DE2359076C2 - 2β,16β-Dipiperidino-5α-androstane und Verfahren zu ihrer Herstellung - Google Patents
2β,16β-Dipiperidino-5α-androstane und Verfahren zu ihrer HerstellungInfo
- Publication number
- DE2359076C2 DE2359076C2 DE2359076A DE2359076A DE2359076C2 DE 2359076 C2 DE2359076 C2 DE 2359076C2 DE 2359076 A DE2359076 A DE 2359076A DE 2359076 A DE2359076 A DE 2359076A DE 2359076 C2 DE2359076 C2 DE 2359076C2
- Authority
- DE
- Germany
- Prior art keywords
- dipiperidino
- androstane
- piperidino
- ether
- added
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0005—Oxygen-containing hetero ring
- C07J71/001—Oxiranes
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB5519172A GB1454749A (en) | 1972-11-29 | 1972-11-29 | 2beta, 16beta-diamino-androstanes and their preparation |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DE2359076A1 DE2359076A1 (de) | 1974-06-06 |
| DE2359076C2 true DE2359076C2 (de) | 1983-12-08 |
Family
ID=10473231
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE2359076A Expired DE2359076C2 (de) | 1972-11-29 | 1973-11-27 | 2β,16β-Dipiperidino-5α-androstane und Verfahren zu ihrer Herstellung |
Country Status (18)
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HU172521B (hu) * | 1975-08-01 | 1978-09-28 | Richter Gedeon Vegyeszet | Sposob poluchenija novykh proizvodnykh triamino-androstana i chetvertichnykh solejj |
| ATE921T1 (de) * | 1978-09-05 | 1982-05-15 | Akzo N.V. | Saeureadditionssalze von 2-beta, 16-beta-bis-piperidino-an drostan-16-beta-monoquaternaeren ammoniumderivaten und diese enthaltende pharmazeutische zusammensetzungen. |
| IE50675B1 (en) * | 1979-12-12 | 1986-06-11 | Akzo Nv | Bis-and mono-quaternary ammonium derivatives of 2beta,16beta-dipiperidino-5alpha-androstanes,processes for their preparation and pharmaceutical preparations |
| IE53463B1 (en) * | 1981-06-15 | 1988-11-23 | Akzo Nv | Mono-and bisquaternary ammonium derivatives of 2 beta,16 beta-d-amino-5 alpha-androstane derivatives and pharmaceutical preparations containing same |
| GB8708886D0 (en) * | 1987-04-14 | 1987-05-20 | Akzo Nv | 2beta-morpholino-androstane derivatives |
| CZ300694A3 (en) * | 1993-12-02 | 1996-05-15 | Akzo Nobel Nv | Substituted 2beta-morpholinandrostane derivatives, process of their preparation, their use for preparing pharmaceutical preparations and pharmaceutical compositions containing thereof |
| US5767112A (en) * | 1994-10-21 | 1998-06-16 | Poli Industria Chimica, S.P.A. | Muscle relaxant pharmaceutical compositions |
| IT1277700B1 (it) * | 1995-12-22 | 1997-11-11 | Poli Ind Chimica Spa | Processo di preparazione di 2-beta, 16-beta-diamino 3-alfa, 17-beta- diacilossi 5-alfaandrostani, bloccanti neuromuscolari a struttura |
| AU2003205244B2 (en) * | 2002-01-18 | 2009-01-08 | Regents Of The University Of Minnesota | Triterpene quaternary salts as biologically active surfactants |
| WO2012147090A1 (en) * | 2011-04-26 | 2012-11-01 | Neon Laboratories Ltd. | Novel process for quaternization of (2p,3a,5a,16p,17p)-2,16-bispiperidino-3,17-diacetoxy-5-androstane |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1138605A (en) * | 1965-02-19 | 1969-01-01 | Organon Labor Ltd | Improvements in or relating to new 2-ß,16-ß-diamino-androstanes |
| FR1468539A (fr) * | 1965-02-19 | 1967-02-03 | Organon Labor Ltd | Nouveaux 2beta, 16beta-diamino-androstanes et procédé pour leur préparation |
-
1972
- 1972-11-29 GB GB5519172A patent/GB1454749A/en not_active Expired
-
1973
- 1973-11-15 ZA ZA738759A patent/ZA738759B/xx unknown
- 1973-11-15 IE IE2064/73A patent/IE38513B1/xx unknown
- 1973-11-22 FI FI733607A patent/FI52349C/fi active
- 1973-11-26 PH PH7315257A patent/PH12359A/en unknown
- 1973-11-26 US US419001A patent/US3872091A/en not_active Expired - Lifetime
- 1973-11-26 FR FR7342036A patent/FR2207724B1/fr not_active Expired
- 1973-11-27 CA CA186,754A patent/CA1018515A/en not_active Expired
- 1973-11-27 DE DE2359076A patent/DE2359076C2/de not_active Expired
- 1973-11-28 ES ES420922A patent/ES420922A1/es not_active Expired
- 1973-11-28 DK DK642473*A patent/DK132500C/da not_active IP Right Cessation
- 1973-11-28 SE SE7316055A patent/SE395460B/xx unknown
- 1973-11-28 NL NL7316237A patent/NL7316237A/xx not_active Application Discontinuation
- 1973-11-28 CH CH1670973A patent/CH605506A5/xx not_active IP Right Cessation
- 1973-11-28 JP JP13333873A patent/JPS546557B2/ja not_active Expired
