -C(CH₃)=C(Br)-CO-O-cyclopentyl, -C(CH₃)=C(Br)-CO-O-cyclohexyl, -C(CH₃)=C(Br)-CO-O-cycloheptyl, -C(CH₃)=C(CN)-COOH, -C(CH₃)=C(CN)-CO-OCH₃, -C(CH₃)=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CN)-CO-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-O-n-C₄H₉, -C(CH₃)=C(CN)-CO-O-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-O-cyclopropyl, -C(CH₃)=C(CN)-CO-O-cyclobutyl, -C(CH₃)=C(CN)-CO-O-cyclopentyl, -C(CH₃)=C(CN)-CO-O-cyclohexyl, -C(CH₃)=C(CN)-CO-O-cycloheptyl, -C(CH₃)=CH-CO-OCH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-OCH(CH₃)-OCH₃, -C(CH₃)=CH-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=CH-CO-OCH₂CH₂-OCH₃, -C(CH₃)=CH-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-OCH₃, - C(CH₃)=C(CH₃)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(C₂H₅)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-O-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=(C₂H₅)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Cl)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Cl)-CO-O-i-C₃H₇, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Cl)-CO-OCH(CH₃)-OC₂H₅, -(CH₃)=C(Cl)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(Br)-CO-O-i-C₃H₇, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OCH₃, -C(CH₃)=C(Br)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(Br)-CO-OCH₂-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂-O-n-C₃H₇, -C(CH₃)=C(CN)-CO-O-i-C₃H₇, -C(CH₃)=C(CN)-CO-OCH(CH₃)OCH₃, -C(CH₃)=C(CN)-CO-OCH(CH₃)-OC₂H₅, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OCH₃, -C(CH₃)=C(CN)-CO-OCH₂CH₂-OC₂H₅, -C(CH₃)=CH-CO-OCH₂-CF₃, -C(CH₃)=CH-CO-OCH₂-CCl₃, -C(CH₃)=CH-CO-OCH₂-oxiranyl, -C(CH₃)=CH-CO-(CH₂)₃-Br,-C(CH₃)=CH-CO-OCH₂-CH=CH₂, -C(CH₃)=CH-CO-OCH₂-C≡CH, -C(CH₃)=CH-CO-OCH₂-CN, -C(CH₃)=CH-CO-OCH₂CH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂-CF₃, -C(CH₃)=C(CH₃)-CO-OCH₂-CCl₃, -C(CH₃)=C(CH₃)-CO-OCH₂-oxiranyl, -C(CH₃)=C(CH₃)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CH₃)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CH₃)-CO-OCH₂-C≡CH, -C(CH₃)=C(CH₃)-CO-OCH₂-CN, -C(CH₃)=C(CH₃)-CO-OCH₂CH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CF₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CCl₃, -C(CH₃)=C(C₂H₅)-CO-OCH₂-oxiranyl, -C(CH₃)=C(C₂H₅)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(C₂H₅)CO-OCH₂-C≡CH, -C(CH₃)=C(C₂H₅)-CO-OCH₂-CN, -C(CH₃)=C(C₂H₅)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂-CF₃, -C(CH₃)=C(Cl)-CO-OCH₂-CCl₃, -C(CH₃)=C(Cl)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Cl)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Cl)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Cl)-CO-OCH₂-C≡CH, -C(CH₃)=C(Cl)-CO-OCH₂-CN, -C(CH₃)=C(Cl)-CO-OCH₂CH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂-CF₃, -C(CH₃)=C(Br)-CO-OCH₂-CCl₃, -C(CH₃)=C(Br)-CO-OCH₂-oxiranyl, -C(CH₃)=C(Br)-CO-O-(CH₂)₃-Br, -C(CH₃)=C(Br)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(Br)-CO-OCH₂-C≡CH, -C(CH₃)=C(Br)-CO-OCH₂-CN, -C(CH₃)=C(Br)-CO-OCH₂CH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂-CF₃, -C(CH₃)=C(CN)-CO-OCH₂-CCl₃, -C(CH₃)=C(CN)-OCH₂-oxiranyl, -C(CH₃)=C(CN)-CO-O(CH₂)₃-Br, -C(CH₃)=C(CN)-CO-OCH₂-CH=CH₂, -C(CH₃)=C(CN)-CO-OCH₂-C≡CH, -C(CH₃)=C(CN)-CO-OCH₂-CN, -C(CH₃)=C(CN)-CO-OCH₂CH₂-CN, -C(CH₃)=CH-CO-CH₃, -C(CH₃)=CH-CO-C₂H₅, -C(CH₃)=CH-CO-n-C₃H₇, -C(CH₃)=CH-CO-i-C₃H₇, -C(CH₃)=CH-CO-n-C₄H₉, -C(CH₃)=CH-CO-tert.-C₄H₉, -C(CH₃)=CH-CO-CH₂Cl, -C(CH₃)=CH-CO-CH₂Br, -C(CH₃)=CH-CO-CHCl₂, -C(CH₃)=CH-CO-CH₂-OCH₃, -C(CH₃)=CH-CO-CH(OCH₃)₂, -C(CH₃)=CH-CO-CH₂-SCH₃, -C(CH₃)=C(CH₃)-CO-CH₃, -C(CH₃)=C(CH₃)-CO-C₂H₅, -C(CH₃)=C(CH₃)-CO-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-CH₂Cl, -C(CH₃)=C(CH₃)-CO-CH₂Br, -C(CH₃)=C(CH₃)-CO-CHCl₂, -C(CH₃)=C(CH₃)-CO-CH₂-OCH₃, -C(CH₃)=C(CH₃)-CO-CH(OCH₃)₂, -C(CH₃)=C(CH₃)-CO-CH₂-SCH₃, -C(CH₃)=C(C₂H₅)-CO-CH₃, -C(CH₃)=C(C₂H₅)-CO-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-CH₂Cl, -C(CH₃)=C(C₂H₅)-CO-CH₂Br, -C(CH₃)=C(C₂H₅)-CO-CHCl₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-OCH₃, -C(CH₃)=C(C₂H₅)-CO-CH(OCH₃)₂, -C(CH₃)=C(C₂H₅)-CO-CH₂-SCH₃, -C(CH₃)=C(Cl)-CO-CH₃, -C(CH₃)=C(Cl)-CO-C₂H₅, -C(CH₃)=C(Cl)-CO-n-C₃H₇, -C(CH₃)=C(Cl)-CO-i-C₃H₇, -C(CH₃)=C(Cl)-CO-n-C₄H₉, -C(CH₃)=C(Cl)-CO-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-CH₂Cl, -C(CH₃)=C(Cl)-CO-CHCl₂, -C(CH₃)=C(Cl)-CO-CH₂-OCH₃, -C(CH₃)=C(Cl)-CO-CH(OCH₃)₂, -C(CH₃)=C(Cl)-CO-CH₂-SCH₃, -C(CH₃)=C(Br)-CO-CH₃, -C(CH₃)=C(Br)-CO-C₂H₅, -C(CH₃)=C(Br)-CO-n-C₃H₇, -C(CH₃)=C(Br)-CO-i-C₃H₇, -C(CH₃)=C(Br)-CO-n-C₄H₉, -C(CH₃)=C(Br)-CO-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-CH₂Cl, -C(CH₃)=C(Br)-CO-CH₂Br, -C(CH₃)=C(Br)-CO-CH₂-OCH₃, -C(CH₃)=C(Br)-CO-CH(OCH₃)₂, -C(CH₃)=C(Br)-CO-CH₂-SCH₃, -C(CH₃)=C(CN)-CO-CH₃, -C(CH₃)=C(CN)-CO-C₂H₅, -C(CH₃)=C(CN)-CO-n-C₃H₇, -C(CH₃)=C(CN)-CO-i-C₃H₇, -C(CH₃)=C(CN)-CO-n-C₄H₉, -C(CH₃)=C(CN)-CO-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-CH₂Cl, -C(CH₃)=C(CN)-CO-CH₂Br, -C(CH₃)=C(CN)-CO-CHCl₂, -C(CH₃)=C(CN)-CO-CH₂-OCH₃, -C(CH₃)=C(CN)-CO-CH(OCH₃)₂, -C(CH₃)=C(CN)-CO-CH₂-SCH₃, -C(CH₃)=CH-CO-C₆H₅, -C(CH₃)=CH-CO-(4-Cl-C₆H₄), -C(CH₃)=C(CH₃)-CO-C₆H₅, -C(CH₃)=C(CH₃)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(C₂H₅)-CO-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-(4-Cl-C₆H₄), -C(CH₃)=C(Cl)-CO-C₆H₅, -C(CH₃)=C(Br)-CO-C₆H₅, -C(CH₃)=C(CN)-CO-C₆H₅, -C(CH₃)=CH-CO-NH₂, -C(CH₃)=CH-CO-NHCH₃, -C(CH₃)=CH-CO-N(CH₃)₂, -C(CH₃)=CH-CO-NH-C₂H₅, -C(CH₃)=CH-CO-N(C₂H₅)₂, -C(CH₃)=CH-CO-NH-n-C₃H₇, -C(CH₃)=CH-CO-NH-i-C₃H₇, -C(CH₃)=CH-CO-NH-tert.-C₄H₉, -C(CH₃)=CH-CO-NH-cyclopropyl, -C(CH₃)=CH-CO-NH-cyclobutyl, -C(CH₃)=CH-CO-NH-cyclopentyl, -C(CH₃)=CH-CO-NH-cyclohexyl, -C(CH₃)=CH-CO-NH-cycloheptyl, -C(CH₃)=CH-CO-NH-cyclooctyl, -C(CH₃)=CH-CO-pyrrolidin-1-yl, -C(CH₃)=CH-CO-piperidin-1-yl, -C(CH₃)=CH-CO-morpholin-4-yl, -C(CH₃)=CH-CO-NH-CH₂CH=CH₂, -C(CH₃)=CH-CO-NH-CH₂C≡CH, -C(CH₃)=CH-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=CH-CO-NH-(CH₂)₂Cl, -C(CH₃)=CH-CO-NH-C₆H₅, -C(CH₃)=C(CH₃)-CO-NH₂, -C(CH₃)=C(CH₃)-CO-NHCH₃, -C(CH₃)=C(CH₃)-CO-N(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-C₂H₅, -C(CH₃)=C(CH₃)-CO-N(C₂H₅)₂, -C(CH₃)=C(CH₃)-CO-NH-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-NH- cyclopropyl, -C(CH₃)=C(CH₃)-CO-NH-cyclobutyl, -C(CH₃)=C(CH₃)-CO-NH-cyclopentyl, -C(CH₃)=C(CH₃)-CO-NH- cyclohexyl, -C(CH₃)=C(CH₃)-CO-NH-cycloheptyl, -C(CH₃)=C(CH₃)-CO-NH-cyclooctyl, -C(CH₃)=C(CH₃)-CO- pyrrolidin-1-yl, -C(CH₃)=C(CH₃)-CO-piperidin-1-yl, -C(CH₃)=C(CH₃)-CO-morpholin-4-yl, -C(CH₃)=C(CH₃)-CO-NH-CH₂CH=C(CH₃)₂, -C(CH₃)=C(CH₃)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CH₃)-CO-NH-C₆H₅, -C(CH₃)=C(C₂H₅)-CO-NH₂, -C(CH₃)=C(C₂H₅)-CO-NHCH₃, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)₂, -C(CH₃)=C(C₂H₅)-CO-NH-C₂H₅, -C(CH₃)=C(C₂H₅)-CO-N(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-NH- cyclopropyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclobutyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclopentyl, -C(CH₃)=C(C₂H₅)-CO-NH-cyclo­ hexyl, -C(CH₃)=C(C₂H₅)-CO-NH-cycloheptyl, -C(CH₃)=C(C₂H₅)-CO-NH- cyclooctyl, -C(CH₃)=C(C₂H₅)-CO-pyrrolidin-1-yl, -C(CH₃)=C(C₂H₅)-CO-piperidin-1-yl, -C(CH₃)=C(C₂H₅)-CO- morpholin-4-yl, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂CH=C(C₂H₅)₂, -C(CH₃)=C(C₂H₅)-CO-NH-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(C₂H₅)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(C₂H₅)-CO-NH-C₆H₅, -C(CH₃)=C(Cl)-CO-NH₂, -C(CH₃)=C(CH₃)=C(Cl)-CO-NHCH₃, -C(CH₃)=C(Cl)-CO-N(CH₃)₂, -C(CH₃)=C(Cl)-CO-NH-C₂H₅, -C(CH₃)=C(Cl)-CO-N(C₂H₅)₂, -C(CH₃)=C(Cl)-CO-NH-n-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-i-C₃H₇, -C(CH₃)=C(Cl)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-NH-cyclopropyl, -C(CH₃)=C(Cl)-CO-NH-cyclobutyl, -C(CH₃)=C(Cl)-CO-NH-cyclopentyl, -C(CH₃)=C(Cl)-CO-NH-cyclohexyl, -C(CH₃)=C(Cl)-CO-NH-cycloheptyl, -C(CH₃)=C(Cl)-CO-NH-cyclooctyl, -C(CH₃)=C(Cl)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Cl)-CO-piperidin-1- yl, -C(CH₃)=C(Cl)-CO-morpholin-4-yl, -C(CH₃)=C(Cl)-CO-NH-CH₂CH=C(Cl)₂, -C(CH₃)=C(Cl)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Cl)-CO-N(CH₃)-CH₂≡CH, -C(CH₃)=C(Cl)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Cl)-CO-NH-C₆H₅, -C(CH₃)=C(Br)-CO-NH₂, -C(CH₃)=C(Br)-CO-NHCH₃, -C(CH₃)=C(Br)-CO-N(CH₃)₂, -C(CH₃)=C(Br)-CO-NH-C₂H₅, -C(CH₃)=C(Br)-CO-N(C₂H₅)₂, -C(CH₃)=C(Br)-CO-NH-n-C₃H₇, -C(CH₃)=C(Br)-CO-NH-i-C₃H₇, -C(CH₃)=C(Br)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-NH-cyclopropyl, -C(CH₃)=C(Br)-CO-NH-cyclobutyl, -C(CH₃)=C(Br)-CO-NH-cyclopentyl, -C(CH₃)=C(Br)-CO-NH-cyclohexyl, -C(CH₃)=C(Br)-CO-NH-cycloheptyl, -C(CH₃)=C(Br)-CO-NH-cyclooctyl, -C(CH₃)=C(Br)-CO-pyrrolidin-1-yl, -C(CH₃)=C(Br)-CO-piperidin-1-yl, -C(CH₃)=C(Br)-CO-morpholin-4-yl, -C(CH₃)=C(Br)-CO-NH-CH₂CH=C(CH₃)=C(Br)-CO-NH-CH₂C≡CH, -C(CH₃)=C(Br)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(Br)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(Br)-CO-NH-C₆H₅, -C(CH₃)=C(CN)-CO-NH₂, -C(CH₃)=C(CN)-CO-NHCH₃, -C(CH₃)=C(CN)-CO-N(CH₃)₂, -C(CH₃)=C(CN)-CO-NH-C₂H₅, -C(CH₃)=C(CN)-CO-N(C₂H₅)₂, -C(CH₃)=C(CN)-CO-NH-n-C₃H₇, -C(CH₃)=C(CN)-CO-NH-i-C₃H₇, -C(CH₃)=C(CN)-CO-NH-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-NH-cyclopropyl, -C(CH₃)=C(CN)-CO-NH-cyclobutyl, -C(CH₃)=C(CN)-CO-NH-cyclopentyl, -C(CH₃)=C(CN)-CO-NH-cyclohexyl, -C(CH₃)=C(CN)-CO-NH-cycloheptyl, -C(CH₃)=C(CN)-CO-NH-cyclooctyl, -C(CH₃)=C(CN)-CO-pyrrolidin-1-yl, -C(CH₃)=C(CN)-CO-piperidin-1-yl, -C(CH₃)=C(CN)-CO-morpholin-4-yl, -C(CH₃)=C(CN)-CO-NH-CH₂CH=C(CN)₂, -C(CH₃)=C(CN)-CO-NH-CH₂C≡CH, -C(CH₃)=C(CN)-CO-N(CH₃)-CH₂C≡CH, -C(CH₃)=C(CH₃)=(CN)-CO-NH-(CH₂)₂Cl, -C(CH₃)=C(CN)-CO-NH-C₆H₅, -C(CH₃)=CH-CO-SCH₃, -C(CH₃)=CH-CO-SC₂H₅, -C(CH₃)=CH-CO-S-n-C₃H₇, -C(CH₃)=CH-CO-S-i-C₃H₇, -C(CH₃)=CH-CO-S-n-C₄H₉, -C(CH₃)=CH-CO-S-tert.-C₄H₉, -C(CH₃)=C(CH₃)-CO-SCH₃, -C(CH₃)=C(CH₃)-CO-SC₂H₅, -C(CH₃)=C(CH₃)CO-S-n-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-i-C₃H₇, -C(CH₃)=C(CH₃)-CO-S-n-C₄H₉, -C(CH₃)=C(CH₃)-CO-S-tert.-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-SCH₃, -C(CH₃)=C(C₂H₅)-CO-SC₂H₅, -C(CH₃)=C(C₂H₅)-CO-S-n-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-i-C₃H₇, -C(CH₃)=C(C₂H₅)-CO-S-n-C₄H₉, -C(CH₃)=C(C₂H₅)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Cl)-CO-SCH₃, -C(CH₃)=C(Cl)-CO-SC₂H₅, -C(CH₃)=C(Cl)-CO-S-n-C₃H₇, -C(CH₃)=C(Cl)-CO-S-i-C₃H₇, -C(CH₃)=C(Cl)-CO-S-n-C₄H₉, -C(CH₃)=C(Cl)-CO-S-tert.-C₄H₉, -C(CH₃)=C(Br)-CO-SCH₃, -C(CH₃)=C(Br)-CO-SC₂H₅, -C(CH₃)=C(Br)-CO-S-n-C₃H₇, -C(CH₃)=C(Br)-CO-S-i-C₃H₇, -C(CH₃)=C(Br)-CO-S-n-C₄H₉, -C(CH₃)=C(Br)-CO-S-tert.-C₄H₉, -C(CH₃)=C(CN)-CO-SCH₃, -C(CH₃)=C(CN)-CO-SC₂H₅, -C(CH₃)=C(CN)-CO-S-n-C₃H₇, -C(CH₃)=C(CN)-CO-S-i-C₃H₇, -C(CH₃)=C(CN)-CO-S-n-C₄H₉, -C(CH₃)=C(CN)-CO-S-tert.-C₄H₉, -C(CH₃)=C(COCH₃)-CO-OCH₃, -C(CH₃)=C(COC₂H₅)-CO-OCH₃, -C(CH₃)=C(CO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COCH₃)-CO-OC₂H₅, -C(CH₃)=C(COC₂H₅)-CO-OC₂H₅, -C(CH₃)=C(CO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COCH₃)-CO-O-n-C₃H₇, -C(CH₃)=C(COC₂H₅)-CO-O-n-C₃H₇, -C(CH₃)=C(CO-n-C₃H₇)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-OCH₃, -C(CH₃)=C(CF₃)-CO-OC₂H₅, -C(CH₃)=C(CF₃)-CO-O-n-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-i-C₃H₇, -C(CH₃)=C(CF₃)-CO-O-n-C₄H₉, -C(CH₃)=C(CF₃)-CO-O-tert.-C₄H₉, -C(CH₃)=C(COOCH₃)₂, -C(CH₃)=C(COOC₂H₅)₂, -C(CH₃)=C(COOCH₃)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)-CO-OCH₃, -C(CH₃)=C(COO-n-C₃H₇)-CO-OC₂H₅, -C(CH₃)=C(COO-n-C₃H₇)₂, -C(CH₃)=CH-CH=CH-COOH, -C(CH₃)=CH-CH=CH-CO-OCH₃, -C(CH₃)=CH-CH=CH-CO-OC₂H₅, -C(CH₃)=CH-CH=C(COOCH₃)₂, -C(CH₃)=CH-CH=C(CN)-CO-OCH₃, -C(CH₃)=CH-CH=C(CN)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CN)CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OCH₃, -C(CH₃)=C(CH₃)-CH=C(CH₃)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Cl)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(Br)-CO-OC₂H₅, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH₂, -C(CH₃)=C(CH₃)-CH=C(CN)-CO-NH-CH₃, -C(CH₃)=CH-(CH₂)₂-COOH, -C(CH₃)=CH-(CH₂)₂-CO-OCH₃, -C(CH₃)=CH-(CH₂)₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(COOCH₃)₂, -C(CH₃)=CH-CH₂-CH(COOC₂H₅)₂, -C(CH₃)=CH-CH₂-CH(CN)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CN)-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OCH₃, -C(CH₃)=CH-CH₂-CH(CH₃)-CO-OC₂H₅, -C(CH₃)=CH-(CH₂)₂- ⁷⁸⁴²⁴ ⁰⁰⁰⁷⁰ ⁵⁵² ⁰⁰¹⁰⁰⁰²⁸⁰⁰⁰⁰⁰00200012000285917831300040 0002004131038 00004 78305 CO-NH₂, -C(CH₃)=CH-(CH₂)₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-COOH, -C(CH₃)=CH-CH₂-CO-OCH₃, -C(CH₃)=CH-CH₂-CO-OC₂H₅, -C(CH₃)=C(COOCH₃)-CH₂-CO-OCH₃, -C(CH₃)=C(COOCH₃)-CH₂-CO-OC₂H₅, -C(CH₃)=CH-CH₂-CO-NH₂, -C(CH₃)=CH-CH₂-CO-NH-CH₃, -C(CH₃)=CH-CH₂-CO-N(CH₃)₂.
Ganz besonders bevorzugt sind Verbindungen I, wobei X¹ und X² Sauerstoff, R¹ Halogen, R² Wasserstoff oder Fluor, R³ C₁-C₆- Alkyl, partiell oder vollständig halogeniertes C₁-C₂-Alkyl, R⁴ C₁-C₆-Alkyl, partiell oder vollständig halogeniertes C₁-C₂-Alkyl, R⁵ Wasserstoff oder R⁴ und R⁵ zusammen eine Tetramethylenkette bedeuten.
Die substituierten 3-Phenylurazile sind auf verschiedene Weise erhältlich, und zwar vorzugsweise nach einem der folgenden Verfahren:
a) Cyclisierung eines Enamin-esters der Formel II oder eines Enamin-carboxylats der Formel III
L¹ bedeutet niedermolekulares Alkyl, vorzugsweise C₁-C₄-Alkyl, oder Phenyl.
In der Regel arbeitet man in einem inerten Lösungs- oder Verdünnungsmittel, vorzugsweise in Gegenwart einer Base.
Als Lösungs- oder Verdünnungsmittel eignen sich inerte aprotische organische Lösungsmittel, beispsielsweise aliphatische oder cyclische Ether wie 1,2-Dimethoxyäthan, Tetrahydrofuran und Dioxan, aromatische Kohlenwasserstoffe wie Benzol, Toluol und Xylole, sowie inerte polare organische Lösungsmittel wie Dimethylformamid oder Dimethylsulfoxid, oder auch Wasser, wobei die polaren Lösungsmittel gegebenenfalls auch als Mischung mit einem unpolaren Kohlenwasserstoff wie n-Hexan verwendet werden können.
Als Basen kommen vorzugsweise Alkalimetallalkoholate, insbesondere Natriumalkoholate wie Natriummethanolat und Natriumethanolat, Alkalimetallhydroxide, insbesondere Natriumhydroxid und Kaliumhydroxid, Alkalimetallcarbonate, insbesondere Natriumcarbonat und Kaliumcarbonat, sowie Alkalimetallhydride, insbesondere Natriumhydrid in Betracht.
Bei der Verwendung von Natriumhydrid ist das Lösungsmittel besonders bevorzugt ein aliphatischer oder cyclischer Ether wie Tetrahydrofuran sowie Dimethylformamid und Dimethylsulfoxid.
Die Menge an Base liegt vorzugsweise zwischen der 0,5- und 2-molaren Menge, bezogen auf die Menge an II oder III.
Im allgemeinen empfiehlt sich eine Reaktionstemperatur zwischen (-78)°C und der Siedetemperatur des Reaktionsgemisches, insbesondere zwischen (-60) und 60°C.
Produkte I, in denen R³ Wasserstoff bedeutet, liegen nach der Cyclisierung je nach der Natur der verwendeten Base in Form des entsprechenden Metallsalzes der allgemeinen Formel Ic
(M⊕=ein Äquivalent eines Metallions, insbesondere ein Alkalimetallion wie Natrium)
vor, beispielsweise im Falle der vorstehend genannten bevorzugten, Alkalimetall enthaltenden Basen in Form des entsprechenden Alkalimetallsalzes. Das Salz kann in an sich bekannter Weise isoliert und gereinigt werden, beispielsweise durch Umkristallisation.
