DD134228A5 - Verfahren zur herstellung von spirooxazolidindionen - Google Patents

Verfahren zur herstellung von spirooxazolidindionen

Info

Publication number
DD134228A5
DD134228A5 DD77202424A DD20242477A DD134228A5 DD 134228 A5 DD134228 A5 DD 134228A5 DD 77202424 A DD77202424 A DD 77202424A DD 20242477 A DD20242477 A DD 20242477A DD 134228 A5 DD134228 A5 DD 134228A5
Authority
DD
German Democratic Republic
Prior art keywords
spirooxazolide
indions
producing
spirooxazolide indions
producing spirooxazolide
Prior art date
Application number
DD77202424A
Other languages
German (de)
English (en)
Inventor
Jean C Miller
Gerald E Gutowski
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of DD134228A5 publication Critical patent/DD134228A5/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • C07D519/04Dimeric indole alkaloids, e.g. vincaleucoblastine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
DD77202424A 1976-12-06 1977-12-06 Verfahren zur herstellung von spirooxazolidindionen DD134228A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/747,575 US4096148A (en) 1976-12-06 1976-12-06 Oxazolidinedione derivatives of Vinca alkaloids

Publications (1)

Publication Number Publication Date
DD134228A5 true DD134228A5 (de) 1979-02-14

Family

ID=25005690

Family Applications (2)

Application Number Title Priority Date Filing Date
DD77202423A DD134227A5 (de) 1976-12-06 1977-12-06 Verfahren zur herstellung von dimeren indoldihydroindoldionen
DD77202424A DD134228A5 (de) 1976-12-06 1977-12-06 Verfahren zur herstellung von spirooxazolidindionen

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DD77202423A DD134227A5 (de) 1976-12-06 1977-12-06 Verfahren zur herstellung von dimeren indoldihydroindoldionen

Country Status (31)

Country Link
US (1) US4096148A (xx)
JP (1) JPS5371100A (xx)
AR (1) AR218467A1 (xx)
AT (2) AT353987B (xx)
AU (1) AU513936B2 (xx)
BE (1) BE861417A (xx)
BG (1) BG33436A3 (xx)
CA (2) CA1082180A (xx)
CH (2) CH634076A5 (xx)
CS (2) CS195344B2 (xx)
DD (2) DD134227A5 (xx)
DE (1) DE2753791A1 (xx)
DK (2) DK144916C (xx)
ES (2) ES464765A1 (xx)
FR (1) FR2372839A1 (xx)
GB (1) GB1590649A (xx)
GR (2) GR67243B (xx)
HK (1) HK57281A (xx)
HU (2) HU180725B (xx)
IE (1) IE46105B1 (xx)
IL (1) IL53506A (xx)
MX (1) MX4326E (xx)
MY (1) MY8200176A (xx)
NL (1) NL7713336A (xx)
NZ (1) NZ185818A (xx)
PL (2) PL106522B1 (xx)
PT (2) PT67343B (xx)
RO (2) RO74137A (xx)
SE (2) SE435930B (xx)
SU (2) SU843753A3 (xx)
ZA (1) ZA777237B (xx)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU181874B (en) * 1977-08-08 1983-11-28 Lilly Co Eli Process for preparing amides of deacetyl-leurosine and deacetyl-leuroformine
US4357334A (en) * 1980-03-20 1982-11-02 Eli Lilly And Company Use of VLB 3-(2-chloroethyl) carboxamide in treating neoplasms
US4362664A (en) * 1980-12-29 1982-12-07 Eli Lilly And Company Vinblastine oxazolidinedione disulfides and related compounds
DE3484691D1 (de) * 1983-04-29 1991-07-18 Omnichem Sa Konjugierte vinblastin-verbindungen und ihre derivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische zusammensetzungen.
HUT76925A (hu) * 1995-04-04 1998-01-28 MTA Enzimológiai Intézet Bisz-indol-származékok, eljárás előállításukra és az azokat tartalmazó gyógyszerkészítmények
EP2266607A3 (en) 1999-10-01 2011-04-20 Immunogen, Inc. Immunoconjugates for treating cancer

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL125835C (xx) * 1960-05-24
HU165986B (xx) * 1973-02-16 1974-12-28
AR204004A1 (es) * 1973-04-02 1975-11-12 Lilly Co Eli Procedimientos para preparar derivados de vinblastina leurosidina y leurocristina
US4012390A (en) * 1974-10-16 1977-03-15 Eli Lilly And Company Vinblastinoic acid

Also Published As

Publication number Publication date
SE436036B (sv) 1984-11-05
NZ185818A (en) 1979-12-11
DD134227A5 (de) 1979-02-14
DK541077A (da) 1978-06-07
PT67343B (en) 1979-04-26
CH634076A5 (de) 1983-01-14
DK145001B (da) 1982-07-26
ATA868877A (de) 1979-05-15
RO74137A (ro) 1981-08-30
DE2753791A1 (de) 1978-06-08
SU843753A3 (ru) 1981-06-30
US4096148A (en) 1978-06-20
SE7713587L (sv) 1978-06-07
SE7713586L (sv) 1978-06-07
DK145001C (da) 1982-12-27
PL106522B1 (pl) 1979-12-31
HU180724B (en) 1983-04-29
DK144916C (da) 1982-12-06
MX4326E (es) 1982-03-24
JPS5371100A (en) 1978-06-24
ZA777237B (en) 1979-07-25
IE46105B1 (en) 1983-02-23
IL53506A (en) 1981-09-13
DK541177A (da) 1978-06-07
GR67243B (xx) 1981-06-25
AU513936B2 (en) 1981-01-15
AR218467A1 (es) 1980-06-13
AT353987B (de) 1979-12-10
CS195344B2 (en) 1980-01-31
ATA868777A (de) 1980-08-15
ES464764A1 (es) 1979-01-01
PT67343A (en) 1977-12-01
NL7713336A (nl) 1978-06-08
CS195343B2 (en) 1980-01-31
SE435930B (sv) 1984-10-29
FR2372839A1 (fr) 1978-06-30
CH632516A5 (de) 1982-10-15
HU180725B (en) 1983-04-29
BG33436A3 (en) 1983-02-15
ES464765A1 (es) 1979-01-01
JPS625160B2 (xx) 1987-02-03
AT361638B (de) 1981-03-25
PL202659A1 (pl) 1978-12-04
HK57281A (en) 1981-11-27
FR2372839B1 (xx) 1981-11-06
CA1103664A (en) 1981-06-23
SU865127A3 (ru) 1981-09-15
IL53506A0 (en) 1978-03-10
GR67244B (xx) 1981-06-25
PL110671B1 (en) 1980-07-31
AU3123077A (en) 1979-06-14
CA1082180A (en) 1980-07-22
DK144916B (da) 1982-07-05
MY8200176A (en) 1982-12-31
GB1590649A (en) 1981-06-03
PT67342B (en) 1979-04-26
RO75391A (ro) 1980-11-30
DE2753791C2 (xx) 1990-08-02
IE46105L (en) 1978-06-06
PL202660A1 (pl) 1978-08-28
PT67342A (en) 1977-12-01
BE861417A (fr) 1978-06-02

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