DE2211019C3 - Geschmacksverbessernde Formulierungen oraler Penicilline - Google Patents
Geschmacksverbessernde Formulierungen oraler PenicillineInfo
- Publication number
- DE2211019C3 DE2211019C3 DE2211019A DE2211019A DE2211019C3 DE 2211019 C3 DE2211019 C3 DE 2211019C3 DE 2211019 A DE2211019 A DE 2211019A DE 2211019 A DE2211019 A DE 2211019A DE 2211019 C3 DE2211019 C3 DE 2211019C3
- Authority
- DE
- Germany
- Prior art keywords
- parts
- taste
- mixed
- dry
- granules
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
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- 235000021096 natural sweeteners Nutrition 0.000 description 1
- QIQXTHQIDYTFRH-UHFFFAOYSA-N octadecanoic acid Chemical compound CCCCCCCCCCCCCCCCCC(O)=O QIQXTHQIDYTFRH-UHFFFAOYSA-N 0.000 description 1
- OQCDKBAXFALNLD-UHFFFAOYSA-N octadecanoic acid Natural products CCCCCCCC(C)CCCCCCCCC(O)=O OQCDKBAXFALNLD-UHFFFAOYSA-N 0.000 description 1
- 239000007968 orange flavor Substances 0.000 description 1
- 239000003531 protein hydrolysate Substances 0.000 description 1
- 229960001153 serine Drugs 0.000 description 1
- 210000002966 serum Anatomy 0.000 description 1
- 238000007873 sieving Methods 0.000 description 1
- WXMKPNITSTVMEF-UHFFFAOYSA-M sodium benzoate Chemical compound [Na+].[O-]C(=O)C1=CC=CC=C1 WXMKPNITSTVMEF-UHFFFAOYSA-M 0.000 description 1
- 235000010234 sodium benzoate Nutrition 0.000 description 1
- 239000004299 sodium benzoate Substances 0.000 description 1
- 235000019812 sodium carboxymethyl cellulose Nutrition 0.000 description 1
- 229920001027 sodium carboxymethylcellulose Polymers 0.000 description 1
- 239000011780 sodium chloride Substances 0.000 description 1
- 229940073490 sodium glutamate Drugs 0.000 description 1
- 239000008117 stearic acid Substances 0.000 description 1
- 229940124530 sulfonamide Drugs 0.000 description 1
- 150000003456 sulfonamides Chemical class 0.000 description 1
- 239000000454 talc Substances 0.000 description 1
- 229910052623 talc Inorganic materials 0.000 description 1
- 239000011975 tartaric acid Substances 0.000 description 1
- 235000002906 tartaric acid Nutrition 0.000 description 1
- 229960002898 threonine Drugs 0.000 description 1
- 238000001291 vacuum drying Methods 0.000 description 1
- 229940088594 vitamin Drugs 0.000 description 1
- 239000011782 vitamin Substances 0.000 description 1
- 235000019195 vitamin supplement Nutrition 0.000 description 1
- 230000008673 vomiting Effects 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/429—Thiazoles condensed with heterocyclic ring systems
- A61K31/43—Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
- A61K9/0007—Effervescent
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1617—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Biophysics (AREA)
- Zoology (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Molecular Biology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Priority Applications (15)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE2211019A DE2211019C3 (de) | 1972-03-08 | 1972-03-08 | Geschmacksverbessernde Formulierungen oraler Penicilline |
| US336478A US3872227A (en) | 1972-03-08 | 1973-02-28 | Formulation for oral administration of penicillins having improved taste properties |
| IL41686A IL41686A (en) | 1972-03-08 | 1973-03-05 | Taste-improving formulations of oral penicillins |
| HUBA2886A HU167988B (enExample) | 1972-03-08 | 1973-03-05 | |
