DE3324403A1 - Androsten-17-dithioketale und diese verbindungen enthaltende arzeimittel - Google Patents

Androsten-17-dithioketale und diese verbindungen enthaltende arzeimittel

Info

Publication number
DE3324403A1
DE3324403A1 DE19833324403 DE3324403A DE3324403A1 DE 3324403 A1 DE3324403 A1 DE 3324403A1 DE 19833324403 DE19833324403 DE 19833324403 DE 3324403 A DE3324403 A DE 3324403A DE 3324403 A1 DE3324403 A1 DE 3324403A1
Authority
DE
Germany
Prior art keywords
dien
thio7
hydroxy
fluoro
androsta
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
DE19833324403
Other languages
German (de)
English (en)
Inventor
Ravi K. Belle Mead N.J. Varma
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
ER Squibb and Sons LLC
Original Assignee
ER Squibb and Sons LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ER Squibb and Sons LLC filed Critical ER Squibb and Sons LLC
Publication of DE3324403A1 publication Critical patent/DE3324403A1/de
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/003—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring the S atom directly linked to a ring carbon atom of the cyclopenta(a)hydrophenanthrene skeleton
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Rheumatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DE19833324403 1982-07-07 1983-07-06 Androsten-17-dithioketale und diese verbindungen enthaltende arzeimittel Ceased DE3324403A1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/396,178 US4447363A (en) 1982-07-07 1982-07-07 Androstene-17-dithioketals

Publications (1)

Publication Number Publication Date
DE3324403A1 true DE3324403A1 (de) 1984-01-12

Family

ID=23566177

Family Applications (1)

Application Number Title Priority Date Filing Date
DE19833324403 Ceased DE3324403A1 (de) 1982-07-07 1983-07-06 Androsten-17-dithioketale und diese verbindungen enthaltende arzeimittel

Country Status (7)

Country Link
US (1) US4447363A (enExample)
JP (1) JPS5921700A (enExample)
CA (1) CA1213271A (enExample)
DE (1) DE3324403A1 (enExample)
FR (1) FR2529893A1 (enExample)
GB (1) GB2123425B (enExample)
IT (1) IT1165458B (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0524813A1 (en) * 1991-07-25 1993-01-27 E.R. SQUIBB & SONS, INC. Selective thioketalization process, process for preparing thioenol ethers from thioketals, and process for the preparation of thioketals

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4528138A (en) * 1984-06-20 1985-07-09 E. R. Squibb & Sons, Inc. 16-Keto-17-substituted thia-17-alkyl(or alkenyl or alkynyl) androstenes
US4529547A (en) * 1984-06-20 1985-07-16 E.R. Squibb & Sons, Inc. 17-(substituted thio)-17-(substituted dithio)androstenes
JPS6284864A (ja) * 1985-10-11 1987-04-18 Akio Nakano ダイカスト機の射出ノズル

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4361559A (en) * 1981-08-20 1982-11-30 E. R. Squibb & Sons, Inc. Antiinflammatory 17,17-bis (substituted thio) androstenes

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4091036A (en) * 1977-05-12 1978-05-23 E. R. Squibb & Sons, Inc. 17-Alkylthio (and arylthio)-1',2',3',4'-tetrahydroandrosteno [16 α, 17 α-b]naphthalenes and derivatives
US4133811A (en) * 1978-02-17 1979-01-09 E. R. Squibb & Sons, Inc. 13-Alkylthio (and arylthio)-11,17-epoxy-17-methyl-18-norandrostenes
US4265815A (en) * 1980-03-31 1981-05-05 E. R. Squibb & Sons, Inc. 17-(Substituted thio)androst-4-ene[16,17,-b]-[1,4]benzodioxin-3-ones

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4361559A (en) * 1981-08-20 1982-11-30 E. R. Squibb & Sons, Inc. Antiinflammatory 17,17-bis (substituted thio) androstenes

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
Arzneimittelforschung/Drug Res. 36 (II), Nr. 12(1986), S. 1782-1787 *
Arzneimittelforschung/Drug Res. 36 (II), Nr. 12(1986), S. 1787-1795 *

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0524813A1 (en) * 1991-07-25 1993-01-27 E.R. SQUIBB & SONS, INC. Selective thioketalization process, process for preparing thioenol ethers from thioketals, and process for the preparation of thioketals

Also Published As

Publication number Publication date
GB2123425B (en) 1986-02-05
GB8318305D0 (en) 1983-08-10
FR2529893A1 (fr) 1984-01-13
GB2123425A (en) 1984-02-01
IT8321969A0 (it) 1983-07-07
CA1213271A (en) 1986-10-28
FR2529893B1 (enExample) 1985-04-26
JPS5921700A (ja) 1984-02-03
US4447363A (en) 1984-05-08
IT1165458B (it) 1987-04-22

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Legal Events

Date Code Title Description
8128 New person/name/address of the agent

Representative=s name: VOSSIUS, V., DIPL.-CHEM. DR.RER.NAT. TAUCHNER, P.,

8110 Request for examination paragraph 44
8131 Rejection