DE3060481D1 - Anthracycline glycosides, methods for the production thereof and therapeutical compositions containing same - Google Patents

Anthracycline glycosides, methods for the production thereof and therapeutical compositions containing same

Info

Publication number
DE3060481D1
DE3060481D1 DE8080100447T DE3060481T DE3060481D1 DE 3060481 D1 DE3060481 D1 DE 3060481D1 DE 8080100447 T DE8080100447 T DE 8080100447T DE 3060481 T DE3060481 T DE 3060481T DE 3060481 D1 DE3060481 D1 DE 3060481D1
Authority
DE
Germany
Prior art keywords
compounds
methods
compositions containing
containing same
production
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
DE8080100447T
Other languages
English (en)
Inventor
Guiseppe Cassinelli
Federico Arcamone
Marco Aurelio Dr Di
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Italia SRL
Original Assignee
Farmitalia Carlo Erba SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farmitalia Carlo Erba SRL filed Critical Farmitalia Carlo Erba SRL
Application granted granted Critical
Publication of DE3060481D1 publication Critical patent/DE3060481D1/de
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/24—Condensed ring systems having three or more rings
    • C07H15/252—Naphthacene radicals, e.g. daunomycins, adriamycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biotechnology (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Furan Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
DE8080100447T 1979-02-02 1980-01-29 Anthracycline glycosides, methods for the production thereof and therapeutical compositions containing same Expired DE3060481D1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB7903700 1979-02-02

Publications (1)

Publication Number Publication Date
DE3060481D1 true DE3060481D1 (en) 1982-07-22

Family

ID=10502917

Family Applications (1)

Application Number Title Priority Date Filing Date
DE8080100447T Expired DE3060481D1 (en) 1979-02-02 1980-01-29 Anthracycline glycosides, methods for the production thereof and therapeutical compositions containing same

Country Status (6)

Country Link
US (1) US4254110A (de)
EP (1) EP0014425B1 (de)
JP (1) JPS55133370A (de)
AT (1) ATE1150T1 (de)
DE (1) DE3060481D1 (de)
DK (1) DK45080A (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4314999A (en) * 1978-07-31 1982-02-09 Proter S.P.A. N-Acyl derivatives of glucosamine having antitumor chemotherapeutic acitivity
ATE15375T1 (de) * 1980-11-01 1985-09-15 Erba Farmitalia Anthracyclin-glycoside, zwischenprodukte, verfahren zu beider herstellung und arzneimittel.
GB2196626B (en) * 1986-10-15 1990-09-19 Erba Farmitalia Antitumor anthracycline glycosides, their preparation, intermediates thereof, and compositions and use therefor
FR2660561B1 (fr) * 1990-04-06 1994-05-13 Technomed International Sonde rectale.
US7388083B2 (en) * 2005-03-07 2008-06-17 Solux Corporation Epimerization of 4′-C bond and modification of 14-CH3-(CO)-fragment in anthracyclin antibiotics
US8802830B2 (en) 2005-12-20 2014-08-12 Solux Corporation Synthesis of epirubicin from 13-dihydrodaunorubicine
US8357785B2 (en) 2008-01-08 2013-01-22 Solux Corporation Method of aralkylation of 4′-hydroxyl group of anthracylins

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL130756C (de) * 1964-03-02
GB1550879A (en) * 1976-12-22 1979-08-22 Farmaceutici Italia Antitumour glycosides
GB1542920A (en) * 1976-12-22 1979-03-28 Farmaceutici Italia Antitumour glycosides
US4181795A (en) * 1978-05-22 1980-01-01 Purdue Research Foundation Daunosamine synthesis

Also Published As

Publication number Publication date
ATE1150T1 (de) 1982-06-15
EP0014425A1 (de) 1980-08-20
EP0014425B1 (de) 1982-06-02
US4254110A (en) 1981-03-03
DK45080A (da) 1980-08-03
JPS6321671B2 (de) 1988-05-09
JPS55133370A (en) 1980-10-17

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Legal Events

Date Code Title Description
8339 Ceased/non-payment of the annual fee