| AT196073A AT326819B (de) | 1972-03-08 | 1973-03-06 | Verfahren zur herstellung geschmackverbessernder formulierungen von phenoxymethylpenicillin, alpha-phenoxy-n-propylpenicillin und alpha-amino-benzylpenicillin bzw. von deren salzen |
| AU52954/73A AU482786B2 (en) | 1973-03-06 | Taste-improving formulations of oral penicillins | |
| NL7303207A NL7303207A (enExample) | 1972-03-08 | 1973-03-07 | |
| IE367/73A IE37378B1 (en) | 1972-03-08 | 1973-03-07 | Taste-improving formulations of oral penicillins |
| DK125173A DK132738C (da) | 1972-03-08 | 1973-03-07 | Fremgangsmade til fremstilling af orale penicillinpreparater med forbedret smag |
| GB1096873A GB1388358A (en) | 1972-03-08 | 1973-03-07 | Taste-improving formulations of oral penicillins |
| ES412387A ES412387A1 (es) | 1972-03-08 | 1973-03-07 | Procedimiento para la obtencion de formulaciones mejoradas del sabor de penicilinas orales. |
| ZA731589A ZA731589B (en) | 1972-03-08 | 1973-03-07 | Taste-improving formulations of oral penicillins |
| JP48026247A JPS4899317A (enExample) | 1972-03-08 | 1973-03-07 | |
| BE128513A BE796446A (fr) | 1972-03-08 | 1973-03-08 | Nouvelles formulations de penicillines orales de gout ameliore |
| FR7308349A FR2181804B1 (enExample) | 1972-03-08 | 1973-03-08 |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE2211019A DE2211019C3 (de) | 1972-03-08 | 1972-03-08 | Geschmacksverbessernde Formulierungen oraler Penicilline |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| DE2211019A1 DE2211019A1 (de) | 1973-09-13 |
| DE2211019B2 DE2211019B2 (de) | 1979-12-20 |
| DE2211019C3 true DE2211019C3 (de) | 1980-08-28 |
Family
ID=5838215
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE2211019A Expired DE2211019C3 (de) | 1972-03-08 | 1972-03-08 | Geschmacksverbessernde Formulierungen oraler Penicilline |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US3872227A (enExample) |
| JP (1) | JPS4899317A (enExample) |
| AT (1) | AT326819B (enExample) |
| BE (1) | BE796446A (enExample) |
| DE (1) | DE2211019C3 (enExample) |
| DK (1) | DK132738C (enExample) |
| ES (1) | ES412387A1 (enExample) |
| FR (1) | FR2181804B1 (enExample) |
| GB (1) | GB1388358A (enExample) |
| HU (1) | HU167988B (enExample) |
| IE (1) | IE37378B1 (enExample) |
| IL (1) | IL41686A (enExample) |
| NL (1) | NL7303207A (enExample) |
| ZA (1) | ZA731589B (enExample) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2832009A1 (de) * | 1978-07-20 | 1980-01-31 | Deutsches Krebsforsch | Verwendung von sarkosin und sarkosinderivaten ls tumorhemmende wirksubstanzen |
| IT1183574B (it) * | 1985-05-08 | 1987-10-22 | Eurand Spa | Metodo per ottenere una sospensione estemporanea omogenea di microcapsule |
| US5670170A (en) * | 1990-04-27 | 1997-09-23 | Beecham Group P.L.C. | Pharamaceutical formulation |
| US5631038A (en) * | 1990-06-01 | 1997-05-20 | Bioresearch, Inc. | Specific eatable taste modifiers |
| US5637618A (en) * | 1990-06-01 | 1997-06-10 | Bioresearch, Inc. | Specific eatable taste modifiers |
| HUT68764A (en) * | 1991-11-27 | 1995-07-28 | Bioresearch Inc | Eatable taste modifiers |
| US5639475A (en) * | 1995-02-03 | 1997-06-17 | Eurand America, Incorporated | Effervescent microcapsules |
| US5622723A (en) * | 1995-02-03 | 1997-04-22 | Eurand America, Incorporated | Procedure for encapsulating chlorpheniramine |
| US7504376B2 (en) * | 1996-08-12 | 2009-03-17 | Natural Alternatives International | Methods and compositions for increasing the anaerobic working capacity in tissues |