- 1973-11-28 NO NO4543/73A patent/NO139088C/no unknown
- 1973-11-29 BE BE138322A patent/BE807988A/xx not_active IP Right Cessation
- 1973-11-29 HU HUAO376A patent/HU168724B/hu unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JPS4993353A (US08088918-20120103-C00476.png) | 1974-09-05 |
| HU168724B (US08088918-20120103-C00476.png) | 1976-07-28 |
| FI52349C (fi) | 1977-08-10 |
| ZA738759B (en) | 1974-10-30 |
| AU6286273A (en) | 1975-05-29 |
| FR2207724A1 (US08088918-20120103-C00476.png) | 1974-06-21 |
| BE807988A (fr) | 1974-05-29 |
| IE38513L (en) | 1974-05-20 |
| SE395460B (sv) | 1977-08-15 |
| DK132500C (da) | 1976-05-17 |
| FR2207724B1 (US08088918-20120103-C00476.png) | 1977-09-02 |
| CA1018515A (en) | 1977-10-04 |
| FI52349B (US08088918-20120103-C00476.png) | 1977-05-02 |
| NO139088B (no) | 1978-09-25 |
| CH605506A5 (US08088918-20120103-C00476.png) | 1978-09-29 |
| NL7316237A (US08088918-20120103-C00476.png) | 1974-05-31 |
| ES420922A1 (es) | 1976-04-01 |
| DE2359076A1 (de) | 1974-06-06 |
| PH12359A (en) | 1979-01-29 |
| JPS546557B2 (US08088918-20120103-C00476.png) | 1979-03-29 |
| NO139088C (no) | 1979-01-03 |
| US3872091A (en) | 1975-03-18 |
| DK132500B (da) | 1975-12-15 |
| GB1454749A (en) | 1976-11-03 |
| IE38513B1 (en) | 1978-03-29 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DE2359076C2 (de) | 2β,16β-Dipiperidino-5α-androstane und Verfahren zu ihrer Herstellung | |
| DE1244777B (de) | Verfahren zur Herstellung von 7alpha-Methyl-16alpha-hydroxy-oestron bzw. -3, 16-diacetat | |
| DE1962757B2 (de) | Evomonosid-Derivate, Verfahren zu deren Herstellung sowie diese enthaltende Arzneimittel | |
| DE1568308B2 (de) | Verfahren zur herstellung von delta hoch 4,9,11-trienen der 19-nor- androstanreihe, 17-oxygenierte 3-oxo- 7 alpha-methyl-delta hoch 4,9,11-19 nor- androstatriene und diese enthaltende pharmazeutische praeparate sowie 3-oxo-7 alpha -methyl-delta hoch 5 (10), 9 (11) -19-nor- androstadiene | |
| CH640247A5 (de) | Steroid-spiro-oxazolidone und verfahren zu ihrer herstellung. | |
| DE1807585C3 (de) | 14,15beta-Epoxycardenolide, Verfahren zu deren Herstellung und diese enthaltende Mittel | |
| DE1947221A1 (de) | 3-Aza-19-hydroxy-3,19-cyclo-A-homosteroide und ein Verfahren zu deren Herstellung | |
| DE1288602B (de) | Verfahren zur Herstellung von Steroidverbindungen | |
| DE1568308C3 (de) | 10.09.65 Schweiz 12624-65 Verfahren zur Herstellung von Delta hoch 4,9,11-Trienen der 19-Norandrostanreihe, 17-oxygenierte 3-Oxo-7 alpha-methyl-Delta hoch 4,9,11-19 norandrostatriene und diese enthaltende pharmazeutische Präparate sowie 3-Oxo-7 alpha -methyl-Delta hoch 5 (10), 9 (11) -19-norandrostadiene | |
| DE1543005C3 (de) | 4-Alkyl-9beta, lOalpha-Delta hoch 4,6-bzw. -Delta hoch 1,4,6 -steroide der Androstanreihe und Verfahren zu deren Herstellung | |
| DE2138426A1 (de) | Neue Steroide und Verfahren zu ihrer Herstellung | |
| AT240540B (de) | Verfahren zur Herstellung von 4-Chlor-Δ<4>-3-ketosteroidverbindungen | |
| DE2438424C2 (de) | Verfahren zur Herstellung von Equilenin und Equileninderivaten | |
| AT275054B (de) | Verfahren zur Herstellung von neuen 9β,10α-Steroiden | |
| DE1468635C (de) | Verfahren zur Herstellung von 12 Acylaminosteroiden | |
| DE1443546C (de) | Verfahren zur Herstellung von 6 Methyl Delta hoch 14 steroiden der Pregnanreihe | |
| AT270893B (de) | Verfahren zur Herstellung von neuen 19-Alkenylsteroiden | |
| DE1443638A1 (de) | Neue 7 alpha-Methyl-androstene und ein Verfahren zu deren Herstellung | |
| DE1445807A1 (de) | Verfahren zur Herstellung von 2-Dehydroemetin | |
| DE1105412B (de) | Verfahren zur Herstellung von ?-3-Keto-6ª-methylsteroiden der Androstan- und Pregnanreihe | |
| DE1220415B (de) | Verfahren zur Herstellung von 19-niedrig-Alkylverbindungen der Androstanreihe | |
| DE1793344A1 (de) | 2-Halogen-18-methyl-1-androstene | |
| DE1094258B (de) | Verfahren zur Herstellung von fluorierten 16-Methylsteroiden | |
| DE1805338A1 (de) | 2,3-Epithio-5d-androst-6-en-steroide | |
| DE2304493A1 (de) | Cyclopenteno-chinolonderivate und verfahren zur herstellung derselben |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| OD | Request for examination | ||
| OD | Request for examination | ||
| D2 | Grant after examination | ||
| 8364 | No opposition during term of opposition | ||
| 8339 | Ceased/non-payment of the annual fee |