Produkte I, in denen R³ Wasserstoff bedeutet, erhält man durch Ansäuern des nach der Cyclisierung erhaltenen Reaktionsgemisches, z. B. mit Salzsäure.
b) Alkylierung oder Acylierung eines substituierten 3-Phenylurazils I, wobei R³ Wasserstoff bedeutet
Die Alkylierung erfolgt normalerweise mit dem Halaogenid, vorzugsweise dem Chlorid oder Bromid, oder dem Sulfat eines Alkans, Alkens, Alkins, Cycloalkans, Cyanoalkans, Halogenalkans, Phenylalkans oder Alkoxyalkans.
Als Acylierungsmittel kommen z. B. Ameisensäure-, Alkancarbonsäure- oder Alkoxycarbonsäurehalogenide in Betracht, wobei jeweils die Chloride und Bromide bevorzugt sind.
Die Alkylierung erfolgt zweckmäßigerweise in Gegenwart eines inerten organischen Lösungsmittels, beispielsweise in einem protischen Lösungsmittel wie niederen Alkoholen, vorzugsweie Ethanol, gegebenenfalls im Gemisch mit Wasser, oder in einem aprotischen Lösungsmittel wie alipahtische oder cyclische Ether, vorzugsweise 1,2-Dimethoxyethan, Tetrahydrofuran und Dioxan, aliphatischen Ketonen, vorzugsweise Aceton, Amiden, vorzugsweise Dimethylformamid, oder Sulfoxiden, vorzugsweise Dimethylsulfoxid.
In einer besonders bevorzugten Ausführungsform alkyliert man das als Salz vorliegende Produkt der Cyclisierung (Methode a) ohne vorherige Isolierung aus der Reaktionsmischung, wobei in diesem Fall noch aus der Cyclisierung der Verbindung II oder III stammende, überschüssige Base, beispielsweise Natriumhydrid, ein Natriumalkoholat oder Natriumcarbonat, vorhanden sein kann. Diese Base wirkt jedoch nicht störend; gewünschtenfalls kann auch noch eine weitere Menge des Verdünnungsmittels, das auch zur Cyclisierung der Verbindung II oder III verwendet wurde, zugesetzt werden.
Die Acylierung mit einem Halogenid kann auf analoge Weise erfolgen, wobei in diesem Fall besonders bevorzugt in einem aprotischen Lösungsmittel und in Gegenwart von Natriumhydrid als Base gearbeitet wird.
Die Reaktionstemperatur liegt im allgemeinen zwischen 0°C und ca. 100°C, vorzugsweise zwischen 0 und 40°C.
c) Substitution eines Halogenatoms am Phenylteil der substituierten 3-Phenylurazile I (R¹=Halogen) durch die Cyanogruppe
Hal bedeutet Halogen, vorzugsweise Chlor oder Brom.
Die Umsetzung erfolgt vorteilhaft in Gegenwart eines aprotischen, polaren Lösungsmittels, beispielsweise eines Alkylnitrils wie Acetonitril, Propionitril und Butyronitrol, eines Alkylharnstoffes wie N,N,N′,N′-Tetramethylharnstoff, eines Dialkylamids wie Dimethylformamid, eines Dialkylsulfoxids wie Dimethylsulfoxid oder in N-Methyl-2-pyrrolidon, 1,2-Dimethyl-imidazolidin-2-on, 1,2-Dimethyl-3,4,5,6-tetrahydro-2(1/h)-pyrimidinon oder Hexamethylphosphorsäuretriamid.
Normalerweise führt man die Reaktion unter Verwendung eines Metallcyanides, insbesondere eines Übergangsmetallcyanides wie Kupfer(I)cyanid, bei erhöhten Temperaturen, vorzugsweise zwischen 150 und 250°C, durch.
Zweckmäßig werden die Edukte in stöchiometrischen Mengen eingesetzt, jedoch kann auch ein Überschuß an Metallcyanid, etwa bis zur 4fachen molaren Menge (bezogen auf die Menge an Edukt I mit R¹=Halogen), vorteilhaft sein.
d) Überführung eines Pyrimidonderivats der Formel IVa oder IVb in einen Enolether Ia oder Ib
Hal bedeutet Chlor oder Brom;
Me⊕ bedeutet ein Äquivalent eines Metallions, insbesondere eines Übergangsmetallions, eines Alkalimetallions wie Natrium und Kalium oder eines Erdalkalimetallions wie Kalzium und Magnesium. Besonders bevorzugt ist Natrium.
Die Umsetzung der Pyrimidonderivate IVa oder IVb mit Alkanolen, Alkenolen, Alkinolen (R3′-OH) oder Alkanthiolen, Alkenthiolen, Alkinthiolen (R3′-SH) erfolgt vorteilhaft in Gegenwart einer organischen Base, wobei Pyridin besonders bevorzugt ist.
Die Menge an Base ist nicht kritisch; normalerweise ist die 0,5- bis 2fache molare Menge, bezogen auf die Menge an IVa oder IVb, ausreichend.
Die Umsetzungen von IVa mit H-X1-R3′ und von IVb mit H-X2-R3′ kann entweder ohne Lösungsmittel in einem Überschuß an R3′-OH bzw. R3′-SH oder in einem Geeigneten inerten organischen Lösungsmittel, z. B. in einem Aromaten wie Toluol und Xylol, in einem Ether wie Diethylether, Tetrahydrofuran und 1,2-Dimethoxyethan, oder in einem halogenierten Kohlenwasserstoff wie Dichlormethan und Chlorbenzol, vorgenommen werden.
Bei Einsatz der Verbindung R3′-OH arbeitet man vorzugsweise ohne Lösungsmittel, und zwar unter Verwendung der 1- bis ca. 150fachen Menge an R3′-OH, bezogen auf die Menge an Pyrimidonderivat IVa oder IVb.
Bei der Reaktionsführung mit einem Salz der Formel M⊕⊖O-R3′ oder M⊕⊖S-R3′ empfehlen sich äquimolare Mengen an Pyrimidonderivat und Salz, jedoch kann auch ein Überschuß an Salz bis etwa 30 mol-% (bezogen auf die Menge an Pyrimidonderivat) vorteilhaft sein.
Normalerweise ist eine Reaktionstemperatur zwischen 0 und 50°C, bevorzugt zwischen 10 und 30°C ausreichend.
Sofern nicht unmittelbar durch die als Methode a) beschriebene Cyclisierung unter basischen Bedingungen herstellbar, können die Salze derjenigen Verbindungen I, in denen R³ Wasserstoff bedeutet, auch in an sich bekannter Weise aus den Produkten der vorliegenden Methode d) erhalten werden. Zu diesem Zweck versetzt man beispielsweise die wäßrige Lösung einer anorganischen oder organischen Base mit dem substituierten 3-Phenylurazil I, bei dem R³ für Wasserstoff steht. Die Salzbildung erfolgt normalerweise bereits bei 20-25°C mit ausreichender Geschwindigkeit.
Besonders vorteilhaft ist es, das Natriumsalz durch Auflösen des 3-Phenylurazils I )R³=Wasserstoff) in wäßriger Natriumhydroxidlösung bei 20-25°C herzustellen, wobei äquivalente Mengen an 3-Phenylurazil und Natriumhydroxid eingesetzt werden. Das Salz des 3-Phenylurazils kann dann z. B. durch Fällen mit einem geeigneten inerten Lösungsmittel oder durch Abdampfen des Lösungsmittels isoliert werden.
Salze der 3-Phenylurazile, deren Metallion kein Alkalimetallion ist, können üblicherweise durch Umsalzen des entsprechenden Alkalimetallsalzes in wäßriger Lösung hergestellt werden. Auf diese Weise lassen sich im allgemeinen 3-Phenylurazil-Metallsalze herstellen, die in Wasser unlöslich sind.
e) Acetalisierung einer Verbindung I, wobei W eine Gruppe -C(=O)-R⁸ bedeutet
Die Acetalisierung erfolgt allgemein in einem inerten aprotischen organischen Lösungsmittel, beispielsweise in einem aliphatischen oder cyclischen Ether wie Diethylether, 1,2-Dimothoxyethan, Tetrahydrofuran und Dioxan, in einem aromatischen Kohlenwasserstoff wie Benzol, Toluol, o-, m-, p-Xylol und Mesitylen oder in einem chlorierten Kohlenwasserstoff wie Methylenchlorid, Chloroform und Chlorbenzol, sofern sie nicht ohne Lösungsmittel in einem Überschuß an H-X³R⁶, H-X⁴R⁷ oder H-X³(R⁶R⁷)X⁴-H durchgeführt wird.
Entstehendes Reaktionswasser kann wie üblich aus dem Reaktionsgemisch entfernt werden, z. B. mittels Wasserabscheidung.
Vorzugsweise führt man die Acetalisierung in Gegenwart einer organischen Säure wie p-Toluolsulfonsäure und/oder einer Lewissäure wie Zinntetrachlorid, Zinn-II-chlorid, Eisen-III-chlorid und Bortrifluoretherat durch, wobei die Menge an Säure normalerweise zwischen 0,5 und 100 mol-%, bezogen auf die Menge an zu acetalisierendem Edukt, liegt.
Die Mengenverhältnisse sind nicht kritisch. Für eine vollständige Umsetzung werden alle Reaktionspartner in etwa stöchiometrischem Verhältnis eingesetzt, bevorzugt verwendet man jedoch einen Überschuß an H-X³R⁶ und H-X⁴R⁷ bzw. H-X³(R⁶R⁷)X⁴-H.
Verwendet man die Edukte H-X³R⁶ und H-X⁴R⁷ bzw. H-X³(R⁶R⁷)X⁴-H gleichzeitig als Verdünnungsmittel, so liegen sie in einem größeren Überschuß vor.
Im allgemeinen arbeitet man bei einer Temperatur zwischen (-78) und 180°C, vorzaugsweise zwischen (-40) und 150°C.
Werden Produktgemische erhalten, z. B., wenn R⁶ und R⁷ keinen gemeinsamen Rest bilden und C³R⁶ und X⁴R⁷ nicht gleich sind, so können diese gewünschtenfalls nach an sich bekannten Methoden wie Kristallisation und Chromatograpie gereinigt und getrennt werden.
Insbesondere Verbindungen der Formel I, wobei W für eine Gruppe -C(R⁸)(X³R⁶)(X⁴R⁷) steht, in der R⁶ und R⁷ keinen gemeinsamen Rest bilden und X³R⁶ und X⁴R⁷ nicht gleich sind, können auch nach anderen literaturbekannte Methoden dargestellt werden (vgl. zum Beispiel Tetrahedron Lett. 32, 467-470 [1991] sowie die dort zitierte Literatur).
f) Acetalspaltung einer Verbindung I, wobei W eine Gruppe -C(R⁸)(X³R⁶)(X⁴R⁷) bedeutet
Die Acetalspaltung kann ohne Säurezusatz in Gegenwart einer Säure, z. B. einer Mineralsäure wie Salzsäure und Schwefelsäure, einer organischen Carbonsäure wie Ameisensäure, Essigsäure, Oxalsäure und Trifluoressigsäure, in Gegenwart eines sauren Ionenaustauschers, wie Amberlite® (Warenzeichen der Fa. "Aldrich") IR120 oder IRC84, oder in Gegenwart eines Übergangsmetallsalzes wie Quecksilber-(II)-oxid, Kupfer-(I)-oxid und Eisen-(III)-chlorid, durchgeführt werden.
Als Lösungs- oder Verdünnungsmittel eignen sich beispielsweise Aromaten wie Benzol, Toluol und o-, m-, p-Xylol, aliphatische oder cyclische Ether wie 1,2-Dimethoxyethan, Diethylether, Tetrahydrofuran und Dioxan, Alkohole wie Methanol, Ethanol und Isopropanol, polare organische Lösungsmittel wie Dimethylformamid, Dimethylsulfoxid und Acetonitril, Ketone wie Aceton und Butanon oder auch Wasser.
Vorzugsweise arbeitet man ohne Lösungsmittel in einem Überschuß der zur Acetalspaltung verwendeten Säure, wobei Ameisensäure besonders bevorzugt ist.
Für eine vollständige Umsetzung werden die Edukte I, wobei W eine Gruppe -C(R⁸)(X³R⁶)(X⁴R⁷) bedeutet; und H₂X⁵ in mindestens stöchiometrischem Verhältnis eingesetzt, jedoch ist auch ein Überschuß an H₂X⁵ bis etwa 200 mol-% möglich.
Die Menge an Säure, Ionenaustauscher oder Übergangsmetallsalz ist nicht kritisch. Im allgemeinen ist eine Menge bis etwa 300 mol-%, bezogen auf die Menge an H₂X⁵, ausreichend.
In der Regel liegt die Reaktionstemperatur zwischen (-78) und 180°C, vorzugsweise zwischen 0°C und der Siedetemperatur des jeweiligen Verdünnungsmittels.
Weitere zur Herstellung der substituierten 3-Phenylurazile I brauchbare Methoden können Houben-Weyl, Handbuch der Org. Chemie, 4. Auflage, Bd. E3, S. 362 ff, entnommen werden.
g) Olefinierung von Verbindungen I (W=-C(R⁸)=O)
Die Reaktion kann mit den folgenden Phosphoryliden Va bis Vd, Phosphoniumsalzen VIa bis VId und Phosphonaten VIIa bis VIId durchgeführt werden:
Phosphorylide V:
R³P=C(R⁹)-CO-R¹⁰ (Va)
R³P=C(R⁹)-CH₂-CO-R¹⁰ (Vb)
R³P=C(R⁹)-C(R¹¹)=C(R¹²)-CO-R¹⁰ (Vc)
R³P=C(R⁹)-CH₂-CH(R¹³)-CO-R¹⁰ (Vd)
Phosphoniumsalze VI:
R₃P⊕-CH(R⁹)-CO-R¹⁰, Hal⊖ (VIa)
R₃P⊕-CH(R⁹)-CH₂-CO-R¹⁰, Hal⊖ (VIb)
R₃P⊕-C(R⁹)-CR¹¹=CR¹²-CO-R¹⁰, Hal⊖ (VIc)
R₃P⊕-C(R⁹)-CH₂-CHR¹³-CO-R¹⁰, Hal⊖ (VId)
Phosphonate VII:
(RO)₂PO-CH(R⁹)-CO-R¹⁰ (VIIa)
(RO)₂PO-CH(R⁹)-CH₂-CO-R¹⁰ (VIIb)
(RO)₂PO-CH(R⁹)-CR¹¹=CR¹²-CO-R¹⁰ (VIIc)
(RO)₂PO-CH(R⁹)-CH₂-CHR¹³-CO-R¹⁰ (VIId)
Wenig geeignet sind diejenigen Phosphorylide Vb und Vd, Phosphoniumsalze VIb und VId sowie Phosphonate VIIb und VIId, bei denen R¹⁰ Wasserstoff, Alkyl oder Cycloalkyl bedeutet.
Die Reste R am Phosphor können gleich oder verschieden sein und stehen beispielsweise für verzweigte oder unverzweigte C₁-C₈- Alkylgruppen, C₅- oder C₆-Cycloalkylgruppen und insbesondere für Phenyl, das weitere (für die Umsetzung inerte Substituenten, beispielsweise C₁-C₄-Alkyl wie Methyl, Ethyl und tert. Butyl, C₁-C₄-Alkoxy wie Methoxy oder Halogen wie Fluor, Chlor und Brom) tragen kann. Bevorzugt sind unsubstituierte Phenylreste, da der für die Herstellung der Phosphorylide V und Phosphoniumsalze VI verwendete Ausgangsstoff Triphenylphosphin besonders kostengünstig ist und zudem das bei den Umsetzungen das sehr reaktionsträge und gut abtrennbare feste Triphenylphospinoxid entsteht.
Zur Herstellung der Phosphonate VII eignen sich beispielsweise die in Houben-Weyl, Methoden der Organischen Chemie, Band E2, 1982, S. 345 ff. beschriebenen Methoden.
Als Lösungsmittel kommen inerte organische Lösungsmittel, z. B. Aromaten wie Toluol und o-, m-, p-Xylol, Ether wie 1,2-Dimethoxyethan, Diethylether, Tetrahydrofuran und Dioxan, polare organische Lösungsmittel wie Dimethylformamid und Dimethylsulfoxid, oder Alkohole wie Methanol, Ethanol und Isopropanol, in Betracht.
Bei der Olefinierung von I, wobei W -C(R⁸)=O bedeutet, mit einem Phosphoniumsalz VI oder einem Phosphonat VII arbeitet man in Gegenwart einer Base, wobei Alkalimetallalkyle wie n-Butyllithium, Alkalimetallhydride und -alkoholate wie Natriumhydrid, Natriumethanolat und Kalium-tert.-butanolat, sowie Alkalimetall- und Erdalkalimetallhydroxide wie Calciumhydroxid, besonders gut geeignet sind.
Für eine vollständige Umsetzung werden alle Reaktionspartner in etwa stöchiometrischem Verhältnis eingesetzt, bevorzugt verwendet man jedoch einen Überschuß an Base bis etwa 10 mol-%.
Im allgemeinen liegt die Reaktionstemperatur zwischen (-40) und 150°C.
Die Verbindungen der Formel V, VI und VII sind bekannt oder lassen sich in auf bekannte Weise darstellen (vgl. z. H. Houben- Weyl, Methoden d. Org. Chemie, Bd. E1, S. 636 ff., Georg Thieme Verlag, Stuttgart 1982, Chem. Ber. 95, 3993 (1962) oder Houben- Weyl, Methoden d. Org. Chemie, Bd. E2, S. 345 ff., Georg Thieme Verlag, Stuttgart 1982).
Eine weitere Möglichkeit zur Darstellung von 3-Phenylurazilen I, wobei W -CR⁸=CR⁹-CO-R¹⁰ bedeutet und R¹⁰ Wasserstoff, Alkyl, Alkenyl, Haloalkyl, Cycloalkyl, Phenyl oder Alkoxyalkyl bedeuten, besteht in der an sich bekannten Aldolkondensation. Hierfür geeignete Bedingungen sind z. B. Nielsen, Org. React. 16, 1 ff. (1968) zu entnehmen.
Als weitere Methode zur Synthese von Verbindungen der Formel I, wobei
W -C(R⁸)=C(R⁹)-CO-R¹⁰, -CH(R⁸)=CH(R⁹)-CO-R¹⁰, -CR⁸=CR¹¹-CH₂-CO-R¹²,
-CR⁸=CR¹¹-CR¹³=CR¹⁴-CO-R¹⁰ oder -CR⁸=CR¹¹-CH₂-CHR¹⁵-CO-R¹²
wobei R⁹ oder R¹¹ Wasserstoff, Cyano, Alkoxycarbonyl oder Alkylcarbonyl bedeuten, kommen sowohl die Knoevenagel-Kondensation als auch die Perkin-Kondensation in Betracht. Geeignete Bedingungen sind z. B. aus Org. React. 1967, 15, 204 ff. (Knoevenagel) bzw. Johnson, Org. React. 1942, 1, 210 ff. (Perkin) ersichtlich.
Verbindungen, in denen R¹⁰ -NR¹⁸R¹⁹ oder -SR¹⁷ bedeuten, lassen sich z. B. in an sich bekannter Weise dadurch herstellen, daß man Verbindungen, in denen R¹⁰ für Hydroxyl steht, in die entsprechenden Säurehalogenide (R¹⁰ bedeutet Halogen) überführt und die Verfahrensprodukte anschließend mit einem entsprechenden Amin H-NR¹⁸R¹⁹ oder Thiol H-SR¹⁷ oder mit einem reaktiven Derivat dieser Verbindungen umsetzt.
h) Umsetzung von Verbindungen I (W = -C(R⁸)=O) mit Aminen, Hydroxylaminen oder Hydrazinen
Die Umsetzung erfolgt normalerweise in einem inerten organischen Lösungs- oder Verdünnungsmittel, z. B. in einem Aromaten wie Toluol und Xylol, in einem chlorierten Kohlenwasserstoff wie Dichlormethan, Chloroform und Chlorbenzol, in einem Ether wie Diethylether, 1,2-Dimethoxyether und Tetrahydrofuran, in einem Alkohol wie Methanol und Ethanol, oder in einem Gemisch der genannten Lösungsmittel.
Liegen die Amine H₂N-R¹⁴ als Salze, z. B. als Hydrochloride oder Oxalate vor, so ist zu ihrer Freisetzung die Zugabe einer Base wie vorzugsweise Natriumcarbonat, Kaliumcarbonat, Natriumhydrogencarbonat, Triethylamin und Pyridin, empfehlenswert.
Das entstehende Reaktionswasser kann gegebenenfalls destillativ oder mit Hilfe eines Wasserabscheiders aus dem Reaktionsgemisch entfernt werden.
Üblicherweise liegt die Reaktionstemperatur zwischen (-30) und 150°C, bevorzugt zwischen 0 und 130°C.
i) Spaltung von Verbindungen I, wobei W -C(R⁸)=N-R¹⁴ bedeutet
Die Spaltung erfolgt lösungsmittelfrei oder in einem inerten Lösungs- oder Verdünnungsmittel mit Wasser oder einem reaktionsfähigen Derivat des Wassers.
Die Umsetzung kann hydrolytisch oder unter oxidativen Bedingungen durchgeführt werden, wobei sich eine Reaktionstemperatur zwischen (-78) und 180°C, vorzugsweise zwischen 0°C und dem Siedepunkt des Verdünnungsmittels empfiehlt.
Als Lösungs- oder Verdünnungsmittel kommen z. B. Aromaten wie Benzol, Toluol und o-, m-, p-Xylol, chlorierte Kohlenwasserstoffe wie Dichlormethan, Chloroform und Chlorbenzol, Ether wie Dialkylether, 1,2-Dimethoxyethan, Tetrahydrofuran und Dioxan, Alkohle wie Methanol und Ethanol, Ketone wie Aceton oder Wasser sowie Gemische der genannten Lösungsmittel, in Betracht.
Zweckmäßigerweise arbeitet man in Gegenwart einer Mineralsäure wie Salzsäure, Bromwasserstoffsäure und Schwefelsäure, einer Carbonsäure wie Essigsäure und Trifluoressigsäure oder einer Sulfonsäure wie p-Toluolsulfonsäure.
Bei der Arbeitsweise unter oxidativen Bedingungen eignen sich insbesondere Oxidationsmittel wie Bleitetraacetat, Natriumhypochlorid und Wasserstoffperoxid.
Gewünschtenfalls kann die Reaktionsführung zusätzlich in Gegenwart eines Katalysators wie Kupfer-(II)-sulfat, Titantetrachlorid und Bortrifluoretherat erfolgen.
Die Mengen an Säure, Oxidationsmittel und Katalysator können in weiten Bereichen variiert werden. Normalerweise liegen sowohl Säure- als auch Katalysatormenge zwischen 5 und 200 mol-%, und die Menge an Oxidationsmittel zwischen 25 und 400 mol-%, bezogen auf die Menge der zu oxidierenden Verbindung.
k) Umsetzung eines substituierten 3-Phenylurazils I, wobei X² Sauerstoff bedeutet, mit einem Schwefelungsreagenz
Die Umsetzung erfolgt in der Regel in einem inerten Lösungsmittel, beispielsweise in einem aromatischen Kohlenwasserstoff wie Toluol und o-, m-, p-Xylol, in einem Ether wie Diethylether, 1,2-Dimethoxyethan und Tetrahydrofuran, oder in einem organischen Amin wie Pyridin.
Als Schwefelungsreagenz eignen sich besonders gut Phosphor(V)- sulfid und 2,4-Bis(4-methoxyphenyl)-1,3,2,4-dithiadiphosphetan- 2,4-dithion ("Lawessons Reagenz").
Die Menge an Schwefelungsreagenz ist nicht kritisch; normalerweise verwendet man die 1- bis 5fache molare Menge, bezogen auf das zu schwefelnde 3-Phenylurazil.
Normalerweise liegt die Reaktionstemperatur zwischen 20 und 200°C, vorzugsweise zwischen 40°C und dem Siedepunkt des Lösungsmittels.
l) Halogenierung eines substituierten 3-Phenylurazils I, wobei R⁵ Wasserstoff bedeutet
Die Halogenierung erfolgt in der Regel in einem inerten organischen Lösungs- oder Verdünnungsmittel. Für die Chlorierung und Bromierung kommen beispielsweise aliphatische Carbonsäure wie Essigsäure, oder chlorierte aliphatische Kohlenwasserstoffe wie Methylenchlorid, Chloroform und Tetrachlorkohlenstoff, in Betracht. Für die Jodierung sind niedrig siedende aliphatische Carbonsäuren wie Essigsäure besonders bevorzugt.
