CZ172399A3 - Piperidinové deriváty, způsob výroby a farmaceutický prostředek - Google Patents
Piperidinové deriváty, způsob výroby a farmaceutický prostředek Download PDFInfo
- Publication number
- CZ172399A3 CZ172399A3 CZ991723A CZ172399A CZ172399A3 CZ 172399 A3 CZ172399 A3 CZ 172399A3 CZ 991723 A CZ991723 A CZ 991723A CZ 172399 A CZ172399 A CZ 172399A CZ 172399 A3 CZ172399 A3 CZ 172399A3
- Authority
- CZ
- Czechia
- Prior art keywords
- compound
- formula
- methyl
- thienyl
- pharmaceutically acceptable
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Psychiatry (AREA)
- Epidemiology (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP96203175 | 1996-11-14 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CZ172399A3 true CZ172399A3 (cs) | 1999-11-17 |
Family
ID=8224578
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CZ991723A CZ172399A3 (cs) | 1996-11-14 | 1997-11-12 | Piperidinové deriváty, způsob výroby a farmaceutický prostředek |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US6288085B1 (tr) |
| EP (1) | EP0941225A1 (tr) |
| JP (1) | JP2001508044A (tr) |
| KR (1) | KR20000053217A (tr) |
| CN (1) | CN1092655C (tr) |
| AR (1) | AR010289A1 (tr) |
| AU (1) | AU722224B2 (tr) |
| BR (1) | BR9713044A (tr) |
| CA (1) | CA2271832A1 (tr) |
| CZ (1) | CZ172399A3 (tr) |
| HU (1) | HUP9904526A3 (tr) |
| IL (1) | IL122072A (tr) |
| NO (1) | NO992302L (tr) |
| NZ (1) | NZ335631A (tr) |
| PL (1) | PL333323A1 (tr) |
| RU (1) | RU2183624C2 (tr) |
| TR (1) | TR199901385T2 (tr) |
| TW (1) | TW374085B (tr) |
| WO (1) | WO1998021206A1 (tr) |
| ZA (1) | ZA979781B (tr) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1999034800A1 (en) * | 1998-01-09 | 1999-07-15 | Akzo Nobel N.V. | Use of phenylthienylmethylene piperidine derivative in the manufacture of a medicament for the treatment of movement disorders |
| WO1999034802A1 (en) * | 1998-01-09 | 1999-07-15 | Akzo Nobel N.V. | Use of phenylthienylmethylene piperidine derivatives in the manufacture of a medicament for the treatment of depression |
| CN100384421C (zh) * | 2002-12-18 | 2008-04-30 | 拜尔农科股份公司 | N-(取代的芳基甲基)-4-(二取代的甲基)哌啶和吡啶 |
| US20060009491A1 (en) * | 2004-06-24 | 2006-01-12 | Incyte Corporation | Amido compounds and their use as pharmaceuticals |
| EA200700117A1 (ru) * | 2004-06-24 | 2007-06-29 | Инсайт Корпорейшн | N-замещенные пиперидины и их применение в качестве фармацевтических препаратов |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL88063C (tr) * | 1950-12-05 | |||
| GB1242169A (en) * | 1969-04-09 | 1971-08-11 | Ucb Sa | Piperidine derivatives |
| GB1320481A (en) * | 1971-01-11 | 1973-06-13 | Pfizer Ltd | Substituted gem-diaryl ethylene derivatives and therapeutic compositions thereof |
| CH587845A5 (en) * | 1973-07-17 | 1977-05-13 | Sandoz Ag | New piperidylidene-benzo-cyclohepta-thiophenes prodn. - by dehydrating corresp. alcohols, useful e.g. as neuroleptics and analgesics |
| US4073912A (en) * | 1976-10-12 | 1978-02-14 | Smithkline Corporation | Piperidylidene derivatives of benzo-fused xanthenes, thioxanthenes and dibenzoxepins and antipsychotic use thereof |
