DE2436149C3 - Verfahren zur Herstellung von 5-Fluorcytosin - Google Patents
Verfahren zur Herstellung von 5-FluorcytosinInfo
- Publication number
- DE2436149C3 DE2436149C3 DE19742436149 DE2436149A DE2436149C3 DE 2436149 C3 DE2436149 C3 DE 2436149C3 DE 19742436149 DE19742436149 DE 19742436149 DE 2436149 A DE2436149 A DE 2436149A DE 2436149 C3 DE2436149 C3 DE 2436149C3
- Authority
- DE
- Germany
- Prior art keywords
- ethoxy
- water
- fluoro
- fluorocytosine
- fluoropyrimidine
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/32—One oxygen, sulfur or nitrogen atom
- C07D239/34—One oxygen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Saccharide Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH1289573A CH579057A5 (ja) | 1973-09-07 | 1973-09-07 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| DE2436149A1 DE2436149A1 (de) | 1975-03-27 |
| DE2436149B2 DE2436149B2 (de) | 1978-10-12 |
| DE2436149C3 true DE2436149C3 (de) | 1979-06-07 |
Family
ID=4387383
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE19742436149 Expired DE2436149C3 (de) | 1973-09-07 | 1974-07-26 | Verfahren zur Herstellung von 5-Fluorcytosin |
Country Status (10)
| Country | Link |
|---|---|
| JP (1) | JPS5050386A (ja) |
| AT (1) | AT331259B (ja) |
| BE (1) | BE819606A (ja) |
| CH (1) | CH579057A5 (ja) |
| DD (1) | DD114263A5 (ja) |
| DE (1) | DE2436149C3 (ja) |
| FR (1) | FR2247457B1 (ja) |
| GB (1) | GB1461184A (ja) |
| NL (1) | NL7410730A (ja) |
| SU (1) | SU578873A3 (ja) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4080455A (en) * | 1975-12-16 | 1978-03-21 | Taisho Pharmaceutical Company Limited | 5-Fluoropyrimidin-4-one compositions |
| PL2562162T3 (pl) * | 2008-01-22 | 2016-01-29 | Dow Agrosciences Llc | Pochodne N-cyjano-4-amino-5-fluoropirymidyny jako fungicydy |
| UA112284C2 (uk) | 2009-08-07 | 2016-08-25 | ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі | Похідні 5-фторпіримідинону |
| UA107671C2 (en) | 2009-08-07 | 2015-02-10 | Dow Agrosciences Llc | N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives |
| UA106889C2 (uk) | 2009-08-07 | 2014-10-27 | ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі | Похідні n1-ацил-5-фторпіримідинону |
| NZ597644A (en) | 2009-08-07 | 2014-05-30 | Dow Agrosciences Llc | N1-sulfonyl-5-fluoropyrimidinone derivatives |
| MX2012007954A (es) | 2010-01-07 | 2012-08-03 | Dow Agrosciences Llc | Tiazolo [5, 4-d] pirimidinas y su uso como agroquimicos. |
| KR102012992B1 (ko) | 2011-08-17 | 2019-08-21 | 아다마 마켓심 리미티드 | 5-플루오로-4-이미노-3-(치환된)-3,4-디히드로피리미딘-2-(1ｈ)-온 유도체 |
| US9321734B2 (en) | 2012-12-28 | 2016-04-26 | Dow Agrosciences Llc | N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2H)-carboxamide derivatives |
| AU2013370470B2 (en) | 2012-12-28 | 2018-05-10 | Adama Makhteshim Ltd. | 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1H)-one derivatives |
| JP6324994B2 (ja) | 2012-12-28 | 2018-05-16 | アダマ・マクテシム・リミテッド | Ｎ−（置換）−５−フルオロ−４−イミノ−３−メチル−２−オキソ−３，４−ジヒドロピリミジン−１（２ｈ）−カルボキシレート誘導体 |
| WO2014105845A1 (en) | 2012-12-31 | 2014-07-03 | Dow Agrosciences Llc | 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides |
| JP6609257B2 (ja) | 2013-12-31 | 2019-11-20 | アダマ・マクテシム・リミテッド | 真菌防除のための相乗的殺真菌性混合物および組成物 |
| SG11201605372QA (en) | 2013-12-31 | 2016-08-30 | Adama Makhteshim Ltd | 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1- (arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation |
-
1973
- 1973-09-07 CH CH1289573A patent/CH579057A5/xx not_active IP Right Cessation
-
1974
- 1974-07-26 DE DE19742436149 patent/DE2436149C3/de not_active Expired
- 1974-08-09 NL NL7410730A patent/NL7410730A/xx unknown
- 1974-09-05 FR FR7430135A patent/FR2247457B1/fr not_active Expired
- 1974-09-05 DD DD18093474A patent/DD114263A5/xx unknown
- 1974-09-05 JP JP10142674A patent/JPS5050386A/ja active Pending
- 1974-09-06 BE BE148257A patent/BE819606A/xx not_active IP Right Cessation
- 1974-09-06 GB GB3901574A patent/GB1461184A/en not_active Expired
- 1974-09-06 SU SU7402057486A patent/SU578873A3/ru active
- 1974-09-06 AT AT720874A patent/AT331259B/de not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| CH579057A5 (ja) | 1976-08-31 |
| ATA720874A (de) | 1975-11-15 |
| BE819606A (fr) | 1975-03-06 |
| DE2436149A1 (de) | 1975-03-27 |
| JPS5050386A (ja) | 1975-05-06 |
| FR2247457A1 (ja) | 1975-05-09 |
| DD114263A5 (ja) | 1975-07-20 |
| SU578873A3 (ru) | 1977-10-30 |
| DE2436149B2 (de) | 1978-10-12 |
| GB1461184A (en) | 1977-01-13 |
| FR2247457B1 (ja) | 1976-10-22 |
| NL7410730A (nl) | 1975-03-11 |
| AT331259B (de) | 1976-08-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| C3 | Grant after two publication steps (3rd publication) | ||
| 8327 | Change in the person/name/address of the patent owner |
Owner name: F. HOFFMANN-LA ROCHE AG, BASEL, CH |
|
| 8328 | Change in the person/name/address of the agent |
Free format text: LEDERER, F., DIPL.-CHEM. DR., 8000 MUENCHEN RIEDERER FRHR. VON PAAR ZU SCHOENAU, A., DIPL.-ING., PAT.-ANWAELTE, 8300 LANDSHUT |