Für die Chlorierung und Bromierung eignen sich insbesondere elementares Chlor bzw. Brom sowie Sulfurylchlorid bzw. Sulfurylbromid, wobei sich eine Reaktionstemperatur zwischen 0 und 60°C, vorzugsweise zwischen 10 und 30°C, empfiehlt.
Gewünschtenfalls kann die Chlorierung und Bromierung in Gegenwart eines säurebindenden Mittels erfolgen, wobei Natriumacetat und tertiäre Amine wie Triethylamin, Dimethylanilin und Pyridin besonders bevorzugt sind.
Als Jodierungsmittel ist elementares Jod besonders bevorzugt, wobei in diesem Fall die Reaktionstemperatur zwischen ca. 0 und 110°C, vorzugsweise zwischen 10 und 30°C, liegt.
Besonders vorteilhaft führt man die Jodierung in Gegenwart einer Mineralsäure wie rauchende Salpetersäure durch.
Die Menge an Halogenierungsmittel ist nicht kritisch; normalerweise verwendet man äquimolare Mengen an Halogenierungsmittel oder einen Überschuß bis etwa 200 mol-%, bezogen auf das zu halogenierende Edukt.
Überschüssiges Jod kann beispielsweise nach der Reaktion mittels gesättigter wäßriger Natriumhydrogensulfitlösung entfernt werden.
m) Reduktion eines substituierten 3-Phenylurazils I, wobei W die Cyanogruppe bedeutet
Die Umsetzung erfolgt zweckmäßig in einem inerten organischen Lösungsmittel, z. B. einem Aromaten wie Toluol und o-, m-, p-Xylol, einem aliphatischen oder cyclischen Ether wie Diethylether, tert.-Butylmethylether, Tetrahydrofuran und Dioxan, einem chlorierten Kohlenwasserstoff wie Methylenchlorid, Chloroform und Chlorbenzol, oder in einer organischen Carbonsäure wie Ameisensäure.
Als Reduktionsmittel eignen sich beispielsweise Wasserstoff oder Metallsalze wie Zinn-(II)-chlorid, Metallhydride wie Diisobutylaluminiumhydrid, Diisopropylaluminiumhydrid, Lithium-trisethoxyaluminiumhydrid und Lithium-bisethoxy-aluminiumhydrid oder Triethylsilan. Bevorzugt ist die Verwendung von Diisobutylaluminiumhydrid, Ameisensäure oder Wasserstoff.
Gewünschtenfalls kann die Reduktion in Gegenwart eines Katalysators, wie Triethyloxoniumtetrafluoroborat oder Raney-Nickel durchgeführt werden.
Arbeitet man ohne Verdünnungsmittel in Ameisensäure als Reduktionsmittel, so kann diese auch in einem größeren Überschuß vorliegen.
Die vorteilhafteste Reaktionstemperatur ist abhängig vom jeweiligen Reduktionsmittel, liegt aber im allgemeinen zwischen (-78) und 150°C.
Die als Ausgangsstoffe benötigten Enamin-Ester der Formel II sind neu, es sei denn, W bedeutet eine Gruppe -CH=CH-CO-OR¹⁴ mit R¹⁴ C₁-C₆-Alkyl oder C₃-C₆-Alkenyl, wenn R⁴ die Trifluormethylgruppe und R⁵ Wasserstoff sind (vgl. US 49 79 982). Sie können ebenfalls als Herbizide eingesetzt werden.
Die Enamin-Ester II können nach an sich bekannten Methoden hergestellt werden, z. B. nach einem der folgenden Verfahren:
Vorzugsweise arbeitet man im wesentlichen wasserfrei in einem inerten Lösungs- oder Verdünnungsmittel, besonders bevorzugt in Gegenwart eines sauren oder basischen Katalysators.
Als Lösungs- oder Verdünnungsmittel kommen insbesondere mit Wasser azeotrop mischbare organische Lösungsmittel, beispielsweise Aromate wie Benzol, Toluol und o-, m-, p-Xylol, halogenierte Kohlenwasserstoffe wie Methylenchlorid, Chloroform, Tetrachlorkohlenstoff und Chlorbenzol, aliphatische und cyclische Ether wie 1,2-Dimethoxyethan, Tetrahydrofuran und Dioxan, oder Cyclohexan, aber auch Alkohole wie Methanol und Ethanol, in Betracht.
Als saure Katalysatoren eignen sich bevorzugt starke Mineralsäuren wie Schwefelsäure und Salzsäure, Phosphor enthaltende Säuren wie Orthophosphorsäure und Polyphosphorsäure, organische Säuren wie p-Toluolsulfonsäure sowie saure Kationenaustauscher wie "Amberlyst 15" (Fluka).
Als basische Katalysatoren eignen sich z. B. Metallhydride wie Natriumhydrid sowie besonders bevorzugt Metallalkoholate wie Natriummethanolat und Ethanolat.
Zweckmäßig setzt man den β-Ketoester VIII und den Phenylharnstoff IX in stöchiometrischem Verhältnis ein oder man arbeitet mit einem geringen Überschuß der einen oder anderen Komponente bis etwa 10 mol-%.
Normalerweise ist eine Katalysatormenge zwischen 0,5 und 50 mol-%, bezogen auf die Menge eines Edukts, ausreichend.
Im allgemeinen erfolgt die Reaktionsführung bei einer Temperatur zwischen 60 und 120°C, zur raschen Entfernung von entstehendem Wasser vorzugsweise bei der Siedetemperatur des Reaktionsgemisches.
L³ bedeutet C₁-C₄-Alkyl oder Phenyl.
Diese Umsetzung kann beispielsweise in einem inerten, mit Wasser mischbaren, organischen Lösungsmittel, beispielsweise einem aliphatischen oder cyclischen Ether wie Diethylether, 1,2-Dimethoxyethan, Tetrahydrofuran und Dioxan, oder einem niederen Alkohol, insbesondere Ethanol, durchgeführt werden, wobei die Reaktionstemperatur normalerweise zwischen 50 und 100°C, vorzugsweise bei der Siedetemperatur des Reaktionsgemisches, liegt.
Die Reaktion kann jedoch auch in einem aromatischen Verdünnungsmittel wie Benzol, Toluol und o-, m-, p-Xylol durchgeführt werden, wobei in diesem Fall der Zusatz entweder eines sauren Katalysators wie Salzsäure und p-Toluolsulfonsäure oder einer Base, z. B. eines Alkalimetallalkoholates wie Natriummethanolat und Natriumethanolat, empfehlenswert ist. Auch bei dieser Verfahrensvariante liegt die Reaktionstemperatur normalerweise zwischen 50 und 100°C, bevorzugt jedoch zwischen 60 und 80°C.
Die Umsetzung erfolgt zweckmäßig in Gegenwart eines im wesentlichen wasserfreiem aprotischen organischen Lösungs- oder Verdünnungsmittel, beispielsweise eines aliphatischen oder cyclischen Ethers wie Diethylether, 1,2-Dimethoxyethan, Tetrahydrofuran und Dioxan, eines aliphatischen oder aromatischen Kohlenwasserstoffs wie n-Hexan, Benzol, Toluol und o-, m-, p-Xylol, eines halogenierten, aliphatischen Kohlenwasserstoffs wie Methylenchlorid, Chloroform, Tetrachlorkohlenstoff, 1,2-Dichlorethan und Chlorbenzol, eines aprotischen, polaren Lösungsmittel wie Dimethylformamid, Hexamethylphosphorsäuretriamid und Dimethylsulfoxid, oder eines Gemisches aus den genannten Solventien.
Gewünschtenfalls kann auch in Gegenwart einer Metallhydridbase wie Natrium- und Kaliumhydrid, eines Alkalimetall- oder Erdalkalimetallalkoholates wie Natriummethanolat, Natriumethanolat und Kalium-tert.-butanolat, oder einer organischen tertiären Base wie Triethylamin und Pyridin gearbeitet werden, wobei die organische Base gleichzeitig als Lösungsmittel dienen kann.
Zweckmäßig setzt man die Edukte in stöchiometrischem Verhältnis ein oder man arbeitet mit einem geringen Überschuß der einen oder anderen Komponente bis etwa 20 mol-%. Arbeitet man ohne Lösungsmittel in Gegenwart einer organischen Base, so liegt diese in einem größeren Überschuß vor.
Die Reaktionstemperatur liegt vorzugsweise im Bereich zwischen (-80) und 50°C, besonders bevorzugt zwischen (-60) und 30°C.
L¹ und L⁴ bedeuten C₁-C₄-Alkyl oder Phenyl.
Diese Reaktion erfolgt zweckmäßig in einem aprotischen, polaren Lösungs- oder Verdünnungsmittel wie Dimethylformamid, 2-Butanon, Dimethylsulfoxid und Acetonitril, und zwar vorteilhaft in Gegenwart einer Base, beispielsweise eines Alkalimetall- oder Erdalkalimetallalkoholats, insbesondere eines Natriumalkanolates wie Natriummethanolat, eines Alkalimetall- oder Erdalkalimetallcarbonates, insbesondere Natriumcarbonat, oder eines Alkalimetallhydrids wie Lithium- und Natriumhydrid.
Normalerweise ist die 1- bis 2fache molare Menge an Base, bezogen auf die Menge eines Edukts, ausreichend.
Die Reaktionstemperatur liegt im allgemeinen zwischen 80 und 180°C, vorzugsweise bei der Siedetemperatur des Reaktionsgemisches.
Bezüglich der Mengenverhältnisse der Edukte gelten die Angaben für Methode n).
In einer besonders bevorzugten Ausführungsform verwendet man ein Natriumalkoholat als Base und destilliert den im Laufe der Reaktion entstehenden Alkohol kontinuierlich ab. Die auf diese Weise hergestellten Enamin-Ester der Formel II können ohne Isolierung aus der Reaktionsmischung gemäß Verfahrensvariante a) zu einem Salz der substituierten 3-Phenylurazile I cyclisiert werden.
Diese Umsetzung erfolgt vorteilhaft in Gegenwart eines im wesentlichen wasserfreien, aprotischen, organischen Lösungs- oder Verdünnungsmittels, gewünschtenfalls in Gegenwart einer Metallhydridbase wie Natrium- und Kaliumhydrid oder einer organischen tertiären Base wie Triethylamin und Pyridin, wobei die organische Base auch als Lösungsmittel dienen kann.
Bezüglich der geeigneten Lösungsmittel und der Mengenverhältnisse gelten die Angaben für Methode o).
Die Reaktionstemperatur liegt in der Regel zwischen (-80) und 150°C, vorzugsweise zwischen (-60)°C und dem jeweiligen Siedepunkt des Lösungsmittels.
Die Enamin-carboxylate der Formel III sind ebenfalls neu und können als Herbizide eingesetzt werden. Sie sind nach an sich bekannten Verfahren herstellbar, beispielsweise aus einem Anilinderivat der Formel XVI nach folgendem Reaktionsschema:
In Gleichung (Gl1) bedeuten R⁴′ und R⁵′ Wasserstoff oder C₁-C₄-Alkyl.
Die Umsetzungen nach Reaktionsgleichung 1 und 2 erfolgen vorzugsweise in einem wasserfreien inerten aprotischen Lösungsmittel, beispielsweise in einem halogenierten Kohlenwasserstoff wie Methylenchlorid, Chloroform, Tetrachlorkohlenstoff und Chlorbenzol, einem aromatischen Kohlenwasserstoff wie Benzol, Toluol und o-, m-, p-Xylol, oder einem aliphatischen oder cyclischen Äther wie Diethylether, Dibutylether, 1,2-Dimethoxyethan, Tetrahydrofuran und Dioxan.
Für die Umsetzung des Lactons XV mit dem Anilinderivat XVI nach Gleichung (Gl1) empfiehlt sich der Zusatz eines basischen Katalysators, z. B. 4-Pyrrolidinopyridin, 4-Dimethylamino-pyridin, 1,2-Diazabicyclo[2,2,2]octan, 1,5-Diazabicyclo[4,3,0]non-5-en, 1,8-Diazabicyclo[5,4,0]undec-7-en oder Diethylamin.
Da die Reaktion exotherm verläuft, ist im allgemeinen eine Reaktionstemperatur zwischen (-10) und 50°C, vorzugsweise zwischen 10 und 30°C, ausreichend.
Für die Reaktion der Verbindungen der Formeln XVIII und XVI miteinander nach Gleichung (Gl2) sind dagegen höhere Temperaturen, etwa zwischen 70 und 140°C, insbesondere zwischen 100 und 120°C, vorteilhaft.
Bei der Umsetzung nach Reaktionsgleichung (Gl3) handelt es sich um eine Aminolyse, die in der Regel entweder ohne Lösungsmittel [vgl. z. B. J. Soc. Dyes Col. 42, 81 (1926), Ber. 64, 970 (1931); Org. Synth., Coll. Vol. IV, 80 (1963) und J.A.C.S. 70, 2402 (1948)] oder in einem inerten wasserfreien Lösungs- oder Verdünnungsmittel, insbesondere in einem aprotischen Solvens, beispielsweise in einem gegebenenfalls halogenierte Aromaten wie Toluol, o-, m-, p-Xylol und Chlorbenzol, durchgeführt wird.
Hierbei empfiehlt sich das Arbeiten in Gegenwart eines basischen Katalysators, z. B. eines höher siedenden Amins [siehe beispielsweise Helv. Chim. Acta 11, 779 (1928) und U.S. 24 16 738] oder Pyridin.
Vorzugsweise liegt die Reaktionstemperatur zwischen etwa 20 und 160°C.
Bei allen drei Herstellungsvarianten setzt man die Edukte zweckmäßigerweise in stöchiometrischem Verhältnis ein oder man arbeitet mit einem geringen Überschuß der einen oder anderen Komponente bis etwa 10 mol-%. Arbeitet man in Gegenwart eines basischen Katalysators, so ist im allgemeinen eine Menge zwischen 0,5 und 200 mol-%, bezogen auf die Menge eines Edukts, ausreichend.
Die anschließende Umsetzung der so hergestellten Verbindungen der Formel XVII mit der Verbindung H₂N-COOL¹ wird vorteilhaft in einem weitgehend wasserfreien Lösungs- oder Verdünnungsmittel bei Normaldruck durchgeführt, besonders bevorzugt in Gegenwart eines sauren Katalysators.
Als Lösungs- oder Verdünnungsmittel kommen insbesondere mit Wasser azeotrop mischbare organische Flüssigkeiten, beispielsweise Aromaten wie Benzol, Toluol und o-, m-, p-Xylol oder halogenierte Kohlenwasserstoffe wie Tetrachlorkohlenstoff und Chlorbenzol, in Betracht.
Geeignete Katalysatoren sind insbesondere starke Mineralsäuren wie Schwefelsäure, organische Säuren wie p-Toluolsulfonsäure, Phosphor enthaltende Säuren wie Orthophosphorsäure und Polyphosphorsäure oder saure Kationenaustauscher wie "Amberlyst 15" (Fluka).
Im allgemeinen liegt die Reaktionstemperatur zwischen etwa 70 und 150°C; zur raschen Entfernung des entstehenden Reaktionswassers arbeitet man jedoch zweckmäßigerweise bei der Siedetemperatur des Solvens.
Die Pyrimidon-Derivate IVa und IVb, von denen Methode d) ausgeht, können durch Halogenierung, vorzugsweise Chlorierung und Bromierung, von 3-Phenylurazilen I, in denen R³ Wasserstoff bedeutet, in Gegenwart eines inerten Lösungs- oder Verdünnungsmittels erhalten werden.
Als Lösungs- oder Verdünnungsmittel kommen insbesondere aprotische organische Flüssigkeiten, beispielsweise aliphatische oder aromatische Kohlenwasserstoffe wie n-Hexan, Benzol, Toluol und o-, m-, p-Xylol, halogenierte aliphatische Kohlenwasserstoffe wie Methylenchlorid, Chloroform und 1,2-Dichlorethan, halogenierte aromatische Kohlenwasserstoffe wie Chlorbenzol, oder tertiäre Amine wie N,N-Dimethylanilin, in Betracht.
Als Halogenierungsmittel eignen sich insbesondere Thionylchlorid, Phosphorpentachlorid, Phosphoroxychlorid, Phosphorpentabromid oder Phosphorylbromid. Besonders vorteilhaft kann auch ein Gemisch aus Phosphorpentachlorid und Phosphoroxychlorid oder aus Phosphorpentabromid und Phosphorylbromid sein, wobei dann ohne Verdünnungsmittel in einem Überschuß an Phosphoroxychlorid oder Phosphorylbromid gearbeitet werden kann.
Bei Verwendung von Thionylchlorid als Halogenierungsmittel empfiehlt es sich, eine katalytische Menge an Dimethylformamid zuzusetzen.
Die Menge an Halogenierungsmittel ist nicht kritisch; für eine vollständige Umsetzung benötigt man mindestens äquimolare Mengen an Halogenierungsmittel und zu halogenierendem Edukt. Es kann jedoch auch ein 1- bis 8facher molarer Überschuß an Halogenierungsmittel vorteilhaft sein.
Die Reaktionstemperaturen liegen im allgemeinen zwischen 0°C und der Rückflußtemperatur des Reaktionsgemisches, vorzugsweise zwischen 20 und 120°C.
Die Verbindungen der Formeln IX, XII, XIII und XIV sind ebenfalls neu. Sie können nach an sich bekannten Methoden hergestellt werden, besonders vorteilhaft aus Verbindungen der Formel XVI:
s) durch "Phosgenierung" und Hydrolyse der Verfahrensprodukte mit Ammoniak
Das Verfahren kann in einem inerten, im wesentlichen wasserfreien Lösungs- oder Verdünnungsmittel oder ohne Lösungsmittel durchgeführt werden, wobei die Verbindungen XVI bevorzugt mit Phosgen oder Chlorameisensäuretrichlormethylester umgesetzt werden.
Als Lösungs- oder Verdünnungsmittel kommen insbesondere aprotische, organische Lösungsmittel, beispielsweise Aromaten wie Toluol und o-, m-, p-Xylol, halogenierte Kohlenwasserstoffe wie Methylenchlorid, Chloroform, 1,2-Dichlorethan und Chlorbenzol, aliphatische oder cyclische Ether wie 1,2-Dimethoxyethan, Tetrahydrofuran und Dioxan, oder Ester wie Essigsäureethylester, sowie Gemische dieser Lösungsmittel, in Betracht.
Je nach eingesetztem Anilinderivat XVI kann der Zusatz einer Base wie Triethylamin vorteilhaft sein, beispielsweise in 0,5- bis 2facher molarer Menge, bezogen auf die Menge an XVI.
Durch Wahl der geeigneten Reaktionsbedingungen lassen sich sowohl die Carbaminsäurechloride XIV als auch die Phenylisocyanate XII erhalten:
So erhält man bei niederen Temperaturen zwischen etwa (-40) und 50°C normalerweise die Carbaminsäurechloride XIV, während weitere Temperaturerhöhung, bis zur Siedetemperatur des Reaktionsgemisches, dagegen überwiegend zur Bildung der Phenylisocyanate XII führt, die mit Ammoniak oder einem reaktiven Derivat des Ammoniaks zu den Phenylharnstoffderivaten IX umgesetzt werden können.
t) durch Umsetzung mit Alkalimetallcyanaten
M⊕ steht für das Äquivalent eines Metallions, insbesondere für ein Alkalimetallion wie Natrium und Kalium.
Die Umsetzung erfolgt in einem inerten Lösungs- oder Verdünnungsmittel, beispielsweise in einem aromatischen Kohlenwasserstoff wie Toluol und o-, m-, p-Xylol, in einem aliphatischen oder cyclischen Ether wie Tetrahydrofuran und Dioxan, in einem niederen Alkohol wie Methanol und Ethanol, in Wasser oder in einem Gemisch der genannten Solventien.
Die Menge an Cyanat ist nicht kritisch; für eine vollständige Umsetzung benötigt man mindestens äquimolare Mengen an Anilinderivat XVI und Cyanat, jedoch kann auch ein Überschuß an Cyanat, bis etwa 100 mol-%, vorteilhaft sein.
Die Reaktionstemperatur liegt im allgemeinen zwischen 0°C und der Rückflußtemperatur des Reaktionsgemisches.
u) durch Umsetzung mit Estern XX
L⁴ steht für C₁-C₄-Alkyl oder Phenyl;
L⁵ steht für Halogen, vorzugsweise Chlor oder Brom, für C₁-C₄- Alkoxy oder Phenoxy.
Als Lösungs- oder Verdünnungsmittel eignen sich beispielsweise aromatische Kohlenwasserstoffe wie Toluol und o-, m-, p-Xylol, halogenierten Kohlenwasserstoffe wie Methylenchlorid, Chloroform, 1,2-Dichlorethan und Chlorbenzol, aliphatische oder cyclische Ethern, wie 1,2-Dimethoxyethan, Tetrahydrofuran und Dioxan, Ester wie Essigsäureethylester, Alkohole wie Methanol und Ethanol, oder Wasser oder Zweiphasengemische aus einem organischen Lösungsmittel und Wasser.
Vorteilhaft verläuft die Umsetzung in Gegenwart einer Base, z. B. eines Alkalimetallhydroxides, -carbonates oder -alkoholates wie Natriumhydroxid, Natriumcarbonat, Natriummethanolat und Natriumethanolat oder eines tertiären Amins wie Pyridin und Triethylamin.
Gewünschtenfalls kann auch ein Katalysator, z. B. eine Lewissäure wie Antimontrichlorid, zugesetzt werden.
Zweckmäßig setzt man die Ausgangsverbindungen und die Base in stöchiometrischem Verhältnis ein, jedoch kann auch die eine oder andere Komponente in einem Überschuß, bis etwa 100 mol-%, vorliegen.
In der Regel beträgt die Katalysatormenge 1 bis 50 mol-%, bevorzugt 2 bis 30 mol-%, bezogen auf die Menge an eingesetztem Anilinderivat XVI.
Im allgemeinen liegt die Reaktionstemperatur zwischen (-40)°C und der Siedetemperatur des Reaktionsgemisches.
Die Ausgangsverbindungen der Formel XVI und deren Herstellung sind aus der Literatur bekannt oder nach an sich bekannten Methoden herstellbar.
Bei den vorstehend genannten Verfahren zur Synthese von substituierten Phenylurazilen I, deren Salzen, Enolethern oder Vorprodukten arbeitet man zweckmäßigerweise unter Normaldruck oder unter dem Eigendruck des jeweiligen Lösungsmittels. Geringerer oder höherer Druck ist möglich, bringt aber normalerweise keine Vorteile.
Sofern nicht anders angegeben, sind die zur Herstellung der substituierten 3-Phenylurazile I, Ia und Ib benötigten Edukte und Reagenzien bekannt oder können nach an sich bekannten Methoden hergestellt werden.
Die Aufarbeitung der jeweiligen Reaktionsgemische erfolgt in der Regel nach an sich bekannten Methoden, beispielsweise durch Entfernen des Lösungsmittels, Verteilen des Rückstandes in einem Gemisch aus Wasser und einem geeigneten organischen Lösungsmittel und Isolieren des Produktes der organischen Phase.
Die substituierten 3-Phenylurazile können bei der Herstellung als Isomerengemische anfallen, die jedoch gewünschtenfalls nach den hierfür üblichen Methoden, z. B. durch Kristallisation oder Chromatographie an einem optisch aktiven Adsorbat, in die reinen Isomeren getrennt werden können. Reine optisch aktive Isomere lassen sich beispielsweise aus entsprechenden optisch aktiven Ausgangsmaterialien synthetisieren.
Die substituierten 3-Phenylurazile I, Ia und Ib eignen sich, sowohl als Isomerengemische als auch in Form der reinen Isomeren, als Herbizide. Im allgemeinen sind sie verträglich und somit selektiv in breitblättrigen Kulturen sowie in monokotylen (einkeimblättrigen) Gewächsen.