| CH690817A5 (de) * | 1996-09-03 | 2001-01-31 | Flachsmann Ag Emil | Verfahren zur Herstellung eines stabilen, homogenen, von Folgeprodukten freien oder nahezu freien Extraktes. |
| ATE445335T1 (de) | 1998-12-23 | 2009-10-15 | Sinai School Medicine | Hemmstoffe zur unterdrückung des bitteren geschmacks |
| EP1424997B1 (en) * | 2001-09-14 | 2007-11-21 | SCOLR, Inc. | Amino acid modulated extended release dosage form |
| JP2006052169A (ja) * | 2004-08-12 | 2006-02-23 | Wakoudou Kk | ゾル状又はゲル状の服薬補助食品 |
| US7455872B2 (en) * | 2005-06-20 | 2008-11-25 | Redpoint Bio Corporation | Compositions and methods for producing a salty taste in foods or beverages |
| US7452563B2 (en) * | 2005-06-20 | 2008-11-18 | Redpoint Bio Corporation | Compositions and methods for producing flavored seasonings that contain reduced quantities of common salt |
| FR2963239B1 (fr) * | 2010-08-02 | 2013-03-08 | Vetalis | Formes galeniques effervescentes solides pour animaux |
| RU2676327C2 (ru) | 2013-07-18 | 2018-12-28 | Сандоз Аг | Порошковые смеси для составов сухого сиропа антибиотика |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR1477464A (fr) * | 1964-12-03 | 1967-04-21 | Bayer Ag | Procédé pour diminuer les altérations de goût et d'odeur des pénicillines |
| GB1291282A (en) * | 1969-03-20 | 1972-10-04 | Pfizer Ltd | Improvements in pharmaceutical compositions |
-
1972
- 1972-03-08 DE DE2211019A patent/DE2211019C3/de not_active Expired
-
1973
- 1973-02-28 US US336478A patent/US3872227A/en not_active Expired - Lifetime
- 1973-03-05 HU HUBA2886A patent/HU167988B/hu unknown
- 1973-03-05 IL IL41686A patent/IL41686A/en unknown
- 1973-03-06 AT AT196073A patent/AT326819B/de not_active IP Right Cessation
- 1973-03-07 ZA ZA731589A patent/ZA731589B/xx unknown
- 1973-03-07 DK DK125173A patent/DK132738C/da active
- 1973-03-07 IE IE367/73A patent/IE37378B1/xx unknown
- 1973-03-07 NL NL7303207A patent/NL7303207A/xx not_active Application Discontinuation
- 1973-03-07 ES ES412387A patent/ES412387A1/es not_active Expired
- 1973-03-07 JP JP48026247A patent/JPS4899317A/ja active Pending
- 1973-03-07 GB GB1096873A patent/GB1388358A/en not_active Expired
- 1973-03-08 FR FR7308349A patent/FR2181804B1/fr not_active Expired
- 1973-03-08 BE BE128513A patent/BE796446A/xx unknown
Non-Patent Citations (2)
| Title |
|---|
| Helwig B. Moderne Artzneimittel, Stuttgart 1976, S. 27. * |
| Ritschel W. A. Die Tablette, Aulendorf 1966, S. 141 * |
Also Published As
| Publication number | Publication date |
|---|---|
| BE796446A (fr) | 1973-09-10 |
| IE37378L (en) | 1973-09-08 |
| FR2181804A1 (enExample) | 1973-12-07 |
| IE37378B1 (en) | 1977-07-06 |
| AT326819B (de) | 1975-12-29 |
| IL41686A0 (en) | 1973-05-31 |
| DK132738C (da) | 1976-07-05 |
| AU5295473A (en) | 1974-09-12 |
| ZA731589B (en) | 1973-11-28 |
| NL7303207A (enExample) | 1973-09-11 |
| ATA196073A (de) | 1975-03-15 |
| JPS4899317A (enExample) | 1973-12-15 |
| DE2211019A1 (de) | 1973-09-13 |
| ES412387A1 (es) | 1976-01-16 |
| HU167988B (enExample) | 1976-02-28 |
| DK132738B (da) | 1976-02-02 |
| GB1388358A (en) | 1975-03-26 |
| DE2211019B2 (de) | 1979-12-20 |
| FR2181804B1 (enExample) | 1976-10-22 |
| US3872227A (en) | 1975-03-18 |
| IL41686A (en) | 1976-10-31 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| C3 | Grant after two publication steps (3rd publication) | ||
| 8339 | Ceased/non-payment of the annual fee |