| US4485107A (en) * | 1982-11-01 | 1984-11-27 | Janssen Pharmaceutica N.V. | [[Bis(aryl)methylene]-1-piperidinyl]alkyl-pyrimidinones |
| US4797489A (en) * | 1987-12-02 | 1989-01-10 | American Home Products Corp. | Adamantyl- and fluorenyl-arylpiperazines and -arylpiperidines |
| GB8900382D0 (en) * | 1989-01-09 | 1989-03-08 | Janssen Pharmaceutica Nv | 2-aminopyrimidinone derivatives |
| EP0465254B1 (en) * | 1990-07-06 | 1996-11-13 | Yoshitomi Pharmaceutical Industries, Ltd. | Fused thiophene compounds and uses thereof |
| US5683998A (en) * | 1991-04-23 | 1997-11-04 | Toray Industries, Inc. | Tricyclic triazolo derivatives, processes for producing the same and the uses of the same |
-
1997
- 1997-10-30 IL IL12207297A patent/IL122072A/xx not_active IP Right Cessation
- 1997-10-30 ZA ZA9709781A patent/ZA979781B/xx unknown
- 1997-11-06 TW TW086116718A patent/TW374085B/zh active
- 1997-11-12 CA CA002271832A patent/CA2271832A1/en not_active Abandoned
- 1997-11-12 HU HU9904526A patent/HUP9904526A3/hu unknown
- 1997-11-12 RU RU99112513/04A patent/RU2183624C2/ru not_active IP Right Cessation
- 1997-11-12 JP JP52218698A patent/JP2001508044A/ja active Pending
- 1997-11-12 CZ CZ991723A patent/CZ172399A3/cs unknown
- 1997-11-12 EP EP97951893A patent/EP0941225A1/en not_active Withdrawn
- 1997-11-12 US US09/308,035 patent/US6288085B1/en not_active Expired - Fee Related
- 1997-11-12 KR KR1019990704185A patent/KR20000053217A/ko not_active Application Discontinuation
- 1997-11-12 TR TR1999/01385T patent/TR199901385T2/tr unknown
- 1997-11-12 BR BR9713044-3A patent/BR9713044A/pt not_active IP Right Cessation
- 1997-11-12 WO PCT/EP1997/006321 patent/WO1998021206A1/en not_active Application Discontinuation
- 1997-11-12 PL PL97333323A patent/PL333323A1/xx unknown
- 1997-11-12 CN CN97180646A patent/CN1092655C/zh not_active Expired - Fee Related
- 1997-11-12 AU AU55520/98A patent/AU722224B2/en not_active Ceased
- 1997-11-12 NZ NZ335631A patent/NZ335631A/xx unknown
- 1997-11-13 AR ARP970105310A patent/AR010289A1/es unknown
-
1999
- 1999-05-12 NO NO992302A patent/NO992302L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| PL333323A1 (en) | 1999-12-06 |
| IL122072A (en) | 2001-03-19 |
| CN1092655C (zh) | 2002-10-16 |
| AU5552098A (en) | 1998-06-03 |
| US6288085B1 (en) | 2001-09-11 |
| KR20000053217A (ko) | 2000-08-25 |
| BR9713044A (pt) | 2000-04-11 |
| ZA979781B (en) | 1998-06-08 |
| NO992302D0 (no) | 1999-05-12 |
| CN1240444A (zh) | 2000-01-05 |
| WO1998021206A1 (en) | 1998-05-22 |
| IL122072A0 (en) | 1998-03-10 |
| EP0941225A1 (en) | 1999-09-15 |
| HUP9904526A3 (en) | 2000-12-28 |
| HUP9904526A2 (hu) | 2000-11-28 |
| TW374085B (en) | 1999-11-11 |
| NO992302L (no) | 1999-05-14 |
| CA2271832A1 (en) | 1998-05-22 |
| TR199901385T2 (tr) | 1999-11-22 |
| NZ335631A (en) | 2000-10-27 |
| AR010289A1 (es) | 2000-06-07 |
| JP2001508044A (ja) | 2001-06-19 |
| AU722224B2 (en) | 2000-07-27 |
| RU2183624C2 (ru) | 2002-06-20 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PD00 | Pending as of 2000-06-30 in czech republic |