In Abhängigkeit von der jeweiligen Applikationsmethode können die substituierten Phenylurazile Ia und Ib bzw. sie enthaltende Mittel in einer Vielzahl von Kulturpflanzen zur Beseitigung unerwünschter Pflanzen eingesetzt werden, wobei die folgenden Kulturen beispielhaft genannt seien:
Botanischer Name
Deutscher Name
Allium cepa
Küchenzwiebel
Ananas comosus Ananas
Arachis hypogaea Erdnuß
Asparagus officinalis Spargel
Beta vulgaris spp. altissima Zuckerrübe
Beta vulgaris spp. rapa Futterrübe
Brassica napus var. napus Raps
Brassica napus var. napobrassica Kohlrübe
Brassica rapa var. silvestris Rüben
Camellia sinensis Teestrauch
Carthamus tinctorius Saflor - Färberdistel
Carya illinoinensis Pekannußbaum
Citrus limon Zitrone
Citrus sinensis Apfelsine, Orange
Coffea arabica (Coffea canephora, Coffea liberica) Kaffee
Cucumis sativus Gurke
Cynodon dactylon Bermudagras
Daucus carota Möhre
Elaeis guineensis Ölpalme
Fragaria vesca Erdbeere
Glycine max Sojabohne
Gossypium hirsutum (Gossypium arboreum, Gossypium herbaceum, Gossypium vitifolium) Baumwolle
Helianthus annuus Sonnenblume
Hevea brasiliensis Parakautschukbaum
Hordeum vulgare Gerste
Humulus lupulus Hopfen
Ipomoea batatas Süßkartoffeln
Juglans regia Walnußbaum
Lens culinaris Linse
Linum usitatissimum Faserlein
Lycopersicon lycopersicum Tomate
Malus spp. Apfel
Manihot esculenta Maniok
Medicago sativa Luzerne
Musa spp. Obst- und Mehlbanane
Nicotiana tabacum (N. rustica) Tabak
Olea europaea Ölbaum
Oryza sativa Reis
Phaseolus lunatus Mondbohne
Phaseolus vulgaris Buschbohnen
Picea abies Rotfichte
Pinus spp. Kiefer
Pisum sativum Gartenerbse
Prunus avium Süßkirsche
Prunus persica Pfirsich
Pyrus communis Birne
Ribes sylvestre Rote Johannisbeere
Ricinus communis Rizinus
Saccharum officinarum Zuckerrohr
Secale cereale Roggen
Solanum tuberosum Kartoffel
Sorghum bicolor (s. vulgare) Mohrenhirse
Theobroma cacao Kakaobaum
Trifolium pratense Rotklee
Triticum aestivum Weizen
Triticum durum Hartweizen
Vicia faba Pferdebohnen
Vitis vinifera Weinrebe
Zea mays Mais
Des weiteren eignen sich die substituierten 3-Phenylurazile I, Ia und Ib auch zur Desiccation und Defoliation von Pflanzen. Als Dessicantien eignen sie sich insbesondere zur Austrocknung der oberirdischen Teile von Kulturpflanzen wie Kartoffel, Raps, Sonnenblume und Sojabohne. Damit wird ein vollständig mechanisiertes Beernten dieser wichtigen Kulturpflanzen ermöglicht.
Von wirtschaftlichem Interesse ist ferner die Ernteerleichterung, die durch das zeitlich konzentrierte Abfallen oder Vermindern der Haftfestigkeit am Baum bei Zitrusfrüchten, Oliven oder bei anderen Arten und Sorten von Kern-, Stein- und Schalenobst ermöglicht wird. Derselbe Mechanismus, das heißt die Förderung der Ausbildung von Trenngewebe zwischen Frucht- bzw. Blatt- und Sproßteil der Pflanze ist auch für ein gut kontrollierbares Entblättern von Nutzpflanzen wie beispielsweise Baumwolle wesentlich.
Außerdem führt die Verkürzung des Zeitintervalls, in dem die einzelnen Baumwollpflanzen reif werden, zu einer erhöhten Faserqualität nach der Ernte.
Abgesehen von ihrer herbiziden und entblätternden Wirkung können einige der substituierten 3-Phenylurazile der Formeln I, Ia und Ib auch als Wachstumsregulatoren oder zur Bekämpfung von Schäd­ lingen aus der Klasse der Insekten, Spinnentiere und Nematoden eingesetzt werden. Sie können im Pflanzenschutz sowie auf dem Hygiene-, Vorratsschutz- und Veterinärsektor zur Bekämpfung von Schädlingen dienen.
Zu den schädlichen Insekten gehören aus der Ordnung der Schmetterlinge (Lepidoptera) beispielsweise Agrotis ypsilon, Agrotis segetum, Alambama argillacea, Anticarsia gemmatalis, Argyresthia conjugella, Autographa gamma, Bupalus piniarius, Cacoecia murinana, Capua reticulana, Cheimatobia brumata, Choristoneura fumiferana, Choristoneura occidentalis, Cirphis unipuncta, Cydia pomonella, Dendrolimus pini, Diaphania nitidalis, Diatracea grandiosella, Earias insulana, Elasmopalpus lignosellus, Eupoecilia ambiguella, Evetria bouliana, Feltia subterranea, Galleria mellonella, Grapholita funebrana, Grapholita molesta, Heliothis armigera, Heliothis virescens, Heliothis zea, Hellula undalis, Hibernia defoliaria, Hyphantria cunea, Hyponomeuta malinellus, Keifferia lycopersicella, Lambdina fiscellaria, Laphygma exigua, Leucoptera coffeella, Leucoptera scitella, Lithocolletis blancardella, Lobesia botrana, Loxostege sticticalis, Lymantria dispar, Lymantria monacha, Lyonetia clerkella, Malacosoma neustria, Mamestra brassicae, Orgyia pseudotsugata, Ostrinia nubilalis, Panolis flamea, Pectinophora gossypiella, Peridroma saucia, Phalera bucephala, Phthorimaea operculella, Phyllocnistis citrella, Pieris brassicae, Plathypena scarbra, Plutella xylostella, Pseudoplusia includens, Phyacionia frustrana, Scrobipalpula absoluta, Sitotroga cerelella, Sparganothis pilleriana, Spodoptera frugiperda, Spodoptera littoralis, Spodoptera litura, Thaumatopoea pityocampa, Tortrix viridana, Trichoplusia ni, Zeiraphera canadensis.
Aus der Ordnung der Käfer (Coleoptera) beispielsweise Agrilus sinuatus, Agriotes lineatus, Agriotes obscurus, Amphimallus solstitialis, Anisandrus dispar, Anthonomus grandis, Anthonomus pomorum, Atomaria linearis, Blastophagus piniperda, Blitophaga undata, Bruchus rufimanus, Bruchus pisorum, Bruchus lentis, Byctiscus betulae, Cassida nebulosa, Cerotoma trifurcata, Ceuthorrhynchus assimilis, Ceuthorrynchus napi, Chaetocnema tibialis, Conoderus vespertinus, Crioceris asparagi, Diabrotica longicornis, Diabrotica 12-punctata, Diabrotica virgifera, Epilachna varivestis, Epitrix hirtipennis, Eutinobothrus brasiliensis, Hylobius abietis, Hypera brunneipennis, Hypera postica, Ips typographus, Lema bilineata, Lema melanopus, Leptinotarsa decemlineata, Limonius californicus, Lissorhoptrus oryzophilus, Melanotus communis, Meligethes aeneus, Melolontha hippocastani, Melolontha melolontha, Onlema oryzae, Ortiorrhynchus sulcatus, Otiorrhynchus ovatus, Phaedon cochleariae, Phyllotreta chrysocephala, Phyllophaga sp., Phyllopertha horticola, Phyllotreta nemorum, Phyllotreta striolata, Popillia japonica, Sitona lineatus, Sitophilus granaria.
Aus der Ordnung der Zweiflügler (Diptera) beispielsweise Aedes aegypti, Aedes vexans, Anastrepha ludens, Anopheles maculipennis, Ceratitis capitata, Chrysomya bezziana, Chrysomya hominivorax, Chrysomya macellaria, Contarinia sorghicola, Cordylobia anthropophaga, Culex pipiens, Dacus cucurbitae, Dacus oleae, Dasineura brassicae, Fannia canicularis, Gasterophilus intestinalis, Glossia morsitans, Haematobia irritans, Haplodiplosis equestris, Hylemyia platura, Hypoderma lineata, Liriomyza sativae, Liriomyza trifolii, Lucilia caprina, Lucilia cuprina, Lucilia sericata, Lycoria pectoralis, Mayetiola destructor, Musca domestica, Muscina stabulans, Oestrus ovis, Oscinella frit, Pegomya hysocyami, Phorbia antiqua, Phorbia brassicae, Phorbia coarctata, Rhagoletis cerasi, Rhagoletis pomonella, Tabanus bovinus, Tipula oleracea, Tipula paludosa.
Aus der Ordnung der Thripse (Thysanoptera) beispielsweise Frankliniella fusca, Frankliniella occidentalis, Frankliniellla tritici, Scirtothrips citri, Thrips oryzae, Thrips palmi, Thrips tabaci.
Aus der Ordnung der Hautflügler (Hymenoptera) beispielsweise Athalia rosae, Atta cephalotes, Atta sexdens, Atta texana, Hoplocampa minuta, Hoplocampa testudinea, Monomorium pharaonis, Solenopsis geminata, Solenopsis invicta.
Aus der Ordnung der Wanzen (Heteroptera) beispielsweise Acrosterum hilare, Blissus leucopterus, Cyrtopeltis notatus Dysdercus cingulatus, Dysdercus intermedius, Eurygaster integriceps, Euchistus impictiventris, Leptoglossus phyllopus, Lygus lineolaris, Lygus pratensis, Nezara viridula, Piesma quadrata, Solubea insularis, Thyanta perditor.
Aus der Ordnung der Pflanzensauger (Homoptera) beispielsweise Acyrthosiphon onobrychis, Adelges laricis, Aphidula nasturtii, Aphis fabae, Aphis pomi, Aphis sambuci, Brachycaudus cardui, Brevicoryne brassicae, Cerosipha gossypii, Dreyfusia nordmannianae, Dreyfusia piceae, Dyasphis radicola, Dysaulacorthum pseudosolani, Empoasca fabae, Macrosiphum avenae, Macrosiphum euphorbiae, Macrosiphon rosae, Megoura viciae, Metopolophium dirhodum, Myzodes persicae, Myzus cerasi, Nilaparvata lugens, Pemphigus bursarius, Perkinsiella saccharicida, Phorodon humuli, Psylla mali, Psylla piri, Rhopalomyzus ascalonicus, Rhopalosiphum maidis, Sappaphis mala, Sappaphis mali, Schizaphis graminum, Schizoneura lanuginosa, Trialeurodes vaporariorum, Viteus vitifolii.
Aus der Ordnung der Termiten (Isoptera) beispielsweise Calotermes flavicollis, Leucotermes flavipes, Reticulitermes lucifugus, Termes natalensis.
Aus der Ordnung der Geradflügler (Orthoptera) beispielsweise Acheta domestica, Blatta orientalis, Blattella germanica, Forficula auricularia, Gryllotalpa gryllotalpa, Locusta migratoria, Melanoplus birittatus, Melanoplus femur-rubrum, Melanoplus mexicanus, Melanoplus sanguinipes, Melanoplus spretus, Nomadacris septemfasciata, Periplaneta americana, Schistocerca americana, Schistocerca peregrina, Stauronotus maroccanus, Tachycines asynamours.
Aus der Klasse der Arachnoidea beispielsweise Spinnentiere (Acarina) wie Amblyomma americanum, Amblyomma variegatum, Argas persicus, Boophilus annulatus, Boophilus decoloratus, Boophilus microplus, Brevipalpus phoenicis, Bryobia praetiosa, Dermacentor silvarum, Eotetranychus carpini, Eriophyes sheldoni, Hyalomma truncatum, Ixodus ricinus, Ixodus rubicundus, Ornithodorus moubata, Otobins megnini, Paratetranychus pilosus, Permanyssus gallinae, Phyllocaptrata oleivora, Polyphagotarsonemus latus, Psoroptes ovis, Rhipicephalus appendiculatus, Rhipicephalus evertsi, Saccoptes scabiei, Tetranychus cinnabarinus, Tetranychus kanzawai, Tetranychus pacificus, Tetranychus telarius, Tetranychus urticae.
Aus der Klasse der Nematoden beispielsweise Wurzelgallen­ nematoden, z. B. Meloidogyne hapla, Meloidogyne incognita, Meloidogyne javanica, Zysten bildende Nematoden, z. B. Globodera rostochiensis, Heterodera avenae, Heterodera glycinae, Heterodera schatii, Heterodera trifolii, Stock- und Blattälchen, z. B. Belonolaimus longicaudatus, Ditylenchus destructor, Ditylenchus dipsaci, Heliocotylenchus multicinctus, Longidorus elongatus, Radopholus similis, Rotylenchus robustus, Trichodorus primitivus, Tylenchorhynchus claytoni, Tylenchorhynchus dubius, Pratylenchus neglectus, Pratylenchus penetrans, Pratylenchus curvitatus, Pratylenchus goodeyi.
Die Wirkstoffe können als solche, in Form ihrer Formulierungen oder den daraus bereiteten Anwendungsformen, z. B. in Form von direkt versprühbaren Lösungen, Pulvern, Suspensionen oder Dispersionen, Emulsionen, Öldispersionen, Pasten, Stäubemitteln, Streumitteln, Granulaten durch Versprühen, Vernebeln, Verstäuben, Verstreuen oder Gießen angewendet werden. Die Anwendungsformen richten sich ganz nach den Verwendungszwecken; sie sollten in jedem Fall möglichst die feinste Verteilung der erfindungsgemäßen Wirkstoffe gewährleisten.
Die Formulierungen werden in bekannter Weise hergestellt, z. B. durch Verstecken des Wirkstoffs mit Lösungsmitteln und/oder Trägerstoffen, gewünschtenfalls unter Verwendung von Emulgier­ mitteln und Dispergiermitteln, wobei im Falle von Wasser als Verdünnungsmittel auch andere organische Lösungsmittel als Hilfslösungsmittel verwendet werden können. Als inerte Hilfs­ stoffe kommen dafür im wesentlichen in Betracht: Mineralölfrak­ tionen von mittlerem bis hohem Siedepunkt wie Kerosin und Diesel­ öl, ferner Kohlenteeröl sowie Öle pflanzlichen oder tierischen Ursprungs, Lösungsmittel wie Aromaten (z. B. Toluol, Xylol), chlorierte Aromaten (z. B. Chlorbenzole), Paraffine (z. B. Erdöl­ fraktionen), Alkohole (z. B. Methanol, Ethanol, Butanol, Cyclo­ hexanol), Ketone (z. B. Cyclohexanon, Isophoron), Amine (z. B. Ethanolamin, N,N-Dimethylformamid, N-Methylpyrrolidon) und Wasser; Trägerstoffe wie natürliche Gesteinsmehle (z. B. Kaoline, Tonerden, Talkum, Kreide) und synthetische Gesteinsmehle (z. B. hochdisperse Kieselsäure, Silikate); Emulgiermittel wie nicht- ionogene und anionische Emulgatoren (z. B. Polyoxyethylen-Fettalkohol- Ether, Alkylsulfonate und Arylsulfonate) und Dispergiermittel wie Ligninsulfitablaugen und Methylcellulose.
Wäßrige Anwendungsformen können aus Emulsionskonzentraten, Dispersionen, Pasten, netzbaren Pulvern oder wasserdispergierbaren Granulaten durch Zusatz von Wasser bereitet werden. Zur Herstellung von Emulsionen, Pasten oder Öldispersionen können die Substrate als solche oder in einem Öl oder Lösungsmittel gelöst, mittels Netz-, Haft-, Dispergier- oder Emulgiermittel in Wasser homogenisiert werden. Es können aber auch aus wirksamer Substanz, Netz-, Haft-, Dispergier- oder Emulgiermittel und eventuell Lösungsmittel oder Öl bestehende Konzentrate hergestellt werden, die zur Verdünnung mit Wasser geeignet sind.
Als oberflächenaktive Stoffe kommen die Alkali-, Erdalkali-, Ammoniumsalze von aromatischen Sulfonsäuren, z. B. Lignin-, Phenol-, Naphthalin- und Dibutylnaphthalinsulfonsäure, sowie von Fettsäuren, Alkyl- und Alkylarylsulfonaten, Alkyl-, Laurylether- und Fettalkoholsulfaten, sowie Salze sulfatierter Hexa-, Hepta- und Octadecanolen, sowie von Fettalkoholglykolether, Kondensationsprodukte von sulfoniertem Naphthalin und seiner Derivate mit Formaldehyd, Kondensationsprodukte des Naphthalins bzw. der Naphthalinsulfonsäuren mit Phenol und Formaldehyd, Polyoxyethylenoctylphenolether, ethoxyliertes Isooctyl-, Octyl- oder Nonylphenol, Alkylphenol-, Tributylphenylpolyglykolether, Alkylarylpolyetheralkohole, Isotridecylalkohol, Fettalkoholethylenoxid- Kondensate, ethoxyliertes Rizinusöl, Polyoxyethylenalkylether oder Polyoxypropylen, Laurylalkoholpolyglykoletheracetat, Sorbitester, Lignin-Sulfitablaugen oder Methylcellulose in Betracht.
Pulver-, Streu- und Stäubemittel können durch Mischen oder gemeinsames Vermahlen der wirksamen Substanzen mit einem festen Trägerstoff hergestellt werden.
Granulate, z. B. Umhüllungs-, Imprägnierungs- und Homogengranulate können durch Bindung der Wirkstoffe an feste Trägerstoffe hergestellt werden. Feste Trägerstoffe sind Mineralerden wie Silicagel, Kieselsäuren, Kieselgele, Silikate, Talkum, Kaolin, Kalkstein, Kalk, Kreide, Bolus, Löß, Ton, Dolomit, Diatomeenerde, Calcium- und Magnesiumsulfat, Magnesiumoxid, gemahlene Kunststoffe, Düngemittel, wie Ammoniumsulfat, Ammoniumphosphat, Ammoniumnitrat, Harnstoffe und pflanzliche Produkte, wie Getreidemehl, Baumrinden-, Holz- und Nußschalenmehl, Cellulosepulver oder andere feste Trägerstoffe.
Die Konzentrationen der Wirkstoffe I, Ia und Ib in den anwendungsfertigen Zubereitungen können in weiten Bereichen variiert werden, etwa zwischen 0,0001 und 95 Gew.-%. Für die Anwendung als Herbizide oder das Pflanzenwachstum regulierende Mittel empfehlen sich Konzentrationen zwischen 0,01 und 95 Gew.-%, vorzugsweise zwischen 0,5 und 90 Gew.-%, Wirkstoff. Für die Anwendung als Insektizide kommen Formulierungen mit 0,0001 bis 10 Gew.-%, vorzugsweise 0,01 bis 1 Gew.-% Wirkstoff, in Betracht. Die Wirkstoffe werden dabei in einer Reinheit von 90% bis 100%, vorzugsweise 95% bis 100% (nach NMR-Spektrum), eingesetzt.
Beispiele für solche Zubereitungen sind:
  • 1. eine Lösung aus 90 Gew.-Teilen der Verbindung Nr. 1.1 und 10 Gew.-Teilen N-Methyl-α-pyrrolidon, die zur Anwendung in Form kleinster Tropfen geeignet ist;
  • II. eine Mischung aus 20 Gew.-Teilen der Verbindung Nr. 1.2, 80 Gew.-Teilen Xylol, 10 Gew.-Teilen des Anlagerungsproduktes von 8 bis 10 Mol Ethylenoxid an 1 Mol Ölsäure-N-monoethanolamid, 5 Gew.-Teilen Calciumsalz der Dodecylbenzolsulfonsäure, 5 Gew.-Teilen des Anlagerungsproduktes und 40 Mol Ethylenoxid an 1 Mol Ricinusöl. Durch feines Verteilen des Gemisches in 100 000 Gew.-Teilen Wasser erhält man eine Dispersion, die 0,02 Gew.-% des Wirkstoffs enthält;
  • III. eine wäßrige Dispersion aus 20 Gew.-Teilen der Verbindung Nr. 3.1, 40 Gew.-Teilen Cyclohexanon, 30 Gew.- Teilen Isobutanol, 20 Gew.-Teilen des Anlagerungsproduktes von 40 mol Ethylenoxid an 1 mol Ricinusöl. Die Mischung dieser Dispersion mit 100 000 Gewichtsteilen Wasser enthält 0,02 Gew.-% des Wirkstoffes;
  • IV. eine wäßrige Dispersion aus 20 Gew.-Teilen der Verbindung Nr. 2.1, 25 Gew.-Teilen Cyclohexanol, 65 Gew.- Teilen einer Mineralölfraktion vom Siedepunkt 210 bis 280°C und 10 Gew.-Teilen des Anlagerungsproduktes von 40 mol Ethylenoxid an 1 mol Ricinusöl. Die Mischung dieser Dispersion mit 100 000 Gew.-Teilen Wasser enthält 0,02% des Wirkstoffes;
  • V. eine in einer Hammermühle vermahlene Mischung aus 80 Gew.-Teilen der Verbindung Nr. 3.1, 3 Gew.-Teilen des Natriumsalzes der Diisobutylnaphthalin-α-sulfonsäure, 10 Gew.-Teilen des Natriumsalzes einer Ligninsulfonsäure aus einer Sulfitablauge und 7 Gew.-Teilen pulverförmigem Kieselsäuregel. Durch feines Verteilen der Mischung in 20 000 Gew.-Teilen Wasser erhält man eine Spritzbrühe, die 0,1 Gew.-% des Wirkstoffs enthält;
  • VI. eine innige Mischung aus 3 Gew.-Teilen der Verbindung Nr. 3.2 und 97 Gew.-Teilen feinteiligem Kaolin. Dieses Stäubemittel enthält 3 Gew.-% Wirkstoff;
  • VII. eine innige Mischung aus 30 Gew.-Teilen der Verbindung Nr. 3.3, 92 Gew.-Teilen pulverförmigem Kieselsäuregel und 8 Gew.-Teilen Paraffinöl, das auf die Oberfläche dieses Kieselsäuregels gesprüht wurde. Diese Aufbereitung gibt dem Wirkstoff eine gute Haftfähigkeit;
  • VIII. eine stabile Dispersion aus 40 Gew.-Teilen der Verbindung Nr. 4.1, 10 Gew.-Teilen des Natriumsalzes eines Phenosulfonsäure-harnstoff-formaldehyd-Kondensates, 2 Gew.-Teilen Kieselgel und 48 Gew.-Teilen Wasser, die weiter verdünnt werden kann;
  • IX. eine stabile ölige Dispersion aus 20 Gew.-Teilen der Verbindung Nr. 1.1, 2 Gew.-Teilen des Calciumsalzes der Dodecylbenzolsulfonsäure, 8 Gew.-Teilen Fettalkoholpolyglykolether, 20 Gew.-Teilen des Natriumsalzes eines Phenolsulfonsäure-harnstoff-formaldehyd-Kondensates und 68 Gew.-Teilen eines paraffinischen Mineralöls;
  • X. eine in einer Hammermühle vermahlene Mischung aus 10 Gew.-Teilen der Verbindung Nr. 2.1, 4 Gew.-Teilen des Natriumsalzes der Diisobutylnaphthalin-α-sulfonsäure, 20 Gew.-Teilen des Natriumsalzes einer Ligninsulfonsäure aus einer Sulfitablauge, 38 Gew.-Teilen Kieselsäuregel und 38 Gew.-Teilen Kaolin. Durch feines Verteilen der Mischung in 10 000 Gew.-Teilen Wasser erhält man eine Spritzbrühe, die 0,1 Gew.-% des Wirkstoffs enthält.
Die Applikation der Wirkstoffe bzw. der herbiziden und das Pflanzenwachstum regulierenden Mittel kann im Vorauflauf- oder im Nachauflaufverfahren erfolgen. Normalerweise werden die Pflanzen mit den Wirkstoffen besprüht oder bestäubt oder die Samen der Testpflanzen mit den Wirkstoffen behandelt. Sind die Wirkstoffe für gewisse Kulturpflanzen weniger verträglich, so können Ausbringungstechniken angewandt werden, bei welchen die herbiziden Mittel mit Hilfe der Spritzgeräte so gespritzt werden, daß die Blätter der empfindlichen Kulturpflanzen nach Möglichkeit nicht getroffen werden, während die Wirkstoffe auf die Blätter darunter wachsender unerwünschter Pflanzen oder die unbedeckte Bodenfläche gelangen (post-directed, lay-by).
Die Aufwandmengen an Wirkstoff betragen je nach Bekämpfungsziel, Jahreszeit, Zielpflanzen und Wachstumsstadium 0,001 bis 5,0, vorzugsweise 0,01 bis 2 kg/ha aktive Substanz (a. S.).
Zur Verbreiterung des Wirkungsspektrums und zur Erzielung synergistischer Effekte können die substituierten 3-Phenylurazile I, Ia und Ib mit zahlreichen Vertretern anderer herbizider oder wachstumsregulierender Wirkstoffgruppen gemischt und gemeinsam ausgebracht werden. Beispielsweise kommen als Mischungspartner Diazine, 4H-3,1-Benzoxazinderivate, Benzothiadiazinone, 2,6-Dinitroaniline, N-Phenylcarbamate, Thiolcarbamate, Halogencarbonsäuren, Triazine, Amide, Harnstoffe, Diphenylether, Triazinone, Uracile, Benzofuranderivate, Cyclohexan-1,3-dionderivate, die in 2-Stellung z. B. eine Carboxy- oder Carbimino-Gruppe tragen, Chinolincarbonsäurederivate, Imidazolinone, Sulfonamide, Sulfonylharnstoffe, Aryloxy-, Heteroaryloxyphenoxypropionsäuren sowie deren Salze, Ester und Amide und andere in Betracht.
Die substituierten 3-Phenylurazile I, Ia und Ib können auch gemeinsam mit anderen Pflanzenschutzmitteln wie Herbiziden, Wachstumsregulatoren, Schädlingsbekämpfungsmittel, Fungiziden und Bakteriziden ausgebracht werden. Diese Mittel können zu den erfindungsgemäßen Mitteln im Gewichtsverhältnis 1 : 100 bis 100 : 1 zugemischt werden, gewünschtenfalls auch erst unmittelbar vor der Anwendung (Tankmix). Von Interesse ist ferner die Mischbarkeit mit Mineralsalzlösungen, welche zur Behebung von Ernährungs- und Spurenelementmängeln eingesetzt werden. Es können auch nicht- phytotoxische Öle und Ölkonzentrate zugesetzt werden.
Herstellungsbeispiele Beispiele 1 3-(4-Chlor-3-(2-chlor-2-ethoxycarbonyl-ethen-1-yl)-phenyl)-2,4- dioxo-6-trifluormethyl-1,2,3,4-tetrahydropyrimidin
Zu einer Suspension von 0,53 g Natriumhydrid in 100 ml Dimethylformamid wurde bei 0-5°C eine Lösung von 3,7 g 3-Amino-4,4,4-trifluor- crotonsäureethylester in 20 ml Toluol gegeben. Nach 30 Minuten rühren wurde die Mischung bei (-30) bis (-25)°C mit einer Lösung von 5,7 g 4-Chlor-3-(α-Chlor-acrylsäureethylester)-phenylisocyanat in 30 ml Toluol versetzt. Man rührte noch 5 Stunden bei etwa 20-25°C und hydrolysierte dann mit 150 ml Wasser. Anschließend neutralisierte man das Reaktionsgemisch mit 10gew.- %iger Salzsäure (pH=7), wonach die wäßrige Phase abgetrennt und zweimal mit je 100 ml Toluol extrahiert wurde. Die vereinigten organischen Phasen wurden dreimal mit je 10 ml Wasser gewaschen, über Natriumsulfat getrocknet und dann eingeengt. Das Rohprodukt wurde mit Diisopropylether verrührt, dann abgetrennt und mit Diisopropylether und Petrolether gewaschen.
Smp.: 202-206°C.
Vorstufe 4-Chlor-3-(α-Chlor-acrylsäureethylester)-phenylisocyanat
Zu einer Suspension von 26,0 g 4-Chlor-3-(α-Chlor-acrylsäureethylester)- anilin in 200 ml Toluol wurde eine Lösung von 13,2 ml Chlorameisensäuretrichlormethylester in 40 ml Toluol gegeben. Die Mischung wurde 14 Std. bei ca. 20-25°C und anschließend noch 10 Std. bei 90-95°C gerührt. Nach Abtrennen des gebildeten Niederschlags wurde das Lösungsmittel unter reduziertem Druck entfernt. Der Rückstand wurde im Hochvakuum getrocknet. Öl.
Analog wurde die folgende Verbindung synthetisiert:
3-(4-Chloro-3-(methoxyoximinomethyl)-phenyl)-2,4-dioxo-6-trifluormet-hyl- 1,2,3,4-tetrahydropyrimidin, Smp.: 221-223°C (Verbindung Nr. 1.2).
Beispiel 2 3-(4-Chloro-3-(1,3-dioxolan-2-yl)-phenyl)-2,4-dioxo-6-trifluormethyl-- 1,2,3,4-tetrahydropyrimidin
Zu einer Suspension von 7,3 g Natriumhydrid in 200 ml Dimethylformamid wurde bei 0 bis 5°C eine Mischung von 51,2 g 3-Amino- 4,4,4-trifluoro-crotonsäureethylester in 150 ml Toluol gegeben. Nach 30 Minuten Rühren versetzte man das Gemisch bei (-30) bis (-25)°C mit einer Lösung von 62,2 g 4-Chloro-3-(1,3-dioxolan-2- yl)-phenylisocyanat in 150 ml Toluol. Nach 5 Stunden Rühren bei ca. 20-25°C hydrolysierte man mit Wasser, wonach die Reaktionsmischung mit 10gew.-%iger Salzsäure neutral gewaschen wurde. Man extrahierte die wäßrige Phase dreimal mit je 100 ml Toluol. Die vereinigten organischen Phasen wurden dreimal mit je 50 ml Wasser gewaschen, dann über Natriumsulfat getrocknet und eingeengt. Das Rohprodukt wurde durch Flash-Chromatographie an Kieselgel (Laufmittel zu Methylenchlorid/Essigester 1 : 1) gereinigt.
Smp.: 180-182°C.
Vorstufe 4-Chloro-3-(1,3-dioxolan-2-yl)-phenylisocyanat
Zu einer Lösung von 3,0 g Chlorameisensäuretrichlormethylester in 50 ml Toluol wurden bei ca. 20-25°C 2,0 g 4-Chloro-3-(1,3-dioxolan- 2-yl)-anilin in 25 ml Essigsäureethylester gegeben. Diese Mischung wurde 2 Std. bei 20-25°C und anschließend noch 5 Std. bei Rückflußtemperatur gerührt. Anschließend engte man das Reaktionsgemisch ein und trocknete den Rückstand im Hochvakuum.
Ausbeute: 2,0 g (Öl).
Beispiel 3 3-(4-Chloro-3-(2-chloro-2-ethoxycarbonyl-ethen-1-yl)-phenyl)-2,4- dioxo-1-methyl-6-trifluoromethyl-1,2,3,4-tetrahydropyrimidin
Zu einer Suspension von 0,31 g Natriumhydrid in 100 ml Dimethylformamid wurde eine Lösung von 4,2 g 3-[4-Chloro-3-[2-chloro-2- ethoxy-carbonyl-ethen-1-yl]-phenyl]-2,4-dioxo-6-trifluormethyl- 1,2,3,4-tetrahydropyrimidin in 30 ml Dimethylformamid gegeben. Nach 1 Std. Rühren wurde eine Lösung von 1,70 g Methyliodid in 20 ml Dimethylformamid zugetropft. Nach 20 Std. Rühren bei etwa 20-25°C entfernte man unter reduziertem Druck die leichter flüchtigen Anteile des Reaktionsgemisches. Der ölige Rückstand wurde mit 150 ml Toluol aufgenommen und dreimal mit je 50 ml Wasser gewaschen, wonach man das Verdünnungsmittel trocknete und unter reduziertem Druck einengte. Das erhaltene Rohprodukt wurde mit Petrolether verrührt, dann wieder abgetrennt, getrocknet und aus Ethanol umkristallisiert. Smp.: 159-160°C.
Analog wurden die folgenden Verbindungen synthetisiert:
3-(4-Chloro-3-(methoxyoximinomethyl)-phenyl)-2,4-dioxo-1-methyl- 6-trifluoromethyl-1,2,3,4-tetrahydropyrimidin: Smp.: 132-134°C (Verbindung Nr. 3.2);
3-(4-Chloro-3-(1,3-dioxolan-2-yl)-phenyl)-2,4-dioxo-1-methyl-6- trifluoromethyl-1,2,3,4-tetrahydropyrimidin: Smp.: 58-60°C (Verbindung Nr. 3.3).
Beispiel 4 3-(4-Chlor-3-formyl-phenyl)-2,4-dioxo-1-methyl-6-trifluormethyl- 1,2,3,4-tetrahydropyrimidin
Zu einer Lösung von 1,9 g 3-(4-Chlor-3-(1,3-dioxolan-2-yl)- phenyl)-2,4-dioxo-1-methyl-6-trifluormethyl-1,2,3,4-tetrahydropyrimi-din in 45 ml Eisessig wurden 5 ml Wasser gegeben. Nach 12 Std. Rühren bei ca. 20-25°C und noch 5 Std. bei 40-50°C rührte man 150 ml in die Mischung. Danach wurde der gebildete Niederschlag abgetrennt, mit Wasser und Petrolether gewaschen und getrocknet. Smp.: 151-153°C.
Anwendungsbeispiele (herbizide Wirksamkeit)
Die herbizide Wirkung der substituierten Phenylurazile I, Ia und Ib ließ sich durch Gewächshausversuche zeigen:
Als Kulturgefäße dienten Plastikblumentöpfe mit lehmigem Sand mit etwa 3,0% Humus als Substrat. Die Samen der Testpflanzen wurden nach Arten getrennt eingesät.
Bei Vorauflaufbehandlung wurden die in Wasser suspendierten oder emulgierten Wirkstoffe direkt nach Einsaat mittels fein verteilender Düsen aufgebracht. Die Gefäße wurden leicht beregnet, um Keimung und Wachstum zu fördern und anschließend mit durchsichtigen Plastikhauben abgedeckt, bis die Pflanzen angewachsen waren. Diese Abdeckung bewirkt ein gleichmäßiges Keimen der Testpflanzen, sofern dies nicht durch die Wirkstoffe beeinträchtigt wurde.
Zum Zwecke der Nachauflaufbehandlung wurden die Testpflanzen bereits in den Versuchsgefäßen angezogen oder einige Tage vorher in die Versuchsgefäße verpflanzt. Die Applikation der in Wasser suspendierten oder emulgierten Wirkstoffe erfolgte je nach Wuchsform erst bei einer Wuchshöhe von 3 bis 15 cm.
Die Pflanzen wurden artenspezifisch bei Temperaturen von 10-25°C bzw. 20-35°C gehalten. Die Versuchsperiode erstreckte sich über 2 bis 4 Wochen. Während dieser Zeit wurden die Pflanzen gepflegt, und ihre Reaktion auf die einzelnen Behandlungen wurde ausgewertet.
Bewertet wurde nach einer Skala von 0 bis 100. Dabei bedeutet 100 kein Aufgang der Pflanzen bzw. völlige Zerstörung zumindest der oberirdischen Teile und 0 keine Schädigung oder normaler Wachstumsverlauf.
Die in den Gewächshausversuchen verwendeten Pflanzen setzten sich aus folgenden Arten zusammen:
Bei einer Aufwandmenge von 0,06 und 0,03 kg/ha lassen sich mit der Verbindung Nr. 3.1 unerwünschte breitblättrige Pflanzen im Nachauflaufverfahren sehr gut bekämpfen.
Anwendungsbeispiele (Defoliationswirkung)
Als Vergleichsmittel diente
A 6,7-Dihydrodipyridol(1,2-alpha:2′,1′-c)pyridilium als Dibromid-Monohydrat-Salz (Common Name: Diquat®).
Das Vergleichsmittel wurde in Form des fertig formulierten Handelsproduktes verwendet.
Als Testpflanzen dienten junge, 4blättrige (ohne Keimblätter) Baumwollpflanzen der Sorte Stoneville 825, die unter Gewächshausbedingungen angezogen wurden (rel. Luftfeuchtigkeit 50 bis 70%; Tag-/Nachttemperatur 27/20°C).
Anwendungsbeispiel 1
Die jungen Baumwollpflanzen wurden tropfnaß mit wäßrigen Aufbereitungen der angegebenen Wirkstoffe (unter Zusatz von 0,15 Gew.-% des Fettalkoholalkoxylats Plurafac LF 700, bezogen auf die Spritzbrühe) blattbehandelt. Die ausgebrachte Wassermenge betrug umgerechnet 1000 l/ha. Nach 13 Tagen wurde die Anzahl abgeworfener Blätter und der Grad der Entblätterung in % bestimmt. Bei den unbehandelten Kontrollpflanzen trat kein Blattfall auf.
Das Ergebnis zeigt, daß die erfindungsgemäßen substituierten 3-Phenylurazile I eine sehr gute entblätternde Wirkung aufweisen und hierbei dem Handelsprodukt A überlegen sind.
Anwendungsbeispiele (insektizide Wirksamkeit)
Die insektizide Wirkung der Verbindungen der allgemeinen Formel I, Ia und Ib ließ sich durch folgende Versuche zeigen:
Die Wirkstoffe wurden
  • a) als 0,1%ige Lösung in Aceton oder
  • b) als 10%ige Emulsion in einem Gemisch aus 70 Gew.-% Cyclohexanol, 20 Gew.-% Nekanil® LN (Lutensol® AP6, Netzmittel mit Emulgier- und Dispergierwirkung auf der Basis ethoxylierter Alkylphenole) und 10 Gew.-% Emulphor® EL (Emulan® EL, Emulgator auf der Basis ethoxylierter Fettalkohole)
aufbereitet und entsprechend der gewünschten Konzentration mit Aceton im Fall von a) bzw. mit Wasser im Fall von b) verdünnt.
Nach Abschluß der Versuche wurde die jeweils niedrigste Konzentration ermittelt, bei der die Verbindungen im Vergleich zu unbehandelten Kontrollversuchen noch eine 80-100%ige Hemmung bzw. Mortalität hervorriefen (Wirkschwelle bzw. Minimalkonzentration).

Claims (23)

1. Substituierte 3-Phenylurazile der allgemeinen Formel I in der die Variablen folgende Bedeutung haben:
X¹, X² Sauerstoff oder Schwefel;
W eine Gruppe -C(R⁸)=X⁵, -C(R⁸)(X³R⁶)(X⁴R⁷), -C(R⁸)=C(R⁹)-CO-R¹⁰,
-C(R⁸)-CH(R⁹)-CO-R¹⁰, -C(R⁸)=C(R⁹)-CH₂-CO-R¹⁰, -C(R⁸)=C(R⁹)-C(R¹¹)=C(R¹²)-CO-R¹⁰ oder
-C(R⁸)=C(R⁹)-CH₂-CH(R¹³)-CO-R¹⁰ mit
X³, X⁴ Sauerstoff oder Schwefel;
X⁵ Sauerstoff, Schwefel oder ein Rest -NR¹⁴, mit
R¹⁴ Wasserstoff, Hydroxyl, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₃-C₇-Cycloalkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆- Alkoxy, C₃-C₆-Alkenyloxy, C₃-C₆-Alkinyloxy, C₅-C₇-Cycloalkoxy, C₅-C₇-Cycloalkenyloxy, partiell oder vollständig halogeniertem C₁-C₆-Alkoxy, partiell oder vollständig halogeniertem C₃-C₆-Alkenyloxy, Hydroxy-C₁-C₆- alkoxy, Cyano-C₁-C₆-alkoxy, C₃-C₇-Cycloalkyl- C₁-C₆-alkoxy, C₁-C₆-Alkoxy-C₁-C₆-alkoxy, C₁-C₆-Alkoxy-C₃-C₆-alkenyloxy, C₁-C₆-Alkylcarbonyloxy, C₁-C₆-Alkoxycarbonyl- C₂-C₆-alkoxy, C₁-C₆-Alkylthio-C₁-C₆-alkoxy, Di-(C₁-C₆-alkyl)-amino-C₁-C₆-alkoxy, Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl, Phenyl-C₁-C₆-alkoxy, Phenyl-C₃-C₆-alkenyloxy oder Phenyl-C₃-C₆- alkinyloxy, wobei jeweils eine oder zwei Methylengruppen der Kohlenstoffketten durch -O-, -S- oder -N(C₁-C₆-Alkyl)- ersetzt sein können und wobei der Phenylring jeweils auch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl,
oder-N(R¹⁵)R¹⁶, wobei
R¹⁵, R¹⁶ Wasserstoff, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, C₃-C₆-Cycloalkyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxycarbonyl oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆- Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl, oder
R¹⁵ und R¹⁶ zusammen mit dem gemeinsamen Stickstoffatom einen gesättigten oder ungesättigten 4-7gliedrigen Heterocyclus, wobei ein Ringglied durch -O-, -S-, -N=, -NH- oder -N(C₁-C₆-Alkyl)- ersetzt sein kann,
bedeuten;
R⁶, R⁷ C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, C₁-C₆- Alkoxy-C₁-C₆-alkyl oder
R⁶ und R⁷ zusammen eine gesättigte oder ungesät­ tigte, zwei- bis viergliedrige Kohlenstoffkette, die einen Oxosubstituenten tragen kann, wobei ein Glied dieser Kette durch ein den Variablen X³ und X⁴ nicht benachbartes Sauerstoff-, Schwefel- oder Stickstoffatom ersetzt sein kann, und wobei die Kohlenstoffkette noch ein bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Amino, Halogen, C₁-C₆-Alkyl, C₂-C₆-Alkenyl, C₁-C₆-Alkoxy, C₃-C₆-Alkenyloxy, C₃-C₆-Alkinyloxy, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, Cyano-C₁-C₆-alkyl, Hydroxy-C₁-C₆-alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₃-C₆-Alkenyloxy-C₁-C₆-alkyl, C₃-C₆-Alkinyloxy- C₁-C₆-alkyl, Carboxy, C₁-C₆-Alkoxycarbonyl und C₁-C₆-Alkyl-carbonyloxy-C₁-C₆-alkyl;
R⁸ Wasserstoff, Cyano, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, partiell oder vollständig haloge­ niertes C₁-C₆-Alkyl, C₃-C₇-Cycloalkyl, C₁-C₆- Alkoxy-C₁-C₆-alkyl oder C₁-C₆-Alkoxycarbonyl;
R⁹, R¹² Wasserstoff, Cyano, Halogen, C₁-C₆-Alkyl, C₁-C₆- Alkoxy, Halogen-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl oder C₁-C₆-Alkoxycarbonyl;
R¹⁰ Wasserstoff, O-R¹⁷, S-R¹⁷, C₁-C₆-Alkyl, das noch einen oder zwei C₁-C₆-Alkoxysubstituenten tragen kann, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₃-C₇- Cycloalkyl, C₁-C₆-Alkylthio-C₁-C₆-alkyl, -N(R¹⁵)R¹⁶ oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆- Alkyl, C₃-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy oder C₁-C₆-Alkoxycarbonyl,
R¹⁷ bedeutet Wasserstoff, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₃-C₇-Cycloalkyl, partiell oder vollständig halogeniertes C₂-C₆-Alkyl, partiell oder vollständig halo­ geniertes C₃-C₆-Alkenyl, Cyano-C₁-C₆-alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl oder C₁-C₆-Alkyl­ oximino-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxycarbonyl oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxy­ carbonyl;
R¹¹ Wasserstoff, Cyano, Halogen, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxycarbonyl, -NR¹⁸R¹⁹, wobei R¹⁸ und R¹⁹ die Bedeutungen von R¹⁵ und R¹⁶ haben, oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogenier­ tem C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl;
R¹³ Wasserstoff, Cyano, C₁-C₆-Alkyl oder C₁-C₆-Alkoxy­ carbonyl;
R¹ Halogen, die Cyano-, Nitro- oder Trifluormethylgruppe;
R² Wasserstoff oder Halogen;
R³ Wasserstoff, eine C₁-C₆-Alkylgruppe, eine C₃-C₆-Alkenyl­ gruppe, eine C₃-C₆-Alkinylgruppe, eine C₃-C₈-Cycloalkyl­ gruppe, eine C₃-C₈-Cycloalkylcarbonylgruppe, eine C₁-C₆- Cyanoalkylgruppe, eine partiell oder vollständig haloge­ nierte C₁-C₆-Alkylgruppe, eine C₁-C₆-Alkoxy-C₁-C₆-alkyl­ gruppe, die Formylgruppe, eine C₁-C₆-Alkanoylgruppe, eine C₁-C₆-Alkoxycarbonylgruppe, eine partiell oder vollständig halogenierte C₁-C₆-Alkylcarbonylgruppe,
eine Gruppe -N(R²⁰)R²¹, wobei R²⁰ und R²¹ für eine der Bedeutungen von R¹⁵ und R¹⁶ stehen,
die Phenylgruppe oder eine Phenyl-C₁-C₆-alkylgruppe, wobei der Phenylring jeweils noch einen bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₂-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl;
R⁴ Wasserstoff, Cyano, Halogen, eine C₁-C₆-Alkylgruppe eine C₂-C₆-Alkenylgruppe, eine C₂-C₆-Alkinylgruppe, eine C₃-C₇- Cycloalkylgruppe, eine partiell oder vollständig haloge­ nierte C₁-C₆-Alkylgruppe, eine C₁-C₆-Hydroxyalkylgruppe, eine C₁-C₆-Cyanoalkylgruppe, eine C₁-C₆-Alkoxy-C₁-C₆-alkyl­ gruppe, eine C₁-C₆-Alkylthio-C₁-C₆-alkylgruppe oder die Phenylgruppe, die noch einen bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₁-C₆-Alkenyl, partiell oder voll­ ständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl;
R⁵ Wasserstoff, Cyano, Nitro, Halogen, eine C₁-C₆-Alkylgruppe, eine C₂-C₆-Alkenylgruppe, eine C₂-C₆-Alkinylgruppe, eine C₃-C₇-Cycloalkylgruppe, eine partiell oder vollständig halo­ genierte C₁-C₆-Alkylgruppe, eine C₁-C₆-Hydroxyalkylgruppe, eine C₁-C₆-Cycloalkylgruppe, eine C₁-C₆-Alkoxy-C₁-C₆-alkyl­ gruppe, eine C₁-C₆-Alkylthio-C₁-C₆-alkylgruppe, die Formyl­ gruppe, eine C₁-C₆-Alkylcarbonylgruppe, eine partiell oder vollständig halogenierte C₁-C₆-Alkylcarbonylgruppe, eine C₁-C₆-Alkoxycarbonylgruppe, eine Gruppe -N(R²²)R²³, wobei R²² und R²³ für eine der Bedeutungen von R¹⁵ und R¹⁶ stehen, die Phenylgruppe, die noch einen bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₂-C₆-Alkenyl, partiell oder voll­ ständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl, oder
R⁴ und R⁵ zusammen eine gesättigte oder ungesättigte 3- oder 4gliedrige Kohlenstoffkette, die gewünschtenfalls ein bis drei Heteroatome als Glieder enthalten kann, ausgewählt aus einer Gruppe bestehend aus 1 oder 2 Sauerstoffatomen, 1 oder 2 Schwefelatomen und 1 bis 3 Stickstoffatomen, wobei die Kette noch ein bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Amino, Halogen, C₁-C₆-Alkyl, C₂-C₆-Alkenyl, C₁-C₆-Alkoxy, C₁-C₆-Alkylthio und C₁-C₆-Alkoxycarbonyl;
mit der Maßgabe, daß nicht gleichzeitig R⁴ die Trifluor­ methylgruppe R⁵ Wasserstoff sein können, wenn W eine Gruppe -CH=CH-CO-R¹⁰ mit R¹⁰ C₁-C₆-Alkoxy oder C₃-C₇-Cycloalkoxy bedeutet,
sowie die Salze und Enolether derjenigen Verbindungen I, bei denen R³ Wasserstoff bedeutet.
2. Verbindungen der allgemeinen Formeln Ia oder Ib in denen die Variablen folgende Bedeutung haben:
X¹, X² Sauerstoff oder Schwefel;
W eine Gruppe -C(R⁸)=X⁵, -C(R⁸)(X³R⁶)(X⁴R⁷),
-C(R⁸)=C(R⁹)-CO-R¹⁰,
-CH(R⁸)-CH(R⁹)-CO-R¹⁰,
-C(R⁸)=C(R⁹)-CH₂-CO-R¹⁰, -C(R⁸)=C(R⁹)-C(R¹¹)=C(R¹²)-CO-R¹⁰ oder
-C(R⁸)=C(R⁹)-CH₂-CH(R¹³)-CO-R¹⁰ mit
X³, X⁴ Sauerstoff oder Schwefel;
X⁵ Sauerstoff, Schwefel oder ein Rest -NR₁₄, mit
R¹⁴ Wasserstoff, Hydroxyl, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₃-C₇-Cycloalkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆- Alkoxy, C₃-C₆-Alkenyloxy, C₃-C₆-Alkinyloxy, C₅-C₇-Cycloalkoxy, C₅-C₇-Cycloalkenyloxy, partiell oder vollständig halogeniertem C₁-C₆-Alkoxy, partiell oder vollständig halo­ geniertem C₃-C₆-Alkenyloxy, Hydroxy-C₁-C₆- alkoxy, Cyano-C₁-C₆-alkoxy, C₃-C₇-Cycloalkyl- C₁-C₆-alkoxy, C₁-C₆-Alkoxy-C₁-C₆-alkoxy, C₁-C₆-Alkoxy-C₃-C₆-alkenyloxy, C₁-C₆-Alkyl­ carbonyloxy, C₁-C₆-Alkoxycarbonyl-C₂-C₆- alkoxy, C₁-C₆-Alkylthio-C₁-C₆-alkoxy, Di-(C₁-C₆-alkyl)-amino-C₁-C₆-alkoxy, Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl, Phenyl-C₁-C₆-alkoxy, Phenyl-C₃-C₆-alkenyloxy oder Phenyl-C₃-C₆- alkinyloxy, wobei jeweils eine oder zwei Methylengruppen der Kohlenstoffketten durch -O-, -S-, oder -N(C₁-C₆-Alkyl)- ersetzt sein können und wobei der Phenylring jeweils auch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, partiell oder vollständig haloge­ niertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl,
oder -N(R¹⁵)R¹⁶, wobei
R¹⁵, R¹⁶ Wasserstoff, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, C₃-C₆-Cycloalkyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆-Alkyl­ carbonyl, C₁-C₆-Alkoxycarbonyl oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, par­ tiell oder vollständig halogeniertem C₁-C₆- Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl, oder
R¹⁵ und R¹⁶ zusammen mit dem gemeinsamen Stickstoffatom einen gesättigten oder unge­ sättigten 4-7gliedrigen Heterocyclus, wobei ein Ringglied durch -O-, -S-, -N=, -NH- oder -N(C₁-C₆-Alkyl)- ersetzt sein kann,
bedeuten;
R⁶, R⁷ C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, C₁-C₆- Alkoxy-C₁-C₆-alkyl oder
R⁶ und R⁷ zusammen eine gesättigte oder ungesät­ tigte, zwei- bis viergliedrige Kohlenstoffkette, die einen Oxosubstituenten tragen kann, wobei ein Glied dieser Kette durch ein den Variablen X³ und X⁴ nicht benachbartes Sauerstoff-, Schwefel- oder Stickstoffatom ersetzt sein kann, und wobei die Kohlenstoffkette noch ein bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Amino, Halogen, C₁-C₆-Alkyl, C₂-C₆- Alkenyl, C₁-C₆-Alkoxy, C₃-C₆-Alkenyloxy, C₃-C₆- Alkinyloxy, partiell oer vollständig halogenier­ tem C₁-C₆-Alkyl, Cyano-C₁-C₆-alkyl, Hydroxy-C₁-C₆- alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₃-C₆-Alkenyl­ oxy-C₁-C₆-alkyl, C₃-C₆-Alkinyloxy-C₁-C₆-alkyl, Carboxy, C₁-C₆-Alkoxycarbonyl und C₁-C₆-Alkyl- carbonyloxy-C₁-C₆-alkyl;
R⁸ Wasserstoff, Cyano, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, partiell oder vollständig haloge­ niertes C₁-C₆-Alkyl, C₃-C₇-Cycloalkyl, C₁-C₆- Alkoxy-C₁-C₆-alkyl oder C₁-C₆-Alkoxycarbonyl
R⁹, R¹² Wasserstoff, Cyano, Halogen, C₁-C₆-Alkyl, C₁-C₆- Alkoxy, Halogen-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl oder C₁-C₆-Alkoxycarbonyl;
R¹⁰ Wasserstoff, O-R¹⁷, S-R¹⁷, C₁-C₆-Alkyl, das noch einen oder zwei C₁-C₆-Alkoxysubstituenten tragen kann, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₃-C₇- Cycloalkyl, C₁-C₆-Alkylthio-C₁-C₆-alkyl,
-N(R¹⁵)R¹⁶ oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆- Alkyl, C₃-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy oder C₁-C₆-Alkoxycarbonyl,
R¹⁷ bedeutet Wasserstoff, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₃-C₇-Cycloalkyl, partiell oder vollständig halogeniertes C₂-C₆-Alkyl, partiell oder vollständig halogeniertes C₃-C₆-Alkenyl, Cyano-C₁-C₆- alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl oder C₁-C₆- Alkyl-oximino-C₁-C₆-alkyl, C₁-C₆-Alkyl- carbonyl, C₁-C₆-Alkoxycarbonyl oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl;
R¹¹ Wasserstoff, Cyano, Halogen, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxycarbonyl, -NR¹⁸R¹⁹, wobei R¹⁸ und R¹⁹ die Bedeutungen von R¹⁵ und R¹⁶ haben, oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyanon, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogenier­ tem C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl;
R¹³ Wasserstoff, Cyano, C₁-C₆-Alkyl oder C₁-C₆-Alkoxy­ carbonyl;
R¹ Halogen, die Cyano-, Nitro- oder Trifluormethylgruppe;
R² Wasserstoff oder Halogen;
R³′ eine C₁-C₆-Alkylgruppe, eine C₃-C₆-Alkenylgruppe oder eine C₃-C₆-Alkinylgruppe;
R⁴ Wasserstoff, Cyano, Halogen, eine C₁-C₆-Alkylgruppe, eine C₂-C₆-Alkenylgruppe, eine C₂-C₆-Alkinylgruppe, eine C₃-C₈- Cycloalkylgruppe, eine partiell oder vollständig halogenierte C₁-C₆-Alkylgruppe, eine C₁-C₆-Hydroxyalkylgruppe, eine C₁-C₆-Cyanoalkylgruppe, eine C₁-C₆-Alkoxy-C₁-C₆-alkylgruppe, eine C₁-C₆-Alkylthio-C₁-C₆-alkylgruppe oder die Phenylgruppe, die noch einen bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₂-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl;
R⁵ Wasserstoff, Cyano, Nitro, Halogen, eine C₁-C₆-Alkylgruppe, eine C₂-C₆-Alkenylgruppe, eine C₂-C₆-Alkinylgruppe, eine C₃-C₇-Cycloalkylgruppe, eine partiell oder vollständig halogenierte C₁-C₆-Alkylgruppe, eine C₁-C₆--Hydroxyalkylgruppe, eine C₁-C₆-Cyanoalkylgruppe, eine C₁-C₆-Alkoxy-C₁-C₆-alkylgruppe, eine C₁-C₆-Alkylthio-C₁-C₆-alkylgruppe, die Formylgruppe, eine C₁-C₆-Alkylcarbonylgruppe, eine partiell oder vollständig halogenierte C₁-C₆-Alkylcarbonylgruppe, eine C₁-C₆-Alkoxycarbonylgruppe, eine Gruppe äN(R²²)R²³, wobei R²² und R²³ für eine der Bedeutungen von R¹⁵ und R¹⁶ stehen, die Phenylgruppe, die noch einen bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₂-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl, oder
R⁴ und R⁵ zusammen eine gesättigte oder ungesättigte 3- oder 4gliedrige Kohlenstoffkette, die ein bis drei Heteroatome als Glieder enthalten kann, ausgewählt aus einer Gruppe bestehend aus 1 oder 2 Sauerstoffatomen, 1 oder 2 Schwefelatomen und 1 bis 3 Stickstoffatomen, wobei die Kette noch ein bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Amino, Halogen, C₁-C₆-Alkyl, C₂-C₆-Alkenyl, C₁-C₆-Alkoxy, C₁-C₆-Alkylthio und C₁-C₆- Alkoxycarbonyl;
mit der Maßgabe, daß nicht gleichzeitig R⁴ die Trifluormethylgruppe R⁵ Wasserstoff sein können, wenn W eine Gruppe -CH=CH-CO-R¹⁰ mit R¹⁰ C₁-C₆-Alkoxy oder C₃-C₆-Cycloalkoxy bedeutet.
3. Verbindungen nach Anspruch 1 oder 2, wobei W die Cyanogruppe, eine Gruppe -C(R⁸)=X⁵, -C(R⁸)(X³R⁶)(X⁴R⁷), -C(R⁸)=C(R⁹)-CO-R¹⁰ oder -CH(R⁸)-CH(R⁹)-CO-R¹⁰ bedeutet.
4. Verbindungen nach Anspruch 1 oder 2, wobei R¹ Wasserstoff oder eine C₁-C₆-Alkylgruppe bedeutet.
5. Verbindungen nach Anspruch 1 oder 2, wobei R¹ Wasserstoff oder Fluor bedeutet.
6. Verbindungen nach Anspruch 1 oder 2, wobei R² Chlor oder Brom bedeutet.
7. Verbindungen nach Anspruch 1 oder 2, wobei R³ eine C₁-C₆- Alkylgruppe bedeutet.
8. Verbindungen nach Anspruch 1 oder 2, wobei R⁴ eine partiell oder vollständig halogenierte C₁-C₆-Alkylgruppe bedeutet.
9. Enamin-Ester der allgemeinen Formel II in der die Variablen folgende Bedeutung haben:
L¹ eine C₁-C₆-Alkylgruppe oder die Phenylgruppe;
X¹ Sauerstoff oder Schwefel;
W eine Gruppe -C(R⁸)=X⁵, -C(R⁸)(X³R⁶)(X⁴R⁷), -C(R⁸)=C(R⁹)-CO-R¹⁰,
-CH(R⁸)-CH(R⁹)-CO-R¹⁰, -C(R⁸)=C(R⁹)-CH₂-CO-R¹⁰, -C(R⁸)=C(R⁹)-C(R¹¹)=C(R¹²)-CO-R¹⁰ oder
-C(R⁸)=C(R⁹)-CH₂-CH(R¹³)-CO-R¹⁰ mit
X³, X⁴ Sauerstoff oder Schwefel;
X⁵ Sauerstoff, Schwefel oder ein Rest -NR¹⁴, mit
R¹⁴ Wasserstoff, Hydroxyl, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₃-C₇-Cycloalkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆- Alkoxy, C₃-C₆-Alkenyloxy, C₃-C₆-Alkinyloxy, C₅-C₇-Cycloalkoxy, C₅-C₇-Cycloalkenyloxy, partiell oder vollständig halogeniertem C₁-C₆-Alkoxy, partiell oder vollständig halogeniertem C₃-C₆-Alkenyloxy, Hydroxy-C₁-C₆- alkoxy, Cyano-C₁-C₆-alkoxy, C₃-C₇-Cycloalkyl- C₁-C₆-alkoxy, C₁-C₆-Alkoxy-C₁-C₆-alkoxy, C₁-C₆-Alkoxy-C₃-C₆-alkenyloxy, C₁-C₆-Alkylcarbonyloxy, C₁-C₆-Alkoxycarbonyl-C₂-C₆- alkoxy, C₁-C₆-Alkylthio-C₁-C₆-alkoxy, Di-(C₁-C₆-alkyl)-amino-C₁-C₆-alkoxy, Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl, Phenyl-C₁-C₆-alkoxy, Phenyl-C₃-C₆-alkenyloxy oder Phenyl-C₃-C₆- alkinyloxy, wobei jeweils eine oder zwei Methylengruppen der Kohlenstoffketten durch -O-, -S- oder -N(C₁-C₆-Alkyl)- ersetzt sein können und wobei der Phenylring jeweils auch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl,
oder -N(R¹⁵)R¹⁶, wobei
R¹⁵, R¹⁶ Wasserstoff, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, C₃-C₆-Cycloalkyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxycarbonyl oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆- Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl, oder
R¹⁵ und R¹⁶ zusammen mit dem gemeinsamen Stickstoffatom einen gesättigten oder ungesättigten 4-7gliedrigen Heterocyclus, wobei ein Ringglied durch -O-, -S-, -N=, -NH- oder -N(C₁-C₆-Alkyl)- ersetzt sein kann,
bedeuten;
R⁶, R⁷ C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, C₁-C₆- Alkoxy-C₁-C₆-alkyl oder
R⁶ und R⁷ zusammen eine gesättigte oder ungesättigte, zwei- bis viergliedrige Kohlenstoffkette, die einen Oxosubstituenten tragen kann, wobei ein Glied dieser Kette durch ein den Variablen X³ und X⁴ nicht benachbartes Sauerstoff-, Schwefel- oder Stickstoffatom ersetzt sein kann, und wobei die Kohlenstoffkette noch ein bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Amino, Halogen, C₁-C₆-Alkyl, C₂-C₆- Alkenyl, C₁-C₆-Alkoxy, C₃-C₆-Alkenyloxy, C₃-C₆- Alkinyloxy, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, Cyano-C₁-C₆-alkyl, Hydroxy-C₁-C₆- alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₃-C₆-Alkenyloxy- C₁-C₆-alkyl, C₃-C₆-Alkinyloxy-C₁-C₆-alkyl, Carboxy, C₁-C₆-Alkoxycarbonyl und C₁-C₆-Alkylcarbonyloxy- C₁-C₆-alkyl;
R⁸ Wasserstoff, Cyano, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₃-C₇-Cycloalkyl, C₁-C₆- Alkoxy-C₁-C₆-alkyl oder C₁-C₆-Alkoxycarbonyl;
R⁹, R¹² Wasserstoff, Cyano, Halogen, C₁-C₆-Alkyl, C₁-C₆- Alkoxy, Halogen-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl oder C₁-C₆-Alkoxycarbonyl;
R¹⁰ Wasserstoff, O-R¹⁷, S-R¹⁷, C₁-C₆-Alkyl, das noch einen oder zwei C₁-C₆-Alkoxysubstituenten tragen kann, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₃-C₇- Cycloalkyl, C₁-C₆-Alkylthio-C₁-C₆-alkyl, -N(R¹⁵)R¹⁶ oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆- Alkyl, C₃-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy oder C₁-C₆-Alkoxycarbonyl,
R¹⁷ bedeutet Wasserstoff, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₃-C₇-Cycloalkyl, partiell oder vollständig halogeniertes C₂-C₆-Alkyl, partiell oder vollständig halogeniertes C₃-C₆-Alkenyl, Cyano-C₁-C₆- alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl oder C₁-C₆- Alkyl-oximino-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxycarbonyl oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl;
R¹¹ Wasserstoff, Cyano, Halogen, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxycarbonyl, -NR¹⁸R¹⁹, wobei R¹⁸ und R¹⁹ die Bedeutungen von R¹⁵ und R¹⁶ haben, oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl;
R¹³ Wasserstoff, Cyano, C₁-C₆-Alkyl oder C₁-C₆-Alkoxycarbonyl;
R¹ Halogen, die Cyano-, Nitro- oder Trifluormethylgruppe;
R² Wasserstoff oder Halogen;
R³ Wasserstoff, eine C₁-C₆-Alkylgruppe, eine C₃-C₆-Alkenylgruppe, eine C₃-C₆-Alkinylgruppe, eine C₃-C₈-Cycloalkylgruppe, eine C₃-C₈-Cycloalkylcarbonylgruppe, eine C₁-C₆- Cyanoalkylgruppe, eine partiell oder vollständig halogenierte C₁-C₆-Alkylgruppe, eine C₁-C₆-Alkoxy-C₁-C₆-alkylgruppe, die Formylgruppe, eine C₁-C₆-Alkanoylgruppe, eine C₁-C₆-Alkoxycarbonylgruppe, eine partiell oder vollständig halogenierte C₁-C₆-Alkylcarbonylgruppe,
eine Gruppe -N(R¹⁰)R²¹, wobei R²⁰ und R²¹ für eine der Bedeutungen von R¹⁵ und R¹⁶ stehen,
die Phenylgruppe oder eine Phenyl-C₁-C₆-alkylgruppe, wobei der Phenylring jeweils noch einen bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₂-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl;
R⁴ Wasserstoff, Cyano, Halogen, eine C₁-C₆-Alkylgruppe, eine C₂-C₆-Alkenylgruppe, eine C₂-C₆-Alkinylgruppe, eine C₃-C₇- Cycloalkylgruppe, eine partiell oder vollständig halogenierte C₁-C₆-Alkylgruppe, eine C₁-C₆-Hydroxyalkylgruppe, eine C₁-C₆-Cyanoalkylgruppe, eine C₁-C₆-Alkoxy-C₁-C₆-alkylgruppe, eine C₁-C₆-Alkylthio-C₁-C₆-alkylgruppe oder die Phenylgruppe, die noch einen bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₂-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl;
R⁵ Wasserstoff, Cyano, Nitro, Halogen, eine C₁-C₆-Alkylgruppe, eine C₂-C₆-Alkenylgruppe, eine C₂-C₆-Alkinylgruppe, eine C₃-C₇-Cycloalkylgruppe, eine partiell oder vollständig halogenierte C₁-C₆-Alkylgruppe, eine C₁-C₆-Hydroxyalkylgruppe, eine C₁-C₆-Cyanoalkylgruppe, eine C₁-C₆-Alkoxy-C₁-C₆-alkylgruppe, eine C₁-C₆-Alkylthio-C₁-C₆-alkylgruppe, die Formylgruppe, eine C₁-C₆-Alkylcarbonylgruppe, eine partiell oder vollständig halogenierte C₁-C₆-Alkylcarbonylgruppe, eine C₁-C₆-Alkoxycarbonylgruppe, eine Gruppe -N(R²²)R²³, wobei R²² und R²³ für eine der Bedeutungen von R¹⁵ und R¹⁶ stehen, die Phenylgruppe, die noch einen bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₂-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl, oder
R⁴ und R⁵ zusammen eine gesättigte oder ungesättigte 3- oder 4gliedrige Kohlenstoffkette, die ein bis drei Heteroatome als Glieder enthalten kann, ausgewählt aus einer Gruppe bestehend aus 1 oder 2 Sauerstoffatomen, 1 oder 2 Schwefelatomen und 1 bis 3 Stickstoffatomen, wobei die Kohlenstoffkette noch ein bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Amino, Halogen, C₁-C₆-Alkyl, C₂-C₆-Alkenyl, C₁-C₆-Alkoxy, C₁-C₆-Alkylthio und C₁-C₆-Alkoxycarbonyl.
10. Enamin-Carboxylate der allgemeinen Formel III in der die Variablen folgende Bedeutung haben:
L¹ eine C₁-C₆-Alkylgruppe oder die Phenylgruppe;
X² Sauerstoff oder Schwefel;
W eine Gruppe -C(R⁸)=X⁵, -C(R⁸)(X³R⁶)(X⁴R⁷), -C(R⁸)=C(R⁹)-CO-R¹⁰,
-CH(R⁸)-CH(R⁹)-CO-R¹⁰, -C(R⁸)=C(R⁹)-CH₂-CO-R¹⁰, -C(R⁸)=C(R⁹)-C(R¹¹)=C(R¹²)-CO-R¹⁰ oder
-C(R⁸)=C(R⁹)-CH₂-CH(R¹³)-CO-R¹⁰ mit
X³, X⁴ Sauerstoff oder Schwefel;
X⁵ Sauerstoff, Schwefel oder ein Rest -NR¹⁴, mit
R¹⁴ Wasserstoff, Hydroxyl, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₃-C₇-Cycloalkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆- Alkoxy, C₃-C₆-Alkenyloxy, C₃-C₆-Alkinyloxy, C₅-C₇-Cycloalkoxy, C₅-C₇-Cycloalkenyloxy, partiell oder vollständig halogeniertem C₁-C₆-Alkoxy, partiell oder vollständig halogeniertem C₃-C₆-Alkenyloxy, Hydroxy-C₁-C₆- alkoxy, Cyano-C₁-C₆-alkoxy, C₃-C₇-Cycloalkyl- C₁-C₆-alkoxy, C₁-C₆-Alkoxy-C₁-C₆-alkoxy, C₁-C₆-Alkoxy-C₃-C₆-alkenyloxy, C₁-C₆-Alkylcarbonyloxy, C₁-C₆-Alkoxycarbonyl-C₂-C₆-alkoxy, C₁-C₆-Alkylthio-C₁-C₆-alkoxy, Di-(C₁-C₆- alkyl)-amino-C₁-C₆-alkoxy, Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl, Phenyl-C₁-C₆-alkoxy, Phenyl- C₃-C₆-alkenyloxy oder Phenyl-C₃-C₆-alkinyloxy, wobei jeweils eine oder zwei Methylengruppen der Kohlenstoffketten durch -O-, -S- oder -N(C₁-C₆-Alkyl)- ersetzt sein können und wobei der Phenylring jeweils auch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl,
oder -N(R¹⁵)R¹⁶, wobei
R¹⁵, R¹⁶ Wasserstoff, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, C₃-C₆-Cycloalkyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxycarbonyl oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆- Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl, oder
R¹⁵ und R¹⁶ zusammen mit dem gemeinsamen Stickstoffatom einen gesättigten oder ungesättigten 4-7gliedrigen Heterocyclus, wobei ein Ringglied durch -O-, -S-, -N=, -NH- oder -N(C₁-C₆-Alkyl)- ersetzt sein kann,
bedeuten;
R⁶, R⁷ C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, C₁-C₆- Alkoxy-C₁-C₆-alkyl oder
R⁶ und R⁷ zusammen eine gesättigte oder ungesättigte, zwei bis viergliedrige Kohlenstoffkette, die einen Oxosubstituenten tragen kann, wobei ein Glied dieser Kette durch ein den Variablen X³ und X⁴ nicht benachbartes Sauerstoff-, Schwefel- oder Stickstoffatom ersetzt sein kann, und wobei die Kohlenstoffkette noch ein bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Amino, Halogen, C₁-C₆-Alkyl, C₂-C₆- Alkenyl, C₁-C₆-Alkoxy, C₃-C₆-Alkenyloxy, C₃-C₆- Alkinyloxy, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, Cyano-C₁-C₆-alkyl, Hydroxy-C₁-C₆- alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₃-C₆-Alkenyloxy- C₁-C₆-alkyl, C₃-C₆-Alkinyloxy-C₁-C₆-alkyl, Carboxy, C₁-C₆-Alkoxycarbonyl und C₁-C₆-Alkylcarbonyloxy- C₁-C₆-alkyl;
R⁸ Wasserstoff, Cyano, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, partiell oder vollständig halogenisiertes C₁-C₆-Alkyl, C₃-C₇-Cycloalkyl, C₁-C₆- Alkoxy-C₁-C₆-alkyl oder C₁-C₆-Alkoxycarbonyl;
R⁹, R¹² Wasserstoff, Cyano, Halogen, C₁-C₆-Alkyl, C₁-C₆- Alkoxy, Halogen-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl oder C₁-C₆-Alkoxycarbonyl;
R¹⁰ Wasserstoff, O-R¹⁷, S-R¹⁷, C₁-C₆-Alkyl, das noch einen oder zwei C₁-C₆-Alkoxysubstituenten tragen kann, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₃-C₇- Cycloalkyl, C₁-C₆-Alkylthio-C₁-C₆-alkyl, -N(R¹⁵)R¹⁶ oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆- Alkyl, C₃-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy oder C₁-C₆-Alkoxycarbonyl,
R¹⁷ bedeutet Wasserstoff, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₃-C₆-Cycloalkyl, partiell oder vollständig halogeniertes C₂-C₆-Alkyl, partiell oder vollständig halogeniertes C₃-C₆-Alkenyl, Cyano-C₁-C₆- alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl oder C₁-C₆- Alkyl-oximino-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxycarbonyl oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl;
R¹¹ Wasserstoff, Cyano, Halogen, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxycarbonyl, -NR¹⁸R¹⁹, wobei R¹⁸ und R¹⁹ die Bedeutungen von R¹⁵ und R¹⁶ haben, oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl;
R¹³ Wasserstoff, Cyano, C₁-C₆-Alkyl oder C₁-C₆-Alkoxycarbonyl;
R¹ Halogen, die Cyano-, Nitro- oder Trifluormethylgruppe;
R² Wasserstoff oder Halogen;
R⁴ Wasserstoff, Cyano, Halogen, eine C₁-C₆-Alkylgruppe, eine C₂-C₆-Alkenylgruppe, eine C₂-C₆-Alkinylgruppe, eine C₃-C₇- Cycloalkylgruppe, eine partiell oder vollständig halogenierte C₁-C₆-Alkylgruppe, eine C₁-C₆-Hydroxyalkylgruppe, eine C₁-C₆-Cyanoalkylgruppe, eine C₁-C₆-Alkoxy-C₁-C₆-alkylgruppe, eine C₁-C₆-Alkylthio-C₁-C₆-alkylgruppe oder die Phenylgruppe, die noch einen bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₂-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl;
R⁵ Wasserstoff, Cyano, Nitro, Halogen, eine C₁-C₆-Alkylgruppe, eine C₂-C₆-Alkenylgruppe, eine C₂-C₆-Alkinylgruppe, eine C₃-C₇-Cycloalkylgruppe, eine partiell oder vollständig halogenierte C₁-C₆-Alkylgruppe, eine C₁-C₆-Hydroxyalkylgruppe, eine C₁-C₆-Cyanoalkylgruppe, eine C₁-C₆-Alkoxy-C₁-C₆-alkylgruppe, eine C₁-C₆-Alkylthio-C₁-C₆-alkylgruppe, die Formylgruppe, eine C₁-C₆-Alkylcarbonylgruppe, eine partiell oder vollständig halogenierte C₁-C₆-Alkylcarbonylgruppe, eine C₁-C₆-Alkoxycarbonylgruppe, eine Gruppe -N(R²²)R²³, wobei R²² und R²³ für eine der Bedeutungen von R¹⁵ und R¹⁶ stehen, die Phenylgruppe, die noch einen bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₂-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl, oder
R⁴ und R⁵ zusammen eine gesättigte oder ungesättigte 3- oder 4gliedrige Kohlenstoffkette, die ein bis drei Heteroatome als Glieder enthalten kann, ausgewählt aus einer Gruppe bestehend aus 1 oder 2 Sauerstoffatomen, 1 oder 2 Schwefelatomen und 1 bis 3 Stickstoffatomen, wobei die Kohlenstoffkette noch ein bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Amino, Halogen, C₁-C₆-Alkyl, C₂-C₆-Alkenyl, C₁-C₆-Alkoxy, C₁-C₆-Alkylthio und C₁-C₆-Alkoxycarbonyl.
11. Pyrimidon-Derivate der allgemeinen Formel IVa oder IVb in der die Variablen folgende Bedeutung haben:
Hal Halogen;
X¹, X² Sauerstoff oder Schwefel;
W eine Gruppe -C(R⁸)=X⁵, -C(R⁸)(X³R⁶)(X⁴R⁷), -C(R⁸)=C(R⁹)-CO-R¹⁰,
-CH(R⁸)-CH(R⁹)-CO-R¹⁰, -C(R⁸)=C(R⁹)-CH₂-CO-R¹⁰, -C(R⁸)=C(R⁹)-C(R¹¹)=C(R¹²)-CO-R¹⁰ oder
-C(R⁸)=C(R⁹)-CH₂-CH(R¹³)-CO-R¹⁰ mit
X³, X⁴ Sauerstoff oder Schwefel;
X⁵ Sauerstoff, Schwefel oder ein Rest -NR¹⁴, mit
R¹⁴ Wasserstoff, Hydroxyl, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₃-C₇-Cycloalkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆- Alkoxy, C₃-C₆-Alkenyloxy, C₃-C₆-Alkinyloxy, C₅-C₇-Cycloalkoxy, C₅-C₇-Cycloalkenyloxy, partiell oder vollständig halogeniertem C₁-C₆-Alkoxy, partiell oder vollständig halogeniertem C₃-C₆-Alkenyloxy, Hydroxy-C₁-C₆- alkoxy, Cyano-C₁-C₆-alkoxy, C₃-C₇-Cycloalkyl- C₁-C₆-alkoxy, C₁-C₆-Alkoxy-C₁-C₆-alkoxy, C₁-C₆-Alkoxy-C₃-C₆-alkenyloxy, C₁-C₆-Alkylcarbonyloxy, C₁-C₆-Alkoxycarbonyl-C₂-C₆-alkoxy, C₁-C₆-Alkylthio-C₁-C₆-alkoxy, Di-(C₁-C₆- alkyl)-amino-C₁-C₆-alkoxy, Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl, Phenyl-C₁-C₆-alkoxy, Phenyl- C₃-C₆-alkenyloxy oder Phenyl-C₃-C₆-alkinyloxy, wobei jeweils eine oder zwei Methylengruppen der Kohlenstoffketten durch -O-, -S- oder -N(C₁-C₆-Alkyl)- ersetzt sein können und wobei der Phenylring jeweils auch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl,
oder -N(R¹⁵)R¹⁶, wobei
R¹⁵, R¹⁶ Wasserstoff, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, C₃-C₆-Cycloalkyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxycarbonyl oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl, oder
R¹⁵ und R¹⁶ zusammen mit dem gemeinsamen Stickstoffatom einen gesättigten oder ungesättigten 4-7gliedrigen Heterocyclus, wobei ein Ringglied durch -O-, -S-, -N=, -NH- oder -N(C₁-C₆-Alkyl)- ersetzt sein kann,
bedeuten;
R⁶, R⁷ C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₁-C₆- Alkoxy-C₁-C₆-alkyl oder
R⁶ und R⁷ zusammen eine gesättigte oder ungesättigte, zwei- bis viergliedrige Kohlenstoffkette, die einen Oxosubstituenten tragen kann, wobei ein Glied dieser Kette durch ein den Variablen X³ und X⁴ nicht benachbartes Sauerstoff-, Schwefel- oder Stickstoffatom ersetzt sein kann, und wobei die Kohlenstoffkette noch ein bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Amino, Halogen, C₁-C₆-Alkyl, C₂-C₆-Alkenyl, C₁-C₆-Alkoxy, C₃-C₆-Alkenyloxy, C₃-C₆-Alkinyloxy, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, Cyano-C₁-C₆-alkyl, Hydroxy-C₁-C₆-alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₃-C₆-Alkenyloxy- C₁-C₆-alkyl, C₃-C₆-Alkinyloxy-C₁-C₆-alkyl, Carboxy, C₁-C₆-Alkoxycarbonyl und C₁-C₆-Alkyl­ carbonyloxy-C₁-C₆-alkyl;
R⁸ Wasserstoff, Cyano, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₃-C₇-Cycloalkyl, C₁-C₆-Alkoxy- C₁-C₆-alkyl oder C₁-C₆-Alkoxycarbonyl;
R⁹, R¹² Wasserstoff, Cyano, Halogen, C₁-C₆-Alkyl, C₁-C₆-Alkoxy, Halogen-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl oder C₁-C₆-Alkoxycarbonyl;
R¹⁰ Wasserstoff, O-R¹⁷, S-R¹⁷, C₁-C₆-Alkyl, das noch einen oder zwei C₁-C₆-Alkoxysubstituenten tragen kann, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₃-C₇-Cycloalkyl, C₁-C₆-Alkylthio-C₁-C₆-alkyl, -N(R¹⁵)R¹⁶ oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy oder C₁-C₆-Alkoxycarbonyl,
R¹⁷ bedeutet Wasserstoff, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, C₃-C₇-Cycloalkyl, partiell oder vollständig halogeniertes C₂-C₆-Alkyl, partiell oder vollständig halogeniertes C₃-C₆-Alkenyl, Cyano-C₁-C₆-alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl oder C₁-C₆-Alkyl­ oximino-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxycarbonyl oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl;
R¹¹ Wasserstoff, Cyano, Halogen, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxycarbonyl, -NR¹⁸R¹⁹, wobei R¹⁸ und R¹⁹ die Bedeutungen von R¹⁵ und R¹⁶ haben, oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl;
R¹³ Wasserstoff, Cyano, C₁-C₆-Alkyl oder C₁-C₆-Alkoxycarbonyl;
R¹ Halogen, die Cyano-, Nitro- oder Trifluormethylgruppe;
R² Wasserstoff oder Halogen;
R⁴ Wasserstoff, Cyano, Halogen, eine C₁-C₆-Alkylgruppe, eine C₂-C₆-Alkenylgruppe, eine C₂-C₆-Alkinylgruppe, eine C₃-C₈- Cycloalkylgruppe, eine partiell oder vollständig halogenierte C₁-C₆-Alkylgruppe, eine C₁-C₆-Hydroxyalkylgruppe, eine C₁-C₆-Cyanoalkylgruppe, eine C₁-C₆-Alkoxy-C₁-C₆-alkylgruppe, eine C₁-C₆-Alkylthio-C₁-C₆-alkylgruppe oder die Phenylgruppe, die noch einen bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₂-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl;
R⁵ Wasserstoff, Cyano, Nitro, Halogen, eine C₁-C₆-Alkylgruppe, eine C₂-C₆-Alkenylgruppe, eine C₂-C₆-Alkinylgruppe, eine C₃-C₇-Cycloalkylgruppe, eine partiell oder vollständig halogenierte C₁-C₆-Alkylgruppe, eine C₁-C₆-Hydroxyalkylgruppe, eine C₁-C₆-Cyanoalkylgruppe, eine C₁-C₆-Alkoxy-C₁-C₆-alkylgruppe, eine C₁-C₆-Alkylthio-C₁-C₆-alkylgruppe, die Formylgruppe, eine C₁-C₆-Alkylcarbonylgruppe, eine partiell oder vollständig halogenierte C₁-C₆-Alkylcarbonylgruppe, eine C₁-C₆-Alkoxycarbonylgruppe, eine Gruppe -N(R²²)R²³, wobei R²² und R²³ für eine der Bedeutungen von R¹⁵ und R¹⁶ stehen, die Phenylgruppe, die noch einen bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₂-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl, oder
R⁴ und R⁵ zusammen eine gesättigte oder ungesättigte 3- oder 4gliedrige Kohlenstoffkette, die ein bis drei Heteroatome als Glieder enthalten kann, ausgewählt aus einer Gruppe bestehend aus 1 oder 2 Sauerstoffatomen, 1 oder 2 Schwefelatomen und 1 bis 3 Stickstoffatomen, wobei die Kette noch ein bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Amino, Halogen, C₁-C₆-Alkyl, C₂-C₆-Alkenyl, C₁-C₆-Alkoxy, C₁-C₆-Alkylthio und C₁-C₆- Alkoxycarbonyl.
12. Phenylharnstoffe der allgemeinen Formel IX in der die Variablen folgende Bedeutung haben:
R¹ Halogen, die Cyano-, Nitro- oder Trifluormethylgruppe;
R² Wasserstoff oder Halogen;
W eine Gruppe -C(R⁸)=X⁵, -C(R⁸)(X³R⁶)(X⁴R⁷), -C(R⁸)=C(R⁹)-CO-R¹⁰,
-CH(R⁸)-CH(R⁹)-CO-R¹⁰, -C(R⁸)=C(R⁹)-CH₂-CO-R¹⁰, -C(R⁸)=C(R⁹)-C(R¹¹)=C(R¹²)-CO-R¹⁰ oder
-C(R⁸)=C(R⁹)-CH₂-CH(R¹³)-CO-R¹⁰ mit
X³, X⁴ Sauerstoff oder Schwefel;
X⁵ Sauerstoff, Schwefel oder ein Rest -NR¹⁴ mit
R¹⁴ Wasserstoff, Hydroxyl, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₃-C₇-Cycloalkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆- Alkoxy, C₃-C₆-Alkenyloxy, C₃-C₆-Alkinyloxy, C₅-C₇-Cycloalkoxy, C₅-C₇-Cycloalkenyloxy, partiell oder vollständig halogeniertem C₁-C₆-Alkoxy, partiell oder vollständig halogeniertem C₃-C₆-Alkenyloxy, Hydroxy-C₁-C₆- alkoxy, Cyano-C₁-C₆-alkoxy, C₃-C₇-Cycloalkyl- C₁-C₆-alkoxy, C₁-C₆-Alkoxy-C₁-C₆-alkoxy, C₁-C₆-Alkoxy-C₃-C₆-alkenyloxy, C₁-C₆-Alkylcarbonyloxy, C₁-C₆-Alkoxycarbonyl-C₂-C₆-alkoxy, C₁-C₆-Alkylthio-C₁-C₆-alkoxy, Di-(C₁-C₆- alkyl)-amino-C₁-C₆-alkoxy, Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl, Phenyl-C₁-C₆-alkoxy, Phenyl- C₃-C₆-alkenyloxy oder Phenyl-C₃-C₆-alkinyloxy, wobei jeweils eine oder zwei Methylengruppen der Kohlenstoffketten durch -O-, -S- oder -N(C₁-C₆-Alkyl)- ersetzt sein können und wobei der Phenylring jeweils auch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl,
oder -N(R¹⁵)R¹⁶, wobei
R¹⁵, R¹⁶ Wasserstoff, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, C₃-C₆-Cycloalkyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxycarbonyl oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆- Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl, oder
R¹⁵ und R¹⁶ zusammen mit dem gemeinsamen Stickstoffatom einen gesättigten oder ungesättigten 4-7gliedrigen Heterocyclus, wobei ein Ringglied durch -O-, -S-, -N=, -NH- oder -N(C₁-C₆-Alkyl)- ersetzt sein kann,
bedeuten;
R⁶, R⁷ C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, C₁-C₆- Alkoxy-C₁-C₆-alkyl oder
R⁶ und R⁷ zusammen eine gesättigte oder ungesättigte, zwei- bis viergliedrige Kohlenstoffkette, die einen Oxosubstituenten tragen kann, wobei ein Glied dieser Kette durch ein den Variablen X³ und X⁴ nicht benachbartes Sauerstoff-, Schwefel- oder Stickstoffatom ersetzt sein kann, und wobei die Kohlenstoffkette noch ein bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Amino, Halogen, C₁-C₆-Alkyl, C₂-C₆- Alkenyl, C₁-C₆-Alkoxy, C₃-C₆-Alkenyloxy, C₃-C₆- Alkinyloxy, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, Cyano-C₁-C₆-alkyl, Hydroxy-C₁-C₆- alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₃-C₆-Alkenyloxy- C₁-C₆-alkyl, C₃-C₆-Alkinyloxy-C₁-C₆-alkyl, Carboxy, C₁-C₆-Alkoxycarbonyl und C₁-C₆-Alkyl­ carbonyloxy-C₁-C₆-alkyl;
R⁸ Wasserstoff, Cyano, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₃-C₇-Cycloalkyl, C₁-C₆-Alkoxy- C₁-C₆-alkyl oder C₁-C₆-Alkoxycarbonyl;
R⁹, R¹² Wasserstoff, Cyano, Halogen, C₁-C₆-Alkyl, C₁-C₆- Alkoxy, Halogen-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl oder C₁-C₆-Alkoxycarbonyl;
R¹⁰ Wasserstoff, O-R¹⁷, S-R¹⁷, C₁-C₆-Alkyl, das noch einen oder zwei C₁-C₆-Alkoxysubstituenten tragen kann, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₃-C₇- Cycloalkyl, C₁-C₆-Alkylthio-C₁-C₆-alkyl, -N(R¹⁵)R¹⁶ oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆- Alkyl, C₃-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy oder C₁-C₆-Alkoxycarbonyl,
R¹⁷ bedeutet Wasserstoff, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₃-C₇-Cycloalkyl, partiell oder vollständig halogeniertes C₂-C₆-Alkyl, partiell oder vollständig halogeniertes C₃-C₆-Alkenyl, Cyano-C₁-C₆- alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl oder C₁-C₆- Alkyl-oximino-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxycarbonyl oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl;
R¹¹ Wasserstoff, Cyano, Halogen, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxycarbonyl, -NR¹⁸R¹⁹, wobei R¹⁸ und R¹⁹ die Bedeutungen von R¹⁵ und R¹⁶ haben, oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl;
R¹³ Wasserstoff, Cyano, C₁-C₆-Alkyl oder C₁-C₆-Alkoxycarbonyl.
13. Phenylisocyanate der allgemeinen Formel XIIa in der die Variablen folgende Bedeutung haben:
R¹ Halogen, die Cyano-, Nitro- oder Trifluormethylgruppe;
R² Wasserstoff oder Halogen;
W eine Gruppe -C(R⁸)=X⁵, -C(R⁸)(X³R⁶)(X⁴R⁷), -C(R⁸)=C(R⁹)-CO-R¹⁰,
-CH(R⁸)-CH(R⁹)-CO-R¹⁰, -C(R⁸)=C(R⁹)-CH₂-CO-R¹⁰, -C(R⁸)=C(R⁹)-C(R¹¹)=C(R¹²)-CO-R¹⁰ oder
-C(R⁸)=C(R⁹)-CH₂-CH(R¹³)-CO-R¹⁰ mit
X³, X⁴ Sauerstoff oder Schwefel;
X⁵ Sauerstoff, Schwefel oder ein Rest -NR¹⁴ mit
R¹⁴ Wasserstoff, Hydroxyl, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₃-C₇-Cycloalkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆- Alkoxy, C₃-C₆-Alkenyloxy, C₃-C₆-Alkinyloxy, C₅-C₇-Cycloalkoxy, C₅-C₇-Cycloalkenyloxy, partiell oder vollständig halogeniertem C₁-C₆-Alkoxy, partiell oder vollständig halogeniertem C₃-C₆-Alkenyloxy, Hydroxy-C₁-C₆- alkoxy, Cyano-C₁-C₆-alkoxy, C₃-C₇-Cycloalkyl- C₁-C₆-alkoxy, C₁-C₆-Alkoxy-C₁-C₆-alkoxy, C₁-C₆-Alkoxy-C₃-C₆-alkenyloxy, C₁-C₆-Alkylcarbonyloxy, C₁-C₆-Alkoxycarbonyl-C₂-C₆-alkoxy, C₁-C₆-Alkylthio-C₁-C₆-alkoxy, Di-(C₁-C₆- alkyl)-amino-C₁-C₆-alkoxy, Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl, Phenyl-C₁-C₆-alkoxy, Phenyl- C₃-C₆-alkenyloxy oder Phenyl-C₃-C₆-alkinyloxy, wobei jeweils eine oder zwei Methylengruppen der Kohlenstoffketten durch -O-, -S- oder -N(C₁-C₆-Alkyl)- ersetzt sein können und wobei der Phenylring jeweils auch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl,
oder -N(R¹⁵)R¹⁶, wobei
R¹⁵, R¹⁶ Wasserstoff, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, C₃-C₆-Cycloalkyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxycarbonyl oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆- Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl, oder
R¹⁵ und R¹⁶ zusammen mit dem gemeinsamen Stickstoffatom einen gesättigten oder ungesättigten 4-7gliedrigen Heterocyclus, wobei ein Ringglied durch -O-, -S-, -N=, -NH- oder -N(C₁-C₆-Alkyl)- ersetzt sein kann,
bedeuten;
R⁶, R⁷ C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, C₁-C₆- Alkoxy-C₁-C₆-alkyl oder
R⁶ und R⁷ zusammen eine gesättigte oder ungesättigte, zwei- bis viergliedrige Kohlenstoffkette, die einen Oxosubstituenten tragen kann, wobei ein Glied dieser Kette durch ein den Variablen X³ und X⁴ nicht benachbartes Sauerstoff-, Schwefel- oder Stickstoffatom ersetzt sein kann, und wobei die Kohlenstoffkette noch ein bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Amino, Halogen, C₁-C₆-Alkyl, C₂-C₆- Alkenyl, C₁-C₆-Alkoxy, C₃-C₆-Alkenyloxy, C₃-C₆- Alkinyloxy, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, Cyano-C₁-C₆-alkyl, Hydroxy-C₁-C₆- alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₃-C₆-Alkenyloxy- C₁-C₆-alkyl, C₃-C₆-Alkinyloxy-C₁-C₆-alkyl, Carboxy, C₁-C₆-Alkoxycarbonyl und C₁-C₆-Alkyl­ carbonyloxy-C₁-C₆-alkyl;
R⁸ Wasserstoff, Cyano, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₃-C₇-Cycloalkyl, C₁-C₆- Alkoxy-C₁-C₆-alkyl oder C₁-C₆-Alkoxycarbonyl;
R⁹, R¹² Wasserstoff, Cyano, Halogen C₁-C₆-Alkyl, C₁-C₆- Alkoxy, Halogen-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl oder C₁-C₆-Alkoxycarbonyl;
R¹⁰ Wasserstoff, O-R¹⁷, S-R¹⁷, C₁-C₆-Alkyl, das noch einen oder zwei C₁-C₆-Alkoxysubstituenten tragen kann, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₃-C₇- Cycloalkyl, C₁-C₆-Alkylthio-C₁-C₆-alkyl, -N(R¹⁵)R¹⁶ oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆- Alkyl, C₃-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy oder C₁-C₆-Alkoxycarbonyl,
R¹⁷ bedeutet Wasserstoff, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₃-C₇-Cycloalkyl, partiell oder vollständig halogeniertes C₂-C₆-Alkyl, partiell oder vollständig halogeniertes C₃-C₆-Alkenyl, Cyano-C₁-C₆-alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl oder C₁-C₆-Alkyl­ oximino-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxycarbonyl oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl;
R¹¹ Wasserstoff, Cyano, Halogen, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxycarbonyl, -NR¹⁸R¹⁹, wobei R¹⁸ und R¹⁹ die Bedeutungen von R¹⁵ und R¹⁶ haben, oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl;
R¹³ Wasserstoff, Cyano, C₁-C₆-Alkyl oder C₁-C₆-Alkoxycarbonyl.
14. N-Phenylurethane der allgemeinen Formel XIII in der die Variablen folgende Bedeutung haben:
L⁴ eine C₁-C₆-Alkylgruppe oder die Phenylgruppe;
R¹ Halogen, die Cyano-, Nitro- oder Trifluormethylgruppe;
R² Wasserstoff oder Halogen;
W eine Gruppe -C(R⁸)=X⁵, -C(R⁸)(X³R⁶)(X⁴R⁷), -C(R⁸)=C(R⁹)-CO-R¹⁰,
-CH(R⁸)-CH(R⁹)-CO-R¹⁰, -C(R⁸)=C(R⁹)-CH₂-CO-R¹⁰, -C(R⁸)=C(R⁹)-C(R¹¹)=C(R¹²)-CO-R¹⁰ oder
-C(R⁸)=C(R⁹)-CH₂-CH(R¹³)-CO-R¹⁰ mit
X³, X⁴ Sauerstoff oder Schwefel;
X⁵ Sauerstoff, Schwefel oder ein Rest -NR¹⁴ mit
R¹⁴ Wasserstoff, Hydroxyl, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₃-C₇-Cycloalkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆- Alkoxy, C₃-C₆-Alkenyloxy, C₃-C₆-Alkinyloxy, C₅-C₇-Cycloalkoxy, C₅-C₇-Cycloalkenyloxy, partiell oder vollständig halogeniertem C₁-C₆-Alkoxy, partiell oder vollständig halogeniertem C₃-C₆-Alkenyloxy, Hydroxy-C₁-C₆- alkoxy, Cyano-C₁-C₆-alkoxy, C₃-C₇-Cycloalkyl- C₁-C₆-alkoxy, C₁-C₆-Alkoxy-C₁-C₆-alkoxy, C₁-C₆-Alkoxy-C₃-C₆-alkenyloxy, C₁-C₆-Alkylcarbonyloxy, C₁-C₆-Alkoxycarbonyl-C₂-C₆-alkoxy, C₁-C₆-Alkylthio-C₁-C₆-alkoxy, Di-(C₁-C₆- alkyl)-amino-C₁-C₆-alkoxy, Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl, Phenyl-C₁-C₆-alkoxy, Phenyl- C₃-C₆-alkenyloxy oder Phenyl-C₃-C₆-alkinyloxy, wobei jeweils eine oder zwei Methylengruppen der Kohlenstoffketten durch -O-, -S- oder -N(C₁-C₆-Alkyl)- ersetzt sein können und wobei der Phenylring jeweils auch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl,
oder -N(R¹⁵)R¹⁶, wobei
R¹⁵, R¹⁶ Wasserstoff, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, C₃-C₆-Cycloalkyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxycarbonyl oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆- Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl, oder
R¹⁵ und R¹⁶ zusammen mit dem gemeinsamen Stickstoffatom einen gesättigten oder ungesättigten 4-7gliedrigen Heterocyclus, wobei ein Ringglied durch -O-, -S-, -N=, -NH- oder -N(C₁-C₆-Alkyl)- ersetzt sein kann,
bedeuten;
R⁶, R⁷ C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, C₁-C₆- Alkoxy-C₁-C₆-alkyl oder
R⁶ und R⁷ zusammen eine gesättigte oder ungesättigte, zwei- bis viergliedrige Kohlenstoffkette, die einen Oxosubstituenten tragen kann, wobei ein Glied dieser Kette durch ein den Variablen X³ und X⁴ nicht benachbartes Sauerstoff-, Schwefel- oder Stickstoffatom ersetzt sein kann, und wobei die Kohlenstoffkette noch ein bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Amino, Halogen, C₁-C₆-Alkyl, C₂-C₆- Alkenyl, C₁-C₆-Alkoxy, C₃-C₆-Alkenyloxy, C₃-C₆- Alkinyloxy, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, Cyano-C₁-C₆-alkyl, Hydroxy-C₁-C₆- alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₃-C₆-Alkenyloxy- C₁-C₆-alkyl, C₃-C₆-Alkinyloxy-C₁-C₆-alkyl, Carboxy, C₁-C₆-Alkoxycarbonyl und C₁-C₆-Alkyl­ carbonyloxy-C₁-C₆-alkyl;
R⁸ Wasserstoff, Cyano, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₃-C₇-Cycloalkyl, C₁-C₆-Alkoxy- C₁-C₆-alkyl oder C₁-C₆-Alkoxycarbonyl;
R⁹, R¹² Wasserstoff, Cyano, Halogen, C₁-C₆-Alkyl, C₁-C₆- Alkoxy, Halogen-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl oder C₁-C₆-Alkoxycarbonyl;
R¹⁰ Wasserstoff, O-R¹⁷, S-R¹⁷, C₁-C₆-Alkyl, das noch einen oder zwei C₁-C₆-Alkoxysubstituenten tragen kann, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₃-C₇- Cycloalkyl, C₁-C₆-Alkylthio-C₁-C₆-alkyl, -N(R¹⁵)R¹⁶ oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆- Alkyl, C₃-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy oder C₁-C₆-Alkoxycarbonyl,
R¹⁷ bedeutet Wasserstoff, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₃-C₇-Cycloalkyl, partiell oder vollständig halogeniertes C₂-C₆-Alkyl, partiell oder vollständig halogeniertes C₃-C₆-Alkenyl, Cyano-C₁-C₆-alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl oder C₁-C₆-Alkyl­ oximino-C₁-C₆-alkyl, C₁-C₆-Alkoxycarbonyl oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl;
R¹¹ Wasserstoff, Cyano, Halogen, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxycarbonyl, -NR¹⁸R¹⁹, wobei R¹⁸ und R¹⁹ die Bedeutungen von R¹⁵ und R¹⁶ haben, oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl;
R¹³ Wasserstoff, Cyano, C₁-C₆-Alkyl oder C₁-C₆-Alkoxycarbonyl.
15. Carbaminsäurechloride der allgemeinen Formel XIV in der die Variablen folgende Bedeutung haben:
R¹ Halogen, die Cyano-, Nitro- oder Trifluormethylgruppe;
R² Wasserstoff oder Halogen;
W eine Gruppe -C(R⁸)=X⁵, -C(R⁸)(X³R⁶)(X⁴R⁷), -C(R⁸)=C(R⁹)-CO-R¹⁰,
-CH(R⁸)-CH(R⁹)-CO-R¹⁰, -C(R⁸)=C(R⁹)-CH₂-CO-R¹⁰, -C(R⁸)=C(R⁹)-C(R¹¹)=C(R¹²)-CO-R¹⁰ oder
-C(R⁸)=C(R⁹)-CH₂-CH(R¹³)-CO-R¹⁰ mit
X³, X⁴ Sauerstoff oder Schwefel;
X⁵ Sauerstoff, Schwefel oder ein Rest -NR¹⁴ mit
R¹⁴ Wasserstoff, Hydroxyl, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₃-C₇-Cycloalkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆- Alkoxy, C₃-C₆-Alkenyloxy, C₃-C₆-Alkinyloxy, C₅-C₇-Cycloalkoxy, C₅-C₇-Cycloalkenyloxy, partiell oder vollständig halogeniertem C₁-C₆-Alkoxy, partiell oder vollständig halogeniertem C₃-C₆-Alkenyloxy, Hydroxy-C₁-C₆- alkoxy, Cyano-C₁-C₆-alkoxy, C₃-C₇-Cycloalkyl- C₁-C₆-alkoxy, C₁-C₆-Alkoxy-C₁-C₆-alkoxy, C₁-C₆-Alkoxy-C₃-C₆-alkenyloxy, C₁-C₆-Alkylcarbonyloxy, C₁-C₆-Alkoxycarbonyl-C₂-C₆-alkoxy, C₁-C₆-Alkylthio-C₁-C₆-alkoxy, Di-(C₁-C₆- alkyl)-amino-C₁-C₆-alkoxy, Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl, Phenyl-C₁-C₆-alkoxy, Phenyl- C₃-C₆-alkenyloxy oder Phenyl-C₃-C₆-alkinyloxy, wobei jeweils eine oder zwei Methylengruppen der Kohlenstoffketten durch -O-, -S- oder -N(C₁-C₆-Alkyl)- ersetzt sein können und wobei der Phenylring jeweils auch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl,
oder -N(R¹⁵)R¹⁶, wobei
R¹⁵, R¹⁶ Wasserstoff, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, C₃-C₆-Cycloalkyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxycarbonyl oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆- Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆- Alkoxycarbonyl, oder
R¹⁵ und R¹⁶ zusammen mit dem gemeinsamen Stickstoffatom einen gesättigten oder ungesättigten 4-7gliedrigen Heterocyclus, wobei ein Ringglied durch -O-, -S-, -N=, -NH- oder -N(C₁-C₆-Alkyl)- ersetzt sein kann,
bedeuten;
R⁶, R⁷ C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, C₁-C₆- Alkoxy-C₁-C₆-alkyl oder
R⁶ und R⁷ zusammen eine gesättigte oder ungesättigte, zwei- bis viergliedrige Kohlenstoffkette, die einen Oxosubstituenten tragen kann, wobei ein Glied dieser Kette durch ein den Variablen X³ und X⁴ nicht benachbartes Sauerstoff-, Schwefel- oder Stickstoffatom ersetzt sein kann, und wobei die Kohlenstoffkette noch ein bis drei Reste tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Amino, Halogen, C₁-C₆-Alkyl, C₂-C₆- Alkenyl, C₁-C₆-Alkoxy, C₃-C₆-Alkenyloxy, C₃-C₆- Alkinyloxy, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, Cyano-C₁-C₆-alkyl, Hydroxy-C₁-C₆- alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₃-C₆-Alkenyloxy- C₁-C₆-alkyl, C₃-C₆-Alkinyloxy-C₁-C₆-alkyl, Carboxy, C₁-C₆-Alkoxycarbonyl und C₁-C₆-Alkyl­ carbonyloxy-C₁-C₆-alkyl;
R⁸ Wasserstoff, Cyano, C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₃-C₇-Cycloalkyl, C₁-C₆- Alkoxy-C₁-C₆-alkyl oder C₁-C₆-Alkoxycarbonyl;
R⁹, R¹² Wasserstoff, Cyano, Halogen C₁-C₆-Alkyl, C₁-C₆- Alkoxy, Halogen-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl oder C₁-C₆-Alkoxycarbonyl;
R¹⁰ Wasserstoff, O-R¹⁷, S-R¹⁷, C₁-C₆-Alkyl, das noch einen oder zwei C₁-C₆-Alkoxysubstituenten tragen kann, C₃-C₆-Alkenyl, C₃-C₆-Alkinyl, partiell oder vollständig halogeniertes C₁-C₆-Alkyl, C₃-C₇- Cycloalkyl, C₁-C₆-Alkylthio-C₁-C₆-alkyl, -N(R¹⁵)R¹⁶ oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆- Alkyl, C₃-C₆-Alkenyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₁-C₆-Alkoxy oder C₁-C₆-Alkoxycarbonyl,
R¹⁷ bedeutet Wasserstoff, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₃-C₇-Cycloalkyl, partiell oder vollständig halogeniertes C₂-C₆-Alkyl, partiell oder vollständig halogeniertes C₃-C₆-Alkenyl, Cyano-C₁-C₆- alkyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl oder C₁-C₆- Alkyl-oximino-C₁-C₆-alkyl, C₁-C₆-Alkoxycarbonyl oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl;
R¹¹ Wasserstoff, Cyano, Halogen, C₁-C₆-Alkyl, C₃-C₆- Alkenyl, C₃-C₆-Alkinyl, C₁-C₆-Alkoxy-C₁-C₆-alkyl, C₁-C₆-Alkylcarbonyl, C₁-C₆-Alkoxycarbonyl, -NR¹⁸R¹⁹, wobei R¹⁸ und R¹⁹ die Bedeutungen von R¹⁵ und R¹⁶ haben, oder Phenyl, das noch einen bis drei Substituenten tragen kann, ausgewählt aus einer Gruppe bestehend aus Cyano, Nitro, Halogen, C₁-C₆-Alkyl, partiell oder vollständig halogeniertem C₁-C₆-Alkyl, C₃-C₆-Alkenyl, C₁-C₆-Alkoxy und C₁-C₆-Alkoxycarbonyl;
R¹³ Wasserstoff, Cyano, C₁-C₆-Alkyl oder C₁-C₆-Alkoxycarbonyl.
16. Herbizides Mittel, enthaltend einen inerten flüssigen oder festen Trägerstoff und eine herbizid wirksame Menge mindestens eines substituierten 3-Phenylurazils der Formel I, Ia oder Ib oder ein Salz oder einen Enolether derjenigen Verbindungen I, in denen R³ Wasserstoff bedeutet.
17. Verfahren zur Bekämpfung von unerwünschtem Pflanzenwuchs, dadurch gekennzeichnet, daß man eine herbizid wirksame Menge eines substituierten 3-Phenylurazils der Formel I, Ia oder Ib oder ein Salz oder einen Enolether derjenigen Verbindungen I, in denen R³ Wasserstoff bedeutet, gemäß Anspruch 1 auf Pflanzen, deren Lebensraum oder auf Saatgut einwirken läßt.
18. Mittel zur Desiccation und Defoliation von Pflanzen, enthaltend neben üblichen Zusatzstoffen eine defoliant und/oder desiccant wirksame Menge mindestens eines substituierten 3-Phenylurazils der Formel I, Ia oder Ib oder ein Salz oder einen Enolether derjenigen Verbindungen I, in denen R³ Wasserstoff bedeutet.
19. Verfahren zur Desiccation und Defoliation von Pflanzen, dadurch gekennzeichnet, daß man eine defoliant und/oder desiccant wirksame Menge eines substituierten 3-Phenylurazils I, Ia oder Ib gemäß den Ansprüchen 1 bis 8 auf die Pflanzen einwirken läßt.
20. Verfahren nach Anspruch 19, dadurch gekennzeichnet, daß man Baumwolle entlaubt.
21. Schädlingsbekämpfungsmittel, enthaltend inerte Trägerstoffe und eine pestizid wirksame Menge mindestens eines substituierten 3-Phenylurazils der Formel I, Ia oder Ib oder eines Salzes oder eines Enolethers derjenigen Verbindungen I, in denen R³ Wasserstoff bedeutet.
22. Verfahren zur Bekämpfung von Schädlingen, dadurch gekennzeichnet, daß man eine pestizid wirksame Menge eines substituierten 3-Phenylurazils der Formel I, Ia oder Ib oder eines Salzes oder eines Enolethers derjenigen Verbindungen I, in denen R³ Wasserstoff bedeutet, gemäß Anspruch 1 auf Schädlinge bzw. ihren Lebensraum einwirken läßt.
23. Verfahren zur Herstellung von substituierten 3-Phenylurazilen I, Ia oder Ib gemäß den Ansprüchen 1 bis 8, dadurch gekennzeichnet, daß man
  • a) einen Enamin-Ester der Formel II oder eine Enamin-Carboxylat der Formel III wobei L¹ eine C₁-C₆-Alkylgruppe oder die Phenylgruppe bedeutet,
    cyclisiert und gewünschtenfalls aus dem erhaltenen Metallsalz mittels Säure das substituierte 3-Phenylurazil I, wobei R³ Wasserstoff bedeutet, freisetzt oder
  • b) ein substituiertes 3-Phenylurazil I, wobei R³ für Wasserstoff steht, alkyliert oder acyliert oder
  • c) ein substituiertes 3-Phenylurazil I, wobei R¹ für Halogen steht, mit einem Metallcyanid umsetzt oder
  • d) ein Pyrimidon-Derivat der Formel IVa oder IVb wobei Hal Halogen bedeutet,
    mit einer Verbindung HO-R3′, HS-R3′, Me⊕⊖OR3′ oder Me⊕⊖SR3′, wobei Me⊕ ein Äquivalent eines Metallions bedeutet, umsetzt oder
  • e) ein substituiertes 3-Phenylurazil I, wobei W eine Gruppe -CO-R⁸ bedeutet, mit Verbindungen H-X³R⁶, H-X⁴R⁷ oder H-X³(R⁴R⁷)X⁴-H acetalisiert oder
  • f) ein substituiertes 3-Phenylurazil I, wobei W eine Gruppe -C(R⁸)(X³R⁶)(X⁴R⁷) bedeutet, einer Acetalspaltung unterwirft oder
  • g) ein substituiertes 3-Phenylurazil I, wobei W eine Gruppe -C(R⁸)=O bedeutet, mit einem Phosphorylid der Formeln Va bis Vd R₃P=CR⁹-CO-R¹⁰ (Va)R₃P=C(R⁹)-CH₂-CO-R¹⁰ (Vb)R₃P=C(R⁹)-C(R¹¹)=C(R¹²)-CO-R¹⁰ (Vc)R₃P=C(R⁹)-CH₂-CHR¹³-CO-R¹⁰ (Vd)wobei R für einen C-organischen Substituenten steht,
    oder mit einem Phosphoniumsalz der Formeln VIa bis VIdR₃P⊕-CH(R⁹)-CO-R¹⁰, Hal⊖ (VIa)R₃P⊕-CH(R⁹)-CH₂-CO-R¹⁰, Hal⊖ (VIb)R₃P⊕-C(R⁹)-CR¹¹=CR¹²-CO-R¹⁰, Hal⊖ (VIc)R₃P⊕-C(R⁹)-CH₂-CHR¹³-CO-R¹⁰, Hal⊖ (VId)wobei Hal für Halogen steht,
    oder mit einem Phosphonat der Formeln VIIa bis VIId(RO)₂PO-CH(R⁹)-CO-R¹⁰ (VIIa)(RO)₂PO-CH(R⁹)-CH₂-CO-R¹⁰ (VIIb)(RO)₂PO-CH(R⁹)-CR¹¹-CR¹²-CO-R¹⁰ (VIIc)(RO)₂PO-CH(R⁹)-CH₂-CHR¹³-CO-R¹⁰ (VIId)umsetzt oder
  • h) ein substituiertes 3-Phenylurazil I, wobei W eine Gruppe -C(R⁸)=O bedeutet, mit einem Amin, Hydroxylamin oder Hydrazin H₂N-R¹⁴ umsetzt oder
  • i) ein substituiertes 3-Phenylurazil I, wobei W eine Gruppe -C(R⁸)=N-R¹⁴ bedeutet, in eine Verbindung I, wobei W für eine Gruppe -C(R⁸)=O steht, spaltet oder
  • k) ein substituiertes 3-Phenylurazil I, wobei X² Sauerstoff bedeutet, mit einem Schwefelungsreagenz umsetzt oder
  • l) ein substituiertes 3-Phenylurazil I, wobei R⁵ Wasserstoff bedeutet, halogeniert oder
  • m) ein substituiertes 3-Phenylurazil I, wobei W die Cyanogruppe bedeutet, reduktiv in eine Verbindung I, wobei W für die Formylgruppe steht, überführt.
DE4131038A 1991-09-20 1991-09-20 Substituierte 3-phenylurazile Withdrawn DE4131038A1 (de)

Priority Applications (13)

Application Number Priority Date Filing Date Title
DE4131038A DE4131038A1 (de) 1991-09-20 1991-09-20 Substituierte 3-phenylurazile
JP50574593A JP3253299B2 (ja) 1991-09-20 1992-09-10 置換3−フェニルウラシル
US08/774,722 US6239074B1 (en) 1991-09-20 1992-09-10 Substituted 3-phenyluracils
CA002119036A CA2119036A1 (en) 1991-09-20 1992-09-10 Substituted 3-phenyluracils
PCT/EP1992/002088 WO1993006090A1 (de) 1991-09-20 1992-09-10 Substituierte-3-phenylurazile als herbizide
BR9206518A BR9206518A (pt) 1991-09-20 1992-09-10 Compostos, processo para sua preparação, composição herbicida e pesticida, processo para combater vegetação indesejável, composição e processo para dessecação e desfolhamento de plantas e processo para o combate de pestes.
HU9400801A HUT70880A (en) 1991-09-20 1992-09-10 Substituted 3-phenyluracils herbicidal composition containing and process for the preparation of activ ingredients
KR1019940700895A KR100260011B1 (ko) 1991-09-20 1992-09-10 제초제로서의 치환 3-페닐우라실
EP92919190A EP0604491A1 (de) 1991-09-20 1992-09-10 Substituierte-3-phenylurazile als herbizide
TW081107305A TW225981B (de) 1991-09-20 1992-09-16
MX9205306A MX9205306A (es) 1991-09-20 1992-09-18 3-feniluracilos sustituidos
ZA927153A ZA927153B (en) 1991-09-20 1992-09-18 Substituted 3-phenylluracils
US09/733,554 US20010031865A1 (en) 1991-09-20 2000-12-04 Substituted 3-phenyluracils

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DE4131038A DE4131038A1 (de) 1991-09-20 1991-09-20 Substituierte 3-phenylurazile

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EP (1) EP0604491A1 (de)
JP (1) JP3253299B2 (de)
KR (1) KR100260011B1 (de)
BR (1) BR9206518A (de)
CA (1) CA2119036A1 (de)
DE (1) DE4131038A1 (de)
HU (1) HUT70880A (de)
MX (1) MX9205306A (de)
TW (1) TW225981B (de)
WO (1) WO1993006090A1 (de)
ZA (1) ZA927153B (de)

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1995025725A1 (en) * 1994-03-21 1995-09-28 Uniroyal Chemical Company, Inc. Pyrimidinyl aryl ketone oximes
WO1996002518A1 (de) * 1994-07-14 1996-02-01 Basf Aktiengesellschaft Substituierte zimtoxim- und zimthydroxamid-derivate
WO1996005179A1 (de) * 1994-08-16 1996-02-22 Basf Aktiengesellschaft Substituierte triazolinone als pflanzenschutzmittel
US5749683A (en) * 1996-09-30 1998-05-12 Northern Logistics, L.L.C. Dry van trailer conversion and material handling method
EP0736014B1 (de) * 1993-12-20 2001-04-04 Bayer Ag N-cyanoaryl-stickstoffheterocyclen mit schwefelhaltigen gruppierungen
US8410176B2 (en) 2009-12-29 2013-04-02 Mapi Pharma Ltd. Intermediate compounds and processes for the preparation of tapentadol and related compounds

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6207830B1 (en) 1987-09-23 2001-03-27 Syngenta Crop Protection, Inc. Process for the production of 3-aryl-uracils
DE4329537A1 (de) * 1993-09-02 1995-03-09 Basf Ag Substituierte 1-Amino-3-phenyluracile
US6057269A (en) * 1995-07-06 2000-05-02 Basf Aktiengesellschaft Benzylhydroxylamines and intermediates used to prepare them
DE19528186A1 (de) * 1995-08-01 1997-02-06 Bayer Ag Substituierte Phenyluracile
AU2651297A (en) * 1996-05-08 1997-11-26 Ihara Chemical Industry Co. Ltd. Indolyl-substituted uracil derivatives and herbicides comprising them as active ingredients
DE19621311A1 (de) * 1996-05-28 1997-12-04 Bayer Ag Substituierte Phenyluracile
DE19649094A1 (de) * 1996-11-27 1998-05-28 Bayer Ag Phenyl-uracil-Derivate
EP0934969B1 (de) * 1997-08-25 2002-11-06 Toray Industries, Inc. Polyesterfolie für elektrische isolierung
US6930101B1 (en) 1999-05-17 2005-08-16 The Regents Of The University Of California Thiazolopyrimidines useful as TNFα inhibitors
DE19932813A1 (de) 1999-07-14 2001-01-18 Bayer Ag Substituierte Phenyluracile
JP4639459B2 (ja) * 1999-11-01 2011-02-23 住友化学株式会社 6−ヒドロキシ−5,6−ジヒドロウラシル化合物
EP1272476A1 (de) * 2000-04-14 2003-01-08 Basf Aktiengesellschaft 2-phenyl-2h-pyridazin-3-one
EP1736052B1 (de) * 2001-05-31 2010-04-21 Sumitomo Chemical Company, Limited Austrocknungsmittel für Stengel und Blätter
BR0117032A (pt) * 2001-05-31 2004-04-20 Sumitomo Chemical Co Reguladores de crescimento de planta para coleta de algodão
PL375299A1 (en) * 2002-07-23 2005-11-28 Basf Aktiengesellschaft 3-heterocyclyl substituted benzoic acid derivatives
WO2008133127A1 (ja) 2007-04-18 2008-11-06 Kissei Pharmaceutical Co., Ltd. 縮合へテロ環誘導体、それを含有する医薬組成物及びその医薬用途
JP5352450B2 (ja) 2007-04-18 2013-11-27 キッセイ薬品工業株式会社 縮合複素環誘導体、それを含有する医薬組成物及びその医薬用途
AR115690A1 (es) * 2018-07-05 2021-02-17 Sumitomo Chemical Co Compuestos de uracilo y composición para el control de artrópodos dañinos que comprende estos compuestos

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS61211178A (ja) * 1985-03-14 1986-09-19 ヤマハ発動機株式会社 自動二輪車のスタンド装置
ZA875466B (en) * 1986-07-31 1988-02-02 F. Hoffmann-La Roche & Co. Aktiengesellschaft Heterocyclic compounds
DE3879915D1 (de) * 1987-06-19 1993-05-06 Ciba Geigy Ag Heterocyclische verbindungen.
JPH02501831A (ja) * 1987-10-22 1990-06-21 チバ ― ガイギー アクチエンゲゼルシャフト 複素環化合物
US4927451A (en) * 1988-12-30 1990-05-22 Uniroyal Chemical Company, Inc. 3-aryldihydrouracils
DE69002792T2 (de) * 1989-05-09 1993-12-09 Sds Biotech Corp Crotonsäureamidderivate und sie enthaltende Insektizide.
DE59007059D1 (de) * 1989-06-29 1994-10-13 Ciba Geigy Ag Heterocyclische verbindungen.
JP2946656B2 (ja) * 1989-07-14 1999-09-06 日産化学工業株式会社 ウラシル誘導体および除草剤
AU627906B2 (en) * 1989-07-14 1992-09-03 Nissan Chemical Industries Ltd. Uracil derivatives and herbicides containing the same as active ingredient
US5084084A (en) * 1989-07-14 1992-01-28 Nissan Chemical Industries Ltd. Uracil derivatives and herbicides containing the same as active ingredient
US4979982A (en) * 1990-02-02 1990-12-25 Uniroyal Chemical Company, Inc. Herbicidal cinnamic ester uracils
US5169430A (en) * 1991-08-09 1992-12-08 Uniroyal Chemical Company, Inc. Benzenesulfonamide derivatives and methods for their production

Cited By (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0736014B1 (de) * 1993-12-20 2001-04-04 Bayer Ag N-cyanoaryl-stickstoffheterocyclen mit schwefelhaltigen gruppierungen
WO1995025725A1 (en) * 1994-03-21 1995-09-28 Uniroyal Chemical Company, Inc. Pyrimidinyl aryl ketone oximes
US5486521A (en) * 1994-03-21 1996-01-23 Uniroyal Chemical Company, Inc. Pyrimidinyl aryl ketone oximes
WO1996002518A1 (de) * 1994-07-14 1996-02-01 Basf Aktiengesellschaft Substituierte zimtoxim- und zimthydroxamid-derivate
WO1996005179A1 (de) * 1994-08-16 1996-02-22 Basf Aktiengesellschaft Substituierte triazolinone als pflanzenschutzmittel
US5885934A (en) * 1994-08-16 1999-03-23 Basf Aktiengesellschaft Substituted triazolinones as crop protection agents
US5749683A (en) * 1996-09-30 1998-05-12 Northern Logistics, L.L.C. Dry van trailer conversion and material handling method
US8410176B2 (en) 2009-12-29 2013-04-02 Mapi Pharma Ltd. Intermediate compounds and processes for the preparation of tapentadol and related compounds

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EP0604491A1 (de) 1994-07-06
US6239074B1 (en) 2001-05-29
HUT70880A (en) 1995-11-28
BR9206518A (pt) 1995-04-25
JPH06510992A (ja) 1994-12-08
JP3253299B2 (ja) 2002-02-04
KR100260011B1 (ko) 2000-08-01
HU9400801D0 (en) 1994-06-28
WO1993006090A1 (de) 1993-04-01
MX9205306A (es) 1993-04-01
CA2119036A1 (en) 1993-04-01
TW225981B (de) 1994-07-01
KR940702490A (ko) 1994-08-20
US20010031865A1 (en) 2001-10-18
ZA927153B (en) 1994-03-18

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